-
2
-
-
70450270900
-
-
C.H.J. Brown, S. Lain, C.H.S. Verma, A.R. Fersht, and D.P. Lane Nat. Rev. Cancer 9 2009 862
-
(2009)
Nat. Rev. Cancer
, vol.9
, pp. 862
-
-
Brown, C.H.J.1
Lain, S.2
Verma, C.H.S.3
Fersht, A.R.4
Lane, D.P.5
-
10
-
-
37549012975
-
-
P. Verhaeghe, N. Azas, M. Gasquet, S. Hutter, C. Ducros, M. Laget, S. Rault, P. Rathelot, and P. Vanelle Bioorg. Med. Chem. Lett. 18 2008 396
-
(2008)
Bioorg. Med. Chem. Lett.
, vol.18
, pp. 396
-
-
Verhaeghe, P.1
Azas, N.2
Gasquet, M.3
Hutter, S.4
Ducros, C.5
Laget, M.6
Rault, S.7
Rathelot, P.8
Vanelle, P.9
-
12
-
-
77949816697
-
-
R.A. Smits, M. Adami, E.P. Istyastono, O.P. Zuiderveld, C.M.E. van Dam, F.J.J. de Kanter, A. Jongejan, G. Coruzzi, R. Leurs, and I.J.P. de Esch J. Med. Chem. 53 2010 2390
-
(2010)
J. Med. Chem.
, vol.53
, pp. 2390
-
-
Smits, R.A.1
Adami, M.2
Istyastono, E.P.3
Zuiderveld, O.P.4
Van Dam, C.M.E.5
De Kanter, F.J.J.6
Jongejan, A.7
Coruzzi, G.8
Leurs, R.9
De Esch, I.J.P.10
-
15
-
-
33644856439
-
-
M.A.H. Ismail, S. Barker, D.A. Abau El Ella, K.A.M. Abouzid, R.A. Toubar, and M.H. Todd J. Med. Chem. 49 2006 1526
-
(2006)
J. Med. Chem.
, vol.49
, pp. 1526
-
-
Ismail, M.A.H.1
Barker, S.2
Abau El Ella, D.A.3
Abouzid, K.A.M.4
Toubar, R.A.5
Todd, M.H.6
-
16
-
-
34250859583
-
-
S. Kasibhatla, V. Baichwal, S.X. Cai, B. Roth, I. Skvortsva, S. Skvortsov, P. Lucas, N.M. English, N. Sirisoma, J. Drewe, A. Pervin, B. Tseng, R.O. Carlson, and C.M. Pleiman Cancer Res. 67 2007 5865
-
(2007)
Cancer Res.
, vol.67
, pp. 5865
-
-
Kasibhatla, S.1
Baichwal, V.2
Cai, S.X.3
Roth, B.4
Skvortsva, I.5
Skvortsov, S.6
Lucas, P.7
English, N.M.8
Sirisoma, N.9
Drewe, J.10
Pervin, A.11
Tseng, B.12
Carlson, R.O.13
Pleiman, C.M.14
-
18
-
-
80052375547
-
-
F. Liu, D.B. Lovejoy, A.A. Hassani, Y. He, J.M. Herold, X. Chen, C.M. Yates, S.V. Frye, P.J. Brown, J. Huang, M. Vedadi, C.H. Arrowsmith, and J. Jin J. Med. Chem. 54 2011 6139
-
(2011)
J. Med. Chem.
, vol.54
, pp. 6139
-
-
Liu, F.1
Lovejoy, D.B.2
Hassani, A.A.3
He, Y.4
Herold, J.M.5
Chen, X.6
Yates, C.M.7
Frye, S.V.8
Brown, P.J.9
Huang, J.10
Vedadi, M.11
Arrowsmith, C.H.12
Jin, J.13
-
19
-
-
77955553428
-
-
EI-Azab, A.S.; Al-Omar, M.A.; Abdel-Aziz, A.A.M.; Abdel-Aziz, N.I.; EI-Sayed, M.A.-A.; Aleisa, A.M.; Sayad-Ahmed, M.M.; Abdel-Hamide, S.G. Eur. J. Med. Chem. 2010, 45, 4188.
