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Volumn 7, Issue 1, 2013, Pages

Organocatalysis in heterocyclic synthesis: DABCO as a mild and efficient catalytic system for the synthesis of a novel class of quinazoline, thiazolo [3,2-a]quinazoline and thiazolo[2,3-b] quinazoline derivatives

Author keywords

DABCO; Organocatalysis; Quinazoline; Thiazolo 2,3 b quinazoline; Thiazolo 3,2 a quinazoline

Indexed keywords


EID: 84877040484     PISSN: None     EISSN: 1752153X     Source Type: Journal    
DOI: 10.1186/1752-153X-7-82     Document Type: Article
Times cited : (10)

References (56)
  • 1
    • 27144529642 scopus 로고    scopus 로고
    • DABCO: An efficient organocatalyst in the ring-opening reactions of aziridines with amines or thiols
    • Wu J, Sun X, Li Y. DABCO: An efficient organocatalyst in the ring-opening reactions of aziridines with amines or thiols. Eur J Org Chem 2005, 20:4271-4275.
    • (2005) Eur J Org Chem , vol.20 , pp. 4271-4275
    • Wu, J.1    Sun, X.2    Li, Y.3
  • 2
    • 80054103144 scopus 로고    scopus 로고
    • DABCO-triggered mild cascade reaction of electron-eficient cyclopentadienone: facile and efficient synthesis of condensed carbocycles
    • Yamguchi K, Eto M, Higashi K, Yoshitake Y, Harano K. DABCO-triggered mild cascade reaction of electron-eficient cyclopentadienone: facile and efficient synthesis of condensed carbocycles. Tetrahedron Lett 2011, 52:6082-6085.
    • (2011) Tetrahedron Lett , vol.52 , pp. 6082-6085
    • Yamguchi, K.1    Eto, M.2    Higashi, K.3    Yoshitake, Y.4    Harano, K.5
  • 3
    • 84864440624 scopus 로고    scopus 로고
    • DABCO-mediated one-pot sequential transformation: convenient access to fluorinated 1H-pyrazol-5(4H)-ones
    • Wu J-W, Li F, Zheng Y, Nie J. DABCO-mediated one-pot sequential transformation: convenient access to fluorinated 1H-pyrazol-5(4H)-ones. Tetrahedron Lett 2012, 53:4828-4831.
    • (2012) Tetrahedron Lett , vol.53 , pp. 4828-4831
    • Wu, J.-W.1    Li, F.2    Zheng, Y.3    Nie, J.4
  • 4
    • 8444252168 scopus 로고    scopus 로고
    • Unveiling reliable catalysts for the asymmetric nitroaldol (Henry) reaction
    • Palomo C, Oiarbide M, Mielgo A. Unveiling reliable catalysts for the asymmetric nitroaldol (Henry) reaction. Angew Chem Int Ed 2004, 43:5442-5444.
    • (2004) Angew Chem Int Ed , vol.43 , pp. 5442-5444
    • Palomo, C.1    Oiarbide, M.2    Mielgo, A.3
  • 5
    • 84864039461 scopus 로고    scopus 로고
    • Direct transition metal-free C-S bond formation: synthesis of 2-aminobenzothiazole derivatives via base-mediated approach
    • Wang R, Yue L, Pan W, Zhao J-J. Direct transition metal-free C-S bond formation: synthesis of 2-aminobenzothiazole derivatives via base-mediated approach. Tetrahedron Lett 2012, 53:4529-4531.
    • (2012) Tetrahedron Lett , vol.53 , pp. 4529-4531
    • Wang, R.1    Yue, L.2    Pan, W.3    Zhao, J.-J.4
  • 6
    • 78649323240 scopus 로고    scopus 로고
    • Synthesis and antitumor activity of some 2,3-disubstituted quinazolin-4(3H)-ones and 4,6-disubstituted-1,2,3,4-tetrahydro- quinazolin-2H-ones
    • 10.1016/j.ejmech.2010.10.008, 21051122
    • Abdel Gawad NM, Georgey HH, Youssef RM, El-Sayed NA. Synthesis and antitumor activity of some 2,3-disubstituted quinazolin-4(3H)-ones and 4,6-disubstituted-1,2,3,4-tetrahydro- quinazolin-2H-ones. Eur J Med Chem 2010, 45:6058-6067. 10.1016/j.ejmech.2010.10.008, 21051122.
