Phenyl-substituted N6-phenyladenosines and N6-phenyl-5',-N- ethylcarboxamidoadenosines with high activity at human adenosine A(2B) receptors

Drug Development Research

Volumn 49, Issue 2, 2000, Pages 85-93

  De Zwart, Maarten ^a,b   De Groote, Miriam ^a   Van Der Klein, Pieter A M ^a   Van Dun, Stephanie ^a   Bronsing, Robert ^a   Von Frijtag Drabbe Künzel, Jacobien K ^a   Ijzerman, Ad P ^a  

^a LEIDEN UNIVERSITY   (Netherlands)

^b LEIDEN UNIVERSITY   (Netherlands)

Author keywords

Adenosine receptor subtypes; Cyclic AMP production at A(2B) receptors; NECA; Radioligand binding

Indexed keywords

ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE A2 RECEPTOR AGONIST; ADENOSINE A2B RECEPTOR;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CHO CELL; DRUG ACTIVITY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; NONHUMAN;

EID: 0033911982     PISSN: 02724391     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1098-2299(200002)49:2<85::AID-DDR2>3.0.CO;2-W     Document Type: Article

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