-
1
-
-
0034112037
-
2 receptor
-
A.E. Alewijnse, H. Timmerman, E.H. Jacobs, M.J. Smit, E. Roovers, and S. Cotecchia The effect of mutations in the DRY motif on the constitutive activity and structural instability of the histamine H(2) receptor Molecular Pharmacology 57 2000 890 898 (Pubitemid 30253371)
-
(2000)
Molecular Pharmacology
, vol.57
, Issue.5
, pp. 890-898
-
-
Alewijnse, A.E.1
Timmerman, H.2
Jacobs, E.H.3
Smit, M.J.4
Roovers, E.5
Cotecchia, S.6
Leurs, R.7
-
2
-
-
0035800850
-
Activation of the beta 2-adrenergic receptor involves disruption of an ionic lock between the cytoplasmic ends of transmembrane segments 3 and 6
-
J.A. Ballesteros, A.D. Jensen, G. Liapakis, S.G. Rasmussen, L. Shi, and U. Gether Activation of the beta 2-adrenergic receptor involves disruption of an ionic lock between the cytoplasmic ends of transmembrane segments 3 and 6 The Journal of Biological Chemistry 276 31 2001 29171 29177
-
(2001)
The Journal of Biological Chemistry
, vol.276
, Issue.31
, pp. 29171-29177
-
-
Ballesteros, J.A.1
Jensen, A.D.2
Liapakis, G.3
Rasmussen, S.G.4
Shi, L.5
Gether, U.6
-
3
-
-
76749100307
-
Preparation of stable isotope-labeled peripheral cannabinoid receptor CB2 by bacterial fermentation
-
C. Berger, J.T. Ho, T. Kimura, S. Hess, K. Gawrisch, and A. Yeliseev Preparation of stable isotope-labeled peripheral cannabinoid receptor CB2 by bacterial fermentation Protein Expression and Purification 70 2010 236 247
-
(2010)
Protein Expression and Purification
, vol.70
, pp. 236-247
-
-
Berger, C.1
Ho, J.T.2
Kimura, T.3
Hess, S.4
Gawrisch, K.5
Yeliseev, A.6
-
4
-
-
50149116588
-
Agonist-induced conformational changes in bovine rhodopsin: Insight into activation of G-protein-coupled receptors
-
S. Bhattacharya, S.E. Hall, and N. Vaidehi Agonist-induced conformational changes in bovine rhodopsin: Insight into activation of G-protein-coupled receptors Journal of Molecular Biology 382 2008 539 555
-
(2008)
Journal of Molecular Biology
, vol.382
, pp. 539-555
-
-
Bhattacharya, S.1
Hall, S.E.2
Vaidehi, N.3
-
5
-
-
36448995359
-
2-adrenergic G protein-coupled receptor
-
DOI 10.1126/science.1150577
-
V. Cherezov, D.M. Rosenbaum, M.A. Hanson, S.G. Rasmussen, F.S. Thian, and T.S. Kobilka High-resolution crystal structure of an engineered human beta2-adrenergic G protein-coupled receptor Science 318 2007 1258 1265 (Pubitemid 350172884)
-
(2007)
Science
, vol.318
, Issue.5854
, pp. 1258-1265
-
-
Cherezov, V.1
Rosenbaum, D.M.2
Hanson, M.A.3
Rasmussen, S.G.F.4
Foon, S.T.5
Kobilka, T.S.6
Choi, H.-J.7
Kuhn, P.8
Weis, W.I.9
Kobilka, B.K.10
Stevens, R.C.11
-
6
-
-
78449305788
-
Structure of the human dopamine D3 receptor in complex with a D2/D3 selective antagonist
-
E.Y. Chien, W. Liu, Q. Zhao, V. Katritch, G.W. Han, and M.A. Hanson Structure of the human dopamine D3 receptor in complex with a D2/D3 selective antagonist Science 330 2010 1091 1095
-
(2010)
Science
, vol.330
, pp. 1091-1095
-
-
Chien, E.Y.1
Liu, W.2
Zhao, Q.3
Katritch, V.4
Han, G.W.5
Hanson, M.A.6
-
7
-
-
84859782842
-
Mistic and TarCF as fusion protein partners for functional expression of the cannabinoid receptor 2 in Escherichia coli
-
A. Chowdhury, R. Feng, Q. Tong, Y. Zhang, and X.-Q. Xie Mistic and TarCF as fusion protein partners for functional expression of the cannabinoid receptor 2 in Escherichia coli Protein Expression and Purification 83 2012 128 134
