Transportable, Chemical Genetic Methodology for the Small Molecule-Mediated Inhibition of Heat Shock Factor 1

ACS Chemical Biology

Volumn 11, Issue 1, 2016, Pages 200-210

  Moore, Christopher L ^a   Dewal, Mahender B ^a,b   Nekongo, Emmanuel E ^a   Santiago, Sebasthian ^a   Lu, Nancy B ^a   Levine, Stuart S ^a   Shoulders, Matthew D ^a  

^a MASSACHUSETTS INSTITUTE OF TECHNOLOGY   (United States)

^b Expansion Technologies   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CHAPERONE; HEAT SHOCK TRANSCRIPTION FACTOR 1; PROTEIN INHIBITOR; PROTEIN VARIANT; DNA BINDING PROTEIN; HEAT SHOCK TRANSCRIPTION FACTOR; MOLECULAR LIBRARY; TRANSCRIPTION FACTOR;

ARTICLE; DOWN REGULATION; EMBRYO; ENZYME INHIBITION; HEAT SHOCK RESPONSE; HEK293 CELL LINE; HUMAN; HUMAN CELL; METHODOLOGY; PLEIOTROPY; PRIORITY JOURNAL; PROTEIN HOMEOSTASIS; UPREGULATION; ANTAGONISTS AND INHIBITORS; CHEMISTRY; DRUG EFFECTS; FLOW CYTOMETRY; GENE EXPRESSION REGULATION; GENETICS; IMMUNOBLOTTING; METABOLISM; MICROARRAY ANALYSIS; MOLECULAR LIBRARY; PHARMACOLOGY; REAL TIME POLYMERASE CHAIN REACTION;

DNA-BINDING PROTEINS; FLOW CYTOMETRY; GENE EXPRESSION REGULATION; HEK293 CELLS; HUMANS; IMMUNOBLOTTING; MICROARRAY ANALYSIS; REAL-TIME POLYMERASE CHAIN REACTION; SMALL MOLECULE LIBRARIES; TRANSCRIPTION FACTORS;

EID: 84955294604     PISSN: 15548929     EISSN: 15548937     Source Type: Journal    
DOI: 10.1021/acschembio.5b00740     Document Type: Article

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