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Volumn , Issue , 2012, Pages 1-252

Essentials of Pharmaceutical Preformulation

Author keywords

[No Author keywords available]

Indexed keywords

BIOCHEMISTRY; DRUG PRODUCTS; STUDENTS;

EID: 84914105462     PISSN: None     EISSN: None     Source Type: Book    
DOI: 10.1002/9781118423226     Document Type: Book
Times cited : (29)

References (165)
  • 1
    • 77953416359 scopus 로고    scopus 로고
    • Separation Science and Technology Series, vol. 8, Academic Press, London
    • Ahuja, S. and Rasmussen, H. (2007) HPLC Method Development for Pharmaceuticals, Separation Science and Technology Series, vol. 8, Academic Press, London. ISBN 0-1237-0540-1.
    • (2007) HPLC Method Development for Pharmaceuticals
    • Ahuja, S.1    Rasmussen, H.2
  • 2
    • 0030647671 scopus 로고    scopus 로고
    • The utility of phase correction in modulated DSC
    • Aubuchon, S.R. and Gill, P.S. (1997) The utility of phase correction in modulated DSC. J. Therm. Anal. Cal., 49, 1039-1044.
    • (1997) J. Therm. Anal. Cal , vol.49 , pp. 1039-1044
    • Aubuchon, S.R.1    Gill, P.S.2
  • 3
    • 0016988717 scopus 로고
    • Acidic potassium dichromate solutions as ultraviolet absorbance standards
    • Burke, R.W. and Mavrodineanu, R. (1976) Acidic potassium dichromate solutions as ultraviolet absorbance standards. J. Res. Natl Bur. Stand. A, 80A, 631-636.
    • (1976) J. Res. Natl Bur. Stand. A , vol.80 A , pp. 631-636
    • Burke, R.W.1    Mavrodineanu, R.2
  • 7
    • 77649234756 scopus 로고    scopus 로고
    • How to improve R&D productivity: the pharmaceutical industry's grand challenge
    • Paul, S.M., Mytelka, D.S., Dunwiddie, C.T. et al. (2010) How to improve R&D productivity: the pharmaceutical industry's grand challenge. Nat. Rev. Drug Disc., 9, 203-214.
    • (2010) Nat. Rev. Drug Disc , vol.9 , pp. 203-214
    • Paul, S.M.1    Mytelka, D.S.2    Dunwiddie, C.T.3
  • 8
    • 0034665153 scopus 로고    scopus 로고
    • Practitioner's guide to method development in thinlayer chromatography
    • Poole, C.F. and Dias, N.C. (2000) Practitioner's guide to method development in thinlayer chromatography. J. Chromatogr. A., 892, 123-142.
    • (2000) J. Chromatogr. A , vol.892 , pp. 123-142
    • Poole, C.F.1    Dias, N.C.2
  • 9
    • 0001419232 scopus 로고
    • Modulated differential scanning calorimetry
    • Reading, M., Luget, A. and Wilson, R. (1994) Modulated differential scanning calorimetry. Thermochim. Acta, 238, 295-307.
    • (1994) Thermochim. Acta , vol.238 , pp. 295-307
    • Reading, M.1    Luget, A.2    Wilson, R.3
  • 10
    • 77955469357 scopus 로고    scopus 로고
    • Modulated temperature differential scanning calorimetry
    • (eds D.Q.M. Craig and M. Reading), CRC Press, Boca Raton, FL
    • Reading, M., Craig, D.Q.M., Murphy, J.R. and Kett, V.L. (2007) Modulated temperature differential scanning calorimetry. In Thermal Analysis of Pharmaceuticals (eds D.Q.M. Craig and M. Reading), CRC Press, Boca Raton, FL. ISBN 0-8247-5814-5.
    • (2007) Thermal Analysis of Pharmaceuticals
    • Reading, M.1    Craig, D.Q.M.2    Murphy, J.R.3    Kett, V.L.4
  • 11
    • 0022026693 scopus 로고
    • Spectral transmittance characteristics of holmium oxide in perchloric acid solution
    • Weidner, V.R., Mavrodineanu, R., and Mielenz, K.D. (1985) Spectral transmittance characteristics of holmium oxide in perchloric acid solution. J. Res. Natl Bur. Stand., 90, 115-125.
    • (1985) J. Res. Natl Bur. Stand , vol.90 , pp. 115-125
    • Weidner, V.R.1    Mavrodineanu, R.2    Mielenz, K.D.3
  • 13
    • 72149101372 scopus 로고    scopus 로고
    • a distribution of drugs: application to drug discovery
    • a distribution of drugs: application to drug discovery. Perspect. Med. Chem., 1, 25-38.
    • (2007) Perspect. Med. Chem , vol.1 , pp. 25-38
    • Manallack, D.T.1
  • 14
    • 36048986392 scopus 로고    scopus 로고
    • a values for pharmaceutical substances
    • (ed. H.B. Brittain), vol. 33, Academic Press, San Diego
    • a values for pharmaceutical substances. In Profiles of Drug Substances, Excipients and Related Methodology (ed. H.B. Brittain), vol. 33, Academic Press, San Diego, pp. 1-726. ISBN 9780-1226-0833-9.
    • (2007) Profiles of Drug Substances, Excipients and Related Methodology , pp. 1-726
    • Prankerd, R.J.1
  • 15
    • 0002293876 scopus 로고
    • The behaviour of carboxylic acids in mixed solvents
    • (ed. B. Pesce), Pergamon Press
    • Shedlovsky, T. (1962) The behaviour of carboxylic acids in mixed solvents. In Electrolytes (ed. B. Pesce), Pergamon Press, pp. 146-151. ISBN 0-0801-3778-4.
    • (1962) Electrolytes , pp. 146-151
    • Shedlovsky, T.1
  • 16
    • 0142028495 scopus 로고    scopus 로고
    • a determination of water-insoluble compounds: validation study in methanol/water mixtures
    • a determination of water-insoluble compounds: validation study in methanol/water mixtures. Int. J. Pharm., 151, 235-248.
    • (1997) Int. J. Pharm , vol.151 , pp. 235-248
    • Takács-Novák, K.1    Box, K.J.2    Avdeef, A.3
  • 17
  • 18
    • 12344335757 scopus 로고    scopus 로고
    • Stability of metronidazole, tetracycline HCl and famotidine alone and in combination
    • Wu, Y. and Fassihi, R. (2005) Stability of metronidazole, tetracycline HCl and famotidine alone and in combination. Int. J. Pharm., 290, 1-13.
    • (2005) Int. J. Pharm , vol.290 , pp. 1-13
    • Wu, Y.1    Fassihi, R.2
  • 19
    • 0001266728 scopus 로고
    • Dissociation constants of some carboxylic acids in mixed aqueous solvents
    • Yasuda, M. (1959) Dissociation constants of some carboxylic acids in mixed aqueous solvents. Bull. Chem. Soc. Jpn, 32, 429-432.
    • (1959) Bull. Chem. Soc. Jpn , vol.32 , pp. 429-432
    • Yasuda, M.1
  • 20
    • 0023547921 scopus 로고
    • A thermodynamic analysis of the Collander equation and establishment of a reference solvent for use in drug partitioning studies
    • Beezer, A.E., Gooch, C.A., Hunter, W.H. and Volpe, P.L. (1987) A thermodynamic analysis of the Collander equation and establishment of a reference solvent for use in drug partitioning studies. J. Pharm. Pharmacol., 39, 774-779.
    • (1987) J. Pharm. Pharmacol , vol.39 , pp. 774-779
    • Beezer, A.E.1    Gooch, C.A.2    Hunter, W.H.3    Volpe, P.L.4
  • 21
    • 0014685056 scopus 로고
    • Partition data of penicillins determined by means of reversed-phase thin-layer chromatography
    • Biagi, G.L., Barbaro, A.M., Gamba, M.F. and Guerra, M.C. (1964) Partition data of penicillins determined by means of reversed-phase thin-layer chromatography. J. Chromatogr. A, 41, 371-379.
    • (1964) J. Chromatogr. A , vol.41 , pp. 371-379
    • Biagi, G.L.1    Barbaro, A.M.2    Gamba, M.F.3    Guerra, M.C.4
  • 22
    • 0014675062 scopus 로고
    • Partition data of cephalosporins determined by means of reversed-phase thin layer chromatography
    • Biagi, G.L., Barbaro, A.M., Guerra, M.C. and Gamba, M.F. (1969) Partition data of cephalosporins determined by means of reversed-phase thin layer chromatography. J. Chromatogr. A, 44, 195-198.
