-
1
-
-
77953416359
-
-
Separation Science and Technology Series, vol. 8, Academic Press, London
-
Ahuja, S. and Rasmussen, H. (2007) HPLC Method Development for Pharmaceuticals, Separation Science and Technology Series, vol. 8, Academic Press, London. ISBN 0-1237-0540-1.
-
(2007)
HPLC Method Development for Pharmaceuticals
-
-
Ahuja, S.1
Rasmussen, H.2
-
2
-
-
0030647671
-
The utility of phase correction in modulated DSC
-
Aubuchon, S.R. and Gill, P.S. (1997) The utility of phase correction in modulated DSC. J. Therm. Anal. Cal., 49, 1039-1044.
-
(1997)
J. Therm. Anal. Cal
, vol.49
, pp. 1039-1044
-
-
Aubuchon, S.R.1
Gill, P.S.2
-
3
-
-
0016988717
-
Acidic potassium dichromate solutions as ultraviolet absorbance standards
-
Burke, R.W. and Mavrodineanu, R. (1976) Acidic potassium dichromate solutions as ultraviolet absorbance standards. J. Res. Natl Bur. Stand. A, 80A, 631-636.
-
(1976)
J. Res. Natl Bur. Stand. A
, vol.80 A
, pp. 631-636
-
-
Burke, R.W.1
Mavrodineanu, R.2
-
7
-
-
77649234756
-
How to improve R&D productivity: the pharmaceutical industry's grand challenge
-
Paul, S.M., Mytelka, D.S., Dunwiddie, C.T. et al. (2010) How to improve R&D productivity: the pharmaceutical industry's grand challenge. Nat. Rev. Drug Disc., 9, 203-214.
-
(2010)
Nat. Rev. Drug Disc
, vol.9
, pp. 203-214
-
-
Paul, S.M.1
Mytelka, D.S.2
Dunwiddie, C.T.3
-
8
-
-
0034665153
-
Practitioner's guide to method development in thinlayer chromatography
-
Poole, C.F. and Dias, N.C. (2000) Practitioner's guide to method development in thinlayer chromatography. J. Chromatogr. A., 892, 123-142.
-
(2000)
J. Chromatogr. A
, vol.892
, pp. 123-142
-
-
Poole, C.F.1
Dias, N.C.2
-
9
-
-
0001419232
-
Modulated differential scanning calorimetry
-
Reading, M., Luget, A. and Wilson, R. (1994) Modulated differential scanning calorimetry. Thermochim. Acta, 238, 295-307.
-
(1994)
Thermochim. Acta
, vol.238
, pp. 295-307
-
-
Reading, M.1
Luget, A.2
Wilson, R.3
-
10
-
-
77955469357
-
Modulated temperature differential scanning calorimetry
-
(eds D.Q.M. Craig and M. Reading), CRC Press, Boca Raton, FL
-
Reading, M., Craig, D.Q.M., Murphy, J.R. and Kett, V.L. (2007) Modulated temperature differential scanning calorimetry. In Thermal Analysis of Pharmaceuticals (eds D.Q.M. Craig and M. Reading), CRC Press, Boca Raton, FL. ISBN 0-8247-5814-5.
-
(2007)
Thermal Analysis of Pharmaceuticals
-
-
Reading, M.1
Craig, D.Q.M.2
Murphy, J.R.3
Kett, V.L.4
-
11
-
-
0022026693
-
Spectral transmittance characteristics of holmium oxide in perchloric acid solution
-
Weidner, V.R., Mavrodineanu, R., and Mielenz, K.D. (1985) Spectral transmittance characteristics of holmium oxide in perchloric acid solution. J. Res. Natl Bur. Stand., 90, 115-125.
-
(1985)
J. Res. Natl Bur. Stand
, vol.90
, pp. 115-125
-
-
Weidner, V.R.1
Mavrodineanu, R.2
Mielenz, K.D.3
-
13
-
-
72149101372
-
a distribution of drugs: application to drug discovery
-
a distribution of drugs: application to drug discovery. Perspect. Med. Chem., 1, 25-38.
-
(2007)
Perspect. Med. Chem
, vol.1
, pp. 25-38
-
-
Manallack, D.T.1
-
14
-
-
36048986392
-
a values for pharmaceutical substances
-
(ed. H.B. Brittain), vol. 33, Academic Press, San Diego
-
a values for pharmaceutical substances. In Profiles of Drug Substances, Excipients and Related Methodology (ed. H.B. Brittain), vol. 33, Academic Press, San Diego, pp. 1-726. ISBN 9780-1226-0833-9.
-
(2007)
Profiles of Drug Substances, Excipients and Related Methodology
, pp. 1-726
-
-
Prankerd, R.J.1
-
15
-
-
0002293876
-
The behaviour of carboxylic acids in mixed solvents
-
(ed. B. Pesce), Pergamon Press
-
Shedlovsky, T. (1962) The behaviour of carboxylic acids in mixed solvents. In Electrolytes (ed. B. Pesce), Pergamon Press, pp. 146-151. ISBN 0-0801-3778-4.
-
(1962)
Electrolytes
, pp. 146-151
-
-
Shedlovsky, T.1
-
16
-
-
0142028495
-
a determination of water-insoluble compounds: validation study in methanol/water mixtures
-
a determination of water-insoluble compounds: validation study in methanol/water mixtures. Int. J. Pharm., 151, 235-248.
-
(1997)
Int. J. Pharm
, vol.151
, pp. 235-248
-
-
Takács-Novák, K.1
Box, K.J.2
Avdeef, A.3
-
17
-
-
0001286790
-
Pharmaceutical preformulation
-
John Wiley & Sons, Ltd, Chichester
-
Wells, J.I. (1988) Pharmaceutical preformulation. In The Physicochemical Properties of Drug Substances, John Wiley & Sons, Ltd, Chichester. ISBN 0-470-21114-8.
-
(1988)
The Physicochemical Properties of Drug Substances
-
-
Wells, J.I.1
-
18
-
-
12344335757
-
Stability of metronidazole, tetracycline HCl and famotidine alone and in combination
-
Wu, Y. and Fassihi, R. (2005) Stability of metronidazole, tetracycline HCl and famotidine alone and in combination. Int. J. Pharm., 290, 1-13.
-
(2005)
Int. J. Pharm
, vol.290
, pp. 1-13
-
-
Wu, Y.1
Fassihi, R.2
-
19
-
-
0001266728
-
Dissociation constants of some carboxylic acids in mixed aqueous solvents
-
Yasuda, M. (1959) Dissociation constants of some carboxylic acids in mixed aqueous solvents. Bull. Chem. Soc. Jpn, 32, 429-432.
-
(1959)
Bull. Chem. Soc. Jpn
, vol.32
, pp. 429-432
-
-
Yasuda, M.1
-
20
-
-
0023547921
-
A thermodynamic analysis of the Collander equation and establishment of a reference solvent for use in drug partitioning studies
-
Beezer, A.E., Gooch, C.A., Hunter, W.H. and Volpe, P.L. (1987) A thermodynamic analysis of the Collander equation and establishment of a reference solvent for use in drug partitioning studies. J. Pharm. Pharmacol., 39, 774-779.
-
(1987)
J. Pharm. Pharmacol
, vol.39
, pp. 774-779
-
-
Beezer, A.E.1
Gooch, C.A.2
Hunter, W.H.3
Volpe, P.L.4
-
21
-
-
0014685056
-
Partition data of penicillins determined by means of reversed-phase thin-layer chromatography
-
Biagi, G.L., Barbaro, A.M., Gamba, M.F. and Guerra, M.C. (1964) Partition data of penicillins determined by means of reversed-phase thin-layer chromatography. J. Chromatogr. A, 41, 371-379.