    • (2010) Eur J Med Chem , vol.45 , pp. 6058-6067
    • Abdel Gawad, N.M.1    Georgey, H.H.2    Youssef, R.M.3    El-Sayed, N.A.4
  • 7
    • 41349085423 scopus 로고    scopus 로고
    • Synthesis of novel 4,6-disubstituted uinazoline derivatives, their anti-inflammatory and anti-cancer activity (cytotoxic) against U937 leukemia cell lines
    • 10.1016/j.ejmech.2007.06.010, 17689837
    • Chandrika PM, Yakaiah T, Rao AR, Narsaiah B, Reddy NC, Sridhar V, Rao JV. Synthesis of novel 4,6-disubstituted uinazoline derivatives, their anti-inflammatory and anti-cancer activity (cytotoxic) against U937 leukemia cell lines. Eur J Med Chem 2008, 43:846-852. 10.1016/j.ejmech.2007.06.010, 17689837.
    • (2008) Eur J Med Chem , vol.43 , pp. 846-852
    • Chandrika, P.M.1    Yakaiah, T.2    Rao, A.R.3    Narsaiah, B.4    Reddy, N.C.5    Sridhar, V.6    Rao, J.V.7
  • 8
    • 84855763252 scopus 로고    scopus 로고
    • Substituted thiazoles V. Synthesis and antitumor activity of novel thiazolo[2,3-b]quinazoline and pyrido[4,3-d]thiazolo[3,2-a]- pyrimidine analogues
    • Al-Omary FAM, Hassan GS, El-Messery SM, El-Subbagh HI. Substituted thiazoles V. Synthesis and antitumor activity of novel thiazolo[2,3-b]quinazoline and pyrido[4,3-d]thiazolo[3,2-a]- pyrimidine analogues. Eur J Med Chem 2012, 47:65-72.
    • (2012) Eur J Med Chem , vol.47 , pp. 65-72
    • Al-Omary, F.A.M.1    Hassan, G.S.2    El-Messery, S.M.3    El-Subbagh, H.I.4
  • 10
    • 42149190240 scopus 로고    scopus 로고
    • Design, synthesis and pharmacological evaluation of hybrid molecules out of quinazolinimines and lipoic acid lead to highly potent and selective butyrylcholinesterase inhibitors with antioxidant properties
    • 10.1016/j.bmc.2008.02.083, 18343673
    • Decker M, Kraus B. Design, synthesis and pharmacological evaluation of hybrid molecules out of quinazolinimines and lipoic acid lead to highly potent and selective butyrylcholinesterase inhibitors with antioxidant properties. Bioorg Med Chem 2008, 16:4252-4261. 10.1016/j.bmc.2008.02.083, 18343673.
    • (2008) Bioorg Med Chem , vol.16 , pp. 4252-4261
    • Decker, M.1    Kraus, B.2
  • 11
    • 60149105200 scopus 로고    scopus 로고
    • Design and synthesis of azolopyrimidoquinolines, pyrimidoquinazolines as anti-oxidant, anti-inflamm- atory and analgesic activities
    • 10.1016/j.ejmech.2008.03.022, 18462840
    • El-Gazzar ABA, Youssef MM, Youssef AMS, Abu-Hashem AA, Badria FA. Design and synthesis of azolopyrimidoquinolines, pyrimidoquinazolines as anti-oxidant, anti-inflamm- atory and analgesic activities. Eur J Med Chem 2009, 44:609-624. 10.1016/j.ejmech.2008.03.022, 18462840.
    • (2009) Eur J Med Chem , vol.44 , pp. 609-624
    • El-Gazzar, A.B.A.1    Youssef, M.M.2    Youssef, A.M.S.3    Abu-Hashem, A.A.4    Badria, F.A.5
  • 12
    • 0242298226 scopus 로고    scopus 로고
    • Some new 2,3,6-trisubstituted quinazolinones as potent anti-inflammatory, analgesic and COX-II inhibitors
    • 10.1016/S0968-0896(03)00501-7, 14604693
    • Kumar A, Sharma S, Bajaj AK, Sharma S, Panwar H, Singh T, Srivastava VK. Some new 2,3,6-trisubstituted quinazolinones as potent anti-inflammatory, analgesic and COX-II inhibitors. Bioorg Med Chem 2003, 11:5293-5299. 10.1016/S0968-0896(03)00501-7, 14604693.