    • (1969) J. Chromatogr. A , vol.44 , pp. 195-198
    • Biagi, G.L.1    Barbaro, A.M.2    Guerra, M.C.3    Gamba, M.F.4
  • 23
    • 0028299385 scopus 로고
    • Determination of lipophilicity by means of reversed-phase thin-layer chromatography. i. Basic aspects and relationship between slope and intercept of TLC equations
    • Biagi, G.L., Barbaro, A.M., Sapone, A. and Recanatini, M. (1994a) Determination of lipophilicity by means of reversed-phase thin-layer chromatography. i. Basic aspects and relationship between slope and intercept of TLC equations. J. Chromatogr. A, 662, 341-361.
    • (1994) J. Chromatogr. A , vol.662 , pp. 341-361
    • Biagi, G.L.1    Barbaro, A.M.2    Sapone, A.3    Recanatini, M.4
  • 24
    • 0028243154 scopus 로고
    • Determination of lipophilicity by means of reversed-phase thin-layer chromatography. ii. Influence of the organic modifier on the slope of the thin-layer chromatographic equation
    • Biagi, G.L., Barbaro, A.M., Sapone, A. and Recanatini, M. (1994b) Determination of lipophilicity by means of reversed-phase thin-layer chromatography. ii. Influence of the organic modifier on the slope of the thin-layer chromatographic equation. J. Chromatogr. A, 669, 246-253.
    • (1994) J. Chromatogr. A , vol.669 , pp. 246-253
    • Biagi, G.L.1    Barbaro, A.M.2    Sapone, A.3    Recanatini, M.4
  • 25
    • 0027997411 scopus 로고
    • Determination of lipophilicity by means of reversed-phase thin-layer chromatography. iii. Study of the TLC equations for a series of ionizable quinolone derivatives
    • Biagi, G.L., Barbaro, A.M. and Recanatini, M. (1994c) Determination of lipophilicity by means of reversed-phase thin-layer chromatography. iii. Study of the TLC equations for a series of ionizable quinolone derivatives. J. Chromatogr. A, 678, 127-137.
    • (1994) J. Chromatogr. A , vol.678 , pp. 127-137
    • Biagi, G.L.1    Barbaro, A.M.2    Recanatini, M.3
  • 26
    • 0015237832 scopus 로고
    • Reversed-phase thin layer chromatography and partition coefficients of penicillins
    • Bird, A.E. and Marshall, C. (1971) Reversed-phase thin layer chromatography and partition coefficients of penicillins. J. Chromatogr. A, 63, 313-319.
    • (1971) J. Chromatogr. A , vol.63 , pp. 313-319
    • Bird, A.E.1    Marshall, C.2
  • 27
    • 0020076112 scopus 로고
    • Partitioning of organic compounds in octanol-water systems
    • Chiou, C.T., Schmedding, D.W. and Manes, M. (1982) Partitioning of organic compounds in octanol-water systems. Environ. Sci. Technol., 16, 4-10.
    • (1982) Environ. Sci. Technol , vol.16 , pp. 4-10
    • Chiou, C.T.1    Schmedding, D.W.2    Manes, M.3
  • 28
    • 0023804237 scopus 로고
    • Measurement of the distribution coefficients of several classes of drug using reversed-phase thin-layer chromatography
    • Jack, D.B., Hawker, J.L., Rooney, L. et al. (1988) Measurement of the distribution coefficients of several classes of drug using reversed-phase thin-layer chromatography. J. Chromatogr. A, 452, 257-264.
    • (1988) J. Chromatogr. A , vol.452 , pp. 257-264
    • Jack, D.B.1    Hawker, J.L.2    Rooney, L.3
  • 29
    • 77955581133 scopus 로고    scopus 로고
    • Revisiting thin-layer chromatography as a lipophilicity determination tool - a comparative study on several techniques with a model solute set
    • Komsta, L., Skibinski, R., Berecka, A. et al. (2010) Revisiting thin-layer chromatography as a lipophilicity determination tool - a comparative study on several techniques with a model solute set. J. Pharm. Biomed. Anal., 53, 911-918.
    • (2010) J. Pharm. Biomed. Anal , vol.53 , pp. 911-918
    • Komsta, L.1    Skibinski, R.2    Berecka, A.3
  • 30
    • 0027818680 scopus 로고
    • Modeling oil-water partitioning and membrane permeation using reversed-phase chromatography
    • Lambert, W.J. (1993) Modeling oil-water partitioning and membrane permeation using reversed-phase chromatography. J. Chromatogr. A, 656, 469-484.
    • (1993) J. Chromatogr. A , vol.656 , pp. 469-484
    • Lambert, W.J.1
  • 31
    • 8644243613 scopus 로고
    • Partition coefficients and their uses
    • Leo, A., Hansch, C. and Elkins, D. (1971) Partition coefficients and their uses. Chem. Rev., 71, 525-616.
    • (1971) Chem. Rev , vol.71 , pp. 525-616
    • Leo, A.1    Hansch, C.2    Elkins, D.3
  • 32
    • 0021124186 scopus 로고
    • General approach for the estimation of octanol/water partition coefficient by reversed-phase high-performance liquid chromatography
    • Valkó, K. (1984) General approach for the estimation of octanol/water partition coefficient by reversed-phase high-performance liquid chromatography. J. Liq. Chromatogr., 7, 1405-1424.
    • (1984) J. Liq. Chromatogr , vol.7 , pp. 1405-1424
    • Valkó, K.1
  • 33
    • 2342635206 scopus 로고    scopus 로고
    • Application of high-performance liquid chromatography based measurements of lipophilicity to model biological distribution
    • Valkó, K. (2004) Application of high-performance liquid chromatography based measurements of lipophilicity to model biological distribution. J. Chromatogr. A, 1037, 299-310.
    • (2004) J. Chromatogr. A , vol.1037 , pp. 299-310
    • Valkó, K.1
  • 34
    • 0027402651 scopus 로고
    • New chromatographic hydrophobicity index (φ0) based on the slope and the intercept of the log K _ versus organic phase concentration plot
    • Valkó, K. and Slégel, P. (1993) New chromatographic hydrophobicity index (φ0) based on the slope and the intercept of the log K _ versus organic phase concentration plot. J. Chromatogr. A, 631, 49-61.
    • (1993) J. Chromatogr. A , vol.631 , pp. 49-61
    • Valkó, K.1    Slégel, P.2
  • 35
    • 0000607945 scopus 로고    scopus 로고
    • Chromatographic hydrophobicity index by fast-gradient RP-HPLC: a high-throughput alternative to log P/log D
    • Valkó, K., Bevan, C. and Reynolds, D. (1997) Chromatographic hydrophobicity index by fast-gradient RP-HPLC: a high-throughput alternative to log P/log D. Anal. Chem., 69, 2022-2029.
    • (1997) Anal. Chem , vol.69 , pp. 2022-2029
    • Valkó, K.1    Bevan, C.2    Reynolds, D.3
  • 36
    • 0022818104 scopus 로고
    • Determination of partition coefficients and aqueous solubilities by reverse phase chromatography - I. Theory and background
    • Weber Jr, W.J., Chin, Y.-P. and Rice, C.P. (1986) Determination of partition coefficients and aqueous solubilities by reverse phase chromatography - I. Theory and background. Water Res., 20, 1433-1442.
    • (1986) Water Res , vol.20 , pp. 1433-1442
    • Weber, W.J.1    Chin, Y.-P.2    Rice, C.P.3
  • 39
    • 0028948839 scopus 로고
    • A theoretical basis for a biopharmaceutical drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability
    • Amidon, G.L., Lennernäs, H., Shah, V.P. and Crison, J.R. (1995) A theoretical basis for a biopharmaceutical drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability. Pharm. Res., 12, 413-420.
    • (1995) Pharm. Res , vol.12 , pp. 413-420
    • Amidon, G.L.1    Lennernäs, H.2    Shah, V.P.3    Crison, J.R.4
  • 40
    • 0033224876 scopus 로고    scopus 로고
    • Solubility of paracetamol in pure solvents
    • Granberg, R.A. and Rasmuson, A.C. (1999) Solubility of paracetamol in pure solvents. J. Chem. Engng Data, 44, 1391-1395.
    • (1999) J. Chem. Engng Data , vol.44 , pp. 1391-1395
    • Granberg, R.A.1    Rasmuson, A.C.2
  • 41
    • 0002177778 scopus 로고
    • Biopharmaceutical considerations in drug formulation design and evaluation
    • Kaplan, S.A. (1972) Biopharmaceutical considerations in drug formulation design and evaluation. Drug Met. Rev., 1, 15-34.