-
(1964)
J. Chromatogr. A
, vol.41
, pp. 371-379
-
-
Biagi, G.L.1
Barbaro, A.M.2
Gamba, M.F.3
Guerra, M.C.4
-
22
-
-
0014675062
-
Partition data of cephalosporins determined by means of reversed-phase thin layer chromatography
-
Biagi, G.L., Barbaro, A.M., Guerra, M.C. and Gamba, M.F. (1969) Partition data of cephalosporins determined by means of reversed-phase thin layer chromatography. J. Chromatogr. A, 44, 195-198.
-
(1969)
J. Chromatogr. A
, vol.44
, pp. 195-198
-
-
Biagi, G.L.1
Barbaro, A.M.2
Guerra, M.C.3
Gamba, M.F.4
-
23
-
-
0028299385
-
Determination of lipophilicity by means of reversed-phase thin-layer chromatography. i. Basic aspects and relationship between slope and intercept of TLC equations
-
Biagi, G.L., Barbaro, A.M., Sapone, A. and Recanatini, M. (1994a) Determination of lipophilicity by means of reversed-phase thin-layer chromatography. i. Basic aspects and relationship between slope and intercept of TLC equations. J. Chromatogr. A, 662, 341-361.
-
(1994)
J. Chromatogr. A
, vol.662
, pp. 341-361
-
-
Biagi, G.L.1
Barbaro, A.M.2
Sapone, A.3
Recanatini, M.4
-
24
-
-
0028243154
-
Determination of lipophilicity by means of reversed-phase thin-layer chromatography. ii. Influence of the organic modifier on the slope of the thin-layer chromatographic equation
-
Biagi, G.L., Barbaro, A.M., Sapone, A. and Recanatini, M. (1994b) Determination of lipophilicity by means of reversed-phase thin-layer chromatography. ii. Influence of the organic modifier on the slope of the thin-layer chromatographic equation. J. Chromatogr. A, 669, 246-253.
-
(1994)
J. Chromatogr. A
, vol.669
, pp. 246-253
-
-
Biagi, G.L.1
Barbaro, A.M.2
Sapone, A.3
Recanatini, M.4
-
25
-
-
0027997411
-
Determination of lipophilicity by means of reversed-phase thin-layer chromatography. iii. Study of the TLC equations for a series of ionizable quinolone derivatives
-
Biagi, G.L., Barbaro, A.M. and Recanatini, M. (1994c) Determination of lipophilicity by means of reversed-phase thin-layer chromatography. iii. Study of the TLC equations for a series of ionizable quinolone derivatives. J. Chromatogr. A, 678, 127-137.
-
(1994)
J. Chromatogr. A
, vol.678
, pp. 127-137
-
-
Biagi, G.L.1
Barbaro, A.M.2
Recanatini, M.3
-
26
-
-
0015237832
-
Reversed-phase thin layer chromatography and partition coefficients of penicillins
-
Bird, A.E. and Marshall, C. (1971) Reversed-phase thin layer chromatography and partition coefficients of penicillins. J. Chromatogr. A, 63, 313-319.
-
(1971)
J. Chromatogr. A
, vol.63
, pp. 313-319
-
-
Bird, A.E.1
Marshall, C.2
-
27
-
-
0020076112
-
Partitioning of organic compounds in octanol-water systems
-
Chiou, C.T., Schmedding, D.W. and Manes, M. (1982) Partitioning of organic compounds in octanol-water systems. Environ. Sci. Technol., 16, 4-10.
-
(1982)
Environ. Sci. Technol
, vol.16
, pp. 4-10
-
-
Chiou, C.T.1
Schmedding, D.W.2
Manes, M.3
-
28
-
-
0023804237
-
Measurement of the distribution coefficients of several classes of drug using reversed-phase thin-layer chromatography
-
Jack, D.B., Hawker, J.L., Rooney, L. et al. (1988) Measurement of the distribution coefficients of several classes of drug using reversed-phase thin-layer chromatography. J. Chromatogr. A, 452, 257-264.
-
(1988)
J. Chromatogr. A
, vol.452
, pp. 257-264
-
-
Jack, D.B.1
Hawker, J.L.2
Rooney, L.3
-
29
-
-
77955581133
-
Revisiting thin-layer chromatography as a lipophilicity determination tool - a comparative study on several techniques with a model solute set
-
Komsta, L., Skibinski, R., Berecka, A. et al. (2010) Revisiting thin-layer chromatography as a lipophilicity determination tool - a comparative study on several techniques with a model solute set. J. Pharm. Biomed. Anal., 53, 911-918.
-
(2010)
J. Pharm. Biomed. Anal
, vol.53
, pp. 911-918
-
-
Komsta, L.1
Skibinski, R.2
Berecka, A.3
-
30
-
-
0027818680
-
Modeling oil-water partitioning and membrane permeation using reversed-phase chromatography
-
Lambert, W.J. (1993) Modeling oil-water partitioning and membrane permeation using reversed-phase chromatography. J. Chromatogr. A, 656, 469-484.
-
(1993)
J. Chromatogr. A
, vol.656
, pp. 469-484
-
-
Lambert, W.J.1
-
31
-
-
8644243613
-
Partition coefficients and their uses
-
Leo, A., Hansch, C. and Elkins, D. (1971) Partition coefficients and their uses. Chem. Rev., 71, 525-616.
-
(1971)
Chem. Rev
, vol.71
, pp. 525-616
-
-
Leo, A.1
Hansch, C.2
Elkins, D.3
-
32
-
-
0021124186
-
General approach for the estimation of octanol/water partition coefficient by reversed-phase high-performance liquid chromatography
-
Valkó, K. (1984) General approach for the estimation of octanol/water partition coefficient by reversed-phase high-performance liquid chromatography. J. Liq. Chromatogr., 7, 1405-1424.
-
(1984)
J. Liq. Chromatogr
, vol.7
, pp. 1405-1424
-
-
Valkó, K.1
-
33
-
-
2342635206
-
Application of high-performance liquid chromatography based measurements of lipophilicity to model biological distribution
-
Valkó, K. (2004) Application of high-performance liquid chromatography based measurements of lipophilicity to model biological distribution. J. Chromatogr. A, 1037, 299-310.
-
(2004)
J. Chromatogr. A
, vol.1037
, pp. 299-310
-
-
Valkó, K.1
-
34
-
-
0027402651
-
New chromatographic hydrophobicity index (φ0) based on the slope and the intercept of the log K _ versus organic phase concentration plot
-
Valkó, K. and Slégel, P. (1993) New chromatographic hydrophobicity index (φ0) based on the slope and the intercept of the log K _ versus organic phase concentration plot. J. Chromatogr. A, 631, 49-61.
-
(1993)
J. Chromatogr. A
, vol.631
, pp. 49-61
-
-
Valkó, K.1
Slégel, P.2
-
35
-
-
0000607945
-
Chromatographic hydrophobicity index by fast-gradient RP-HPLC: a high-throughput alternative to log P/log D
-
Valkó, K., Bevan, C. and Reynolds, D. (1997) Chromatographic hydrophobicity index by fast-gradient RP-HPLC: a high-throughput alternative to log P/log D. Anal. Chem., 69, 2022-2029.