-
(2010)
Eur. J. Med. Chem.
, vol.45
, pp. 4188
-
-
Ei-Azab, A.S.1
Al-Omar, M.A.2
Abdel-Aziz, A.A.M.3
Abdel-Aziz, N.I.4
Ei-Sayed, A.M.-A.5
Aleisa, A.M.6
Sayad-Ahmed, M.M.7
Abdel-Hamide, S.G.8
-
21
-
-
41349085423
-
-
P.M. Chandrika, T. Yakaiah, A.R.R. Rao, B. Narsaiah, N.C. Reddy, V. Srindar, and J.V. Rao Eur. J. Med. Chem. 43 2008 846
-
(2008)
Eur. J. Med. Chem.
, vol.43
, pp. 846
-
-
Chandrika, P.M.1
Yakaiah, T.2
Rao, A.R.R.3
Narsaiah, B.4
Reddy, N.C.5
Srindar, V.6
Rao, J.V.7
-
22
-
-
64249139659
-
-
A.M. Al-Obaid, S.G.A. Abdel-Hamide, H.A. El-Kashef, A.A.-M. Abdel-Aziz, A.S. El-Azad, H.A. Al-Khamees, and H.I. El-Subbagh Eur. J. Med. Chem. 44 2009 2379
-
(2009)
Eur. J. Med. Chem.
, vol.44
, pp. 2379
-
-
Al-Obaid, A.M.1
Abdel-Hamide, S.G.A.2
El-Kashef, H.A.3
Abdel-Aziz, A.A.-M.4
El-Azad, A.S.5
Al-Khamees, H.A.6
El-Subbagh, H.I.7
-
23
-
-
71749092646
-
-
M. Li, A. Jung, U. Ganswindt, P. Marini, A. Friedl, P.T. Daniel, K. Lauber, V. Jendrossek, and C. Belka Biochem. Pharmacol. 79 2010 122
-
(2010)
Biochem. Pharmacol.
, vol.79
, pp. 122
-
-
Li, M.1
Jung, A.2
Ganswindt, U.3
Marini, P.4
Friedl, A.5
Daniel, P.T.6
Lauber, K.7
Jendrossek, V.8
Belka, C.9
-
24
-
-
65149091722
-
-
N. Sirisoma, A. Pervin, H. Zhang, S. Jiang, J.A. Willardsen, M.B. Anderson, G. Mather, C.M. Pleiman, S. Kasibhatla, B. Tseng, J. Drewe, and S.X. Cai J. Med. Chem. 52 2009 2341
-
(2009)
J. Med. Chem.
, vol.52
, pp. 2341
-
-
Sirisoma, N.1
Pervin, A.2
Zhang, H.3
Jiang, S.4
Willardsen, J.A.5
Anderson, M.B.6
Mather, G.7
Pleiman, C.M.8
Kasibhatla, S.9
Tseng, B.10
Drewe, J.11
Cai, S.X.12
-
25
-
-
77949486119
-
-
N. Sirisoma, A. Pervin, H. Zhang, S. Jiang, W.J. Adam, M.B. Anderson, G. Mather, C.M. Pleiman, S. Kasibhatla, B. Tseng, J. Drewe, and S.X. Cai Bioorg. Med. Chem. Lett. 20 2010 2330
-
(2010)
Bioorg. Med. Chem. Lett.
, vol.20
, pp. 2330
-
-
Sirisoma, N.1
Pervin, A.2
Zhang, H.3
Jiang, S.4
Adam, W.J.5
Anderson, M.B.6
Mather, G.7
Pleiman, C.M.8
Kasibhatla, S.9
Tseng, B.10
Drewe, J.11
Cai, S.X.12
-
26
-
-
79952486230
-
-
A. Garofalo, L. Goossens, A. Lemoine, S. Ravez, P. Six, M. Howsam, A. Farce, and P. Depreux Med. Chem. Commun. 2 2011 65
-
(2011)
Med. Chem. Commun.
