Characterization and inhibition by a wide range of xenobiotics of organic anion excretion by primary human hepatocytes

Biochemical Pharmacology

Volumn 60, Issue 12, 2000, Pages 1967-1975

  Payen, Léa ^a   Courtois, Arnaud ^a   Campion, Jean Pierre ^a   Guillouzo, André ^a   Fardel, Olivier ^a  

^a INSERM   (France)

Author keywords

Carboxy 2',7' dichlorofluorescein; Efflux; Human hepatocytes; Multidrug resistance protein (MRP); Primary culture

Indexed keywords

ABC TRANSPORTER; ANION; CARRIER PROTEIN; CYCLOSPORIN A; FLUORESCEIN DERIVATIVE; GLIBENCLAMIDE; GLYCOPROTEIN P; INDOMETACIN; MULTIDRUG RESISTANCE PROTEIN; ORGANIC COMPOUND; PROBENECID; RIFAMPICIN; RNA; VERLUKAST; VINBLASTINE; XENOBIOTIC AGENT;

ADULT; ANION TRANSPORT; ARTICLE; CELL MEMBRANE TRANSPORT; CONTROLLED STUDY; CULTURE MEDIUM; DRUG DETOXIFICATION; DRUG ELIMINATION; DRUG TRANSPORT; HUMAN; HUMAN CELL; LIVER CELL; LIVER METABOLISM; NORTHERN BLOTTING; PRIORITY JOURNAL; PROTEIN EXPRESSION; TEMPERATURE DEPENDENCE; WESTERN BLOTTING; XENOBIOTIC METABOLISM;

EID: 0034672539     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-2952(00)00496-2     Document Type: Article

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