-
(1997)
Anal. Chem
, vol.69
, pp. 2022-2029
-
-
Valkó, K.1
Bevan, C.2
Reynolds, D.3
-
36
-
-
0022818104
-
Determination of partition coefficients and aqueous solubilities by reverse phase chromatography - I. Theory and background
-
Weber Jr, W.J., Chin, Y.-P. and Rice, C.P. (1986) Determination of partition coefficients and aqueous solubilities by reverse phase chromatography - I. Theory and background. Water Res., 20, 1433-1442.
-
(1986)
Water Res
, vol.20
, pp. 1433-1442
-
-
Weber, W.J.1
Chin, Y.-P.2
Rice, C.P.3
-
39
-
-
0028948839
-
A theoretical basis for a biopharmaceutical drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability
-
Amidon, G.L., Lennernäs, H., Shah, V.P. and Crison, J.R. (1995) A theoretical basis for a biopharmaceutical drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability. Pharm. Res., 12, 413-420.
-
(1995)
Pharm. Res
, vol.12
, pp. 413-420
-
-
Amidon, G.L.1
Lennernäs, H.2
Shah, V.P.3
Crison, J.R.4
-
40
-
-
0033224876
-
Solubility of paracetamol in pure solvents
-
Granberg, R.A. and Rasmuson, A.C. (1999) Solubility of paracetamol in pure solvents. J. Chem. Engng Data, 44, 1391-1395.
-
(1999)
J. Chem. Engng Data
, vol.44
, pp. 1391-1395
-
-
Granberg, R.A.1
Rasmuson, A.C.2
-
41
-
-
0002177778
-
Biopharmaceutical considerations in drug formulation design and evaluation
-
Kaplan, S.A. (1972) Biopharmaceutical considerations in drug formulation design and evaluation. Drug Met. Rev., 1, 15-34.
-
(1972)
Drug Met. Rev
, vol.1
, pp. 15-34
-
-
Kaplan, S.A.1
-
42
-
-
0030886937
-
Managing the drug discovery/development interface
-
Kennedy, T. (1997) Managing the drug discovery/development interface. Drug Disc. Today, 2, 436-444.
-
(1997)
Drug Disc. Today
, vol.2
, pp. 436-444
-
-
Kennedy, T.1
-
43
-
-
0000882284
-
Purity determination by differential scanning calorimetry
-
Marti, E.E. (1972) Purity determination by differential scanning calorimetry. Thermochim. Acta, 5, 173-220.
-
(1972)
Thermochim. Acta
, vol.5
, pp. 173-220
-
-
Marti, E.E.1
-
44
-
-
66049083443
-
Temperature and solvent effects in the solubility of some pharmaceutical compounds: measurements and modeling
-
Mota, F.L., Carneiro, A.P., Queimada, A.J. et al. (2009) Temperature and solvent effects in the solubility of some pharmaceutical compounds: measurements and modeling. Eur. J. Pharm. Sci., 37, 499-507.
-
(2009)
Eur. J. Pharm. Sci
, vol.37
, pp. 499-507
-
-
Mota, F.L.1
Carneiro, A.P.2
Queimada, A.J.3
-
45
-
-
0026733159
-
Solid state properties of drugs. I. Estimation of heat capacities for fusion and thermodynamic functions for solution from aqueous solubility-temperature dependence measurements
-
Prankerd, R.J. (1992) Solid state properties of drugs. I. Estimation of heat capacities for fusion and thermodynamic functions for solution from aqueous solubility-temperature dependence measurements. Int. J. Pharm., 84, 233-244.
-
(1992)
Int. J. Pharm
, vol.84
, pp. 233-244
-
-
Prankerd, R.J.1
-
46
-
-
0019809124
-
Difference in physic-chemical properties between crystalline and non-crystalline 9,3__-diacetylmidecamycin
-
Sato, T., Okada, A., Sekiguchi, K. and Tsuda, Y. (1981) Difference in physic-chemical properties between crystalline and non-crystalline 9,3__-diacetylmidecamycin. Chem. Pharm. Bull., 29, 2675-2682.
-
(1981)
Chem. Pharm. Bull
, vol.29
, pp. 2675-2682
-
-
Sato, T.1
Okada, A.2
Sekiguchi, K.3
Tsuda, Y.4
-
47
-
-
33947091552
-
Simple equation for linearization of data in differential scanning calorimetric purity determinations
-
Sondack, D.L. (1972) Simple equation for linearization of data in differential scanning calorimetric purity determinations. Anal. Chem., 44, 888.
-
(1972)
Anal. Chem
, vol.44
, pp. 888
-
-
Sondack, D.L.1
-
48
-
-
34447536520
-
When poor solubility becomes an issue: from early stage to proof of concept
-
Stegemann, S., Leveiller, F., Franchi, D. et al. (2007) When poor solubility becomes an issue: from early stage to proof of concept. Eur. J. Pharm. Sci., 31, 249-261.
-
(2007)
Eur. J. Pharm. Sci
, vol.31
, pp. 249-261
-
-
Stegemann, S.1
Leveiller, F.2
Franchi, D.3
-
49
-
-
77955248335
-
The biowaiver extension for BCS class III drugs: the effect of dissolution rate on the bioequivalence of BCS class III immediate-release drugs predicted by computer simulation
-
Tsume, Y. and Amidon, G.L. (2010) The biowaiver extension for BCS class III drugs: the effect of dissolution rate on the bioequivalence of BCS class III immediate-release drugs predicted by computer simulation. Molec. Pharm., 7, 1235-1243.
-
(2010)
Molec. Pharm
, vol.7
, pp. 1235-1243
-
-
Tsume, Y.1
Amidon, G.L.2
-
50
-
-
0021233407
-
Purity determinations of drugs with differential scanning calorimetry (DSC) - a critical review
-
van Dooren, A.A. and Müller, B.W. (1984) Purity determinations of drugs with differential scanning calorimetry (DSC) - a critical review. Int. J. Pharm., 20, 217-233.
-
(1984)
Int. J. Pharm
, vol.20
, pp. 217-233
-
-
Van Dooren, A.A.1
Müller, B.W.2
-
52
-
-
0002642747
-
Reaktionsgeschwindigkeit in heterogenen systemen
-
Brunner, E. (1904) Reaktionsgeschwindigkeit in heterogenen systemen. Z. Phys. Chem., 43, 56-102.
-
(1904)
Z. Phys. Chem
, vol.43
, pp. 56-102
-
-
Brunner, E.1
-
53
-
-
33747348812
-
Über die Auflösungsgeschwindigkeit fester Körper
-
Brunner, E. and Tolloczko, S. (1900) Über die Auflösungsgeschwindigkeit fester Körper. Z. Phys. Chem., 35, 283-290.
-
(1900)
Z. Phys. Chem
, vol.35
, pp. 283-290
-
-
Brunner, E.1
Tolloczko, S.2
-
54
-
-
0000354093
-
Significance of liquid-film coefficients in gas absorption
-
Danckwerts, P.V. (1951) Significance of liquid-film coefficients in gas absorption. Ind. Engng Chem., 43, 1460-1467.
-
(1951)
Ind. Engng Chem
, vol.43
, pp. 1460-1467
-
-
Danckwerts, P.V.1
-
55
-
-
33747373878
-
Acentury of dissolution research: from Noyes and Whitney to the biopharmaceutical classification system
-
Dokoumetzidis, A. and Macheras, P. (2006)Acentury of dissolution research: from Noyes and Whitney to the biopharmaceutical classification system. Int. J. Pharm., 321, 1-11.