, vol.2
, pp. 65
-
-
Garofalo, A.1
Goossens, L.2
Lemoine, A.3
Ravez, S.4
Six, P.5
Howsam, M.6
Farce, A.7
Depreux, P.8
-
28
-
-
79957802327
-
-
R.D. Li, X. Zhang, Q.Y. Li, Z.M. Ge, and R.T. Li Bioorg. Med. Chem. Lett. 21 2011 3637
-
(2011)
Bioorg. Med. Chem. Lett.
, vol.21
, pp. 3637
-
-
Li, R.D.1
Zhang, X.2
Li, Q.Y.3
Ge, Z.M.4
Li, R.T.5
-
29
-
-
79952801118
-
-
O. Cruz-López, A. Conejo-García, M.C. Núñez, M. Kimatrai, M.E. García-Rubiño, F. Morales, V. Gómez-Pérez, and J.M. Campos Curr. Med. Chem. 18 2011 943
-
(2011)
Curr. Med. Chem.
, vol.18
, pp. 943
-
-
Cruz-López, O.1
Conejo-García, A.2
Núñez, M.C.3
Kimatrai, M.4
García-Rubiño, M.E.5
Morales, F.6
Gómez-Pérez, V.7
Campos, J.M.8
-
30
-
-
49449111557
-
-
G.M. Chinigo, M. Paige, S. Grindrod, E. Hamel, S. Dakshanamurthy, M. Chruszcz, W. Minor, and M.L. Brown J. Med. Chem. 51 2008 4620
-
(2008)
J. Med. Chem.
, vol.51
, pp. 4620
-
-
Chinigo, G.M.1
Paige, M.2
Grindrod, S.3
Hamel, E.4
Dakshanamurthy, S.5
Chruszcz, M.6
Minor, W.7
Brown, M.L.8
-
31
-
-
60349113216
-
-
T. Sardon, T. Cottin, J. Xu, A. Giannis, and I. Vernos ChemBiolChem 10 2009 464
-
(2009)
ChemBiolChem
, vol.10
, pp. 464
-
-
Sardon, T.1
Cottin, T.2
Xu, J.3
Giannis, A.4
Vernos, I.5
-
32
-
-
66349114286
-
-
D. Bebbington, H. Binch, J.-D. Charrier, S. Everitt, D. Fraysse, J. Golec, D. Kay, R. Knegtel, C. Mak, F. Mazzei, A. Miller, M. Mortimore, M. O'Donnell, S. Patel, F. Pierard, J. Pinder, J. Pollard, S. Ramaya, D. Robinson, A. Rutherford, J. Studley, and J. Westcott Bioorg. Med. Chem. Lett. 19 2009 3586
-
(2009)
Bioorg. Med. Chem. Lett.
, vol.19
, pp. 3586
-
-
Bebbington, D.1
Binch, H.2
Charrier, J.-D.3
Everitt, S.4
Fraysse, D.5
Golec, J.6
Kay, D.7
Knegtel, R.8
Mak, C.9
Mazzei, F.10
Miller, A.11
Mortimore, M.12
O'Donnell, M.13
Patel, S.14
Pierard, F.15
Pinder, J.16
Pollard, J.17
Ramaya, S.18
Robinson, D.19
Rutherford, A.20
Studley, J.21
Westcott, J.22
more..
-
33
-
-
77955555432
-
-
S.L. Cao, Y. Wang, L. Zhu, J. Liao, Y.W. Guo, L.L. Chen, H.Q. Liu, and X. Xu Eur. J. Med. Chem. 45 2010 3850
-
(2010)
Eur. J. Med. Chem.