    • (2003) Bioorg Med Chem , vol.11 , pp. 5293-5299
    • Kumar, A.1    Sharma, S.2    Bajaj, A.K.3    Sharma, S.4    Panwar, H.5    Singh, T.6    Srivastava, V.K.7
  • 13
    • 77954313516 scopus 로고    scopus 로고
    • Synthesis of some new 4(3H)-quinazolinone-2-carboxaldehyde thiosemicarbazones and their metal complexes and a study on their anticonvulsant, analgesic, cytotoxic and antimicrobial activities
    • 10.1016/j.ejmech.2010.04.020, 20510483
    • Aly MM, Mohamed YA, El-Bayouki KM, Basyouni WM, Abbas SY. Synthesis of some new 4(3H)-quinazolinone-2-carboxaldehyde thiosemicarbazones and their metal complexes and a study on their anticonvulsant, analgesic, cytotoxic and antimicrobial activities. Eur J Med Chem 2010, 45:3365-3373. 10.1016/j.ejmech.2010.04.020, 20510483.
    • (2010) Eur J Med Chem , vol.45 , pp. 3365-3373
    • Aly, M.M.1    Mohamed, Y.A.2    El-Bayouki, K.M.3    Basyouni, W.M.4    Abbas, S.Y.5
  • 14
    • 0033395476 scopus 로고    scopus 로고
    • Synthesis antibacterial antifungal and anti-HIV evaluation of Schiff and Mannich bases of isatin derivatives with 3-amino-2-methylmercapto quinazolin-4(3H)-one
    • 10.1016/S0031-6865(99)00010-2, 10748620
    • Pandeya SN, Sriram D, Nath G, Clercq ED. Synthesis antibacterial antifungal and anti-HIV evaluation of Schiff and Mannich bases of isatin derivatives with 3-amino-2-methylmercapto quinazolin-4(3H)-one. Pharm Acta Helv 1999, 74:11-17. 10.1016/S0031-6865(99)00010-2, 10748620.
    • (1999) Pharm Acta Helv , vol.74 , pp. 11-17
    • Pandeya, S.N.1    Sriram, D.2    Nath, G.3    Clercq, E.D.4
  • 15
    • 36248960362 scopus 로고    scopus 로고
    • Synthesis, antibacterial, and anti-HIV activities of 3-[5-amino-6-(2,3-dichlorophenyl)-[1,2,4]triazin-3-yl]-6,8-dibromo-2-substituted-3H-quin- azolin-4-one
    • Selvam P, Girija K, Nagarajan G, De Clerco E. Synthesis, antibacterial, and anti-HIV activities of 3-[5-amino-6-(2,3-dichlorophenyl)-[1,2,4]triazin-3-yl]-6,8-dibromo-2-substituted-3H-quin- azolin-4-one. Indian J Pharm Sci 2005, 67:484-487.
    • (2005) Indian J Pharm Sci , vol.67 , pp. 484-487
    • Selvam, P.1    Girija, K.2    Nagarajan, G.3    De Clerco, E.4
  • 16
    • 0033837451 scopus 로고    scopus 로고
    • Synthesis and evaluation of some new fluorinated hydroquinazoline derivatives as antifungal agents
    • Ghorab MM, Abdel-Gawad SM, El-Gaby MSA. Synthesis and evaluation of some new fluorinated hydroquinazoline derivatives as antifungal agents. II Farmaco 2000, 55:249-255.
    • (2000) II Farmaco , vol.55 , pp. 249-255
    • Ghorab, M.M.1    Abdel-Gawad, S.M.2    El-Gaby, M.S.A.3
  • 18
    • 34047188045 scopus 로고    scopus 로고
    • Synthesis and antihypertensive activity of novel 3-benzyl-2-substituted-3H-[1,2,4]triazolo[5,1-b]quinazolin-9-ones
    • 10.1016/j.bmc.2007.03.007, 17391966
    • Alagarsamy V, Pathak US. Synthesis and antihypertensive activity of novel 3-benzyl-2-substituted-3H-[1,2,4]triazolo[5,1-b]quinazolin-9-ones. Bioorg Med Chem 2007, 15:3457-3462. 10.1016/j.bmc.2007.03.007, 17391966.
