Agonist trapping by GABAA receptor channels

Journal of Neuroscience

Volumn 21, Issue 23, 2001, Pages 9083-9091

  Bianchi, M T ^a   Macdonald, R L ^a  

^a VANDERBILT UNIVERSITY   (United States)

Author keywords

Concentration jump; Deactivation; Diazepam; GABA binding; GABAA receptor; Inverse agonist

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID RECEPTOR; BICUCULLINE; DIAZEPAM; 4 AMINOBUTYRIC ACID A RECEPTOR; 4 AMINOBUTYRIC ACID RECEPTOR BLOCKING AGENT; 4 AMINOBUTYRIC ACID RECEPTOR STIMULATING AGENT; LIGAND; PROTEIN SUBUNIT;

ARTICLE; CHANNEL GATING; CONTROLLED STUDY; DRUG RECEPTOR BINDING; GABAERGIC SYSTEM; HUMAN; HUMAN CELL; MEMBRANE CHANNEL; POSTSYNAPTIC INHIBITION; PRIORITY JOURNAL; RECEPTOR OCCUPANCY; SYNAPSE; ANIMAL; BINDING COMPETITION; BINDING SITE; CELL LINE; CYTOLOGY; DRUG EFFECT; DRUG POTENTIATION; FIBROBLAST; GENE EXPRESSION; GENETIC TRANSFECTION; GENETICS; ION TRANSPORT; KIDNEY; METABOLISM; PATCH CLAMP; PHYSIOLOGY; RAT; SITE DIRECTED MUTAGENESIS;

ANIMALS; BINDING SITES; BINDING, COMPETITIVE; CELL LINE; FIBROBLASTS; GABA AGONISTS; GABA ANTAGONISTS; GAMMA-AMINOBUTYRIC ACID; GENE EXPRESSION; HUMANS; ION CHANNEL GATING; ION TRANSPORT; KIDNEY; LIGANDS; MUTAGENESIS, SITE-DIRECTED; PATCH-CLAMP TECHNIQUES; PROTEIN SUBUNITS; RATS; RECEPTORS, GABA-A; TRANSFECTION;

EID: 0035529012     PISSN: 02706474     EISSN: None     Source Type: Journal    
DOI: 10.1523/jneurosci.21-23-09083.2001     Document Type: Article

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