-
(2012)
Protein Expression and Purification
, vol.83
, pp. 128-134
-
-
Chowdhury, A.1
Feng, R.2
Tong, Q.3
Zhang, Y.4
Xie, X.-Q.5
-
8
-
-
34548438468
-
Activation of G Protein-Coupled Receptors
-
DOI 10.1016/S0065-3233(07)74004-4, PII S0065323307740044, Mechanisms and Pathways of Heterotrimeric G Protein Signaling
-
X. Deupi, and B. Kobilka Activation of G protein-coupled receptors Advances in Protein Chemistry 74 2007 137 166 (Pubitemid 47369749)
-
(2007)
Advances in Protein Chemistry
, vol.74
, pp. 137-166
-
-
Deupi, X.1
Kobilka, B.2
-
9
-
-
34147102293
-
G-protein-coupled receptors: An update
-
DOI 10.1111/j.1365-201X.2007.01689.x
-
B.B. Fredholm, T. Hokfelt, and G. Milligan G-protein-coupled receptors: An update Acta Physiologica (Oxford, England) 190 2007 3 7 (Pubitemid 46570172)
-
(2007)
Acta Physiologica
, vol.190
, Issue.1
, pp. 3-7
-
-
Fredholm, B.B.1
Hokfelt, T.2
Milligan, G.3
-
10
-
-
0038024615
-
The G-protein-coupled receptors in the human genome form five main families. Phylogenetic analysis, paralogon groups, and fingerprints
-
DOI 10.1124/mol.63.6.1256
-
R. Fredriksson, M.C. Lagerstrom, L.G. Lundin, and H.B. Schioth The G-protein-coupled receptors in the human genome form five main families. Phylogenetic analysis, paralogon groups, and fingerprints Molecular Pharmacology 63 2003 1256 1272 (Pubitemid 36627220)
-
(2003)
Molecular Pharmacology
, vol.63
, Issue.6
, pp. 1256-1272
-
-
Fredriksson, R.1
Lagerstrom, M.C.2
Lundin, L.-G.3
Schioth, H.B.4
-
11
-
-
0141811657
-
1 angiotensin receptor activation and signaling
-
DOI 10.1210/en.2002-0135
-
Z. Gaborik, G. Jagadeesh, M. Zhang, A. Spat, K.J. Catt, and L. Hunyady The role of a conserved region of the second intracellular loop in AT1 angiotensin receptor activation and signaling Endocrinology 144 2003 2220 2228 (Pubitemid 36629870)
-
(2003)
Endocrinology
, vol.144
, Issue.6
, pp. 2220-2228
-
-
Gaborik, Z.1
Jagadeesh, G.2
Zhang, M.3
Spat, A.4
Catt, K.J.5
Hunyady, L.6
-
12
-
-
0031018485
-
Structural instability of a constitutively active G protein-coupled receptor. Agonist-independent activation due to conformational flexibility
-
DOI 10.1074/jbc.272.5.2587
-
U. Gether, J.A. Ballesteros, R. Seifert, E. Sanders-Bush, H. Weinstein, and B.K. Kobilka Structural instability of a constitutively active G protein-coupled receptor. Agonist-independent activation due to conformational flexibility The Journal of Biological Chemistry 272 1997 2587 2590 (Pubitemid 27053295)
-
(1997)
Journal of Biological Chemistry
, vol.272
, Issue.5
, pp. 2587-2590
-
-
Gether, U.1
Ballesteros, J.A.2
Seifert, R.3
Sanders-Bush, E.4
Weinstein, H.5
Kobilka, B.K.6
-
13
-
-
78650526380
-
Highly conserved tyrosine stabilizes the active state of rhodopsin
-
J.A. Goncalves, K. South, S. Ahuja, E. Zaitseva, C.A. Opefi, and M. Eilers Highly conserved tyrosine stabilizes the active state of rhodopsin Proceedings of the National Academy of Sciences of the United States of America 107 46 2010 19861 19866
-
(2010)
Proceedings of the National Academy of Sciences of the United States of America
, vol.107
, Issue.46
, pp. 19861-19866
-
-
Goncalves, J.A.1
South, K.2
Ahuja, S.3
Zaitseva, E.4
Opefi, C.A.5
