-
1
-
-
22544476852
-
Vancomycin-resistant staphylococci and enterococci: Epidemiology and control
-
Tenover, F. C.; McDonald, L. C. Vancomycin-resistant staphylococci and enterococci: epidemiology and control. Curr. Opin. Infect. Dis. 2005, 18, 300-305. (Pubitemid 41017633)
-
(2005)
Current Opinion in Infectious Diseases
, vol.18
, Issue.4
, pp. 300-305
-
-
Tenover, F.C.1
Clifford McDonald, L.2
-
2
-
-
0345869924
-
Synergistic effects of anacardic acids and methicillin against methicillin resistant Staphylococcus aureus
-
DOI 10.1016/j.bmc.2003.10.046
-
Muroi, H.; Nihei, K.; Tsujimoto, K.; Kubo, I. Synergistic effects of anacardic acids and methicillin against methicillin resistant Staphylococcus aureus. Bioorg. Med. Chem. 2004, 12, 583-587. (Pubitemid 38102228)
-
(2004)
Bioorganic and Medicinal Chemistry
, vol.12
, Issue.3
, pp. 583-587
-
-
Muroi, H.1
Nihei, K.-I.2
Tsujimoto, K.3
Kubo, I.4
-
3
-
-
33645855871
-
Similarity in drugs: Reflections on analogue design
-
Wermuth, C. G. Similarity in drugs: reflections on analogue design. Drug Discov. Today 2006, 11, 348-354.
-
(2006)
Drug Discov. Today
, vol.11
, pp. 348-354
-
-
Wermuth, C.G.1
-
4
-
-
0016805624
-
Substituted thiazolidones: Selective inhibition of nicotinamide adenine dinucleotide-dependent oxidations and evaluation of their cns activity
-
Chaudhari, S. K.; Verma, M.; Chaturvedi, A. K.; Parmar, S. S. Substituted thiazolidones: Selective inhibition of nicotinamide adenine dinucleotide-dependent oxidations and evaluation of their cns activity. J. Pharm. Sci. 1975, 64, 614-617.
-
(1975)
J. Pharm. Sci.
, vol.64
, pp. 614-617
-
-
Chaudhari, S.K.1
Verma, M.2
Chaturvedi, A.K.3
Parmar, S.S.4
-
5
-
-
0017273664
-
CNS depressant activity of pyrimidylthiazolidones and their selective inhibition of NAD-dependent pyruvate oxidation
-
Chaudhary, M.; Parmar, S. S.; Chaudhary, S. K.; Chaturvedi, A. K.; Rama Sastry, B. V. CNS depressant activity of pyrimidylthiazolidones and their selective inhibition of NAD-dependent pyruvate oxidation. J. Pharm. Sci. 1976, 65, 443-446.
-
(1976)
J. Pharm. Sci.
, vol.65
, pp. 443-446
-
-
Chaudhary, M.1
Parmar, S.S.2
Chaudhary, S.K.3
Chaturvedi, A.K.4
Rama Sastry, B.V.5
-
6
-
-
0041831030
-
Novel inhibitors of an emerging target in Mycobacterium tuberculosis; substituted thiazolidinones as inhibitors of dTDP-rhamnose synthesis
-
DOI 10.1016/S0960-894X(03)00673-5
-
Babaoglu, K.; Page, M. A.; Jones, V. C.; McNeil, M. R.; Dong, C.; Naismith, J. H.; Lee, R. E. Novel inhibitors of an emerging target in mycobacterium tuberculosis; substituted thiazolidinones as inhibitors of dTDP-rhamnose synthesis. Bioorg. Med. Chem. Lett. 2003, 13, 3227-3230. (Pubitemid 37093833)
-
(2003)
Bioorganic and Medicinal Chemistry Letters
, vol.13
, Issue.19
, pp. 3227-3230
-
-
Babaoglu, K.1
Page, M.A.2
Jones, V.C.3
McNeil, M.R.4
Dong, C.5
Naismith, J.H.6
Lee, R.E.7
-
7
-
-
0015342854
-
Substituted thiazolidones as anticonvulsants
-
Dwivedi, C.; Gupta, T. K.; Parmar, S. S. Substituted thiazolidones as anticonvulsants. J. Med. Chem. 1972, 15, 553-554.
