BAY60-6583 acts as a partial agonist at adenosine A2B receptors

Journal of Pharmacology and Experimental Therapeutics

Volumn 349, Issue 3, 2014, Pages 427-436

  Hinz, Sonja ^a   Lacher, Svenja K ^a   Seibt, Benjamin F ^a   Müller, Christa E ^a  

^a UNIVERSITY OF BONN   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE A2B RECEPTOR; ADENOSINE RECEPTOR STIMULATING AGENT; BAY 60 6583; CYCLIC AMP; UNCLASSIFIED DRUG; [2 [[6 AMINO 3,5 DICYANO 4 [4 (CYCLOPROPYLMETHOXY)PHENYL]PYRIDIN 2 YL]SULFANYL]ACETAMIDE];

ARTICLE; BINDING AFFINITY; BIOACCUMULATION; CALCIUM MOBILIZATION ASSAY; CONTROLLED STUDY; DRUG EFFICACY; DRUG POTENCY; DRUG PROTEIN BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; EMBRYO; HEK293 CELL LINE; HUMAN; HUMAN CELL; IN VITRO STUDY; JURKAT CELL LINE; LIGAND BINDING; PRIORITY JOURNAL; PROTEIN EXPRESSION;

ADENOSINE A2 RECEPTOR AGONISTS; AMINOPYRIDINES; ANIMALS; CHO CELLS; CRICETULUS; CYCLIC AMP; DRUG PARTIAL AGONISM; HEK293 CELLS; HUMANS; JURKAT CELLS; LIGANDS; PROTEIN BINDING; RECEPTOR, ADENOSINE A2B; TRANSFECTION;

EID: 84901236562     PISSN: 00223565     EISSN: 15210103     Source Type: Journal    
DOI: 10.1124/jpet.113.210849     Document Type: Article

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