-
(2006)
Int. J. Pharm
, vol.321
, pp. 1-11
-
-
Dokoumetzidis, A.1
Macheras, P.2
-
56
-
-
0033805179
-
In vitro-in vivo correlations for lipophilic, poorly water-soluble drugs
-
Dressman, J.B. and Reppas, C. (2000) In vitro-in vivo correlations for lipophilic, poorly water-soluble drugs. Eur. J. Pharm. Sci., 11, S73-S80.
-
(2000)
Eur. J. Pharm. Sci
, vol.11
, pp. S73-S80
-
-
Dressman, J.B.1
Reppas, C.2
-
57
-
-
84962061517
-
The mini paddle apparatus - a useful tool in the early developmental stage? Experiences with immediate-release dosage forms
-
Klein, S. (2006) The mini paddle apparatus - a useful tool in the early developmental stage? Experiences with immediate-release dosage forms. Dissol. Technol., 13, 6-11.
-
(2006)
Dissol. Technol
, vol.13
, pp. 6-11
-
-
Klein, S.1
-
58
-
-
23844475290
-
Effect of chloride ion on dissolution of different salt forms of haloperidol, a model basic drug
-
Li, S., Doyle, P., Metz, S. et al. (2005) Effect of chloride ion on dissolution of different salt forms of haloperidol, a model basic drug. J. Pharm. Sci., 94, 2224-2231.
-
(2005)
J. Pharm. Sci
, vol.94
, pp. 2224-2231
-
-
Li, S.1
Doyle, P.2
Metz, S.3
-
59
-
-
0030927353
-
Characterization of fluids from the stomach and proximal jejunum in men and women
-
Lindahl, A., Ungell, A.L. and Lennernas, H. (1997) Characterization of fluids from the stomach and proximal jejunum in men and women. Pharm. Res., 14, 497-502.
-
(1997)
Pharm. Res
, vol.14
, pp. 497-502
-
-
Lindahl, A.1
Ungell, A.L.2
Lennernas, H.3
-
60
-
-
43249121029
-
Gut instincts: explorations in intestinal physiology and drug delivery
-
McConnell, E.L. Fadda, H.M. and Basit, A.W. (2008) Gut instincts: explorations in intestinal physiology and drug delivery. Int. J. Pharm., 364, 213-226.
-
(2008)
Int. J. Pharm
, vol.364
, pp. 213-226
-
-
McConnell, E.L.1
Fadda, H.M.2
Basit, A.W.3
-
61
-
-
0002642747
-
Theorie der Reaktionsgeschwindigkeit in Heterogenen Systemen
-
Nernst, W. (1904) Theorie der Reaktionsgeschwindigkeit in Heterogenen Systemen. Z. Phys. Chem., 47, 52-55.
-
(1904)
Z. Phys. Chem
, vol.47
, pp. 52-55
-
-
Nernst, W.1
-
62
-
-
33947487639
-
The rate of solution of solid substances in their own solutions
-
Noyes, A.A. and Whitney, W.R. (1897) The rate of solution of solid substances in their own solutions. J. Am. Chem. Soc., 19, 930-934.
-
(1897)
J. Am. Chem. Soc
, vol.19
, pp. 930-934
-
-
Noyes, A.A.1
Whitney, W.R.2
-
63
-
-
27744515754
-
Intestinal fluid volumes and transit of dosage forms as assessed by magnetic resonance imaging
-
Schiller, C., Fröhlich, C.-P., Giessmann, T. et al. (2005) Intestinal fluid volumes and transit of dosage forms as assessed by magnetic resonance imaging. Ailment Pharmacol. Theory, 22, 971-979.
-
(2005)
Ailment Pharmacol. Theory
, vol.22
, pp. 971-979
-
-
Schiller, C.1
Fröhlich, C.-P.2
Giessmann, T.3
-
64
-
-
0021944082
-
Effect of diffusion layer pH and solubility on the dissolution rate of pharmaceutical acids and their sodium salts. II: salicylic acid, theophylline and benzoic acid
-
Serajuddin, A.T.M. and Jarowski, C.I. (1985) Effect of diffusion layer pH and solubility on the dissolution rate of pharmaceutical acids and their sodium salts. II: salicylic acid, theophylline and benzoic acid. J. Pharm. Sci., 74, 148-154.
-
(1985)
J. Pharm. Sci
, vol.74
, pp. 148-154
-
-
Serajuddin, A.T.M.1
Jarowski, C.I.2
-
65
-
-
0043283915
-
Measurement of intrinsic drug dissolution using two types of apparatus
-
Viegas, T.X., Curatella, R.U., Van Winkle, L.L. and Brinker, G. (2001) Measurement of intrinsic drug dissolution using two types of apparatus. Pharm Technol., 25, 44-43.
-
(2001)
Pharm Technol
, vol.25
, pp. 44-43
-
-
Viegas, T.X.1
Curatella, R.U.2
Van Winkle, L.L.3
Brinker, G.4
-
66
-
-
33747336372
-
Über die Geschwindigkeit Molekularer und Chemischer Reaktionen in Heterogenen Systemen
-
Wilderman, M. (1909) Über die Geschwindigkeit Molekularer und Chemischer Reaktionen in Heterogenen Systemen. Erster Teil. Z. Phys. Chem., 66, 445-495.
-
(1909)
Erster Teil. Z. Phys. Chem
, vol.66
, pp. 445-495
-
-
Wilderman, M.1
-
67
-
-
33748503596
-
The ionization constant of water over wide ranges of temperature and density
-
Bandura, A.V. and Lvov, S.N. (2005) The ionization constant of water over wide ranges of temperature and density. J. Phys. Chem. Ref. Data, 35, 15-30.
-
(2005)
J. Phys. Chem. Ref. Data
, vol.35
, pp. 15-30
-
-
Bandura, A.V.1
Lvov, S.N.2
-
68
-
-
0017623487
-
Pharmaceutical salts
-
Berge, S.M., Bighley, L.D. and Monkhouse, D.C. (1977) Pharmaceutical salts. J. Pharm. Sci., 66, 1-19.
-
(1977)
J. Pharm. Sci
, vol.66
, pp. 1-19
-
-
Berge, S.M.1
Bighley, L.D.2
Monkhouse, D.C.3
-
69
-
-
25844524863
-
Tape and layer structures in cocrystals of some di- and tricarboxylic acids with 4,4_-bipyridines and isonicotinamide. From binary to ternary cocrystals
-
Bhogala, B.R., Basavoju, S. and Nangia, A. (2005) Tape and layer structures in cocrystals of some di- and tricarboxylic acids with 4,4_-bipyridines and isonicotinamide. From binary to ternary cocrystals. Crys. Engng Commun., 7, 551-562.
-
(2005)
Crys. Engng Commun
, vol.7
, pp. 551-562
-
-
Bhogala, B.R.1
Basavoju, S.2
Nangia, A.3
-
70
-
-
0018412446
-
Solubility of doxycycline in aqueous solution
-
Bogardus, J.B. and Blackwood, R.K. (1979) Solubility of doxycycline in aqueous solution. J. Pharm. Sci., 68, 188-194.
-
(1979)
J. Pharm. Sci
, vol.68
, pp. 188-194
-
-
Bogardus, J.B.1
Blackwood, R.K.2
-
71
-
-
40149094922
-
Strategy for the prediction and selection of drug substance salt forms
-
Brittain, H.G. (2007) Strategy for the prediction and selection of drug substance salt forms. Pharm. Technol., 31, 78-88.