    • (1972) Drug Met. Rev , vol.1 , pp. 15-34
    • Kaplan, S.A.1
  • 42
    • 0030886937 scopus 로고    scopus 로고
    • Managing the drug discovery/development interface
    • Kennedy, T. (1997) Managing the drug discovery/development interface. Drug Disc. Today, 2, 436-444.
    • (1997) Drug Disc. Today , vol.2 , pp. 436-444
    • Kennedy, T.1
  • 43
    • 0000882284 scopus 로고
    • Purity determination by differential scanning calorimetry
    • Marti, E.E. (1972) Purity determination by differential scanning calorimetry. Thermochim. Acta, 5, 173-220.
    • (1972) Thermochim. Acta , vol.5 , pp. 173-220
    • Marti, E.E.1
  • 44
    • 66049083443 scopus 로고    scopus 로고
    • Temperature and solvent effects in the solubility of some pharmaceutical compounds: measurements and modeling
    • Mota, F.L., Carneiro, A.P., Queimada, A.J. et al. (2009) Temperature and solvent effects in the solubility of some pharmaceutical compounds: measurements and modeling. Eur. J. Pharm. Sci., 37, 499-507.
    • (2009) Eur. J. Pharm. Sci , vol.37 , pp. 499-507
    • Mota, F.L.1    Carneiro, A.P.2    Queimada, A.J.3
  • 45
    • 0026733159 scopus 로고
    • Solid state properties of drugs. I. Estimation of heat capacities for fusion and thermodynamic functions for solution from aqueous solubility-temperature dependence measurements
    • Prankerd, R.J. (1992) Solid state properties of drugs. I. Estimation of heat capacities for fusion and thermodynamic functions for solution from aqueous solubility-temperature dependence measurements. Int. J. Pharm., 84, 233-244.
    • (1992) Int. J. Pharm , vol.84 , pp. 233-244
    • Prankerd, R.J.1
  • 46
    • 0019809124 scopus 로고
    • Difference in physic-chemical properties between crystalline and non-crystalline 9,3__-diacetylmidecamycin
    • Sato, T., Okada, A., Sekiguchi, K. and Tsuda, Y. (1981) Difference in physic-chemical properties between crystalline and non-crystalline 9,3__-diacetylmidecamycin. Chem. Pharm. Bull., 29, 2675-2682.
    • (1981) Chem. Pharm. Bull , vol.29 , pp. 2675-2682
    • Sato, T.1    Okada, A.2    Sekiguchi, K.3    Tsuda, Y.4
  • 47
    • 33947091552 scopus 로고
    • Simple equation for linearization of data in differential scanning calorimetric purity determinations
    • Sondack, D.L. (1972) Simple equation for linearization of data in differential scanning calorimetric purity determinations. Anal. Chem., 44, 888.
    • (1972) Anal. Chem , vol.44 , pp. 888
    • Sondack, D.L.1
  • 48
    • 34447536520 scopus 로고    scopus 로고
    • When poor solubility becomes an issue: from early stage to proof of concept
    • Stegemann, S., Leveiller, F., Franchi, D. et al. (2007) When poor solubility becomes an issue: from early stage to proof of concept. Eur. J. Pharm. Sci., 31, 249-261.
    • (2007) Eur. J. Pharm. Sci , vol.31 , pp. 249-261
    • Stegemann, S.1    Leveiller, F.2    Franchi, D.3
  • 49
    • 77955248335 scopus 로고    scopus 로고
    • The biowaiver extension for BCS class III drugs: the effect of dissolution rate on the bioequivalence of BCS class III immediate-release drugs predicted by computer simulation
    • Tsume, Y. and Amidon, G.L. (2010) The biowaiver extension for BCS class III drugs: the effect of dissolution rate on the bioequivalence of BCS class III immediate-release drugs predicted by computer simulation. Molec. Pharm., 7, 1235-1243.
    • (2010) Molec. Pharm , vol.7 , pp. 1235-1243
    • Tsume, Y.1    Amidon, G.L.2
  • 50
    • 0021233407 scopus 로고
    • Purity determinations of drugs with differential scanning calorimetry (DSC) - a critical review
    • van Dooren, A.A. and Müller, B.W. (1984) Purity determinations of drugs with differential scanning calorimetry (DSC) - a critical review. Int. J. Pharm., 20, 217-233.
    • (1984) Int. J. Pharm , vol.20 , pp. 217-233
    • Van Dooren, A.A.1    Müller, B.W.2
  • 52
    • 0002642747 scopus 로고
    • Reaktionsgeschwindigkeit in heterogenen systemen
    • Brunner, E. (1904) Reaktionsgeschwindigkeit in heterogenen systemen. Z. Phys. Chem., 43, 56-102.
    • (1904) Z. Phys. Chem , vol.43 , pp. 56-102
    • Brunner, E.1
  • 53
    • 33747348812 scopus 로고
    • Über die Auflösungsgeschwindigkeit fester Körper
    • Brunner, E. and Tolloczko, S. (1900) Über die Auflösungsgeschwindigkeit fester Körper. Z. Phys. Chem., 35, 283-290.
    • (1900) Z. Phys. Chem , vol.35 , pp. 283-290
    • Brunner, E.1    Tolloczko, S.2
  • 54
    • 0000354093 scopus 로고
    • Significance of liquid-film coefficients in gas absorption
    • Danckwerts, P.V. (1951) Significance of liquid-film coefficients in gas absorption. Ind. Engng Chem., 43, 1460-1467.
    • (1951) Ind. Engng Chem , vol.43 , pp. 1460-1467
    • Danckwerts, P.V.1
  • 55
    • 33747373878 scopus 로고    scopus 로고
    • Acentury of dissolution research: from Noyes and Whitney to the biopharmaceutical classification system
    • Dokoumetzidis, A. and Macheras, P. (2006)Acentury of dissolution research: from Noyes and Whitney to the biopharmaceutical classification system. Int. J. Pharm., 321, 1-11.
    • (2006) Int. J. Pharm , vol.321 , pp. 1-11
    • Dokoumetzidis, A.1    Macheras, P.2
  • 56
    • 0033805179 scopus 로고    scopus 로고
    • In vitro-in vivo correlations for lipophilic, poorly water-soluble drugs
    • Dressman, J.B. and Reppas, C. (2000) In vitro-in vivo correlations for lipophilic, poorly water-soluble drugs. Eur. J. Pharm. Sci., 11, S73-S80.
    • (2000) Eur. J. Pharm. Sci , vol.11 , pp. S73-S80
    • Dressman, J.B.1    Reppas, C.2
  • 57
    • 84962061517 scopus 로고    scopus 로고
    • The mini paddle apparatus - a useful tool in the early developmental stage? Experiences with immediate-release dosage forms
    • Klein, S. (2006) The mini paddle apparatus - a useful tool in the early developmental stage? Experiences with immediate-release dosage forms. Dissol. Technol., 13, 6-11.
    • (2006) Dissol. Technol , vol.13 , pp. 6-11
    • Klein, S.1
  • 58
    • 23844475290 scopus 로고    scopus 로고
    • Effect of chloride ion on dissolution of different salt forms of haloperidol, a model basic drug
    • Li, S., Doyle, P., Metz, S. et al. (2005) Effect of chloride ion on dissolution of different salt forms of haloperidol, a model basic drug. J. Pharm. Sci., 94, 2224-2231.
    • (2005) J. Pharm. Sci , vol.94 , pp. 2224-2231
    • Li, S.1    Doyle, P.2    Metz, S.3
  • 59
    • 0030927353 scopus 로고    scopus 로고
    • Characterization of fluids from the stomach and proximal jejunum in men and women
    • Lindahl, A., Ungell, A.L. and Lennernas, H. (1997) Characterization of fluids from the stomach and proximal jejunum in men and women. Pharm. Res., 14, 497-502.
    • (1997) Pharm. Res , vol.14 , pp. 497-502
    • Lindahl, A.1    Ungell, A.L.2    Lennernas, H.3
  • 60
    • 43249121029 scopus 로고    scopus 로고
    • Gut instincts: explorations in intestinal physiology and drug delivery
    • McConnell, E.L. Fadda, H.M. and Basit, A.W. (2008) Gut instincts: explorations in intestinal physiology and drug delivery. Int. J. Pharm., 364, 213-226.
    • (2008) Int. J. Pharm , vol.364 , pp. 213-226
    • McConnell, E.L.1    Fadda, H.M.2    Basit, A.W.3
  • 61
    • 0002642747 scopus 로고
    • Theorie der Reaktionsgeschwindigkeit in Heterogenen Systemen
    • Nernst, W. (1904) Theorie der Reaktionsgeschwindigkeit in Heterogenen Systemen. Z. Phys. Chem., 47, 52-55.