Eilers, M.6
-
14
-
-
77952921531
-
A lipid pathway for ligand binding is necessary for a cannabinoid G protein-coupled receptor
-
D.P. Hurst, A. Grossfield, D.L. Lynch, S. Feller, T.D. Romo, and K. Gawrisch A lipid pathway for ligand binding is necessary for a cannabinoid G protein-coupled receptor The Journal of Biological Chemistry 285 2010 17954 17964
-
(2010)
The Journal of Biological Chemistry
, vol.285
, pp. 17954-17964
-
-
Hurst, D.P.1
Grossfield, A.2
Lynch, D.L.3
Feller, S.4
Romo, T.D.5
Gawrisch, K.6
-
15
-
-
56749103466
-
The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist
-
V.P. Jaakola, M.T. Griffith, M.A. Hanson, V. Cherezov, E.Y. Chien, and J.R. Lane The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist Science 322 2008 1211 1217
-
(2008)
Science
, vol.322
, pp. 1211-1217
-
-
Jaakola, V.P.1
Griffith, M.T.2
Hanson, M.A.3
Cherezov, V.4
Chien, E.Y.5
Lane, J.R.6
-
16
-
-
26444467486
-
Linking agonist binding to histamine H1 receptor activation
-
A. Jongejan, M. Bruysters, J.A. Ballesteros, E. Haaksma, R.A. Bakker, and L. Pardo Linking agonist binding to histamine H1 receptor activation Nature Chemical Biology 1 2005 98 103
-
(2005)
Nature Chemical Biology
, vol.1
, pp. 98-103
-
-
Jongejan, A.1
Bruysters, M.2
Ballesteros, J.A.3
Haaksma, E.4
Bakker, R.A.5
Pardo, L.6
-
17
-
-
34447633368
-
Conformational complexity of G-protein-coupled receptors
-
DOI 10.1016/j.tips.2007.06.003, PII S0165614707001459, Allosterism and Collateral Efficacy
-
B.K. Kobilka, and X. Deupi Conformational complexity of G-protein-coupled receptors Trends in Pharmacological Sciences 28 2007 397 406 (Pubitemid 47087966)
-
(2007)
Trends in Pharmacological Sciences
, vol.28
, Issue.8
, pp. 397-406
-
-
Kobilka, B.K.1
Deupi, X.2
-
18
-
-
36448944318
-
Expression and purification of CB2 for NMR studies in micellar solution
-
DOI 10.2174/092986607782541051
-
D. Krepkiy, K. Gawrisch, and A. Yeliseev Expression and purification of CB2 for NMR studies in micellar solution Protein and Peptide Letters 14 2007 1031 1037 (Pubitemid 350164242)
-
(2007)
Protein and Peptide Letters
, vol.14
, Issue.10
, pp. 1031-1037
-
-
Krepkiy, D.1
Gawrisch, K.2
Yeliseev, A.3
-
19
-
-
0029832901
-
Transmembrane regions V and VI of the human luteinizing hormone receptor are required for constitutive activation by a mutation in the third intracellular loop
-
DOI 10.1074/jbc.271.37.22470
-
M. Kudo, Y. Osuga, B.K. Kobilka, and A.J. Hsueh Transmembrane regions V and VI of the human luteinizing hormone receptor are required for constitutive activation by a mutation in the third intracellular loop The Journal of Biological Chemistry 271 1996 22470 22478 (Pubitemid 26304683)
-
(1996)
Journal of Biological Chemistry
, vol.271
, Issue.37
, pp. 22470-22478
-
-
Kudo, M.1
Osuga, Y.2
Kobilka, B.K.3
Hsueh, A.J.W.4
-
20
-
-
37849186561
-
Cannabinoid CB1 receptor recognition of endocannabinoids via the lipid bilayer: Molecular dynamics simulations of CB1 transmembrane helix 6 and anandamide in a phospholipid bilayer
-
DOI 10.1007/s10822-006-9068-9
-
D.L. Lynch, and P.H. Reggio Cannabinoid CB1 receptor recognition of endocannabinoids via the lipid bilayer: molecular dynamics simulations of CB1 transmembrane helix 6 and anandamide in a phospholipid bilayer Journal of Computer-Aided Molecular Design 20 2006 495 509 (Pubitemid 44823886)