-
(1972)
J. Med. Chem.
, vol.15
, pp. 553-554
-
-
Dwivedi, C.1
Gupta, T.K.2
Parmar, S.S.3
-
8
-
-
0015261681
-
Substituted thiazolidones and their selective inhibition of nicotinamide-adenine dinucleotide dependent oxidations
-
Parmar, S. S.; Dwivedi, C.; Chaudhari, A.; Gupta, T. K. Substituted thiazolidones and their selective inhibition of nicotinamide-adenine dinucleotide dependent oxidations. J. Med. Chem. 1972, 15, 99-101.
-
(1972)
J. Med. Chem.
, vol.15
, pp. 99-101
-
-
Parmar, S.S.1
Dwivedi, C.2
Chaudhari, A.3
Gupta, T.K.4
-
9
-
-
34250159079
-
Synthesis and antimicrobial evaluation of some new thiazole, thiazolidinone and thiazoline derivatives starting from 1-chloro-3,4- dihydronaphthalene-2-carboxaldehyde
-
DOI 10.1016/j.ejmech.2006.12.025, PII S0223523407000268
-
Bondock, S.; Khalifa, W.; Fadda, A. A. Synthesis and antimicrobial evaluation of some new thiazole, thiazolidinone and thiazoline derivatives starting from 1-chloro-3, 4-dihydronaphthalene-2-carboxaldehyde. Eur. J. Med. Chem. 2007, 42, 948-954. (Pubitemid 46907334)
-
(2007)
European Journal of Medicinal Chemistry
, vol.42
, Issue.7
, pp. 948-954
-
-
Bondock, S.1
Khalifa, W.2
Fadda, A.A.3
-
10
-
-
41649108430
-
2-Heteroarylimino-5-benzylidene-4-thiazolidinones analogues of 2-thiazolylimino-5-benzylidene-4-thiazolidinones with antimicrobial activity: Synthesis and structure-activity relationship
-
DOI 10.1016/j.bmc.2008.02.001, PII S0968089608000941
-
Vicini, P.; Geronikaki, A.; Incerti, M.; Zani, F.; Dearden, J.; Hewitt, M. 2-Heteroarylimino-5-benzylidene-4-thiazolidinones analogues of 2-thiazolylimino-5-benzylidene-4-thiazolidinones with antimicrobial activity: Synthesis and structure-activity relationship. Bioorg. Med. Chem. 2008, 16, 3714-3724. (Pubitemid 351484039)
-
(2008)
Bioorganic and Medicinal Chemistry
, vol.16
, Issue.7
, pp. 3714-3724
-
-
Vicini, P.1
Geronikaki, A.2
Incerti, M.3
Zani, F.4
Dearden, J.5
Hewitt, M.6
-
11
-
-
5344259691
-
Synthesis and antiproliferative activity of 2-aryl-4-oxo-thiazolidin-3- yl- amides for prostate cancer
-
DOI 10.1016/j.bmcl.2004.08.029, PII S0960894X04010376
-
Gududuru, V.; Hurh, E.; Dalton, J. T.; Miller, D. D. Synthesis and antiproliferative activity of 2-aryl-4-oxo-thiazolidin-3-yl-amides for prostate cancer. Bioorg. Med. Chem. Lett. 2004, 14, 5289-5293. (Pubitemid 39348915)
-
(2004)
Bioorganic and Medicinal Chemistry Letters
, vol.14
, Issue.21
, pp. 5289-5293
-
-
Gududuru, V.1
Hurh, E.2
Dalton, J.T.3
Miller, D.D.4
-
12
-
-
23244463167
-
In vitro antiproliferative activity against human colon cancer cell lines of representative 4-thiazolidinones. Part I
-
DOI 10.1016/j.bmcl.2005.05.093, PII S0960894X05006967
-
Ottanà, R.; Carotti, S.; Maccari, R.; Landini, I.; Chiricosta, G.; Caciagli, B.; Vigorita, M. G.; Mini, E. In vitro antiproliferative activity against human colon cancer cell lines of representative 4-thiazolidinones. Part I. Bioorg. Med. Chem. Lett. 2005, 15, 3930-3933. (Pubitemid 41095497)
