SCOPUS 정보 검색 플랫폼

Volumn 19, Issue 23, 2011, Pages 7093-7099

Design, synthesis and biological evaluation of cycloalkyl arylpyrimidines (CAPYs) as HIV-1 NNRTIs

(9) Gu, Shuang Xi a Yang, Shi Qiong a He, Qiu Qin a Ma, Xiao Dong a Chen, Fen Er a Dai, Hui Fang a Clercq, Erik De b Balzarini, Jan b Pannecouque, Christophe b

a FUDAN UNIVERSITY (China)

b REGA INSTITUTE FOR MEDICAL RESEARCH (Belgium)

Author keywords

CAPYs; DAPYs; HIV 1 reverse transcriptase; NNRTIs; Structure activity relationships

Indexed keywords

4 [[4 (CYCLOHEXYLAMINO) 5 METHYLPYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOHEXYLAMINO) 6 METHYLPYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOHEXYLAMINO)PYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOHEXYLOXY) 5 METHYLPYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOHEXYLOXY) 6 METHYLPYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOHEXYLOXY)PYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOHEXYLTHIO) 5 METHYLPYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOHEXYLTHIO) 6 METHYLPYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOHEXYLTHIO)PYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOPENTYLAMINO) 5 METHYLPYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOPENTYLAMINO) 6 METHYLPYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOPENTYLAMINO)PYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOPENTYLOXY) 5 METHYLPYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOPENTYLOXY) 6 METHYLPYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOPENTYLOXY)PYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOPROPYLAMINO) 5 METHYLPYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOPROPYLAMINO) 6 METHYLPYRIMIDIN 2 YL]AMINO]BENZONITRILE; 4 [[4 (CYCLOPROPYLAMINO)PYRIMIDIN 2 YL]AMINO]BENZONITRILE; CYCLOALKYL ARYLPYRIMIDINE DERIVATIVE; DELAVIRDINE; EFAVIRENZ; ETRAVIRINE; NEVIRAPINE; NONNUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITOR; PYRIMIDINE DERIVATIVE; UNCLASSIFIED DRUG; ZIDOVUDINE;

ANTIVIRAL ACTIVITY; ARTICLE; CONTROLLED STUDY; CYTOPATHOGENIC EFFECT; DRUG CYTOTOXICITY; DRUG DESIGN; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN IMMUNODEFICIENCY VIRUS 1; IN VITRO STUDY; MOLECULAR MODEL; STRUCTURE ACTIVITY RELATION;

ANTI-HIV AGENTS; HIV REVERSE TRANSCRIPTASE; HIV-1; HUMANS; MODELS, MOLECULAR; PYRIMIDINES; REVERSE TRANSCRIPTASE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 80655146742 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2011.10.002 Document Type: Article

Times cited : (23)

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