OATP1B1/1B3 activity in plated primary human hepatocytes over time in culture

Biochemical Pharmacology

Volumn 82, Issue 9, 2011, Pages 1219-1226

  Ulvestad, Maria ^a,b,c   Björquist, Petter ^c   Molden, Espen ^b   Sberg, Anders ^b   Andersson, Tommy B ^a,d  

^a ASTRAZENECA R AND D   (Sweden)

^b UNIVERSITY OF OSLO   (Norway)

^c Cellartis AB   (Sweden)

^d KAROLINSKA INSTITUTE   (Sweden)

Author keywords

Hepatocytes; OATP1B1; OATP1B3; Pharmacokinetics; Transporters

Indexed keywords

ESTRADIOL; ORGANIC ANION TRANSPORTER; ORGANIC ANION TRANSPORTER 2; ORGANIC ANION TRANSPORTING POLYPEPTIDE 1B1; ORGANIC ANION TRANSPORTING POLYPEPTIDE 1B3; PROTEIN SLCO1B3; UNCLASSIFIED DRUG;

ARTICLE; CELL CULTURE; CELL MEMBRANE; CONFOCAL MICROSCOPY; CONTROLLED STUDY; GENE EXPRESSION; GENOTYPE; HUMAN; HUMAN CELL; HUMAN TISSUE; LIVER CELL; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN LOCALIZATION;

ADULT; AGED; CELLS, CULTURED; ESTRADIOL; FEMALE; GENE EXPRESSION REGULATION; GENOTYPE; HEPATOCYTES; HUMANS; MALE; MIDDLE AGED; ORGANIC ANION TRANSPORTERS; ORGANIC ANION TRANSPORTERS, SODIUM-INDEPENDENT; TIME FACTORS;

EID: 80054002189     PISSN: 00062952     EISSN: 18732968     Source Type: Journal    
DOI: 10.1016/j.bcp.2011.07.076     Document Type: Article

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