-
(2005)
Bioorganic and Medicinal Chemistry Letters
, vol.15
, Issue.17
, pp. 3930-3933
-
-
Ottana, R.1
Carotti, S.2
Maccari, R.3
Landini, I.4
Chiricosta, G.5
Caciagli, B.6
Vigorita, M.G.7
Mini, E.8
-
13
-
-
0034518811
-
QSAR studies on antihistaminic activity of some thiazolidine-4-ones
-
Agrawal, V. K.; Sachan, S.; Khadikar, P. V. QSAR studies on antihistaminic activity of some thiazolidine-4-ones. Acta Pharm. 2000, 50, 281-290. (Pubitemid 32049539)
-
(2000)
Acta Pharmaceutica
, vol.50
, Issue.4
, pp. 281-290
-
-
Agrawal, V.K.1
Sachan, S.2
Khadikar, P.V.3
-
14
-
-
0032863170
-
1-histamine antagonists
-
DOI 10.1016/S0014-827X(99)00064-6, PII S0014827X99000646
-
Diurno, M. V.; Mazzoni, O.; Correale, G.; Monterrey, I. G.; Calignano, A.; La Rana, G.; Bolognese, A. Synthesis and structure-activity relationships of 2-(substituted phenyl)-3-[3-(N, Ndimethylamino) - propyl]-1, 3-thiazolidin-4-ones acting as H1-histamine antagonists. II Farmaco 1999, 54, 579-583. (Pubitemid 29462617)
-
(1999)
Farmaco
, vol.54
, Issue.9
, pp. 579-583
-
-
Diurno, M.V.1
Mazzoni, O.2
Correale, G.3
Gomez Monterrey, I.4
Calignano, A.5
La Rana, G.6
Bolognese, A.7
-
15
-
-
72149105339
-
Novel 4-thiazolidinone derivatives as potential antifungal and antibacterial drugs
-
Omar, K.; Geronikaki, A.; Zoumpoulakis, P.; Camoutsis, C.; Sokovic, M.; Ciric, A.; Glamoclija, J.; Novel 4-thiazolidinone derivatives as potential antifungal and antibacterial drugs. Bioorg. Med. Chem. 2010, 18, 426-432.
-
(2010)
Bioorg. Med. Chem.
, vol.18
, pp. 426-432
-
-
Omar, K.1
Geronikaki, A.2
Zoumpoulakis, P.3
Camoutsis, C.4
Sokovic, M.5
Ciric, A.6
Glamoclija, J.7
-
16
-
-
0037334476
-
Chiral 3,3′-(1,2-Ethanediyl)-bis[2-(3,4-dimethoxyphenyl)-4- thiazolidinones] with anti-inflammatory activity. Part 11: Evaluation of COX-2 selectivity and modelling
-
DOI 10.1016/S0968-0896(02)00518-7, PII S0968089602005187
-
Vigorita, M. G.; Ottanà, R.; Monforte, F.; Maccari, R.; Monforte, M. T.; Trovato, A.; Taviano, M. F.; Miceli, N.; De Luca, G.; Alcaro, S.; Ortuso, F. Chiral 3, 3'-(1, 2-ethanediyl)-bis[2-(3, 4-dimethoxyphenyl)-4- thiazolidinones] with anti-inflammatory activity. Part 11: Evaluation of COX-2 selectivity and modeling. Bioorg. Med. Chem. 2003, 11, 999-1006. (Pubitemid 36287059)
-
(2003)
Bioorganic and Medicinal Chemistry
, vol.11
, Issue.6
, pp. 999-1006
-
-
Vigorita, M.G.1
Ottana, R.2
Monforte, F.3
Maccari, R.4
Monforte, M.T.5
Trovato, A.6
Taviano, M.F.7
Miceli, N.8
De Luca, G.9
Alcaro, S.10
Ortuso, F.11
-
17
-
-
27644537621
-
2-(Aryl)-3-furan-2-ylmethyl-thiazolidin-4-ones as selective HIV-RT Inhibitors
-
DOI 10.1016/j.bmc.2005.07.063, PII S0968089605007285
-
Rawal, R. K.; Prabhakar, Y. S.; Katti, S. B.; De Clercq, E. 2-(Aryl)-3-furan-2-ylmethyl-thiazolidin-4-ones as selective HIV-RT Inhibitors. Bioorg. Med. Chem. 2005, 13, 6771-6776. (Pubitemid 41571222)