-
(2006)
Journal of Computer-Aided Molecular Design
, vol.20
, Issue.7-8
, pp. 495-509
-
-
Lynch, D.L.1
Reggio, P.H.2
-
21
-
-
9144224914
-
1 receptor activation
-
DOI 10.1074/jbc.M406648200
-
S.D. McAllister, D.P. Hurst, J. Barnett-Norris, D. Lynch, P.H. Reggio, and M.E. Abood Structural mimicry in class A G protein-coupled receptor rotamer toggle switches: The importance of the F3.36(201)/W6.48(357) interaction in cannabinoid CB1 receptor activation The Journal of Biological Chemistry 279 2004 48024 48037 (Pubitemid 39540955)
-
(2004)
Journal of Biological Chemistry
, vol.279
, Issue.46
, pp. 48024-48037
-
-
McAllister, S.D.1
Hurst, D.P.2
Barnett-Norris, J.3
Lynch, D.4
Reggio, P.H.5
Abood, M.E.6
-
22
-
-
0242522905
-
1 Receptor Constitutes an Agonist/Inverse Agonist Binding Region
-
DOI 10.1021/jm0302647
-
S.D. McAllister, G. Rizvi, S. Anavi-Goffer, D.P. Hurst, J. Barnett-Norris, and D.L. Lynch An aromatic microdomain at the cannabinoid CB(1) receptor constitutes an agonist/inverse agonist binding region Journal of Medicinal Chemistry 46 2003 5139 5152 (Pubitemid 37414184)
-
(2003)
Journal of Medicinal Chemistry
, vol.46
, Issue.24
, pp. 5139-5152
-
-
McAllister, S.D.1
Rizvi, G.2
Anavi-Goffer, S.3
Hurst, D.P.4
Barnett-Norris, J.5
Lynch, D.L.6
Reggio, P.H.7
Abood, M.E.8
-
23
-
-
0037020296
-
Functional immobilization of a ligand-activated G-protein-coupled receptor
-
DOI 10.1002/1439-7633(20021004)3:10<993::AID-CBIC993>3.0.CO;2-Y
-
L. Neumann, T. Wohland, R.J. Whelan, R.N. Zare, and B.K. Kobilka Functional immobilization of a ligand-activated G-protein-coupled receptor Chembiochem 3 2002 993 998 (Pubitemid 35177752)
-
(2002)
ChemBioChem
, vol.3
, Issue.10
, pp. 993-998
-
-
Neumann, L.1
Wohland, T.2
Whelan, R.J.3
Zare, R.N.4
Kobilka, B.K.5
-
24
-
-
65449161390
-
Ligand binding and micro-switches in 7TM receptor structures
-
R. Nygaard, T.M. Frimurer, B. Holst, M.M. Rosenkilde, and T.W. Schwartz Ligand binding and micro-switches in 7TM receptor structures Trends in Pharmacological Sciences 30 2009 249 259
-
(2009)
Trends in Pharmacological Sciences
, vol.30
, pp. 249-259
-
-
Nygaard, R.1
Frimurer, T.M.2
Holst, B.3
Rosenkilde, M.M.4
Schwartz, T.W.5
-
25
-
-
82955248059
-
Uncovering the intimate relationship between lipids, cholesterol and GPCR activation
-
J. Oates, and A. Watts Uncovering the intimate relationship between lipids, cholesterol and GPCR activation Current Opinion in Structural Biology 21 2011 802 807
-
(2011)
Current Opinion in Structural Biology
, vol.21
, pp. 802-807
-
-
Oates, J.1
Watts, A.2
-
26
-
-
36248970132
-
2 adrenergic G-protein-coupled receptor
-
DOI 10.1038/nature06325, PII NATURE06325
-
S.G. Rasmussen, H.J. Choi, D.M. Rosenbaum, T.S. Kobilka, F.S. Thian, and P.C. Edwards Crystal structure of the human beta2 adrenergic G-protein-coupled receptor Nature 450 2007 383 387 (Pubitemid 350126755)
-
(2007)
Nature
, vol.450
, Issue.7168
, pp. 383-387
-
-
Rasmussen, S.G.F.1
Choi, H.-J.2
Rosenbaum, D.M.3
Kobilka, T.S.4
Thian, F.S.5
Edwards, P.C.6
Burghammer, M.7
Ratnala, V.R.P.8
Sanishvili, R.9
Fischetti, R.F.10
Schertler, G.F.X.11
Weis, W.I.12
Kobilka, B.K.13
-
27
-
-
36448978229
-
2-adrenergic receptor function
-
DOI 10.1126/science.1150609