    • (1904) Z. Phys. Chem , vol.47 , pp. 52-55
    • Nernst, W.1
  • 62
    • 33947487639 scopus 로고
    • The rate of solution of solid substances in their own solutions
    • Noyes, A.A. and Whitney, W.R. (1897) The rate of solution of solid substances in their own solutions. J. Am. Chem. Soc., 19, 930-934.
    • (1897) J. Am. Chem. Soc , vol.19 , pp. 930-934
    • Noyes, A.A.1    Whitney, W.R.2
  • 63
    • 27744515754 scopus 로고    scopus 로고
    • Intestinal fluid volumes and transit of dosage forms as assessed by magnetic resonance imaging
    • Schiller, C., Fröhlich, C.-P., Giessmann, T. et al. (2005) Intestinal fluid volumes and transit of dosage forms as assessed by magnetic resonance imaging. Ailment Pharmacol. Theory, 22, 971-979.
    • (2005) Ailment Pharmacol. Theory , vol.22 , pp. 971-979
    • Schiller, C.1    Fröhlich, C.-P.2    Giessmann, T.3
  • 64
    • 0021944082 scopus 로고
    • Effect of diffusion layer pH and solubility on the dissolution rate of pharmaceutical acids and their sodium salts. II: salicylic acid, theophylline and benzoic acid
    • Serajuddin, A.T.M. and Jarowski, C.I. (1985) Effect of diffusion layer pH and solubility on the dissolution rate of pharmaceutical acids and their sodium salts. II: salicylic acid, theophylline and benzoic acid. J. Pharm. Sci., 74, 148-154.
    • (1985) J. Pharm. Sci , vol.74 , pp. 148-154
    • Serajuddin, A.T.M.1    Jarowski, C.I.2
  • 65
    • 0043283915 scopus 로고    scopus 로고
    • Measurement of intrinsic drug dissolution using two types of apparatus
    • Viegas, T.X., Curatella, R.U., Van Winkle, L.L. and Brinker, G. (2001) Measurement of intrinsic drug dissolution using two types of apparatus. Pharm Technol., 25, 44-43.
    • (2001) Pharm Technol , vol.25 , pp. 44-43
    • Viegas, T.X.1    Curatella, R.U.2    Van Winkle, L.L.3    Brinker, G.4
  • 66
    • 33747336372 scopus 로고
    • Über die Geschwindigkeit Molekularer und Chemischer Reaktionen in Heterogenen Systemen
    • Wilderman, M. (1909) Über die Geschwindigkeit Molekularer und Chemischer Reaktionen in Heterogenen Systemen. Erster Teil. Z. Phys. Chem., 66, 445-495.
    • (1909) Erster Teil. Z. Phys. Chem , vol.66 , pp. 445-495
    • Wilderman, M.1
  • 67
    • 33748503596 scopus 로고    scopus 로고
    • The ionization constant of water over wide ranges of temperature and density
    • Bandura, A.V. and Lvov, S.N. (2005) The ionization constant of water over wide ranges of temperature and density. J. Phys. Chem. Ref. Data, 35, 15-30.
    • (2005) J. Phys. Chem. Ref. Data , vol.35 , pp. 15-30
    • Bandura, A.V.1    Lvov, S.N.2
  • 69
    • 25844524863 scopus 로고    scopus 로고
    • Tape and layer structures in cocrystals of some di- and tricarboxylic acids with 4,4_-bipyridines and isonicotinamide. From binary to ternary cocrystals
    • Bhogala, B.R., Basavoju, S. and Nangia, A. (2005) Tape and layer structures in cocrystals of some di- and tricarboxylic acids with 4,4_-bipyridines and isonicotinamide. From binary to ternary cocrystals. Crys. Engng Commun., 7, 551-562.
    • (2005) Crys. Engng Commun , vol.7 , pp. 551-562
    • Bhogala, B.R.1    Basavoju, S.2    Nangia, A.3
  • 70
    • 0018412446 scopus 로고
    • Solubility of doxycycline in aqueous solution
    • Bogardus, J.B. and Blackwood, R.K. (1979) Solubility of doxycycline in aqueous solution. J. Pharm. Sci., 68, 188-194.
    • (1979) J. Pharm. Sci , vol.68 , pp. 188-194
    • Bogardus, J.B.1    Blackwood, R.K.2
  • 71
    • 40149094922 scopus 로고    scopus 로고
    • Strategy for the prediction and selection of drug substance salt forms
    • Brittain, H.G. (2007) Strategy for the prediction and selection of drug substance salt forms. Pharm. Technol., 31, 78-88.
    • (2007) Pharm. Technol , vol.31 , pp. 78-88
    • Brittain, H.G.1
  • 72
    • 84882389982 scopus 로고    scopus 로고
    • Introduction and overview to the preformulation development of solid dosage forms
    • (eds M.C. Adeyeye and H.G. Brittain), Informa Healthcare, New York
    • Brittain, H.G. (2008) Introduction and overview to the preformulation development of solid dosage forms. In Preformulation in Solid Dosage Form Development (eds M.C. Adeyeye and H.G. Brittain), Informa Healthcare, New York. ISBN 0-8247-5809-9.
    • (2008) Preformulation in Solid Dosage Form Development
    • Brittain, H.G.1
  • 73
    • 34250791543 scopus 로고    scopus 로고
    • The salt-cocrystal continuum: the influence of crystal structure on ionization state
    • Childs, S.L., Stahly, G.P. and Park, A. (2007) The salt-cocrystal continuum: the influence of crystal structure on ionization state. Molec. Pharm., 4, 323-338.
    • (2007) Molec. Pharm , vol.4 , pp. 323-338
    • Childs, S.L.1    Stahly, G.P.2    Park, A.3
  • 74
    • 0027997464 scopus 로고
    • A budesonide prodrug accelerates treatment of colitis in rats
    • Cui, N., Friend, D.R. and Fedorak, R.N. (1994) A budesonide prodrug accelerates treatment of colitis in rats. Gut, 35, 1439-1446.
    • (1994) Gut , vol.35 , pp. 1439-1446
    • Cui, N.1    Friend, D.R.2    Fedorak, R.N.3
  • 75
    • 0642312376 scopus 로고    scopus 로고
    • Synthesis and in vitro properties of prednisolone 21-sulfate sodium as a colon-specific prodrug of prednisolone
    • Doh, M.J., Jung, Y.J., Kim, I.H. et al. (2003) Synthesis and in vitro properties of prednisolone 21-sulfate sodium as a colon-specific prodrug of prednisolone. Arch. Pharm. Res., 26, 258-263.
    • (2003) Arch. Pharm. Res , vol.26 , pp. 258-263
    • Doh, M.J.1    Jung, Y.J.2    Kim, I.H.3
  • 76
    • 0024536377 scopus 로고
    • Microenvironmental pH control of drug dissolution
    • Doherty, C. and York, P. (1989) Microenvironmental pH control of drug dissolution. Int. J. Pharm., 50, 223-232.
    • (1989) Int. J. Pharm , vol.50 , pp. 223-232
    • Doherty, C.1    York, P.2
  • 77
    • 0034713306 scopus 로고    scopus 로고
    • Influence of admixed citric acid on the release profile of pelanserin hydrochloride from HPMC matrix tablets
    • Espinoza, R., Hong, E. and Villafuerte, L. (2000) Influence of admixed citric acid on the release profile of pelanserin hydrochloride from HPMC matrix tablets. Int. J. Pharm., 201, 165-173.
    • (2000) Int. J. Pharm , vol.201 , pp. 165-173
    • Espinoza, R.1    Hong, E.2    Villafuerte, L.3
  • 78
    • 0029890220 scopus 로고    scopus 로고
    • Factors affecting the dissolution of diclofenac salts
    • Fini, A., Fazio, G., Fernández Hervás, M.-J. et al. (1996) Factors affecting the dissolution of diclofenac salts. Eur. J. Pharm. Sci., 4, 231-238.
    • (1996) Eur. J. Pharm. Sci , vol.4 , pp. 231-238
    • Fini, A.1    Fazio, G.2    Fernández Hervás, M.-J.3
  • 79
    • 33749451891 scopus 로고    scopus 로고
    • Ionization states in the microenvironment of solid dosage forms: effect of formulation variables and processing
    • Govindarajan, R., Zinchuk, A., Hancock, B. et al. (2006) Ionization states in the microenvironment of solid dosage forms: effect of formulation variables and processing. Pharm. Res., 23, 2454-2468.