    • (2007) Bioorg Med Chem , vol.15 , pp. 3457-3462
    • Alagarsamy, V.1    Pathak, U.S.2
  • 19
    • 68949149073 scopus 로고    scopus 로고
    • Design and synthesis of novel substituted quinazoline derivatives as antileishmanial agents
    • 10.1016/j.bmcl.2009.07.081, 19692240
    • Agarwal KC, Sharma V, Shakya N, Gupta S. Design and synthesis of novel substituted quinazoline derivatives as antileishmanial agents. Bioorg Med Chem Lett 2009, 19:5474-5477. 10.1016/j.bmcl.2009.07.081, 19692240.
    • (2009) Bioorg Med Chem Lett , vol.19 , pp. 5474-5477
    • Agarwal, K.C.1    Sharma, V.2    Shakya, N.3    Gupta, S.4
  • 20
    • 70349770548 scopus 로고    scopus 로고
    • Synthesis, anticonvulsant and CNS depressant activity of some new bioactive 1-(4-substituted-phenyl)-3-(4-oxo-2- phenyl/ethyl-4H-quinazolin-3-yl)urea
    • 10.1016/j.ejmech.2009.05.008, 19674817
    • Kashawa SK, Kashawa V, Mishra P, Jain NK, Stables JP. Synthesis, anticonvulsant and CNS depressant activity of some new bioactive 1-(4-substituted-phenyl)-3-(4-oxo-2- phenyl/ethyl-4H-quinazolin-3-yl)urea. Eur J Med Chem 2009, 44:4335-4343. 10.1016/j.ejmech.2009.05.008, 19674817.
    • (2009) Eur J Med Chem , vol.44 , pp. 4335-4343
    • Kashawa, S.K.1    Kashawa, V.2    Mishra, P.3    Jain, N.K.4    Stables, J.P.5
  • 22
    • 72149105339 scopus 로고    scopus 로고
    • Novel 4-thiazolidinone derivatives as potential antifungal and antibacterial drugs
    • 10.1016/j.bmc.2009.10.041, 19914077
    • Omar K, Geronikaki A, Zoumpoulakis P, Camoutsis C, Sokovic M, Ciric A, Glamoclija J. Novel 4-thiazolidinone derivatives as potential antifungal and antibacterial drugs. Bioorg Med Chem 2010, 18:426-432. 10.1016/j.bmc.2009.10.041, 19914077.
    • (2010) Bioorg Med Chem , vol.18 , pp. 426-432
    • Omar, K.1    Geronikaki, A.2    Zoumpoulakis, P.3    Camoutsis, C.4    Sokovic, M.5    Ciric, A.6    Glamoclija, J.7
  • 23
    • 79958256411 scopus 로고    scopus 로고
    • Synthesis of new chalcone derivatives bearing 2,4-thiazolidinedione and benzoic acid moieties as potential anti-bacterial agents
    • 10.1016/j.ejmech.2011.05.012, 21624712
    • Liu X, Zheng C, Sun L, Liu X, Piao H. Synthesis of new chalcone derivatives bearing 2,4-thiazolidinedione and benzoic acid moieties as potential anti-bacterial agents. Eur J Med Chem 2011, 46:3469-3473. 10.1016/j.ejmech.2011.05.012, 21624712.
    • (2011) Eur J Med Chem , vol.46 , pp. 3469-3473
    • Liu, X.1    Zheng, C.2    Sun, L.3    Liu, X.4    Piao, H.5
  • 24
    • 77955552993 scopus 로고    scopus 로고
    • Conventional and microwave assisted synthesis of some new N-[(4-oxo-2-substituted aryl-1,3-thiazolidine)acetamidyl]-5-nitroindazoles and its antimicrobial activity
    • 10.1016/j.ejmech.2010.04.029, 20570024
    • Upadhyay A, Srivastava SK, Srivastava SD. Conventional and microwave assisted synthesis of some new N-[(4-oxo-2-substituted aryl-1,3-thiazolidine)acetamidyl]-5-nitroindazoles and its antimicrobial activity. Eur J Med Chem 2010, 45:3541-3548. 10.1016/j.ejmech.2010.04.029, 20570024.