-
D.M. Rosenbaum, V. Cherezov, M.A. Hanson, S.G. Rasmussen, F.S. Thian, and T.S. Kobilka GPCR engineering yields high-resolution structural insights into beta2-adrenergic receptor function Science 318 2007 1266 1273 (Pubitemid 350172885)
-
(2007)
Science
, vol.318
, Issue.5854
, pp. 1266-1273
-
-
Rosenbaum, D.M.1
Cherezov, V.2
Hanson, M.A.3
Rasmussen, S.G.F.4
Foon, S.T.5
Kobilka, T.S.6
Choi, H.-J.7
Yao, X.-J.8
Weis, W.I.9
Stevens, R.C.10
Kobilka, B.K.11
-
28
-
-
0029897495
-
Constitutively active mutants of the α(1B)-adrenergic receptor: Role of highly conserved polar amino acids in receptor activation
-
A. Scheer, F. Fanelli, T. Costa, P.G. De Benedetti, and S. Cotecchia Constitutively active mutants of the alpha 1B-adrenergic receptor: Role of highly conserved polar amino acids in receptor activation The EMBO Journal 15 1996 3566 3578 (Pubitemid 26239769)
-
(1996)
EMBO Journal
, vol.15
, Issue.14
, pp. 3566-3578
-
-
Scheer, A.1
Fanelli, F.2
Costa, T.3
De Benedetti, P.G.4
Cotecchia, S.5
-
29
-
-
0030614337
-
The activation process of the alpha1B-adrenergic receptor: Potential role of protonation and hydrophobicity of a highly conserved aspartate
-
A. Scheer, F. Fanelli, T. Costa, P.G. De Benedetti, and S. Cotecchia The activation process of the alpha1B-adrenergic receptor: Potential role of protonation and hydrophobicity of a highly conserved aspartate Proceedings of the National Academy of Sciences of the United States of America 94 1997 808 813
-
(1997)
Proceedings of the National Academy of Sciences of the United States of America
, vol.94
, pp. 808-813
-
-
Scheer, A.1
Fanelli, F.2
Costa, T.3
De Benedetti, P.G.4
Cotecchia, S.5
-
30
-
-
77951055595
-
Impact of the DRY motif and the missing "ionic lock" on constitutive activity and G-protein coupling of the human histamine H4 receptor
-
E.H. Schneider, D. Schnell, A. Strasser, S. Dove, and R. Seifert Impact of the DRY motif and the missing "ionic lock" on constitutive activity and G-protein coupling of the human histamine H4 receptor The Journal of Pharmacology and Experimental Therapeutics 333 2 2010 382 392
-
(2010)
The Journal of Pharmacology and Experimental Therapeutics
, vol.333
, Issue.2
, pp. 382-392
-
-
Schneider, E.H.1
Schnell, D.2
Strasser, A.3
Dove, S.4
Seifert, R.5
-
31
-
-
33144459843
-
Molecular mechanism of 7TM receptor activation - A global toggle switch model
-
DOI 10.1146/annurev.pharmtox.46.120604.141218
-
T.W. Schwartz, T.M. Frimurer, B. Holst, M.M. Rosenkilde, and C.E. Elling Molecular mechanism of 7TM receptor activation-A global toggle switch model Annual Review of Pharmacology and Toxicology 46 2006 481 519 (Pubitemid 43271198)
-
(2006)
Annual Review of Pharmacology and Toxicology
, vol.46
, pp. 481-519
-
-
Schwartz, T.W.1
Frimurer, T.M.2
Holst, B.3
Rosenkilde, M.M.4
Elling, C.E.5
-
32
-
-
0037174606
-
β2 adrenergic receptor activation: Modulation of the proline kink in transmembrane 6 by a rotamer toggle switch
-
DOI 10.1074/jbc.M206801200
-
L. Shi, G. Liapakis, R. Xu, F. Guarnieri, J.A. Ballesteros, and J.A. Javitch Beta2 adrenergic receptor activation. Modulation of the proline kink in transmembrane 6 by a rotamer toggle switch The Journal of Biological Chemistry 277 2002 40989 40996 (Pubitemid 35215688)
-
(2002)