    • (2006) Pharm. Res , vol.23 , pp. 2454-2468
    • Govindarajan, R.1    Zinchuk, A.2    Hancock, B.3
  • 80
    • 77956367297 scopus 로고    scopus 로고
    • Impact of counterion on the chemical stability of crystalline salts of procaine
    • Guerrieri, P., Jarring, K. and Taylor, L.S. (2010) Impact of counterion on the chemical stability of crystalline salts of procaine. J. Pharm. Sci., 99, 3719-3730.
    • (2010) J. Pharm. Sci , vol.99 , pp. 3719-3730
    • Guerrieri, P.1    Jarring, K.2    Taylor, L.S.3
  • 81
    • 0027449074 scopus 로고
    • In-vitro evaluation of dexamethasone-beta-D-glucuronide for colon-specific drug-delivery
    • Haeberlin, B., Rubas, W., Nolen, H.W. and Friend, D.R. (1993) In-vitro evaluation of dexamethasone-beta-D-glucuronide for colon-specific drug-delivery. Pharm. Res., 10, 1553-1562.
    • (1993) Pharm. Res , vol.10 , pp. 1553-1562
    • Haeberlin, B.1    Rubas, W.2    Nolen, H.W.3    Friend, D.R.4
  • 82
    • 0015702659 scopus 로고
    • The dependence of paracetamol absorption on the rate of gastric emptying
    • Heading, R.C., Nimmo, J., Prescott, L.F. and Tothill, P. (1973) The dependence of paracetamol absorption on the rate of gastric emptying. Br. J. Pharmac., 47, 415-421.
    • (1973) Br. J. Pharmac , vol.47 , pp. 415-421
    • Heading, R.C.1    Nimmo, J.2    Prescott, L.F.3    Tothill, P.4
  • 83
    • 1042264121 scopus 로고    scopus 로고
    • Impact of solid state properties on developability assessment of drug candidates
    • Huang, L.-F. and Tong, W.-Q. (2004) Impact of solid state properties on developability assessment of drug candidates. Adv. Drug. Del. Rev., 56, 321-334.
    • (2004) Adv. Drug. Del. Rev , vol.56 , pp. 321-334
    • Huang, L.-F.1    Tong, W.-Q.2
  • 85
    • 0021806456 scopus 로고
    • Clinical pharmacokinetics of sulphasalazine, its metabolites and other prodrugs for 5-aminosalicylic acid
    • Klotz, U. (1985) Clinical pharmacokinetics of sulphasalazine, its metabolites and other prodrugs for 5-aminosalicylic acid. Clin. Pharmacokinet., 10, 285-302.
    • (1985) Clin. Pharmacokinet , vol.10 , pp. 285-302
    • Klotz, U.1
  • 86
    • 0015449031 scopus 로고
    • Solubility of organic hydrochlorides
    • Kramer, S.F. and Flynn, G.L. (1972) Solubility of organic hydrochlorides. J. Pharm. Sci., 61, 1896-1904.
    • (1972) J. Pharm. Sci , vol.61 , pp. 1896-1904
    • Kramer, S.F.1    Flynn, G.L.2
  • 87
    • 40949126942 scopus 로고    scopus 로고
    • Salt selection in drug development
    • Kumar, L., Amin, A. and Bansal, A.K. (2008) Salt selection in drug development. Pharm. Technol., 32 (3), 128-142.
    • (2008) Pharm. Technol , vol.32 , Issue.3 , pp. 128-142
    • Kumar, L.1    Amin, A.2    Bansal, A.K.3
  • 89
    • 23844499379 scopus 로고    scopus 로고
    • IV-IVC considerations in the development of immediate-release oral dosage form
    • Li, S.F., He, H.D., Parthiban, L.J. et al. (2005a) IV-IVC considerations in the development of immediate-release oral dosage form. J. Pharm. Sci., 94, 1396-1417.
    • (2005) J. Pharm. Sci , vol.94 , pp. 1396-1417
    • Li, S.F.1    He, H.D.2    Parthiban, L.J.3
  • 90
    • 18044381309 scopus 로고    scopus 로고
    • Investigation of solubility and dissolution of a free base and two different salt forms as a function of pH
    • Li, S., Wong, S.M., Sethia, S. et al. (2005b) Investigation of solubility and dissolution of a free base and two different salt forms as a function of pH. Pharm. Res., 22, 628-635.
    • (2005) Pharm. Res , vol.22 , pp. 628-635
    • Li, S.1    Wong, S.M.2    Sethia, S.3
  • 91
    • 0028339856 scopus 로고
    • Permeation of diclofenac salts through silicone membrane - a mechanistic study of percutaneous-absorption of ionizable drugs
    • Maitani, Y., Kugo, M. and Nagai, T. (1994) Permeation of diclofenac salts through silicone membrane - a mechanistic study of percutaneous-absorption of ionizable drugs. Chem. Pharm. Bull., 42, 1297-1301.
    • (1994) Chem. Pharm. Bull , vol.42 , pp. 1297-1301
    • Maitani, Y.1    Kugo, M.2    Nagai, T.3
  • 92
    • 0028219710 scopus 로고
    • An integrated approach to the selection of optimal salt form for a new drug candidate
    • Morris, K.R., Fakes, M.G., Thakur, A.B. et al. (1994) An integrated approach to the selection of optimal salt form for a new drug candidate. Int. J. Pharm., 105, 209-217.
    • (1994) Int. J. Pharm , vol.105 , pp. 209-217
    • Morris, K.R.1    Fakes, M.G.2    Thakur, A.B.3
  • 93
    • 70449176963 scopus 로고
    • Solution rate of theophylline salts and effects from oral administration
    • Nelson, E. (1957) Solution rate of theophylline salts and effects from oral administration. J. Am. Pharm. Soc. Sci. Ed., 46, 607-614.
    • (1957) J. Am. Pharm. Soc. Sci. Ed , vol.46 , pp. 607-614
    • Nelson, E.1
  • 94
    • 3142736454 scopus 로고    scopus 로고
    • The effect of citric acid added to hydroxypropyl methylcellulose (HPMC) matrix tablets on the release of vinpocetine
    • Nie, S., Pan, W., Li, X. and Wu, X. (2004) The effect of citric acid added to hydroxypropyl methylcellulose (HPMC) matrix tablets on the release of vinpocetine. Drug Dev. Ind. Pharm., 30, 627-635.
    • (2004) Drug Dev. Ind. Pharm , vol.30 , pp. 627-635
    • Nie, S.1    Pan, W.2    Li, X.3    Wu, X.4
  • 95
    • 77953716351 scopus 로고    scopus 로고
    • Pharmaceutical salts: a formulation trick or a clinical conundrum?
    • Patel, A., Jones, S.A., Ferro, A. and Patel, N. (2009) Pharmaceutical salts: a formulation trick or a clinical conundrum? Br. J. Cardiol., 16, 281-286.
    • (2009) Br. J. Cardiol , vol.16 , pp. 281-286
    • Patel, A.1    Jones, S.A.2    Ferro, A.3    Patel, N.4
  • 97
    • 0346104829 scopus 로고    scopus 로고
    • Salt selection and simultaneous polymorphism assessment via high-throughput crystallization. The case of sertraline
    • Remenar, J.F., MacPhee, J.M., Larson, B.K. et al. (2003) Salt selection and simultaneous polymorphism assessment via high-throughput crystallization. The case of sertraline. Org. Proc. Res. Dev., 7, 990-996.
    • (2003) Org. Proc. Res. Dev , vol.7 , pp. 990-996
    • Remenar, J.F.1    MacPhee, J.M.2    Larson, B.K.3
  • 98
    • 0033403992 scopus 로고    scopus 로고
    • Tablet dissolution affected by a moisture mediated solid-state interaction between drug and disintegrant
    • Rohrs, B.R., Thamann, T.J., Gao, P. et al. (1999) Tablet dissolution affected by a moisture mediated solid-state interaction between drug and disintegrant. Pharm. Res., 16, 1850-1856.
    • (1999) Pharm. Res , vol.16 , pp. 1850-1856
    • Rohrs, B.R.1    Thamann, T.J.2    Gao, P.3
  • 99
    • 0028088918 scopus 로고
    • pH related changes in the absorption of dipyridamole in the elderly
    • Russell, T.L., Berardi, R.R., Barnett, J.L. et al. (1994) pH related changes in the absorption of dipyridamole in the elderly. Pharm. Res., 11, 136-143.
    • (1994) Pharm. Res , vol.11 , pp. 136-143
    • Russell, T.L.1    Berardi, R.R.2    Barnett, J.L.3
  • 100
  • 101
    • 34548032742 scopus 로고    scopus 로고
    • Salt formation to improve drug solubility
    • Serajuddin, A.T.M. (2007) Salt formation to improve drug solubility. Adv. Drug Del. Rev., 59, 603-616.