-
(2007)
Pharm. Technol
, vol.31
, pp. 78-88
-
-
Brittain, H.G.1
-
72
-
-
84882389982
-
Introduction and overview to the preformulation development of solid dosage forms
-
(eds M.C. Adeyeye and H.G. Brittain), Informa Healthcare, New York
-
Brittain, H.G. (2008) Introduction and overview to the preformulation development of solid dosage forms. In Preformulation in Solid Dosage Form Development (eds M.C. Adeyeye and H.G. Brittain), Informa Healthcare, New York. ISBN 0-8247-5809-9.
-
(2008)
Preformulation in Solid Dosage Form Development
-
-
Brittain, H.G.1
-
73
-
-
34250791543
-
The salt-cocrystal continuum: the influence of crystal structure on ionization state
-
Childs, S.L., Stahly, G.P. and Park, A. (2007) The salt-cocrystal continuum: the influence of crystal structure on ionization state. Molec. Pharm., 4, 323-338.
-
(2007)
Molec. Pharm
, vol.4
, pp. 323-338
-
-
Childs, S.L.1
Stahly, G.P.2
Park, A.3
-
74
-
-
0027997464
-
A budesonide prodrug accelerates treatment of colitis in rats
-
Cui, N., Friend, D.R. and Fedorak, R.N. (1994) A budesonide prodrug accelerates treatment of colitis in rats. Gut, 35, 1439-1446.
-
(1994)
Gut
, vol.35
, pp. 1439-1446
-
-
Cui, N.1
Friend, D.R.2
Fedorak, R.N.3
-
75
-
-
0642312376
-
Synthesis and in vitro properties of prednisolone 21-sulfate sodium as a colon-specific prodrug of prednisolone
-
Doh, M.J., Jung, Y.J., Kim, I.H. et al. (2003) Synthesis and in vitro properties of prednisolone 21-sulfate sodium as a colon-specific prodrug of prednisolone. Arch. Pharm. Res., 26, 258-263.
-
(2003)
Arch. Pharm. Res
, vol.26
, pp. 258-263
-
-
Doh, M.J.1
Jung, Y.J.2
Kim, I.H.3
-
76
-
-
0024536377
-
Microenvironmental pH control of drug dissolution
-
Doherty, C. and York, P. (1989) Microenvironmental pH control of drug dissolution. Int. J. Pharm., 50, 223-232.
-
(1989)
Int. J. Pharm
, vol.50
, pp. 223-232
-
-
Doherty, C.1
York, P.2
-
77
-
-
0034713306
-
Influence of admixed citric acid on the release profile of pelanserin hydrochloride from HPMC matrix tablets
-
Espinoza, R., Hong, E. and Villafuerte, L. (2000) Influence of admixed citric acid on the release profile of pelanserin hydrochloride from HPMC matrix tablets. Int. J. Pharm., 201, 165-173.
-
(2000)
Int. J. Pharm
, vol.201
, pp. 165-173
-
-
Espinoza, R.1
Hong, E.2
Villafuerte, L.3
-
78
-
-
0029890220
-
Factors affecting the dissolution of diclofenac salts
-
Fini, A., Fazio, G., Fernández Hervás, M.-J. et al. (1996) Factors affecting the dissolution of diclofenac salts. Eur. J. Pharm. Sci., 4, 231-238.
-
(1996)
Eur. J. Pharm. Sci
, vol.4
, pp. 231-238
-
-
Fini, A.1
Fazio, G.2
Fernández Hervás, M.-J.3
-
79
-
-
33749451891
-
Ionization states in the microenvironment of solid dosage forms: effect of formulation variables and processing
-
Govindarajan, R., Zinchuk, A., Hancock, B. et al. (2006) Ionization states in the microenvironment of solid dosage forms: effect of formulation variables and processing. Pharm. Res., 23, 2454-2468.
-
(2006)
Pharm. Res
, vol.23
, pp. 2454-2468
-
-
Govindarajan, R.1
Zinchuk, A.2
Hancock, B.3
-
80
-
-
77956367297
-
Impact of counterion on the chemical stability of crystalline salts of procaine
-
Guerrieri, P., Jarring, K. and Taylor, L.S. (2010) Impact of counterion on the chemical stability of crystalline salts of procaine. J. Pharm. Sci., 99, 3719-3730.
-
(2010)
J. Pharm. Sci
, vol.99
, pp. 3719-3730
-
-
Guerrieri, P.1
Jarring, K.2
Taylor, L.S.3
-
81
-
-
0027449074
-
In-vitro evaluation of dexamethasone-beta-D-glucuronide for colon-specific drug-delivery
-
Haeberlin, B., Rubas, W., Nolen, H.W. and Friend, D.R. (1993) In-vitro evaluation of dexamethasone-beta-D-glucuronide for colon-specific drug-delivery. Pharm. Res., 10, 1553-1562.
-
(1993)
Pharm. Res
, vol.10
, pp. 1553-1562
-
-
Haeberlin, B.1
Rubas, W.2
Nolen, H.W.3
Friend, D.R.4
-
82
-
-
0015702659
-
The dependence of paracetamol absorption on the rate of gastric emptying
-
Heading, R.C., Nimmo, J., Prescott, L.F. and Tothill, P. (1973) The dependence of paracetamol absorption on the rate of gastric emptying. Br. J. Pharmac., 47, 415-421.
-
(1973)
Br. J. Pharmac
, vol.47
, pp. 415-421
-
-
Heading, R.C.1
Nimmo, J.2
Prescott, L.F.3
Tothill, P.4
-
83
-
-
1042264121
-
Impact of solid state properties on developability assessment of drug candidates
-
Huang, L.-F. and Tong, W.-Q. (2004) Impact of solid state properties on developability assessment of drug candidates. Adv. Drug. Del. Rev., 56, 321-334.
-
(2004)
Adv. Drug. Del. Rev
, vol.56
, pp. 321-334
-
-
Huang, L.-F.1
Tong, W.-Q.2
-
85
-
-
0021806456
-
Clinical pharmacokinetics of sulphasalazine, its metabolites and other prodrugs for 5-aminosalicylic acid
-
Klotz, U. (1985) Clinical pharmacokinetics of sulphasalazine, its metabolites and other prodrugs for 5-aminosalicylic acid. Clin. Pharmacokinet., 10, 285-302.
-
(1985)
Clin. Pharmacokinet
, vol.10
, pp. 285-302
-
-
Klotz, U.1
-
86
-
-
0015449031
-
Solubility of organic hydrochlorides
-
Kramer, S.F. and Flynn, G.L. (1972) Solubility of organic hydrochlorides. J. Pharm. Sci., 61, 1896-1904.
-
(1972)
J. Pharm. Sci
, vol.61
, pp. 1896-1904
-
-
Kramer, S.F.1
Flynn, G.L.2
-
87
-
-
40949126942
-
Salt selection in drug development
-
Kumar, L., Amin, A. and Bansal, A.K. (2008) Salt selection in drug development. Pharm. Technol., 32 (3), 128-142.
-
(2008)
Pharm. Technol
, vol.32
, Issue.3
, pp. 128-142
-
-
Kumar, L.1
Amin, A.2
Bansal, A.K.3
-
88
-
-
0003409952
-
-
6th edn, Lippincott, Williams and Wilkins, Baltimore, MD
-
Lemke, T.L., Williams, D.A., Roche, V.F. and Zito, S.W. (eds) (2008) Foye's Principles of Medicinal Chemistry, 6th edn, Lippincott, Williams and Wilkins, Baltimore, MD. ISBN 978-0-7817-6879-5.