-
(2005)
Bioorganic and Medicinal Chemistry
, vol.13
, Issue.24
, pp. 6771-6776
-
-
Rawal, R.K.1
Prabhakar, Y.S.2
Katti, S.B.3
De Clercq, E.4
-
18
-
-
0032890436
-
Effects of CP-060S, a novel cardioprotective drug, on cardiac function and myocardial oxygen consumption
-
DOI 10.1016/S0306-3623(98)00062-7, PII S0306362398000627
-
Suzuki, Y.; Akima, M.; Tamura, K. Effects of CP-060S, a novel cardioprotective drug, on cardiac function and myocardial oxygen consumption. Gen. Pharmacol. 1999, 32, 57-63. (Pubitemid 28540791)
-
(1999)
General Pharmacology
, vol.32
, Issue.1
, pp. 57-63
-
-
Suzuki, Y.1
Akima, M.2
Tamura, K.3
-
19
-
-
77953872987
-
Monastrol analogs: A synthesis of pyrazolo-pyridine, benzopyranopyrazolopyridine, and oxygen-bridged azolopyrimidine derivatives and their biological screening
-
Svetlik, J.; Veizerová, L.; Mayer, T. U.; Catarinella, M. Monastrol analogs: A synthesis of pyrazolo-pyridine, benzopyranopyrazolopyridine, and oxygen-bridged azolopyrimidine derivatives and their biological screening. Bioorg. Med. Chem. Lett. 2010, 20, 4073-4076.
-
(2010)
Bioorg. Med. Chem. Lett.
, vol.20
, pp. 4073-4076
-
-
Svetlik, J.1
Veizerová, L.2
Mayer, T.U.3
Catarinella, M.4
-
20
-
-
33645122408
-
Indiplon is a high-affinity positive allosteric modulator with selectivity for alpha1 subunit-containing GABAA receptors
-
Petroski, R. E.; Pomeroy, J. E.; Das, R.; Bowman, H.; Yang, W.; Chen, A. P.; Foster, A. C. Indiplon is a high-affinity positive allosteric modulator with selectivity for alpha1 subunit-containing GABAA receptors. J. Pharmacol. Exp. Ther. 2006, 317, 369-377.
-
(2006)
J. Pharmacol. Exp. Ther.
, vol.317
, pp. 369-377
-
-
Petroski, R.E.1
Pomeroy, J.E.2
Das, R.3
Bowman, H.4
Yang, W.5
Chen, A.P.6
Foster, A.C.7
-
21
-
-
33644762019
-
Comparative cue generalization profiles of L-838,417, SL651498, zolpidem, CL218,872, ocinaplon, bretazenil, zopiclone, and various benzodiazepines in chlordiazepoxide and zolpidem drug discrimination
-
DOI 10.1124/jpet.105.094003
-
Mirza, N. R.; Rodgers, R. J.; Mathiasen, L. S. Comparative cue generalization profiles of L-838, 417, SL651498, zolpidem, CL218, 872, ocinaplon, bretazenil, zopiclone, and various benzodiazepines in chlordiazepoxide and zolpidem drug discrimination. J. Pharmacol. Exp. Ther. 2006, 316, 1291-1299. (Pubitemid 43345305)
-
(2006)
Journal of Pharmacology and Experimental Therapeutics
, vol.316
, Issue.3
, pp. 1291-1299
-
-
Mirza, N.R.1
Rodgers, R.J.2
Mathiasen, L.S.3
-
22
-
-
0034321609
-
Zaleplon: A pyrazolopyrimidine sedative-hypnotic agent for the treatment of insomnia
-
Weitzel, K. W.; Wickman, J. M.; Augustin, S. G.; Strom, J. G. Zaleplon: A pyrazolopyrimidine sedative-hypnotic agent for the treatment of insomnia. Clin. Ther. 2000, 22, 1254-1267.
-
(2000)
Clin. Ther.
