SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 1, 2011, Pages 200-203

In vitro evaluation of 5-arylidene-2-thioxo-4-thiazolidinones active as aldose reductase inhibitors

(6) MacCari, Rosanna a Corso, Antonella Del b Giglio, Marco a Moschini, Roberta b Mura, Umberto b Ottanà, Rosaria a

a UNIVERSITY OF MESSINA (Italy)

b UNIVERSITY OF PISA (Italy)

Author keywords

4 Thiazolidinones; Aldose reductase; Diabetes complications; Enzyme inhibition

Indexed keywords

(5 ARYLIDENE 4 OXO 2 THIOXOTHIAZOLIDIN 3 YL)ACETIC ACID; 5 ARYLIDENE 2 THIOXO 4 THIAZOLIDINONE DERIVATIVE; ALDOSE REDUCTASE INHIBITOR; EPALRESTAT; SORBINIL; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CONCENTRATION RESPONSE; DRUG EFFICACY; DRUG POTENCY; ENZYME INHIBITION; IN VITRO STUDY; STRUCTURE ACTIVITY RELATION;

EID: 78650513550 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2010.11.041 Document Type: Article

Times cited : (59)

References (36)

1
- 0023899991
- P.F. Kador Med. Res. Rev. 8 1988 325
- (1988) Med. Res. Rev. , vol.8 , pp. 325
- Kador, P.F.¹

2
- 0031920049
- C. Yabe-Nishimura Pharmacol. Rev. 50 1998 21
- (1998) Pharmacol. Rev. , vol.50 , pp. 21
- Yabe-Nishimura, C.¹

3
- 0035856980
- M. Brownlee Nature 414 2001 813
- (2001) Nature , vol.414 , pp. 813
- Brownlee, M.¹

4
- 7044247670
- K.V. Ramana, B. Friedrich, S. Srivastava, A. Bhatnagar, and S.K. Srivastava Diabetes 53 2004 2910
- (2004) Diabetes , vol.53 , pp. 2910
- Ramana, K.V.¹ Friedrich, B.² Srivastava, S.³ Bhatnagar, A.⁴ Srivastava, S.K.⁵

5
- 18844369302
- S.K. Srivastava, K.V. Ramana, and A. Bhatnagar Endocr. Rev. 26 2005 380
- (2005) Endocr. Rev. , vol.26 , pp. 380
- Srivastava, S.K.¹ Ramana, K.V.² Bhatnagar, A.³

6
- 47049121292
- C.A. Gleissner, E. Galkina, J.L. Nadler, and K. Ley Drug Discovery Today Dis. Mech. 4 2007 131
- (2007) Drug Discovery Today Dis. Mech. , vol.4 , pp. 131
- Gleissner, C.A.¹ Galkina, E.² Nadler, J.L.³ Ley, K.⁴

7
- 0032511583
- UK Prospective Diabetes Study (UKPDS) Group D.
- R.C. Turner, R.R. Holman, C.A. Cull, I.M. Stratton, D.R. Matthews, V. Frighi, S.E. Manley, A. Neil, H. McElroy, D. Wright, E. Kohner, C. Fox, D. Hadden UK Prospective Diabetes Study (UKPDS) Group Lancet 352 1998 837
- (1998) Lancet , vol.352 , pp. 837
- Turner, R.C.¹ Holman, R.R.² Cull, C.A.³ Stratton, I.M.⁴ Matthews, D.R.⁵ Frighi, V.⁶ Manley, S.E.⁷ Neil, A.⁸ McElroy, H.⁹ Wright, D.¹⁰ Kohner, E.¹¹ Fox, C.¹² Hadden, D.¹³

8
- 33749321231
- D. Zozulinska, and B. Wierusz-Wysocka Diabetes Res. Clin. Pract. 74S 2006 S12
- (2006) Diabetes Res. Clin. Pract. , vol.74 , pp. 12
- Zozulinska, D.¹ Wierusz-Wysocka, B.²