, vol.45
, pp. 3850
-
-
Cao, S.L.1
Wang, Y.2
Zhu, L.3
Liao, J.4
Guo, Y.W.5
Chen, L.L.6
Liu, H.Q.7
Xu, X.8
-
34
-
-
49449113807
-
-
N. Sirisoma, S. Kasibhatla, A. Pervin, H. Zhang, S. Jiang, J.A. Willardsen, M.B. Anderson, V. Baichwal, G.G. Mather, K. Jessing, R. Hussain, K. Hoang, C.M. Pleiman, B. Tseng, J. Drewe, and S.X. Cai J. Med. Chem. 51 2008 4771
-
(2008)
J. Med. Chem.
, vol.51
, pp. 4771
-
-
Sirisoma, N.1
Kasibhatla, S.2
Pervin, A.3
Zhang, H.4
Jiang, S.5
Willardsen, J.A.6
Anderson, M.B.7
Baichwal, V.8
Mather, G.G.9
Jessing, K.10
Hussain, R.11
Hoang, K.12
Pleiman, C.M.13
Tseng, B.14
Drewe, J.15
Cai, S.X.16
-
35
-
-
71249164372
-
-
K.A. Olaussen, F. Commo, M. Tailler, L. Lacroix, I. Vitale, S.Q. Raza, C. Richon, P. Dessen, V. Lazar, J.C. Soria, and G. Kroemer Oncogene 28 2009 4249
-
(2009)
Oncogene
, vol.28
, pp. 4249
-
-
Olaussen, K.A.1
Commo, F.2
Tailler, M.3
Lacroix, L.4
Vitale, I.5
Raza, S.Q.6
Richon, C.7
Dessen, P.8
Lazar, V.9
Soria, J.C.10
Kroemer, G.11
-
36
-
-
38549175764
-
-
S.Y. Hong, K.W. Kwak, C.K. Ryu, S.J. Kang, and K.H. Chung Bioorg. Med. Chem. 16 2008 644
-
(2008)
Bioorg. Med. Chem.
, vol.16
, pp. 644
-
-
Hong, S.Y.1
Kwak, K.W.2
Ryu, C.K.3
Kang, S.J.4
Chung, K.H.5
-
40
-
-
81255208414
-
-
P. Bandyopadhyay, M. Sathe, S. Ponmariappan, A. Sharma, P. Sharma, A.K. Srivastava, and M.P. Kaushik Bioorg. Med. Chem. Lett. 21 2011 7306
-
(2011)
Bioorg. Med. Chem. Lett.
, vol.21
, pp. 7306
-
-
Bandyopadhyay, P.1
Sathe, M.2
Ponmariappan, S.3
Sharma, A.4
Sharma, P.5
Srivastava, A.K.6
Kaushik, M.P.7
-
41
-
-
34247333034
-
-
J.Y. Xu, Y. Zeng, Q. Ran, Z. Wei, Y. Bi, Q.H. He, Q.J. Wang, S. Hu, J. Zhang, M.Y. Tang, W.Y. Hua, and X.M. Wu Bioorg. Med. Chem. Lett. 17 2007 2921
-
(2007)
Bioorg. Med. Chem. Lett.
, vol.17
, pp. 2921
-
-
Xu, J.Y.1
Zeng, Y.2
Ran, Q.3
Wei, Z.4
Bi, Y.5
He, Q.H.6
Wang, Q.J.7
Hu, S.8
Zhang, J.9
Tang, M.Y.10
Hua, W.Y.11
Wu, X.M.12
-
42
-
-
0027175627
-
-
K. Taniguchi, S. Shigenaga, T. Ogahara, T. Fujitsu, and M. Matsuo Chem. Pharm. Bull. 41 1993 301
-
(1993)
Chem. Pharm. Bull.
, vol.41
, pp. 301
-
-
Taniguchi, K.1
Shigenaga, S.2
Ogahara, T.3
Fujitsu, T.4
Matsuo, M.5
-
43
-
-
33745038028
-
-
S.E. Soto, R.V. Molina, F.A. Crespo, J.V. Galicia, H.O. DIaz, M.T. Piedra, and G.N. Vazquez Life Sci. 79 2006 430
-
(2006)
Life Sci.
, vol.79
, pp. 430
-
-
Soto, S.E.1
Molina, R.V.2
Crespo, F.A.3
Galicia, J.V.4
Diaz, H.O.5
Piedra, M.T.6
Vazquez, G.N.7
-
44
-
-
34248647896
-
-
K. Starcevic, M. Kralj, K. Ester, I. Sabol, M. Grce, K. Pavelic, and G.K. Zamola Bioorg. Med. Chem. 15 2007 4419
-
(2007)
Bioorg. Med. Chem.