Journal of Biological Chemistry
, vol.277
, Issue.43
, pp. 40989-40996
-
-
Shi, L.1
Liapakis, G.2
Xu, R.3
Guarnieri, F.4
Ballesteros, J.A.5
Javitch, J.A.6
-
33
-
-
79960070651
-
Structure of the human histamine H1 receptor complex with doxepin
-
T. Shimamura, M. Shiroishi, S. Weyand, H. Tsujimoto, G. Winter, and V. Katritch Structure of the human histamine H1 receptor complex with doxepin Nature 475 2011 65 70
-
(2011)
Nature
, vol.475
, pp. 65-70
-
-
Shimamura, T.1
Shiroishi, M.2
Weyand, S.3
Tsujimoto, H.4
Winter, G.5
Katritch, V.6
-
34
-
-
0037020273
-
Crystal structure of rhodopsin: A G-protein-coupled receptor
-
DOI 10.1002/1439-7633(20021004)3:10<963::AID-CBIC963>3.0.CO;2-9
-
R.E. Stenkamp, D.C. Teller, and K. Palczewski Crystal structure of rhodopsin: A G-protein-coupled receptor Chembiochem 3 2002 963 967 (Pubitemid 35177747)
-
(2002)
ChemBioChem
, vol.3
, Issue.10
, pp. 963-967
-
-
Stenkamp, R.E.1
Teller, D.C.2
Palczewski, K.3
-
35
-
-
20444499405
-
2 adrenoceptor binding site with catechol reveals differences in binding and activation by agonists and partial agonists
-
DOI 10.1074/jbc.M502352200
-
G. Swaminath, X. Deupi, T.W. Lee, W. Zhu, F.S. Thian, and T.S. Kobilka Probing the beta2 adrenoceptor binding site with catechol reveals differences in binding and activation by agonists and partial agonists The Journal of Biological Chemistry 280 2005 22165 22171 (Pubitemid 40827872)
-
(2005)
Journal of Biological Chemistry
, vol.280
, Issue.23
, pp. 22165-22171
-
-
Swaminath, G.1
Deupi, X.2
Lee, T.W.3
Zhu, W.4
Thian, F.S.5
Kobilka, T.S.6
Kobilka, B.7
-
36
-
-
0345791508
-
2 adrenoceptor. Kinetic evidence for intermediate conformational states
-
DOI 10.1074/jbc.M310888200
-
G. Swaminath, Y. Xiang, T.W. Lee, J. Steenhuis, C. Parnot, and B.K. Kobilka Sequential binding of agonists to the beta2 adrenoceptor. Kinetic evidence for intermediate conformational states The Journal of Biological Chemistry 279 2004 686 691 (Pubitemid 38044873)
-
(2004)
Journal of Biological Chemistry
, vol.279
, Issue.1
, pp. 686-691
-
-
Swaminath, G.1
Xiang, Y.2
Lee, T.W.3
Steenhuis, J.4
Parnot, C.5
Kobilka, B.K.6
-
37
-
-
41949112361
-
Toward Deciphering the Code to Aminergic G Protein-Coupled Receptor Drug Design
-
DOI 10.1016/j.chembiol.2008.03.004, PII S1074552108001154
-
E.S. Tan, E.S. Groban, M.P. Jacobson, and T.S. Scanlan Toward deciphering the code to aminergic G protein-coupled receptor drug design Chemical Biology 15 2008 343 353 (Pubitemid 351508426)
-
(2008)
Chemistry and Biology
, vol.15
, Issue.4
, pp. 343-353
-
-
Tan, E.S.1
Groban, E.S.2
Jacobson, M.P.3
Scanlan, T.S.4
-
38
-
-
84858164791
-
Action of molecular switches in GPCRs - Theoretical and experimental studies
-
B. Trzaskowski, D. Latek, S. Yuan, U. Ghoshdastider, A. Debinski, and S. Filipek Action of molecular switches in GPCRs - Theoretical and experimental studies Current Medicinal Chemistry 19 2012 1090 1109
-
(2012)
Current Medicinal Chemistry
, vol.19
, pp. 1090-1109
-
-
Trzaskowski, B.1
Latek, D.2
Yuan, S.3
Ghoshdastider, U.4
Debinski, A.5
Filipek, S.6
-
39
-
-
80055007016
-
Dissecting the functions of conserved prolines within transmembrane helices of the D2 dopamine receptor
-