    • (2007) Adv. Drug Del. Rev , vol.59 , pp. 603-616
    • Serajuddin, A.T.M.1
  • 102
    • 0021944082 scopus 로고
    • Effect of diffusion layer pH and solubility on the dissolution rate of pharmaceutical acids and their sodium salts. II: salicylic acid, theophylline and benzoic acid
    • Serajuddin, A.T.M. and Jarowski, C.I. (1985) Effect of diffusion layer pH and solubility on the dissolution rate of pharmaceutical acids and their sodium salts. II: salicylic acid, theophylline and benzoic acid. J. Pharm. Sci., 74, 148-154.
    • (1985) J. Pharm. Sci , vol.74 , pp. 148-154
    • Serajuddin, A.T.M.1    Jarowski, C.I.2
  • 103
    • 33747179333 scopus 로고    scopus 로고
    • Strategies for the design of hydrophilic matrix tablets with controlled microenvironmental pH
    • Siepe, S., Lueckel, B., Kramer, A. et al. (2006) Strategies for the design of hydrophilic matrix tablets with controlled microenvironmental pH. Int. J. Pharm., 316, 14-20.
    • (2006) Int. J. Pharm , vol.316 , pp. 14-20
    • Siepe, S.1    Lueckel, B.2    Kramer, A.3
  • 105
    • 79952224350 scopus 로고    scopus 로고
    • Physical stability of weak bases in the solid-state
    • Stephenson, G.A., Aburub, A. and Woods, T.A. (2011) Physical stability of weak bases in the solid-state. J. Pharm. Sci., 100, 1607-1617.
    • (2011) J. Pharm. Sci , vol.100 , pp. 1607-1617
    • Stephenson, G.A.1    Aburub, A.2    Woods, T.A.3
  • 106
    • 0034660109 scopus 로고    scopus 로고
    • pH-independent release of a weakly basic drug from water-insoluble and -soluble matrix tablets
    • Streubel, A., Siepmann, J., Dashevsky, A. and Bodmeier, R. (2000) pH-independent release of a weakly basic drug from water-insoluble and -soluble matrix tablets. J. Cont. Rel., 67, 101-110.
    • (2000) J. Cont. Rel , vol.67 , pp. 101-110
    • Streubel, A.1    Siepmann, J.2    Dashevsky, A.3    Bodmeier, R.4
  • 107
    • 77954759851 scopus 로고    scopus 로고
    • The influence of aqueous content in small scale salt screening - improving hit rate for weakly basic, low solubility drugs
    • Tarsa, P.B., Towler, C.S., Woollam, G. and Berghausen, J. (2010) The influence of aqueous content in small scale salt screening - improving hit rate for weakly basic, low solubility drugs. Eur. J. Pharm. Sci., 41, 23-30.
    • (2010) Eur. J. Pharm. Sci , vol.41 , pp. 23-30
    • Tarsa, P.B.1    Towler, C.S.2    Woollam, G.3    Berghausen, J.4
  • 108
    • 0027194762 scopus 로고
    • Effects of temperature and relative humidity on the solid-state chemical stability of ranitidine hydrochloride
    • Teraoka, R., Otsuka, M. and Matsuda, Y. (1993) Effects of temperature and relative humidity on the solid-state chemical stability of ranitidine hydrochloride. J. Pharm. Sci., 82 (1993) 601-604.
    • (1993) J. Pharm. Sci , vol.82 , Issue.1993 , pp. 601-604
    • Teraoka, R.1    Otsuka, M.2    Matsuda, Y.3
  • 109
    • 52249114680 scopus 로고    scopus 로고
    • Modulation of microenvironmental pH and crystallinity of ionizable telmisartan using alkalizers in solid dispersions for controlled release
    • Tran, P.H.L., Thanh, H.T. and Lee, B.-J. (2008) Modulation of microenvironmental pH and crystallinity of ionizable telmisartan using alkalizers in solid dispersions for controlled release. J. Cont. Rel., 129, 59-65.
    • (2008) J. Cont. Rel , vol.129 , pp. 59-65
    • Tran, P.H.L.1    Thanh, H.T.2    Lee, B.-J.3
  • 110
    • 14844320556 scopus 로고    scopus 로고
    • Influence of micro-environmental pH on the gel layer and release of a basic drug from various hydrophilic matrices
    • Varma, M.V.S., Kaushal, A.M. and Garg, S. (2005) Influence of micro-environmental pH on the gel layer and release of a basic drug from various hydrophilic matrices. J. Cont. Rel., 103, 499-510.
    • (2005) J. Cont. Rel , vol.103 , pp. 499-510
    • Varma, M.V.S.1    Kaushal, A.M.2    Garg, S.3
  • 112
    • 0025297596 scopus 로고
    • Application of gastric aciditycontrolled beagle dog to bioavailability study of cinnarizine
    • Yamada, I., Goda, T., Kawata, M. and Ogawa, K. (1990) Application of gastric aciditycontrolled beagle dog to bioavailability study of cinnarizine. Yakugaku Zasshi, 110, 280-285.
    • (1990) Yakugaku Zasshi , vol.110 , pp. 280-285
    • Yamada, I.1    Goda, T.2    Kawata, M.3    Ogawa, K.4
  • 113
    • 34248596026 scopus 로고    scopus 로고
    • Stabilization of the maleate salt of a basic drug by adjustment of microenvironment pH in solid dosage form
    • Zannou, E.A., Yatindra, Q.J., Joshi, M. and Serajuddin, A.T.M. (2007) Stabilization of the maleate salt of a basic drug by adjustment of microenvironment pH in solid dosage form. Int. J. Pharm., 337, 210-218.
    • (2007) Int. J. Pharm , vol.337 , pp. 210-218
    • Zannou, E.A.1    Yatindra, Q.J.2    Joshi, M.3    Serajuddin, A.T.M.4
  • 114
    • 0014104395 scopus 로고
    • Effect of polymorphism on the absorption of chloramphenicol from chloramphenicol palmitate
    • Aguiar, A.J., Krc Jr, J., Kinkel, A.W. and Samyn, J.C. (1967) Effect of polymorphism on the absorption of chloramphenicol from chloramphenicol palmitate. J. Pharm. Sci., 56, 847-853.
    • (1967) J. Pharm. Sci , vol.56 , pp. 847-853
    • Aguiar, A.J.1    Krc, J.2    Kinkel, A.W.3    Samyn, J.C.4
  • 115
    • 0002634817 scopus 로고
    • Mémoire sur les syst 'emes form' es par les points distribués régulièrement sur un plan ou dans l'espace
    • Bravais, A. (1850)Mémoire sur les syst 'emes form' es par les points distribués régulièrement sur un plan ou dans l'espace. J. Ecole Polytech., 19, 1-128.
    • (1850) J. Ecole Polytech , vol.19 , pp. 1-128
    • Bravais, A.1
  • 116
    • 77954864086 scopus 로고    scopus 로고
    • Characterisation of paracetamol Form III with rapid-heating DSC
    • Gaisford, S., Buanz, A.B.M. and Jethwa, N. (2010) Characterisation of paracetamol Form III with rapid-heating DSC. J. Pharm. Biomed. Anal., 53, 366-370.
    • (2010) J. Pharm. Biomed. Anal , vol.53 , pp. 366-370
    • Gaisford, S.1    Buanz, A.B.M.2    Jethwa, N.3
  • 118
    • 0002425795 scopus 로고    scopus 로고
    • Theory and origin of polymorphism
    • (ed. H.G. Brittain), Informa Healthcare
    • Grant, D.J.W. (1999) Theory and origin of polymorphism. In Polymorphism in Pharmaceutical Solids (ed. H.G. Brittain), Informa Healthcare. ISBN 0-8247-0237-3.
    • (1999) Polymorphism in Pharmaceutical Solids
    • Grant, D.J.W.1
  • 120
    • 38349160391 scopus 로고    scopus 로고
    • The use of high-speed differential scanning calorimetry (Hyper-DSC) in the study of pharmaceutical polymorphs
    • McGregor, C. and Bines, E. (2008) The use of high-speed differential scanning calorimetry (Hyper-DSC) in the study of pharmaceutical polymorphs. Int. J. Pharm., 350, 48-52.