-
(2008)
Foye's Principles of Medicinal Chemistry
-
-
Lemke, T.L.1
Williams, D.A.2
Roche, V.F.3
Zito, S.W.4
-
89
-
-
23844499379
-
IV-IVC considerations in the development of immediate-release oral dosage form
-
Li, S.F., He, H.D., Parthiban, L.J. et al. (2005a) IV-IVC considerations in the development of immediate-release oral dosage form. J. Pharm. Sci., 94, 1396-1417.
-
(2005)
J. Pharm. Sci
, vol.94
, pp. 1396-1417
-
-
Li, S.F.1
He, H.D.2
Parthiban, L.J.3
-
90
-
-
18044381309
-
Investigation of solubility and dissolution of a free base and two different salt forms as a function of pH
-
Li, S., Wong, S.M., Sethia, S. et al. (2005b) Investigation of solubility and dissolution of a free base and two different salt forms as a function of pH. Pharm. Res., 22, 628-635.
-
(2005)
Pharm. Res
, vol.22
, pp. 628-635
-
-
Li, S.1
Wong, S.M.2
Sethia, S.3
-
91
-
-
0028339856
-
Permeation of diclofenac salts through silicone membrane - a mechanistic study of percutaneous-absorption of ionizable drugs
-
Maitani, Y., Kugo, M. and Nagai, T. (1994) Permeation of diclofenac salts through silicone membrane - a mechanistic study of percutaneous-absorption of ionizable drugs. Chem. Pharm. Bull., 42, 1297-1301.
-
(1994)
Chem. Pharm. Bull
, vol.42
, pp. 1297-1301
-
-
Maitani, Y.1
Kugo, M.2
Nagai, T.3
-
92
-
-
0028219710
-
An integrated approach to the selection of optimal salt form for a new drug candidate
-
Morris, K.R., Fakes, M.G., Thakur, A.B. et al. (1994) An integrated approach to the selection of optimal salt form for a new drug candidate. Int. J. Pharm., 105, 209-217.
-
(1994)
Int. J. Pharm
, vol.105
, pp. 209-217
-
-
Morris, K.R.1
Fakes, M.G.2
Thakur, A.B.3
-
93
-
-
70449176963
-
Solution rate of theophylline salts and effects from oral administration
-
Nelson, E. (1957) Solution rate of theophylline salts and effects from oral administration. J. Am. Pharm. Soc. Sci. Ed., 46, 607-614.
-
(1957)
J. Am. Pharm. Soc. Sci. Ed
, vol.46
, pp. 607-614
-
-
Nelson, E.1
-
94
-
-
3142736454
-
The effect of citric acid added to hydroxypropyl methylcellulose (HPMC) matrix tablets on the release of vinpocetine
-
Nie, S., Pan, W., Li, X. and Wu, X. (2004) The effect of citric acid added to hydroxypropyl methylcellulose (HPMC) matrix tablets on the release of vinpocetine. Drug Dev. Ind. Pharm., 30, 627-635.
-
(2004)
Drug Dev. Ind. Pharm
, vol.30
, pp. 627-635
-
-
Nie, S.1
Pan, W.2
Li, X.3
Wu, X.4
-
95
-
-
77953716351
-
Pharmaceutical salts: a formulation trick or a clinical conundrum?
-
Patel, A., Jones, S.A., Ferro, A. and Patel, N. (2009) Pharmaceutical salts: a formulation trick or a clinical conundrum? Br. J. Cardiol., 16, 281-286.
-
(2009)
Br. J. Cardiol
, vol.16
, pp. 281-286
-
-
Patel, A.1
Jones, S.A.2
Ferro, A.3
Patel, N.4
-
96
-
-
1042271498
-
Solubility and dissolution of weak acids, bases and salts
-
(eds P.H. Stahl and C.G. Wermuth), revised 2nd edn, Wiley-VCH
-
Pudipeddi, M., Serajuddin, A.T.M., Grant, D.J.W. and Stahl, P.H. (2011) Solubility and dissolution of weak acids, bases and salts. In Handbook of Pharmaceutical Salts. Properties, Selection and Use (eds P.H. Stahl and C.G. Wermuth), revised 2nd edn, Wiley-VCH. ISBN 3-906-39051-9.
-
(2011)
Handbook of Pharmaceutical Salts. Properties, Selection and Use
-
-
Pudipeddi, M.1
Serajuddin, A.T.M.2
Grant, D.J.W.3
Stahl, P.H.4
-
97
-
-
0346104829
-
Salt selection and simultaneous polymorphism assessment via high-throughput crystallization. The case of sertraline
-
Remenar, J.F., MacPhee, J.M., Larson, B.K. et al. (2003) Salt selection and simultaneous polymorphism assessment via high-throughput crystallization. The case of sertraline. Org. Proc. Res. Dev., 7, 990-996.
-
(2003)
Org. Proc. Res. Dev
, vol.7
, pp. 990-996
-
-
Remenar, J.F.1
MacPhee, J.M.2
Larson, B.K.3
-
98
-
-
0033403992
-
Tablet dissolution affected by a moisture mediated solid-state interaction between drug and disintegrant
-
Rohrs, B.R., Thamann, T.J., Gao, P. et al. (1999) Tablet dissolution affected by a moisture mediated solid-state interaction between drug and disintegrant. Pharm. Res., 16, 1850-1856.
-
(1999)
Pharm. Res
, vol.16
, pp. 1850-1856
-
-
Rohrs, B.R.1
Thamann, T.J.2
Gao, P.3
-
99
-
-
0028088918
-
pH related changes in the absorption of dipyridamole in the elderly
-
Russell, T.L., Berardi, R.R., Barnett, J.L. et al. (1994) pH related changes in the absorption of dipyridamole in the elderly. Pharm. Res., 11, 136-143.
-
(1994)
Pharm. Res
, vol.11
, pp. 136-143
-
-
Russell, T.L.1
Berardi, R.R.2
Barnett, J.L.3
-
100
-
-
3042555864
-
Ion-pairs of ibuprofen: increased membrane diffusion
-
Sarveiya, V., Templeton, J.F. and Benson, H.A.E. (2004) Ion-pairs of ibuprofen: increased membrane diffusion. J. Pharm. Pharmacol., 56, 717-724.
-
(2004)
J. Pharm. Pharmacol
, vol.56
, pp. 717-724
-
-
Sarveiya, V.1
Templeton, J.F.2
Benson, H.A.E.3
-
101
-
-
34548032742
-
Salt formation to improve drug solubility
-
Serajuddin, A.T.M. (2007) Salt formation to improve drug solubility. Adv. Drug Del. Rev., 59, 603-616.
-
(2007)
Adv. Drug Del. Rev
, vol.59
, pp. 603-616
-
-
Serajuddin, A.T.M.1
-
102
-
-
0021944082
-
Effect of diffusion layer pH and solubility on the dissolution rate of pharmaceutical acids and their sodium salts. II: salicylic acid, theophylline and benzoic acid
-
Serajuddin, A.T.M. and Jarowski, C.I. (1985) Effect of diffusion layer pH and solubility on the dissolution rate of pharmaceutical acids and their sodium salts. II: salicylic acid, theophylline and benzoic acid. J. Pharm. Sci., 74, 148-154.
