Fully automated synthesis and initial PET evaluation of [11C]PBR28

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 19, 2009, Pages 5636-5639

  Wang, Min ^a   Yoder, Karmen K ^a   Gao, Mingzhang ^a   Mock, Bruce H ^a   Xu, Xiao Ming ^a   Saykin, Andrew J ^a   Hutchins, Gary D ^a   Zheng, Qi Huang ^a  

^a INDIANA UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

11C PBR28; Brain imaging; Positron emission tomography (PET); Radiosynthesis; Translocator protein (TSPO); Traumatic brain injury (TBI)

Indexed keywords

N (2 METHOXYBENZYL) N (4 PHENOXYPYRIDIN 3 YL)ACETAMIDE C 11; RADIOLIGAND; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DRUG FORMULATION; DRUG PURIFICATION; DRUG SYNTHESIS; FEMALE; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; METHYLATION; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; RADIOACTIVITY; RAT;

ANIMALS; CARBON RADIOISOTOPES; CARRIER PROTEINS; FEMALE; GABA-A RECEPTOR ANTAGONISTS; LIGANDS; POSITRON-EMISSION TOMOGRAPHY; PYRIMIDINES; RADIOPHARMACEUTICALS; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, GABA-A;

ANIMALIA;

EID: 69949102160     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2009.08.051     Document Type: Article

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