    • (2010) Eur J Med Chem , vol.45 , pp. 3541-3548
    • Upadhyay, A.1    Srivastava, S.K.2    Srivastava, S.D.3
  • 25
    • 79954622755 scopus 로고    scopus 로고
    • Indentification of thiazolidinones spiro-fused to indolin-2-ones as potent and selective inhibitors of the mycobacterium tuberculosis protein tyrosine phosphatase B
    • Vintonyak VK, Warburg K, Kruse H, Grimme S, Hubel K, Rauh D, Waldmann H. Indentification of thiazolidinones spiro-fused to indolin-2-ones as potent and selective inhibitors of the mycobacterium tuberculosis protein tyrosine phosphatase B. Angew Chem 2010, 122:6038-6041.
    • (2010) Angew Chem , vol.122 , pp. 6038-6041
    • Vintonyak, V.K.1    Warburg, K.2    Kruse, H.3    Grimme, S.4    Hubel, K.5    Rauh, D.6    Waldmann, H.7
  • 26
    • 79958296582 scopus 로고    scopus 로고
    • Design, synthesis and biological evaluation of novel 4-thiazolidinones containing indolin-2-one moiety as potential antitumor agent
    • 10.1016/j.ejmech.2011.05.017, 21621880
    • Wang S, Zhao Y, Zhang G, Lv Y, Zhang N, Gong P. Design, synthesis and biological evaluation of novel 4-thiazolidinones containing indolin-2-one moiety as potential antitumor agent. Eur J Med Chem 2011, 46:3509-3518. 10.1016/j.ejmech.2011.05.017, 21621880.
    • (2011) Eur J Med Chem , vol.46 , pp. 3509-3518
    • Wang, S.1    Zhao, Y.2    Zhang, G.3    Lv, Y.4    Zhang, N.5    Gong, P.6
  • 27
    • 72049095834 scopus 로고    scopus 로고
    • Design, synthesis and biological evaluation of thiazolidinone derivatives as potential EGFR and HER-2 kinase inhibitors
    • 10.1016/j.bmc.2009.10.051, 19914835
    • Lv P, Zhou C, Chen J, Liu P, Wang K, Mao W, Li H, Yang Y, Xiong J, Zhu H. Design, synthesis and biological evaluation of thiazolidinone derivatives as potential EGFR and HER-2 kinase inhibitors. Bioorg Med Chem 2010, 18:314-319. 10.1016/j.bmc.2009.10.051, 19914835.
    • (2010) Bioorg Med Chem , vol.18 , pp. 314-319
    • Lv, P.1    Zhou, C.2    Chen, J.3    Liu, P.4    Wang, K.5    Mao, W.6    Li, H.7    Yang, Y.8    Xiong, J.9    Zhu, H.10
  • 28
    • 77957844111 scopus 로고    scopus 로고
    • Synthesis and anticancer activity evaluation of 4-thiazolidinones containing benzothiazole moiety
    • 10.1016/j.ejmech.2010.08.008, 20810193
    • Havrylyuk D, Mosula L, Zimenkovsky B, Vasylenko O, Gzella A, Lesyk R. Synthesis and anticancer activity evaluation of 4-thiazolidinones containing benzothiazole moiety. Eur J Med Chem 2010, 45:5012-5021. 10.1016/j.ejmech.2010.08.008, 20810193.
    • (2010) Eur J Med Chem , vol.45 , pp. 5012-5021
    • Havrylyuk, D.1    Mosula, L.2    Zimenkovsky, B.3    Vasylenko, O.4    Gzella, A.5    Lesyk, R.6
  • 29
    • 78650513550 scopus 로고    scopus 로고
    • In vitro evaluation of 5-arylidene-2-thioxo-4-thiazolidinones active as aldose reductase inhibitors
    • 10.1016/j.bmcl.2010.11.041, 21129963
    • Maccari R, Corso AD, Giglio M, Moschini R, Mura U, Ottana R. In vitro evaluation of 5-arylidene-2-thioxo-4-thiazolidinones active as aldose reductase inhibitors. Bioorg Med Chem Lett 2011, 21:200-203. 10.1016/j.bmcl.2010.11.041, 21129963.