-
(1985)
J. Pharm. Sci
, vol.74
, pp. 148-154
-
-
Serajuddin, A.T.M.1
Jarowski, C.I.2
-
103
-
-
33747179333
-
Strategies for the design of hydrophilic matrix tablets with controlled microenvironmental pH
-
Siepe, S., Lueckel, B., Kramer, A. et al. (2006) Strategies for the design of hydrophilic matrix tablets with controlled microenvironmental pH. Int. J. Pharm., 316, 14-20.
-
(2006)
Int. J. Pharm
, vol.316
, pp. 14-20
-
-
Siepe, S.1
Lueckel, B.2
Kramer, A.3
-
105
-
-
79952224350
-
Physical stability of weak bases in the solid-state
-
Stephenson, G.A., Aburub, A. and Woods, T.A. (2011) Physical stability of weak bases in the solid-state. J. Pharm. Sci., 100, 1607-1617.
-
(2011)
J. Pharm. Sci
, vol.100
, pp. 1607-1617
-
-
Stephenson, G.A.1
Aburub, A.2
Woods, T.A.3
-
106
-
-
0034660109
-
pH-independent release of a weakly basic drug from water-insoluble and -soluble matrix tablets
-
Streubel, A., Siepmann, J., Dashevsky, A. and Bodmeier, R. (2000) pH-independent release of a weakly basic drug from water-insoluble and -soluble matrix tablets. J. Cont. Rel., 67, 101-110.
-
(2000)
J. Cont. Rel
, vol.67
, pp. 101-110
-
-
Streubel, A.1
Siepmann, J.2
Dashevsky, A.3
Bodmeier, R.4
-
107
-
-
77954759851
-
The influence of aqueous content in small scale salt screening - improving hit rate for weakly basic, low solubility drugs
-
Tarsa, P.B., Towler, C.S., Woollam, G. and Berghausen, J. (2010) The influence of aqueous content in small scale salt screening - improving hit rate for weakly basic, low solubility drugs. Eur. J. Pharm. Sci., 41, 23-30.
-
(2010)
Eur. J. Pharm. Sci
, vol.41
, pp. 23-30
-
-
Tarsa, P.B.1
Towler, C.S.2
Woollam, G.3
Berghausen, J.4
-
108
-
-
0027194762
-
Effects of temperature and relative humidity on the solid-state chemical stability of ranitidine hydrochloride
-
Teraoka, R., Otsuka, M. and Matsuda, Y. (1993) Effects of temperature and relative humidity on the solid-state chemical stability of ranitidine hydrochloride. J. Pharm. Sci., 82 (1993) 601-604.
-
(1993)
J. Pharm. Sci
, vol.82
, Issue.1993
, pp. 601-604
-
-
Teraoka, R.1
Otsuka, M.2
Matsuda, Y.3
-
109
-
-
52249114680
-
Modulation of microenvironmental pH and crystallinity of ionizable telmisartan using alkalizers in solid dispersions for controlled release
-
Tran, P.H.L., Thanh, H.T. and Lee, B.-J. (2008) Modulation of microenvironmental pH and crystallinity of ionizable telmisartan using alkalizers in solid dispersions for controlled release. J. Cont. Rel., 129, 59-65.
-
(2008)
J. Cont. Rel
, vol.129
, pp. 59-65
-
-
Tran, P.H.L.1
Thanh, H.T.2
Lee, B.-J.3
-
110
-
-
14844320556
-
Influence of micro-environmental pH on the gel layer and release of a basic drug from various hydrophilic matrices
-
Varma, M.V.S., Kaushal, A.M. and Garg, S. (2005) Influence of micro-environmental pH on the gel layer and release of a basic drug from various hydrophilic matrices. J. Cont. Rel., 103, 499-510.
-
(2005)
J. Cont. Rel
, vol.103
, pp. 499-510
-
-
Varma, M.V.S.1
Kaushal, A.M.2
Garg, S.3
-
112
-
-
0025297596
-
Application of gastric aciditycontrolled beagle dog to bioavailability study of cinnarizine
-
Yamada, I., Goda, T., Kawata, M. and Ogawa, K. (1990) Application of gastric aciditycontrolled beagle dog to bioavailability study of cinnarizine. Yakugaku Zasshi, 110, 280-285.
-
(1990)
Yakugaku Zasshi
, vol.110
, pp. 280-285
-
-
Yamada, I.1
Goda, T.2
Kawata, M.3
Ogawa, K.4
-
113
-
-
34248596026
-
Stabilization of the maleate salt of a basic drug by adjustment of microenvironment pH in solid dosage form
-
Zannou, E.A., Yatindra, Q.J., Joshi, M. and Serajuddin, A.T.M. (2007) Stabilization of the maleate salt of a basic drug by adjustment of microenvironment pH in solid dosage form. Int. J. Pharm., 337, 210-218.
-
(2007)
Int. J. Pharm
, vol.337
, pp. 210-218
-
-
Zannou, E.A.1
Yatindra, Q.J.2
Joshi, M.3
Serajuddin, A.T.M.4
-
114
-
-
0014104395
-
Effect of polymorphism on the absorption of chloramphenicol from chloramphenicol palmitate
-
Aguiar, A.J., Krc Jr, J., Kinkel, A.W. and Samyn, J.C. (1967) Effect of polymorphism on the absorption of chloramphenicol from chloramphenicol palmitate. J. Pharm. Sci., 56, 847-853.
-
(1967)
J. Pharm. Sci
, vol.56
, pp. 847-853
-
-
Aguiar, A.J.1
Krc, J.2
Kinkel, A.W.3
Samyn, J.C.4
-
115
-
-
0002634817
-
Mémoire sur les syst 'emes form' es par les points distribués régulièrement sur un plan ou dans l'espace
-
Bravais, A. (1850)Mémoire sur les syst 'emes form' es par les points distribués régulièrement sur un plan ou dans l'espace. J. Ecole Polytech., 19, 1-128.
-
(1850)
J. Ecole Polytech
, vol.19
, pp. 1-128
-
-
Bravais, A.1
-
116
-
-
77954864086
-
Characterisation of paracetamol Form III with rapid-heating DSC
-
Gaisford, S., Buanz, A.B.M. and Jethwa, N. (2010) Characterisation of paracetamol Form III with rapid-heating DSC. J. Pharm. Biomed. Anal., 53, 366-370.
-
(2010)
J. Pharm. Biomed. Anal
, vol.53
, pp. 366-370
-
-
Gaisford, S.1
Buanz, A.B.M.2
Jethwa, N.3
-
118
-
-
0002425795
-
Theory and origin of polymorphism
-
(ed. H.G. Brittain), Informa Healthcare
-
Grant, D.J.W. (1999) Theory and origin of polymorphism. In Polymorphism in Pharmaceutical Solids (ed. H.G. Brittain), Informa Healthcare. ISBN 0-8247-0237-3.
-
(1999)
Polymorphism in Pharmaceutical Solids
-
-
Grant, D.J.W.1
-
120
-
-
38349160391
-
The use of high-speed differential scanning calorimetry (Hyper-DSC) in the study of pharmaceutical polymorphs
-
McGregor, C. and Bines, E. (2008) The use of high-speed differential scanning calorimetry (Hyper-DSC) in the study of pharmaceutical polymorphs. Int. J. Pharm., 350, 48-52.
