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Bioorganic and Medicinal Chemistry Letters

Volumn 25, Issue 9, 2015, Pages 1965-1970

Synthesis of [11C]GSK1482160 as a new PET agent for targeting P2X7 receptor

(5) Gao, Mingzhang a Wang, Min a Green, Mark A a Hutchins, Gary D a Zheng, Qi Huang a

a INDIANA UNIVERSITY SCHOOL OF MEDICINE (United States)

Author keywords

Neuroinflammation; P2X7 receptor; Positron emission tomography (PET); Radiosynthesis; 11C GSK1482160

Indexed keywords

CARBON; N-(2-CHLORO-3-(TRIFLUOROMETHYL)BENZYL)-N-METHYL-5-OXOPYRROLIDINE-2-CARBOXAMIDE; P2XR RECEPTOR, HUMAN; PURINERGIC P2X7 RECEPTOR; PYROGLUTAMIC ACID; RADIOPHARMACEUTICAL AGENT;

CHEMICAL STRUCTURE; CHEMISTRY; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HUMAN; METABOLISM; MOLECULAR IMAGING; POSITRON EMISSION TOMOGRAPHY; SOLID PHASE EXTRACTION; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

CARBON RADIOISOTOPES; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; HUMANS; MOLECULAR IMAGING; MOLECULAR STRUCTURE; POSITRON-EMISSION TOMOGRAPHY; PYRROLIDONECARBOXYLIC ACID; RADIOPHARMACEUTICALS; RECEPTORS, PURINERGIC P2X7; SOLID PHASE EXTRACTION; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84930928841 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2015.03.021 Document Type: Article

Times cited : (67)

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