Docking of 1,4-benzodiazepines in the α1/γ 2 GABAA receptor modulator site

Molecular Pharmacology

Volumn 76, Issue 2, 2009, Pages 440-450

  Berezhnoy, D ^a   Gibbs, T T ^a   Farb, David H ^a  

^a BOSTON UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; 4 AMINOBUTYRIC ACID A RECEPTOR ALPHA1; 4 AMINOBUTYRIC ACID A RECEPTOR GAMMA2; ACETYLCHOLINE BINDING PROTEIN; BENZODIAZEPINE DERIVATIVE; BINDING PROTEIN; DIAZEPAM; FLUNITRAZEPAM; ION CHANNEL; UNCLASSIFIED DRUG;

AFFINITY LABELING; ARTICLE; BINDING AFFINITY; BINDING SITE; DRUG BINDING; GENE MUTATION; LYMNAEA; LYMNEA STAGNALIS; MOLECULAR DOCKING; NUCLEOTIDE SEQUENCE; PRIORITY JOURNAL; PROTEIN CONFORMATION; PROTEIN STRUCTURE; SIMULATION; STEREOSPECIFICITY; STRUCTURE ACTIVITY RELATION;

ALLOSTERIC REGULATION; ANIMALS; BENZODIAZEPINES; BINDING SITES; LIGANDS; MODELS, MOLECULAR; PROTEIN BINDING; RATS; RECEPTORS, GABA-A; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 67650815229     PISSN: 0026895X     EISSN: 15210111     Source Type: Journal    
DOI: 10.1124/mol.109.054650     Document Type: Article

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