, vol.22
, pp. 1254-1267
-
-
Weitzel, K.W.1
Wickman, J.M.2
Augustin, S.G.3
Strom, J.G.4
-
23
-
-
0037124207
-
Pyrazolo[3,4-d]pyrimidines containing an extended 3-substituent as potent inhibitors of Lck - A selectivity insight
-
DOI 10.1016/S0960-894X(02)00196-8, PII S0960894X02001968
-
Burchat, A. F.; Calderwood, D. J.; Friedman, M. M.; Hirst, G. C.; Li, B.; Rafferty, P.; Ritter, K.; Skinner, B. S. Pyrazolo[3, 4-d]pyrimidines containing an extended 3-substituent as potent inhibitors of Lck-A selectivity insight. Bioorg. Med. Chem. Lett. 2002, 12, 1687-1690. (Pubitemid 34569272)
-
(2002)
Bioorganic and Medicinal Chemistry Letters
, vol.12
, Issue.12
, pp. 1687-1690
-
-
Burchat, A.F.1
Calderwood, D.J.2
Friedman, M.M.3
Hirst, G.C.4
Li, B.5
Rafferty, P.6
Ritter, K.7
Skinner, B.S.8
-
24
-
-
33748868675
-
4-(Imidazol-1-yl) thiazol-2-yl phenylamines. A novel Class of highly potent colchicine site binding tubulin inhibitors: Synthesis and cytotoxic activity on selected human cancer cell lines
-
Siavosh, M.; Andreas, S.; Heymo, H.; Emerich, E.; Thomas, B.; Mathias, S.; Thomas, M.; Josef, S. F.; Thomas, B. L. [4-(Imidazol-1-yl) thiazol-2-yl]phenylamines. a novel Class of highly potent colchicine site binding tubulin inhibitors: Synthesis and cytotoxic activity on selected human cancer cell lines. J. Med. Chem. 2006, 49, 5769-5776.
-
(2006)
J. Med. Chem.
, vol.49
, pp. 5769-5776
-
-
Siavosh, M.1
Andreas, S.2
Heymo, H.3
Emerich, E.4
Thomas, B.5
Mathias, S.6
Thomas, M.7
Josef, S.F.8
Thomas, B.L.9
-
25
-
-
38149094889
-
Synthesis and antimicrobial screening of 5-arylidene-2-imino-4- thiazolidinones
-
Chavan, A. A.; Pai, N. R.; Synthesis and antimicrobial screening of 5-arylidene-2-imino-4-thiazolidinones. ARKIVOC 2007, 16, 148-155.
-
(2007)
ARKIVOC
, vol.16
, pp. 148-155
-
-
Chavan, A.A.1
Pai, N.R.2
-
26
-
-
33646071514
-
Synthesis and antimicrobial activity of novel 2-thiazolylimino-5- arylidene-4-thiazolidinones
-
Vicini, P.; Geronikaki, A.; Anastasia, K.; Incerti, M.; Zani, F. Synthesis and antimicrobial activity of novel 2-thiazolylimino-5-arylidene-4- thiazolidinones. Bioorg. Med. Chem. 2006, 14, 3859-3864.
-
(2006)
Bioorg. Med. Chem.
, vol.14
, pp. 3859-3864
-
-
Vicini, P.1
Geronikaki, A.2
Anastasia, K.3
Incerti, M.4
Zani, F.5
-
27
-
-
22544462555
-
Synthetic and theoretical aspects of new dimroth rearrangement of 6-aminopyran-2-ones to 6-hydroxypyridin-2-ones via carbamoyl ketenes
-
DOI 10.1002/ejoc.200400875
-
Subbotina, J. O.; Fabian, W. M. F.; Tarasov, E. V.; Volkova, N. N.; Bakulev, V. A. Synthetic and Theoretical Aspects of New Dimroth Rearrangement of 6-Aminopyran-2-ones to 6-Hydroxypyridin-2-ones via Carbamoyl Ketenes. Eur. J. Org. Chem. 2005, 2914-2923. (Pubitemid 41018408)
-
(2005)
European Journal of Organic Chemistry
, Issue.14
, pp. 2914-2923
-
-
Subbotina, J.O.1
Fabian, W.M.F.2
Tarasov, E.V.3
Volkova, N.N.4
Bakulev, V.A.5
-
28
-
-
84860330558
-
2-Aminothiophenes as building blocks in heterocyclic synthesis: Synthesis and antimicrobial evaluation of a new class of pyrido[1, 2-a]thieno[3, 2-e]pyrimidine, quinoline and pyridin-2-one derivatives
-
Behbehani, H.; Ibrahim, H. M.; Makhseed, S.; Elnagdi, M. H.; Mahmoud, H. 2-Aminothiophenes as building blocks in heterocyclic synthesis: Synthesis and antimicrobial evaluation of a new class of pyrido[1, 2-a]thieno[3, 2-e]pyrimidine, quinoline and pyridin-2-one derivatives. Eur. J. Med. Chem. 2012, 52, 61-65.