9
- 2342466734
- S. Wild, G. Roglic, A. Green, R. Sicree, and H. King Diabetes Care 27 2004 1047
- (2004) Diabetes Care , vol.27 , pp. 1047
- Wild, S.¹ Roglic, G.² Green, A.³ Sicree, R.⁴ King, H.⁵

10
- 34249732513
- R. Tammali, K.V. Ramana, and S.K. Srivastava Cancer Lett. 252 2007 299
- (2007) Cancer Lett. , vol.252 , pp. 299
- Tammali, R.¹ Ramana, K.V.² Srivastava, S.K.³

11
- 65649103414
- P. Alexiou, K. Pegklidou, M. Chatzopoulou, I. Nicolaou, and V.J. Demopoulos Curr. Med. Chem. 16 2009 734
- (2009) Curr. Med. Chem. , vol.16 , pp. 734
- Alexiou, P.¹ Pegklidou, K.² Chatzopoulou, M.³ Nicolaou, I.⁴ Demopoulos, V.J.⁵

12
- 70749089191
- K.V. Ramana, and S.K. Srivastava Int. J. Biochem. Cell Biol. 42 2010 17
- (2010) Int. J. Biochem. Cell Biol. , vol.42 , pp. 17
- Ramana, K.V.¹ Srivastava, S.K.²

13
- 0030751728
- L. Costantino, G. Rastelli, G. Cignarella, P. Vianello, and D. Barlocco Exp. Opin. Ther. Patents 7 1997 843
- (1997) Exp. Opin. Ther. Patents , vol.7 , pp. 843
- Costantino, L.¹ Rastelli, G.² Cignarella, G.³ Vianello, P.⁴ Barlocco, D.⁵

14
- 2442516583
- S. Miyamoto Chem. Biol. Inform. J. 2 2002 74
- (2002) Chem. Biol. Inform. J. , vol.2 , pp. 74
- Miyamoto, S.¹

15
- 0042309876
- S. Suzen, and E. Buyukbingol Curr. Med. Chem. 10 2003 1329
- (2003) Curr. Med. Chem. , vol.10 , pp. 1329
- Suzen, S.¹ Buyukbingol, E.²

16
- 0031570301
- A. Urzhumtsev, F. Tête-Favier, A. Mitschler, J. Barbanton, P. Barth, L. Urzhumtseva, J.F. Biellmann, A. Podjarny, and D. Moras Structure 5 1997 601
- (1997) Structure , vol.5 , pp. 601
- Urzhumtsev, A.¹ Tête-Favier, F.² Mitschler, A.³ Barbanton, J.⁴ Barth, P.⁵ Urzhumtseva, L.⁶ Biellmann, J.F.⁷ Podjarny, A.⁸ Moras, D.⁹

17
- 0032578366
- O. El-Kabbani, D.K. Wilson, J.M. Petrash, and F.A. Quiocho Mol. Vis. 4 1998 19
- (1998) Mol. Vis. , vol.4 , pp. 19
- El-Kabbani, O.¹ Wilson, D.K.² Petrash, J.M.³ Quiocho, F.A.⁴

18
- 2542571016
- E.I. Howard, R. Sanishvili, R.E. Cachau, A. Mitschler, B. Chevrier, P. Barth, V. Lamour, M. Van Zandt, E. Sibley, C. Bon, D. Moras, T.R. Schneider, A. Joachimiak, and A. Podjarny Proteins 55 2004 792
- (2004) Proteins , vol.55 , pp. 792
- Howard, E.I.¹ Sanishvili, R.² Cachau, R.E.³ Mitschler, A.⁴ Chevrier, B.⁵ Barth, P.⁶ Lamour, V.⁷ Van Zandt, M.⁸ Sibley, E.⁹ Bon, C.¹⁰ Moras, D.¹¹ Schneider, T.R.¹² Joachimiak, A.¹³ Podjarny, A.¹⁴