, vol.15
, pp. 4419
-
-
Starcevic, K.1
Kralj, M.2
Ester, K.3
Sabol, I.4
Grce, M.5
Pavelic, K.6
Zamola, G.K.7
-
45
-
-
0346671323
-
-
T. Fonseca, B. Gigante, M.M. Marques, L.T. Gilchrist, and E.D. Clercq Bioorg. Med. Chem. 12 2004 103
-
(2004)
Bioorg. Med. Chem.
, vol.12
, pp. 103
-
-
Fonseca, T.1
Gigante, B.2
Marques, M.M.3
Gilchrist, L.T.4
Clercq, E.D.5
-
46
-
-
34250159880
-
-
R.J. Snow, A. Abeywardane, S. Campbell, J. Lord, M.A. Kashem, H.H. Khine, J. King, J.A. Kowalski, S.S. Pullen, T. Roma, G.P. Roth, C.R. Sarko, N.S. Wilson, M.S. Winters, J.P. Wolak, and C.L. Cywin Bioorg. Med. Chem. Lett. 17 2007 3660
-
(2007)
Bioorg. Med. Chem. Lett.
, vol.17
, pp. 3660
-
-
Snow, R.J.1
Abeywardane, A.2
Campbell, S.3
Lord, J.4
Kashem, M.A.5
Khine, H.H.6
King, J.7
Kowalski, J.A.8
Pullen, S.S.9
Roma, T.10
Roth, G.P.11
Sarko, C.R.12
Wilson, N.S.13
Winters, M.S.14
Wolak, J.P.15
Cywin, C.L.16
-
47
-
-
1342324016
-
-
G. Lewaire, C. Delescluse, M. Pralavorio, N. Ledirac, P. Lesca, and R. Rahmani Life Sci. 74 2004 2265
-
(2004)
Life Sci.
, vol.74
, pp. 2265
-
-
Lewaire, G.1
Delescluse, C.2
Pralavorio, M.3
Ledirac, N.4
Lesca, P.5
Rahmani, R.6
-
49
-
-
79956151545
-
-
Z. Sun, H. Wang, K. Wen, Y. Li, and E. Fan J. Org. Chem. 76 2011 4149
-
(2011)
J. Org. Chem.
, vol.76
, pp. 4149
-
-
Sun, Z.1
Wang, H.2
Wen, K.3
Li, Y.4
Fan, E.5
-
50
-
-
84891496457
-
-
Crystallographic data for the structural analysis have been deposited at the Cambridge Crystallographic Data Centre, CCDC No. 928250 (E-mail: deposit@ccdc.cam.ac.uk).
-
-
-
-
52
-
-
0025775062
-
-
A. Monks, D. Schudiero, P. Skehan, R. Shoemaker, K. Paull, D. Vistica, C. Hose, J. Langley, P. Cronise, A. Vaigro-Wolff, M. Gray-Goodrich, H. Campbell, J. Mayo, and M. Boyd J. Natl. Cancer Inst. 83 1991 757
-
(1991)
J. Natl. Cancer Inst.
, vol.83
, pp. 757
-
-
Monks, A.1
Schudiero, D.2
Skehan, P.3
Shoemaker, R.4
Paull, K.5
Vistica, D.6
Hose, C.7
Langley, J.8
Cronise, P.9
Vaigro-Wolff, A.10
Gray-Goodrich, M.11
Campbell, H.12
Mayo, J.13
Boyd, M.14
-
56
-
-
84865102002
-
-
references therein
-
C. Bailly Chem. Rev. 112 2012 3611 and references therein
-
(2012)
Chem. Rev.
, vol.112
, pp. 3611
-
-
Bailly, C.1
-
57
-
-
67650682519
-
-
references therein
-
Y. Pommier Chem. Rev. 109 2009 2894 and references therein
-
(2009)
Chem. Rev.
, vol.109
, pp. 2894
-
-
Pommier, Y.1
|