    • (2011) Bioorg Med Chem Lett , vol.21 , pp. 200-203
    • Maccari, R.1    Corso, A.D.2    Giglio, M.3    Moschini, R.4    Mura, U.5    Ottana, R.6
  • 30
    • 47949096992 scopus 로고    scopus 로고
    • Design and synthesis of 2-(2,6-dibromophenyl)-3-heteroaryl-1,3-thiazolidin-4-ones as anti-HIV agents
    • 10.1016/j.ejmech.2007.12.015, 18242784
    • Rawal RK, Tripathi R, Katti SB, Pannecouque C, De Clercq E. Design and synthesis of 2-(2,6-dibromophenyl)-3-heteroaryl-1,3-thiazolidin-4-ones as anti-HIV agents. Eur J Med Chem 2008, 43:2800-2806. 10.1016/j.ejmech.2007.12.015, 18242784.
    • (2008) Eur J Med Chem , vol.43 , pp. 2800-2806
    • Rawal, R.K.1    Tripathi, R.2    Katti, S.B.3    Pannecouque, C.4    De Clercq, E.5
  • 32
    • 77952043774 scopus 로고    scopus 로고
    • Design, synthesis, and interaction study of quinazoline-2(1H)-thione derivatives as novel potential Bcl-xL inhibitors
    • 10.1021/jm901004c, 20405848
    • Feng Y, Ding X, Chen T, Chen L, Liu F, Jia X, Luo X, Shen X, Chen K, Jiang H, Wang H, Liu H, Liu D. Design, synthesis, and interaction study of quinazoline-2(1H)-thione derivatives as novel potential Bcl-xL inhibitors. J Med Chem 2010, 53:3465-3479. 10.1021/jm901004c, 20405848.
    • (2010) J Med Chem , vol.53 , pp. 3465-3479
    • Feng, Y.1    Ding, X.2    Chen, T.3    Chen, L.4    Liu, F.5    Jia, X.6    Luo, X.7    Shen, X.8    Chen, K.9    Jiang, H.10    Wang, H.11    Liu, H.12    Liu, D.13
  • 33
    • 36649034033 scopus 로고    scopus 로고
    • Efficient solid-phase synthesis of 3-substituted-5-Oxo-5H-thiazolo[2,3-b]quinazoline-8-carboxamides under mild conditions with two diversity positions
    • 10.1021/cc700122a, 2569825, 17907790
    • Bouillon I, Krchnak V. Efficient solid-phase synthesis of 3-substituted-5-Oxo-5H-thiazolo[2,3-b]quinazoline-8-carboxamides under mild conditions with two diversity positions. J Comb Chem 2007, 9:912-915. 10.1021/cc700122a, 2569825, 17907790.
    • (2007) J Comb Chem , vol.9 , pp. 912-915
    • Bouillon, I.1    Krchnak, V.2
  • 34
    • 45949085044 scopus 로고    scopus 로고
    • Novel 9-oxo-thiazolo[5,4-f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: synthesis, biological evaluation and molecular modeling studies
    • 10.1016/j.ejmech.2007.09.020, 17981370
    • Loge C, Testard A, Thierry V, Lozach O, Blairvacq M, Robert J-M, Meijer L, Besson T. Novel 9-oxo-thiazolo[5,4-f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: synthesis, biological evaluation and molecular modeling studies. Eur J Med Chem 2008, 43:1469-1477. 10.1016/j.ejmech.2007.09.020, 17981370.