19
- 2642569349
- C.A. Sotriffer, O. Krämer, and G. Klebe Proteins 56 2004 52
- (2004) Proteins , vol.56 , pp. 52
- Sotriffer, C.A.¹ Krämer, O.² Klebe, G.³

20
- 0032959371
- L. Costantino, G. Rastelli, P. Vianello, G. Cignarella, and D. Barlocco Med. Res. Rev. 19 1999 3
- (1999) Med. Res. Rev. , vol.19 , pp. 3
- Costantino, L.¹ Rastelli, G.² Vianello, P.³ Cignarella, G.⁴ Barlocco, D.⁵

21
- 0020526445
- R. Kikkawa, I. Hatanaka, H. Yasuda, N. Kobayashi, Y. Shigeta, H. Terashima, T. Morimura, and M. Tsuboshima Diabetologia 24 1983 290
- (1983) Diabetologia , vol.24 , pp. 290
- Kikkawa, R.¹ Hatanaka, I.² Yasuda, H.³ Kobayashi, N.⁴ Shigeta, Y.⁵ Terashima, H.⁶ Morimura, T.⁷ Tsuboshima, M.⁸

22
- 0021276233
- H. Terashima, K. Hama, R. Yamamoto, M. Tsuboshima, R. Kikkawa, I. Hatanaka, and Y. Shigeta J. Pharmacol. Exp. Ther. 229 1984 226
- (1984) J. Pharmacol. Exp. Ther. , vol.229 , pp. 226
- Terashima, H.¹ Hama, K.² Yamamoto, R.³ Tsuboshima, M.⁴ Kikkawa, R.⁵ Hatanaka, I.⁶ Shigeta, Y.⁷

23
- 42949097094
- M.A. Ramirez, and N.L. Borja Pharmacotherapy 28 2008 646
- (2008) Pharmacotherapy , vol.28 , pp. 646
- Ramirez, M.A.¹ Borja, N.L.²

24
- 49649122550
- N. Hotta, R. Kawamori, Y. Atsumi, M. Baba, H. Kishikawa, J. Nakamura, S. Oikawa, N. Yamada, H. Yasuda, and Y. Shigeta Diabetes Med. 25 2008 818
- (2008) Diabetes Med. , vol.25 , pp. 818
- Hotta, N.¹ Kawamori, R.² Atsumi, Y.³ Baba, M.⁴ Kishikawa, H.⁵ Nakamura, J.⁶ Oikawa, S.⁷ Yamada, N.⁸ Yasuda, H.⁹ Shigeta, Y.¹⁰

25
- 0032548075
- P. Fresneau, M. Cussac, J. Morand, B. Szymonski, D. Tranqui, and G. Leclerc J. Med. Chem. 41 1998 4706
- (1998) J. Med. Chem. , vol.41 , pp. 4706
- Fresneau, P.¹ Cussac, M.² Morand, J.³ Szymonski, B.⁴ Tranqui, D.⁵ Leclerc, G.⁶

26
- 15244355411
- R. Maccari, R. Ottan, C. Curinga, M.G. Vigorita, D. Rakowitz, T. Steindl, and T. Langer Bioorg. Med. Chem. 13 2005 2809
- (2005) Bioorg. Med. Chem. , vol.13 , pp. 2809
- MacCari, R.¹ Ottan, R.² Curinga, C.³ Vigorita, M.G.⁴ Rakowitz, D.⁵ Steindl, T.⁶ Langer, T.⁷

27
- 34250337361
- R. Maccari, R. Ottan, R. Ciurleo, M.G. Vigorita, D. Rakowitz, T. Steindl, and T. Langer Bioorg. Med. Chem. Lett. 17 2007 3886
- (2007) Bioorg. Med. Chem. Lett. , vol.17 , pp. 3886
- MacCari, R.¹ Ottan, R.² Ciurleo, R.³ Vigorita, M.G.⁴ Rakowitz, D.⁵ Steindl, T.⁶ Langer, T.⁷