    • (2008) Int. J. Pharm , vol.350 , pp. 48-52
    • McGregor, C.1    Bines, E.2
  • 121
    • 3543008927 scopus 로고    scopus 로고
    • The use of high-speed differential scanning calorimetry (DSC) to study the thermal properties of carbamazepine polymorphs
    • McGregor, C., Saunders, M. and Buckton, G. (2004) The use of high-speed differential scanning calorimetry (DSC) to study the thermal properties of carbamazepine polymorphs. Thermochim. Acta, 417, 231-237.
    • (2004) Thermochim. Acta , vol.417 , pp. 231-237
    • McGregor, C.1    Saunders, M.2    Buckton, G.3
  • 122
    • 0004294969 scopus 로고    scopus 로고
    • 4th edn, Butterworth-Heinemann, Oxford
    • Mullin, J.W. (2001) Crystallization, 4th edn, Butterworth-Heinemann, Oxford. ISBN 0-7506-4833-3.
    • (2001) Crystallization
    • Mullin, J.W.1
  • 123
    • 0031473049 scopus 로고    scopus 로고
    • Characterization and interconversion of polymorphs of premafloxacin, a new quinolone antibiotic
    • Schinzer, W.C., Bergren, M.S. and Aldrich, D.S. (1997) Characterization and interconversion of polymorphs of premafloxacin, a new quinolone antibiotic. J. Pharm. Sci., 86, 1426-1431.
    • (1997) J. Pharm. Sci , vol.86 , pp. 1426-1431
    • Schinzer, W.C.1    Bergren, M.S.2    Aldrich, D.S.3
  • 124
    • 0242288839 scopus 로고    scopus 로고
    • Influence of mechanical activation on the physical stability of salbutamol sulphate
    • Brodka-Pfeiffer, K., Langguth, P., Graß, P. and Häusler, H. (2003) Influence of mechanical activation on the physical stability of salbutamol sulphate. Eur. J. Pharm. Biopharm., 56, 393-400.
    • (2003) Eur. J. Pharm. Biopharm , vol.56 , pp. 393-400
    • Brodka-Pfeiffer, K.1    Langguth, P.2    Graß, P.3    Häusler, H.4
  • 125
    • 0034946478 scopus 로고    scopus 로고
    • Quantifying amorphous content of lactose using parallel beam X-ray powder diffraction and whole pattern fitting
    • Chen, X., Bates, S. and Morris, K.R. (2001) Quantifying amorphous content of lactose using parallel beam X-ray powder diffraction and whole pattern fitting. J. Pharm. Biomed. Anal., 26, 63-72.
    • (2001) J. Pharm. Biomed. Anal , vol.26 , pp. 63-72
    • Chen, X.1    Bates, S.2    Morris, K.R.3
  • 126
    • 34548455941 scopus 로고    scopus 로고
    • Comparison of quantitative methods for analysis of polyphasic pharmaceuticals
    • Giron, D., Monnier, S., Mutz, M. et al. (2007) Comparison of quantitative methods for analysis of polyphasic pharmaceuticals. J. Therm. Anal. Cal., 89, 729-743.
    • (2007) J. Therm. Anal. Cal , vol.89 , pp. 729-743
    • Giron, D.1    Monnier, S.2    Mutz, M.3
  • 127
    • 0032722007 scopus 로고    scopus 로고
    • The use of MTDSC to assess the amorphous phase content of a micronised drug substance
    • Guinot, S. and Leveiller, F. (1999) The use of MTDSC to assess the amorphous phase content of a micronised drug substance. Int. J. Pharm., 192, 63-75.
    • (1999) Int. J. Pharm , vol.192 , pp. 63-75
    • Guinot, S.1    Leveiller, F.2
  • 128
    • 85056318483 scopus 로고    scopus 로고
    • Comments on 'An approach to estimate the amorphous content of pharmaceutical powders using calorimetry with no calibration standards'
    • Hancock, B.C. (1998) Comments on 'An approach to estimate the amorphous content of pharmaceutical powders using calorimetry with no calibration standards'. Int. J. Pharm., 160, 131-133.
    • (1998) Int. J. Pharm , vol.160 , pp. 131-133
    • Hancock, B.C.1
  • 129
    • 0034633897 scopus 로고    scopus 로고
    • The quantification of small degrees of disorder in lactose using solution calorimetry
    • Hogan, S.E. and Buckton, G. (2000) The quantification of small degrees of disorder in lactose using solution calorimetry. Int. J. Pharm., 207, 57-64.
    • (2000) Int. J. Pharm , vol.207 , pp. 57-64
    • Hogan, S.E.1    Buckton, G.2
  • 130
    • 20344362926 scopus 로고    scopus 로고
    • Calorimetric investigation of the structural relaxation of amorphous materials: evaluating validity of the methodologies
    • Kawakami, K. and Pikal, M.J. (2005) Calorimetric investigation of the structural relaxation of amorphous materials: evaluating validity of the methodologies. J. Pharm. Sci., 94, 948-965.
    • (2005) J. Pharm. Sci , vol.94 , pp. 948-965
    • Kawakami, K.1    Pikal, M.J.2
  • 131
    • 29244470558 scopus 로고    scopus 로고
    • Quantification of low levels of amorphous content in sucrose by hyperDSC
    • Lappalainen, M., Pitkänen, I. and Harjunen, K. (2006) Quantification of low levels of amorphous content in sucrose by hyperDSC. Int. J. Pharm., 307, 150-155.
    • (2006) Int. J. Pharm , vol.307 , pp. 150-155
    • Lappalainen, M.1    Pitkänen, I.2    Harjunen, K.3
  • 132
    • 0037074074 scopus 로고    scopus 로고
    • Quantification of low levels (<10%) of amorphous content in micronised active batches using dynamic vapour sorption and isothermal microcalorimetry
    • Mackin, L., Zanon, R., Park, J.M. et al. (2002) Quantification of low levels (<10%) of amorphous content in micronised active batches using dynamic vapour sorption and isothermal microcalorimetry. Int. J. Pharm., 231, 227-236.
    • (2002) Int. J. Pharm , vol.231 , pp. 227-236
    • Mackin, L.1    Zanon, R.2    Park, J.M.3
  • 133
    • 0034950053 scopus 로고    scopus 로고
    • The use of inverse phase gas chromatography to measure the surface energy of crystalline, amorphous and recently milled lactose
    • Newell, H.E., Buckton, G., Butler, D.A. et al. (2001) The use of inverse phase gas chromatography to measure the surface energy of crystalline, amorphous and recently milled lactose. Pharm. Res., 18, 662-666.
    • (2001) Pharm. Res , vol.18 , pp. 662-666
    • Newell, H.E.1    Buckton, G.2    Butler, D.A.3
  • 134
    • 80052267239 scopus 로고    scopus 로고
    • Application and use of isothermal calorimetry in pharmaceutical development
    • O'Neill, M.A.A. and Gaisford, S. (2011) Application and use of isothermal calorimetry in pharmaceutical development. Int. J. Pharm., 417, 83-93.
    • (2011) Int. J. Pharm , vol.417 , pp. 83-93
    • O'Neill, M.A.A.1    Gaisford, S.2
  • 136
    • 0030901259 scopus 로고    scopus 로고
    • An approach to estimate the amorphous content of pharmaceutical powders using calorimetry with no calibration standards
    • Phillips, E.M. (1997) An approach to estimate the amorphous content of pharmaceutical powders using calorimetry with no calibration standards. Int. J. Pharm., 149, 267-271.
    • (1997) Int. J. Pharm , vol.149 , pp. 267-271
    • Phillips, E.M.1
  • 137
    • 23444462493 scopus 로고    scopus 로고
    • Calorimetric determination of amorphous content in lactose: a note on the preparation of calibration curves
    • Ramos, R., Gaisford, S. and Buckton, G. (2005) Calorimetric determination of amorphous content in lactose: a note on the preparation of calibration curves. Int. J. Pharm., 300, 13-21.
    • (2005) Int. J. Pharm , vol.300 , pp. 13-21
    • Ramos, R.1    Gaisford, S.2    Buckton, G.3
  • 138
    • 0032703825 scopus 로고    scopus 로고
    • The detection of amorphous material in a nominally crystalline drug using modulated temperature DSC - a case study
    • Saklatvala, R., Royall, P.G. and Craig, D.Q.M. (1999) The detection of amorphous material in a nominally crystalline drug using modulated temperature DSC - a case study. Int. J. Pharm., 192, 55-62.
    • (1999) Int. J. Pharm , vol.192 , pp. 55-62
    • Saklatvala, R.1    Royall, P.G.2    Craig, D.Q.M.3
  • 139
    • 1842557588 scopus 로고    scopus 로고
    • The potential of high speed DSC (hyper-DSC) for the detection and quantification of small amounts of amorphous content in predominantly crystalline samples
    • Saunders, M., Podluii, K., Shergill, S. et al. (2004) The potential of high speed DSC (hyper-DSC) for the detection and quantification of small amounts of amorphous content in predominantly crystalline samples. Int. J. Pharm., 274, 35-40.
