The effect of mutations in the DRY motif on the constitutive activity and structural instability of the histamine H2 receptor

Molecular Pharmacology

Volumn 57, Issue 5, 2000, Pages 890-898

  Alewijnse, Astrid E ^a   Timmerman, Henk ^a   Jacobs, Edwin H ^a   Smit, Martine J ^a   Roovers, Edwin ^a   Cotecchia, Susanna ^b   Leurs, Rob ^a,c  

^a VU UNIVERSITY AMSTERDAM   (Netherlands)

^b UNIVERSITY OF LAUSANNE   (Switzerland)

^c NONE   (Netherlands)

Author keywords

[No Author keywords available]

Indexed keywords

ADRENERGIC RECEPTOR; AMINO ACID; ARGININE; BURIMAMIDE; CIMETIDINE; CYCLIC AMP; FAMOTIDINE; G PROTEIN COUPLED RECEPTOR; HISTAMINE H2 RECEPTOR; RANITIDINE; TIOTIDINE;

ANIMAL CELL; ARTICLE; CERCOPITHECIDAE; CONTROLLED STUDY; HUMAN; HUMAN CELL; MUTATION; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING; SIGNAL TRANSDUCTION;

AMINO ACID MOTIFS; AMINO ACID SEQUENCE; ANIMALS; ARGININE; CELLS, CULTURED; CRICETINAE; HUMANS; LIGANDS; MOLECULAR SEQUENCE DATA; MUTAGENESIS, SITE-DIRECTED; PROTEIN CONFORMATION; RANITIDINE; RECEPTORS, ADRENERGIC, ALPHA-1; RECEPTORS, HISTAMINE H2; SIGNAL TRANSDUCTION;

EID: 0034112037     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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