28
- 44449137462
- R. Maccari, R. Ottan, R. Ciurleo, D. Rakowitz, B. Matuszczak, C. Laggner, and T. Langer Bioorg. Med. Chem. 16 2008 5840
- (2008) Bioorg. Med. Chem. , vol.16 , pp. 5840
- MacCari, R.¹ Ottan, R.² Ciurleo, R.³ Rakowitz, D.⁴ Matuszczak, B.⁵ Laggner, C.⁶ Langer, T.⁷

29
- 0036169268
- G. Bruno, L. Costantino, C. Curinga, R. Maccari, F. Monforte, F. Nicol, R. Ottan, and M.G. Vigorita Bioorg. Med. Chem. 10 2002 1077
- (2002) Bioorg. Med. Chem. , vol.10 , pp. 1077
- Bruno, G.¹ Costantino, L.² Curinga, C.³ MacCari, R.⁴ Monforte, F.⁵ Nicol, F.⁶ Ottan, R.⁷ Vigorita, M.G.⁸

30
- 77953137883
- R. Maccari, R. Ciurleo, M. Giglio, M. Cappiello, R. Moschini, A. Del Corso, U. Mura, and R. Ottan Bioorg. Med. Chem. 18 2010 4049
- (2010) Bioorg. Med. Chem. , vol.18 , pp. 4049
- MacCari, R.¹ Ciurleo, R.² Giglio, M.³ Cappiello, M.⁴ Moschini, R.⁵ Del Corso, A.⁶ Mura, U.⁷ Ottan, R.⁸

31
- 78650515354
- SciFinder, https://scifinder.cas.org.

32
- 78650515144
- Bue-Valleskey, J. M.; Hunden, D. C.; Jones, C. D.; Panetta, J. A.; Shaw, W. N. U.S. 1996, US 5523314.
- Bue-Valleskey, J. M.; Hunden, D. C.; Jones, C. D.; Panetta, J. A.; Shaw, W. N. U.S. 1996, US 5523314.

33
- 78650514807
- Kaarsholm, N. C.; Madsen, P.; Schlein, M.; Olsen, H. B.; Havelund, S.; Steensgaard, D. B.; Ludvigsen, S.; Jakobsen, P.; Petersen, A. K.; Schluckebier, G. PCT Int. Appl. WO 2004056347, 2004.
- Kaarsholm, N. C.; Madsen, P.; Schlein, M.; Olsen, H. B.; Havelund, S.; Steensgaard, D. B.; Ludvigsen, S.; Jakobsen, P.; Petersen, A. K.; Schluckebier, G. PCT Int. Appl. WO 2004056347, 2004.

34
- 58549100461
- A.J. Russell, I.M. Westwood, M.H.J. Crawford, J. Robinson, A. Kawamura, C. Redfield, N. Laurieri, E.D. Lowe, S.G. Davies, and E. Sim Bioorg. Med. Chem. 17 2009 905
- (2009) Bioorg. Med. Chem. , vol.17 , pp. 905
- Russell, A.J.¹ Westwood, I.M.² Crawford, M.H.J.³ Robinson, J.⁴ Kawamura, A.⁵ Redfield, C.⁶ Laurieri, N.⁷ Lowe, E.D.⁸ Davies, S.G.⁹ Sim, E.¹⁰

35
- 0025667192
- A. Del Corso, D. Barsacchi, M. Giannessi, M.G. Tozzi, M. Camici, J.L. Houben, M. Zandomeneghi, and U. Mura Arch. Biochem. Biophys. 283 1990 512
- (1990) Arch. Biochem. Biophys. , vol.283 , pp. 512
- Del Corso, A.¹ Barsacchi, D.² Giannessi, M.³ Tozzi, M.G.⁴ Camici, M.⁵ Houben, J.L.⁶ Zandomeneghi, M.⁷ Mura, U.⁸

36
- 78650511173
- Values calculated by means of the freely accessible web tool Marvin Calculator Plugins
- a and molecular polarizability values of compounds 1-4 are available in the Supplementary data.

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.