SCOPUS 정보 검색 플랫폼

Volumn 18, Issue 14, 2010, Pages 5039-5047

Hybrid diarylbenzopyrimidine non-nucleoside reverse transcriptase inhibitors as promising new leads for improved anti-HIV-1 chemotherapy

(8) Zeng, Zhao Sen a He, Qiu Qin a Liang, Yong Hong a Feng, Xiao Qing a Chen, Fen Er a Clercq, Erik De b Balzarini, Jan b Pannecouque, Christophe b

a FUDAN UNIVERSITY (China)

b REGA INSTITUTE FOR MEDICAL RESEARCH (Belgium)

Author keywords

DABPs; HIV 1 Reverse transcriptase; Molecular hybridization; NNRTIs; SAR

Indexed keywords

3 CHLORO 4 [2 (4 CYANOPHENYLAMINO)QUINAZOLIN 4 YLOXY] 5 METHOXYBENZONITRILE; 4 [2 (4 CYANOPHENYLAMINO)QUINAZOLIN 4 YLOXY] 3,5 DIMETHYLBENZONITRILE; 6 CHLORO 4 (2 CYCLOPROPYLVINYL) 3,4 DIHYDRO 4 TRIFLUOROMETHYL 2(1H) QUINAZOLINONE; BENZENE DERIVATIVE; DELAVIRDINE; EFAVIRENZ; ETRAVIRINE; NEVIRAPINE; NONNUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITOR; POLYCYCLIC AROMATIC HYDROCARBON DERIVATIVE; PYRIMIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIVIRAL ACTIVITY; ARTICLE; DRUG POTENCY; DRUG SELECTIVITY; HUMAN IMMUNODEFICIENCY VIRUS 1; HYBRID; MOLECULAR HYBRIDIZATION; NONHUMAN; STEREOCHEMISTRY; VIRUS MUTANT; VIRUS STRAIN; WILD TYPE;

ANTI-HIV AGENTS; CELL LINE; CELL SURVIVAL; HIV INFECTIONS; HIV REVERSE TRANSCRIPTASE; HIV-1; HUMANS; MODELS, MOLECULAR; PROTEIN BINDING; PYRIDAZINES; QUINAZOLINES; REVERSE TRANSCRIPTASE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 77955316010 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2010.05.081 Document Type: Article

Times cited : (38)

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