-
(2012)
Eur. J. Med. Chem.
, vol.52
, pp. 61-65
-
-
Behbehani, H.1
Ibrahim, H.M.2
Makhseed, S.3
Elnagdi, M.H.4
Mahmoud, H.5
-
29
-
-
79953192257
-
Studies with 3-oxoalkanonitriles: Reactivity of 3-oxo-(1-methylindoloyl) propanenitrile
-
Behbehani, H.; Ibrahim, H. M.; Makhseed, S. Studies with 3-oxoalkanonitriles: Reactivity of 3-oxo-(1-methylindoloyl) propanenitrile. Heterocycles 2009, 78, 3081-3090.
-
(2009)
Heterocycles
, vol.78
, pp. 3081-3090
-
-
Behbehani, H.1
Ibrahim, H.M.2
Makhseed, S.3
-
30
-
-
84862995792
-
-
Crystallographic data for 7c ref. CCDC 875772 can be obtained on request from the director, Cambridge Crystallographic Data Center, 12 Union Road, Cambridge CB2 1EW, UK
-
Crystallographic data for 7c (ref. CCDC 875772) can be obtained on request from the director, Cambridge Crystallographic Data Center, 12 Union Road, Cambridge CB2 1EW, UK.
-
-
-
-
31
-
-
84862997221
-
-
Crystallographic data for 8b ref. CCDC 874404 can be obtained on request from the director, Cambridge Crystallographic Data Center, 12 Union Road, Cambridge CB2 1EW, UK
-
Crystallographic data for 8b (ref. CCDC 874404) can be obtained on request from the director, Cambridge Crystallographic Data Center, 12 Union Road, Cambridge CB2 1EW, UK.
-
-
-
-
32
-
-
84862995795
-
-
Crystallographic data for 11 ref. CCDC 880545 can be obtained on request from the director, Cambridge Crystallographic Data Center, 12 Union Road, Cambridge CB2 1EW, UK
-
Crystallographic data for 11 (ref. CCDC 880545) can be obtained on request from the director, Cambridge Crystallographic Data Center, 12 Union Road, Cambridge CB2 1EW, UK.
-
-
-
-
33
-
-
84862995794
-
-
Crystallographic data for 14 ref. CCDC 880544 can be obtained on request from the director, Cambridge Crystallographic Data Center, 12 Union Road, Cambridge CB2 1EW, UK
-
Crystallographic data for 14 (ref. CCDC 880544) can be obtained on request from the director, Cambridge Crystallographic Data Center, 12 Union Road, Cambridge CB2 1EW, UK.
-
-
-
-
34
-
-
77953464768
-
Synthesis of 7-substituted pyrazolo[1, 5-a]-pyrimidine-3-carboxamides as potential non benzodiazepine hypnotics
-
Behbehani, H.; Ibrahim, H. M.; Makhseed, S. Synthesis of 7-substituted pyrazolo[1, 5-a]-pyrimidine-3-carboxamides as potential non benzodiazepine hypnotics. ARKIVOC 2010, 2, 267-282.
-
(2010)
ARKIVOC
, vol.2
, pp. 267-282
-
-
Behbehani, H.1
Ibrahim, H.M.2
Makhseed, S.3
-
35
-
-
77956190209
-
Synthesis and primary cytotoxicity evaluation of new 5-benzylidene-2, 4-thiazolidinedione derivatives
-
Patil, V.; Tilekar, K.; Mehendale-Munj, S.; Mohan, R.; Ramaa, C. S. Synthesis and primary cytotoxicity evaluation of new 5-benzylidene-2, 4-thiazolidinedione derivatives. Eur. J. Med. Chem. 2010, 45, 4539-4544.
-
(2010)
Eur. J. Med. Chem.
, vol.45
, pp. 4539-4544
-
-
Patil, V.1
Tilekar, K.2
Mehendale-Munj, S.3
Mohan, R.4
Ramaa, C.S.5
|