E.B. Van Arnam, H.A. Lester, and D.A. Dougherty Dissecting the functions of conserved prolines within transmembrane helices of the D2 dopamine receptor ACS Chemical Biology 6 2011 1063 1068
-
(2011)
ACS Chemical Biology
, vol.6
, pp. 1063-1068
-
-
Van Arnam, E.B.1
Lester, H.A.2
Dougherty, D.A.3
-
40
-
-
47949129742
-
Structure of a beta1-adrenergic G-protein-coupled receptor
-
T. Warne, M.J. Serrano-Vega, J.G. Baker, R. Moukhametzianov, P.C. Edwards, and R. Henderson Structure of a beta1-adrenergic G-protein-coupled receptor Nature 454 2008 486 491
-
(2008)
Nature
, vol.454
, pp. 486-491
-
-
Warne, T.1
Serrano-Vega, M.J.2
Baker, J.G.3
Moukhametzianov, R.4
Edwards, P.C.5
Henderson, R.6
-
43
-
-
79954782236
-
-
F. Xu, H. Wu, V. Katritch, G.W. Han, K.A. Jacobson, and Z.G. Gao Structure of an agonist-bound human A2A adenosine receptor. Science 332 2011 322 327
-
(2011)
Structure of An Agonist-bound Human A2A Adenosine Receptor. Science
, vol.332
, pp. 322-327
-
-
Xu, F.1
Wu, H.2
Katritch, V.3
Han, G.W.4
Jacobson, K.A.5
Gao, Z.G.6
-
44
-
-
33746382921
-
2-adrenoceptor
-
DOI 10.1038/nchembio801, PII NCHEMBIO801
-
X. Yao, C. Parnot, X. Deupi, V.R. Ratnala, G. Swaminath, and D. Farrens Coupling ligand structure to specific conformational switches in the beta2-adrenoceptor Nature Chemical Biology 2 2006 417 422 (Pubitemid 44114919)
-
(2006)
Nature Chemical Biology
, vol.2
, Issue.8
, pp. 417-422
-
-
Yao, X.1
Parnot, C.2
Deupi, X.3
Ratnala, V.R.P.4
Swaminath, G.5
Farrens, D.6
Kobilka, B.7
-
45
-
-
25844443463
-
Expression of human peripheral cannabinoid receptor for structural studies
-
DOI 10.1110/ps.051550305
-
A.A. Yeliseev, K.K. Wong, O. Soubias, and K. Gawrisch Expression of human peripheral cannabinoid receptor for structural studies Protein Science 14 2005 2638 2653 (Pubitemid 41395590)
-
(2005)
Protein Science
, vol.14
, Issue.10
, pp. 2638-2653
-
-
Yeliseev, A.A.1
Wong, K.K.2
Soubias, O.3
Gawrisch, K.4
-
46
-
-
77952355281
-
NMR analyses of the interaction between CCR5 and its ligand using functional reconstitution of CCR5 in lipid bilayers
-
C. Yoshiura, Y. Kofuku, T. Ueda, Y. Mase, M. Yokogawa, and M. Osawa NMR analyses of the interaction between CCR5 and its ligand using functional reconstitution of CCR5 in lipid bilayers Journal of the American Chemical Society 132 2010 6768 6777
-
(2010)
Journal of the American Chemical Society
, vol.132
, pp. 6768-6777
-
-
Yoshiura, C.1
Kofuku, Y.2
Ueda, T.3
Mase, Y.4
Yokogawa, M.5
Osawa, M.6
-
47
-
-
42749091750
-
Biosynthesis, purification, and characterization of a cannabinoid receptor 2 fragment (CB2(271-326))
-
Y. Zhang, and X.-Q. Xie Biosynthesis, purification, and characterization of a cannabinoid receptor 2 fragment (CB2(271-326)) Protein Expression and Purification 59 2008 249 257
-
(2008)
Protein Expression and Purification
, vol.59
, pp. 249-257
-
-
Zhang, Y.1
Xie, X.-Q.2
-
48
-
-
16844373364
-
Biosynthesis and purification of a hydrophobic peptide from transmembrane domains of G-protein-coupled CB2 receptor
-
H. Zheng, J. Zhao, S. Wang, C.M. Lin, T. Chen, and D.H. Jones Biosynthesis and purification of a hydrophobic peptide from transmembrane domains of G-protein-coupled CB2 receptor Journal of Peptide Research 65 2005 450 458
-
(2005)
Journal of Peptide Research
, vol.65
, pp. 450-458
-
-
Zheng, H.1
Zhao, J.2
Wang, S.3
Lin, C.M.4
Chen, T.5
Jones, D.H.6
|