    • (2008) Eur J Med Chem , vol.43 , pp. 1469-1477
    • Loge, C.1    Testard, A.2    Thierry, V.3    Lozach, O.4    Blairvacq, M.5    Robert, J.-M.6    Meijer, L.7    Besson, T.8
  • 36
    • 77949346933 scopus 로고    scopus 로고
    • Design, synthesis, and evaluation of 2-methyl- and 2-amino-N-aryl-4,5-dihydrothiazolo[4,5-h]quinazolin-8-amines as ring-constrained 2-anilino-4-(thiazol-5-yl)pyrimidine cyclin-dependent kinase inhibitors
    • 10.1021/jm901660c, 20146435
    • McIntyre NA, McInnes C, Griffiths G, Barnett AL, Kontopidis G, Slawin AMZ, Jackson W, Thomas M, Zheleva DI, Wang S, Blake DG, Westwood NJ, Fischer PM. Design, synthesis, and evaluation of 2-methyl- and 2-amino-N-aryl-4,5-dihydrothiazolo[4,5-h]quinazolin-8-amines as ring-constrained 2-anilino-4-(thiazol-5-yl)pyrimidine cyclin-dependent kinase inhibitors. J Med Chem 2010, 53:2136-2145. 10.1021/jm901660c, 20146435.
    • (2010) J Med Chem , vol.53 , pp. 2136-2145
    • McIntyre, N.A.1    McInnes, C.2    Griffiths, G.3    Barnett, A.L.4    Kontopidis, G.5    Slawin, A.M.Z.6    Jackson, W.7    Thomas, M.8    Zheleva, D.I.9    Wang, S.10    Blake, D.G.11    Westwood, N.J.12    Fischer, P.M.13
  • 37
    • 56049121230 scopus 로고    scopus 로고
    • Thermal reaction of 3aH,5H-thiazolo[5,4-c]quinoline-2,4-diones an easy pathway to 4-amino-1H-quinoline-2-ones and novel 6H-thiazolo[3,4-c]quinazoline-3,5-diones
    • Mrkvicka V, Klasek A, Kimmel R, Pevee A, Kosmrlj J. Thermal reaction of 3aH,5H-thiazolo[5,4-c]quinoline-2,4-diones an easy pathway to 4-amino-1H-quinoline-2-ones and novel 6H-thiazolo[3,4-c]quinazoline-3,5-diones. ARKIVOC 2008, 14:289-302.
    • (2008) ARKIVOC , vol.14 , pp. 289-302
    • Mrkvicka, V.1    Klasek, A.2    Kimmel, R.3    Pevee, A.4    Kosmrlj, J.5
  • 38
    • 0034525453 scopus 로고    scopus 로고
    • Synthesis and in vitro antitumour activity evaluation of 1-aryl-1H,3H-thiazolo[4,3-b]quinazolines
    • 10.1016/S0223-5234(00)01195-8, 11248410
    • Grasso S, Micale N, Monforte A-M, Monforte P, Polimeni S, Zappala M. Synthesis and in vitro antitumour activity evaluation of 1-aryl-1H,3H-thiazolo[4,3-b]quinazolines. Eur J Med Chem 2000, 35:1115-1119. 10.1016/S0223-5234(00)01195-8, 11248410.
    • (2000) Eur J Med Chem , vol.35 , pp. 1115-1119
    • Grasso, S.1    Micale, N.2    Monforte, A.-M.3    Monforte, P.4    Polimeni, S.5    Zappala, M.6
  • 39
    • 79952632056 scopus 로고    scopus 로고
    • Regioselective syntheses of 1-aryl-substituted-5H-[1,3]thiazolo[3,2-a]quinazoline-5-ones during Sonogashira coupling
    • Bakherad M, Keivanloo A, Kalantar Z, Keley V. Regioselective syntheses of 1-aryl-substituted-5H-[1,3]thiazolo[3,2-a]quinazoline-5-ones during Sonogashira coupling. Phosphorus Sulfur Silicon Relat Elem 2011, 186:464-470.
    • (2011) Phosphorus Sulfur Silicon Relat Elem , vol.186 , pp. 464-470
    • Bakherad, M.1    Keivanloo, A.2    Kalantar, Z.3    Keley, V.4
  • 40
    • 0025361796 scopus 로고
    • Heterocyclic systems containing bridgehead nitrogen atom. Part LXIV. Synthesis of 7-methylthiazolo[3,2-a]quinazolines
    • Jain KK, Rout SP, Pujari HK. Heterocyclic systems containing bridgehead nitrogen atom. Part LXIV. Synthesis of 7-methylthiazolo[3,2-a]quinazolines. Indian J Chem Sect B 1990, 29B:379-80.