    • (2004) Int. J. Pharm , vol.274 , pp. 35-40
    • Saunders, M.1    Podluii, K.2    Shergill, S.3
  • 140
    • 77954312924 scopus 로고    scopus 로고
    • Determination of low levels of amorphous content in inhalation grade lactose by moisture sorption isotherms
    • Vollenbroek, J., Hebbink, G.A., Ziffels, S. and Steckel, H. (2010) Determination of low levels of amorphous content in inhalation grade lactose by moisture sorption isotherms. Int. J. Pharm., 395, 62-70.
    • (2010) Int. J. Pharm , vol.395 , pp. 62-70
    • Vollenbroek, J.1    Hebbink, G.A.2    Ziffels, S.3    Steckel, H.4
  • 141
    • 0014699523 scopus 로고
    • Non-symmetrical dielectric relaxation behaviour arising from a simple empirical decay function
    • Williams, G. and Watts, D.C. (1970) Non-symmetrical dielectric relaxation behaviour arising from a simple empirical decay function. Trans. Fara. Soc., 66, 80-85.
    • (1970) Trans. Fara. Soc , vol.66 , pp. 80-85
    • Williams, G.1    Watts, D.C.2
  • 143
    • 37049148254 scopus 로고
    • Mechanism and kinetics of carboxylic ester hydrolysis and carboxyl esterification
    • Day, J.N.E. and Ingold, C.K. (1941) Mechanism and kinetics of carboxylic ester hydrolysis and carboxyl esterification. Trans. Faraday Soc., 37, 686-705.
    • (1941) Trans. Faraday Soc , vol.37 , pp. 686-705
    • Day, J.N.E.1    Ingold, C.K.2
  • 144
    • 50249162817 scopus 로고
    • Autoxidation of etheric oils used in pharmacy
    • Fryklöf, L.-E. (1954) Autoxidation of etheric oils used in pharmacy. Farm. Rev., 53, 317-335.
    • (1954) Farm. Rev , vol.53 , pp. 317-335
    • Fryklöf, L.-E.1
  • 145
    • 0017437920 scopus 로고
    • Humidity fixed of binary saturated aqueous solutions
    • Greenspan, L. (1977) Humidity fixed of binary saturated aqueous solutions. J. Res. Natl Bur. Stand., 81A (1977) 89-96.
    • (1977) J. Res. Natl Bur. Stand , vol.81 A , Issue.1977 , pp. 89-96
    • Greenspan, L.1
  • 146
    • 0344014812 scopus 로고
    • Storage conditions for stability testing (Part 2)
    • Grimm, W. (1986) Storage conditions for stability testing (Part 2). Drugs Made in Germany, 29, 39-47.
    • (1986) Drugs Made in Germany , vol.29 , pp. 39-47
    • Grimm, W.1
  • 147
    • 0031954253 scopus 로고    scopus 로고
    • Extension of the International Conference on Harmonisation Tripartite Guidelines for stability testing of new drug substances and products to countries of Climatic Zones III and IV
    • Grimm, W. (1998) Extension of the International Conference on Harmonisation Tripartite Guidelines for stability testing of new drug substances and products to countries of Climatic Zones III and IV. Drug Dev. Ind. Pharm., 24, 313-325.
    • (1998) Drug Dev. Ind. Pharm , vol.24 , pp. 313-325
    • Grimm, W.1
  • 151
    • 84949755804 scopus 로고
    • Processed photographic colour films and paper prints -methods for measuring image stability
    • ISO 10977 (1993) Photography. Processed photographic colour films and paper prints -methods for measuring image stability.
    • (1993) Photography
  • 152
    • 0033051354 scopus 로고    scopus 로고
    • Trends in stability testing, with emphasis on stability during distribution and storage
    • Kommanaboyina, B. and Rhodes, C.T. (1999) Trends in stability testing, with emphasis on stability during distribution and storage. Drug. Dev. Ind. Pharm., 25, 857-868.
    • (1999) Drug. Dev. Ind. Pharm , vol.25 , pp. 857-868
    • Kommanaboyina, B.1    Rhodes, C.T.2
  • 153
    • 34250459937 scopus 로고
    • Stability of d-cycloserine in aqueous solutions at high concentrations
    • Kondrat'eva, A.P., Bruns, B.P. and Libinson, G.S. (1971) Stability of d-cycloserine in aqueous solutions at high concentrations. Pharm. Chem. J., 5, 356-360.
    • (1971) Pharm. Chem. J , vol.5 , pp. 356-360
    • Kondrat'eva, A.P.1    Bruns, B.P.2    Libinson, G.S.3
  • 154
    • 0019850513 scopus 로고
    • Stability of procaine hydrochloride in a buffered cardioplegia formulation
    • Loucas, S.P., Mehl, B., Litwak, R.S. and Jurado, R.A. (1981) Stability of procaine hydrochloride in a buffered cardioplegia formulation. Am. J. Hosp. Pharm., 38, 1924-1928.
    • (1981) Am. J. Hosp. Pharm , vol.38 , pp. 1924-1928
    • Loucas, S.P.1    Mehl, B.2    Litwak, R.S.3    Jurado, R.A.4
  • 156
    • 33846385383 scopus 로고    scopus 로고
    • Modification of the crystal habit of celecoxib for improved processability
    • Banga, S., Chawla, G., Varandani, D. and Mehta, B.R. (2007) Modification of the crystal habit of celecoxib for improved processability. J. Pharm. Pharmacol., 59, 29-39.
    • (2007) J. Pharm. Pharmacol , vol.59 , pp. 29-39
    • Banga, S.1    Chawla, G.2    Varandani, D.3    Mehta, B.R.4
  • 157
    • 0035206815 scopus 로고    scopus 로고
    • Particle size distribution, Part 1, representations of particle shape, size and distribution
    • Brittain, H.G. (2001) Particle size distribution, Part 1, representations of particle shape, size and distribution. Pharm. Technol., 25, 38-45.
    • (2001) Pharm. Technol , vol.25 , pp. 38-45
    • Brittain, H.G.1
  • 158
    • 0026749510 scopus 로고
    • Crystal habit modifications and altered tableting characteristics
    • Kaul, D., Nguyen, N.T. and Venkataram, S. (1992) Crystal habit modifications and altered tableting characteristics. Int. J. Pharm., 88, 345-350.
    • (1992) Int. J. Pharm , vol.88 , pp. 345-350
    • Kaul, D.1    Nguyen, N.T.2    Venkataram, S.3
  • 159
    • 0037026268 scopus 로고    scopus 로고
    • Crystal habit and tableting behavior
    • Rasenack, N. andMüller, B.W. (2002) Crystal habit and tableting behavior. Int. J. Pharm., 244, 45-57.
    • (2002) Int. J. Pharm , vol.244 , pp. 45-57
    • Rasenack, N.1    Müller, B.W.2
  • 160
    • 0000496231 scopus 로고
    • Evaluating flow properties of solids
    • Carr, R.L. (1965) Evaluating flow properties of solids. Chem. Engng, 72, 163-167.
    • (1965) Chem. Engng , vol.72 , pp. 163-167
    • Carr, R.L.1
  • 161
    • 0002737830 scopus 로고
    • Friction conditions in a mass of metal powder
    • Hausner, H.H. (1967) Friction conditions in a mass of metal powder. Int. J. Powder Metall., 3, 7-13.
    • (1967) Int. J. Powder Metall , vol.3 , pp. 7-13
    • Hausner, H.H.1
  • 162
    • 84984087501 scopus 로고
    • Some angular properties of magnesia and their relevance to material handling
    • Jones, T.M. and Pilpel, N. (1966) Some angular properties of magnesia and their relevance to material handling. J. Pharm. Pharmacol., 18, 182T.
    • (1966) J. Pharm. Pharmacol , vol.18 , pp. 182T
    • Jones, T.M.1    Pilpel, N.2
  • 164
    • 0028025198 scopus 로고
    • Effect of moisture sorption on tableting characteristics of spray dried (15% amorphous) lactose
    • Sebhatu, T., Elamin, A.A. and Ahlneck, C. (1994) Effect of moisture sorption on tableting characteristics of spray dried (15% amorphous) lactose. Pharm. Res., 11, 1233-1238.
    • (1994) Pharm. Res , vol.11 , pp. 1233-1238
    • Sebhatu, T.1    Elamin, A.A.2    Ahlneck, C.3


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