    • (1990) Indian J Chem Sect B , vol.29 B , pp. 379-380
    • Jain, K.K.1    Rout, S.P.2    Pujari, H.K.3
  • 41
    • 79953210705 scopus 로고    scopus 로고
    • Applications of 2-arylhydrazononitriles in synthesis: preparation of new indole containing 1,2,3-triazole, pyrazole and pyrazolo[1,5-a]pyrimidine derivatives and evaluation of their antimicrobial activities
    • 10.1016/j.ejmech.2011.02.040, 21397366
    • Behbehani H, Ibrahim HM, Makhseed S, Mahmoud H. Applications of 2-arylhydrazononitriles in synthesis: preparation of new indole containing 1,2,3-triazole, pyrazole and pyrazolo[1,5-a]pyrimidine derivatives and evaluation of their antimicrobial activities. Eur J Med Chem 2011, 46:1813-1820. 10.1016/j.ejmech.2011.02.040, 21397366.
    • (2011) Eur J Med Chem , vol.46 , pp. 1813-1820
    • Behbehani, H.1    Ibrahim, H.M.2    Makhseed, S.3    Mahmoud, H.4
  • 42
    • 84860330558 scopus 로고    scopus 로고
    • 2-Aminothiophenes as building blocks in heterocyclic synthesis: synthesis and antimicrobial evaluation of a new class of pyrido[1,2-a]thieno[3,2-e]pyrimidine, quinoline and pyridin-2-one derivatives
    • Behbehani H, Ibrahim HM, Makhseed S, Elnagdi MH, Mahmoud H. 2-Aminothiophenes as building blocks in heterocyclic synthesis: synthesis and antimicrobial evaluation of a new class of pyrido[1,2-a]thieno[3,2-e]pyrimidine, quinoline and pyridin-2-one derivatives. Eur J Med Chem 2012, 52:61-65.
    • (2012) Eur J Med Chem , vol.52 , pp. 61-65
    • Behbehani, H.1    Ibrahim, H.M.2    Makhseed, S.3    Elnagdi, M.H.4    Mahmoud, H.5
  • 43
    • 84862998685 scopus 로고    scopus 로고
    • 4-Thiazolidinones in heterocyclic synthesis: synthesis of novel enaminones, azolopyrimidines and 2-Arylimino-5-arylidene-4-thiazolidinones
    • 10.3390/molecules17066362, 22634845
    • Behbehani H, Ibrahim HM. 4-Thiazolidinones in heterocyclic synthesis: synthesis of novel enaminones, azolopyrimidines and 2-Arylimino-5-arylidene-4-thiazolidinones. Molecules 2012, 17:6362-6385. 10.3390/molecules17066362, 22634845.
    • (2012) Molecules , vol.17 , pp. 6362-6385
    • Behbehani, H.1    Ibrahim, H.M.2
  • 44
    • 33646071514 scopus 로고    scopus 로고
    • Synthesis and antimicrobial activity of novel 2-thiazolylimino-5-arylidene-4-thiazolidinones
    • 10.1016/j.bmc.2006.01.043, 16488614
    • Vicini P, Geronikaki A, Anastasia K, Incerti M, Zani F. Synthesis and antimicrobial activity of novel 2-thiazolylimino-5-arylidene-4-thiazolidinones. Bioorg Med Chem 2006, 14:3859-3864. 10.1016/j.bmc.2006.01.043, 16488614.
    • (2006) Bioorg Med Chem , vol.14 , pp. 3859-3864
    • Vicini, P.1    Geronikaki, A.2    Anastasia, K.3    Incerti, M.4    Zani, F.5
  • 45
    • 0034325907 scopus 로고    scopus 로고
    • New synthesis of 2-alkylthio-4-oxo-3,4-dihydroquinazolines, 2-alkylthioquinazolines, as well as, their hetero analogues
    • Gruner M, Rehwald M, Eckert K, Gewald K. New synthesis of 2-alkylthio-4-oxo-3,4-dihydroquinazolines, 2-alkylthioquinazolines, as well as, their hetero analogues. Heterocycles 2000, 53:2363-2377.
    • (2000) Heterocycles , vol.53 , pp. 2363-2377
    • Gruner, M.1    Rehwald, M.2    Eckert, K.3    Gewald, K.4


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