-
(2008)
Int. J. Pharm
, vol.350
, pp. 48-52
-
-
McGregor, C.1
Bines, E.2
-
121
-
-
3543008927
-
The use of high-speed differential scanning calorimetry (DSC) to study the thermal properties of carbamazepine polymorphs
-
McGregor, C., Saunders, M. and Buckton, G. (2004) The use of high-speed differential scanning calorimetry (DSC) to study the thermal properties of carbamazepine polymorphs. Thermochim. Acta, 417, 231-237.
-
(2004)
Thermochim. Acta
, vol.417
, pp. 231-237
-
-
McGregor, C.1
Saunders, M.2
Buckton, G.3
-
122
-
-
0004294969
-
-
4th edn, Butterworth-Heinemann, Oxford
-
Mullin, J.W. (2001) Crystallization, 4th edn, Butterworth-Heinemann, Oxford. ISBN 0-7506-4833-3.
-
(2001)
Crystallization
-
-
Mullin, J.W.1
-
123
-
-
0031473049
-
Characterization and interconversion of polymorphs of premafloxacin, a new quinolone antibiotic
-
Schinzer, W.C., Bergren, M.S. and Aldrich, D.S. (1997) Characterization and interconversion of polymorphs of premafloxacin, a new quinolone antibiotic. J. Pharm. Sci., 86, 1426-1431.
-
(1997)
J. Pharm. Sci
, vol.86
, pp. 1426-1431
-
-
Schinzer, W.C.1
Bergren, M.S.2
Aldrich, D.S.3
-
124
-
-
0242288839
-
Influence of mechanical activation on the physical stability of salbutamol sulphate
-
Brodka-Pfeiffer, K., Langguth, P., Graß, P. and Häusler, H. (2003) Influence of mechanical activation on the physical stability of salbutamol sulphate. Eur. J. Pharm. Biopharm., 56, 393-400.
-
(2003)
Eur. J. Pharm. Biopharm
, vol.56
, pp. 393-400
-
-
Brodka-Pfeiffer, K.1
Langguth, P.2
Graß, P.3
Häusler, H.4
-
125
-
-
0034946478
-
Quantifying amorphous content of lactose using parallel beam X-ray powder diffraction and whole pattern fitting
-
Chen, X., Bates, S. and Morris, K.R. (2001) Quantifying amorphous content of lactose using parallel beam X-ray powder diffraction and whole pattern fitting. J. Pharm. Biomed. Anal., 26, 63-72.
-
(2001)
J. Pharm. Biomed. Anal
, vol.26
, pp. 63-72
-
-
Chen, X.1
Bates, S.2
Morris, K.R.3
-
126
-
-
34548455941
-
Comparison of quantitative methods for analysis of polyphasic pharmaceuticals
-
Giron, D., Monnier, S., Mutz, M. et al. (2007) Comparison of quantitative methods for analysis of polyphasic pharmaceuticals. J. Therm. Anal. Cal., 89, 729-743.
-
(2007)
J. Therm. Anal. Cal
, vol.89
, pp. 729-743
-
-
Giron, D.1
Monnier, S.2
Mutz, M.3
-
127
-
-
0032722007
-
The use of MTDSC to assess the amorphous phase content of a micronised drug substance
-
Guinot, S. and Leveiller, F. (1999) The use of MTDSC to assess the amorphous phase content of a micronised drug substance. Int. J. Pharm., 192, 63-75.
-
(1999)
Int. J. Pharm
, vol.192
, pp. 63-75
-
-
Guinot, S.1
Leveiller, F.2
-
128
-
-
85056318483
-
Comments on 'An approach to estimate the amorphous content of pharmaceutical powders using calorimetry with no calibration standards'
-
Hancock, B.C. (1998) Comments on 'An approach to estimate the amorphous content of pharmaceutical powders using calorimetry with no calibration standards'. Int. J. Pharm., 160, 131-133.
-
(1998)
Int. J. Pharm
, vol.160
, pp. 131-133
-
-
Hancock, B.C.1
-
129
-
-
0034633897
-
The quantification of small degrees of disorder in lactose using solution calorimetry
-
Hogan, S.E. and Buckton, G. (2000) The quantification of small degrees of disorder in lactose using solution calorimetry. Int. J. Pharm., 207, 57-64.
-
(2000)
Int. J. Pharm
, vol.207
, pp. 57-64
-
-
Hogan, S.E.1
Buckton, G.2
-
130
-
-
20344362926
-
Calorimetric investigation of the structural relaxation of amorphous materials: evaluating validity of the methodologies
-
Kawakami, K. and Pikal, M.J. (2005) Calorimetric investigation of the structural relaxation of amorphous materials: evaluating validity of the methodologies. J. Pharm. Sci., 94, 948-965.
-
(2005)
J. Pharm. Sci
, vol.94
, pp. 948-965
-
-
Kawakami, K.1
Pikal, M.J.2
-
131
-
-
29244470558
-
Quantification of low levels of amorphous content in sucrose by hyperDSC
-
Lappalainen, M., Pitkänen, I. and Harjunen, K. (2006) Quantification of low levels of amorphous content in sucrose by hyperDSC. Int. J. Pharm., 307, 150-155.
-
(2006)
Int. J. Pharm
, vol.307
, pp. 150-155
-
-
Lappalainen, M.1
Pitkänen, I.2
Harjunen, K.3
-
132
-
-
0037074074
-
Quantification of low levels (<10%) of amorphous content in micronised active batches using dynamic vapour sorption and isothermal microcalorimetry
-
Mackin, L., Zanon, R., Park, J.M. et al. (2002) Quantification of low levels (<10%) of amorphous content in micronised active batches using dynamic vapour sorption and isothermal microcalorimetry. Int. J. Pharm., 231, 227-236.
-
(2002)
Int. J. Pharm
, vol.231
, pp. 227-236
-
-
Mackin, L.1
Zanon, R.2
Park, J.M.3
-
133
-
-
0034950053
-
The use of inverse phase gas chromatography to measure the surface energy of crystalline, amorphous and recently milled lactose
-
Newell, H.E., Buckton, G., Butler, D.A. et al. (2001) The use of inverse phase gas chromatography to measure the surface energy of crystalline, amorphous and recently milled lactose. Pharm. Res., 18, 662-666.
-
(2001)
Pharm. Res
, vol.18
, pp. 662-666
-
-
Newell, H.E.1
Buckton, G.2
Butler, D.A.3
-
134
-
-
80052267239
-
Application and use of isothermal calorimetry in pharmaceutical development
-
O'Neill, M.A.A. and Gaisford, S. (2011) Application and use of isothermal calorimetry in pharmaceutical development. Int. J. Pharm., 417, 83-93.
-
(2011)
Int. J. Pharm
, vol.417
, pp. 83-93
-
-
O'Neill, M.A.A.1
Gaisford, S.2
-
136
-
-
0030901259
-
An approach to estimate the amorphous content of pharmaceutical powders using calorimetry with no calibration standards
-
Phillips, E.M. (1997) An approach to estimate the amorphous content of pharmaceutical powders using calorimetry with no calibration standards. Int. J. Pharm., 149, 267-271.
-
(1997)
Int. J. Pharm
, vol.149
, pp. 267-271
-
-
Phillips, E.M.1
-
137
-
-
23444462493
-
Calorimetric determination of amorphous content in lactose: a note on the preparation of calibration curves
-
Ramos, R., Gaisford, S. and Buckton, G. (2005) Calorimetric determination of amorphous content in lactose: a note on the preparation of calibration curves. Int. J. Pharm., 300, 13-21.
-
(2005)
Int. J. Pharm
, vol.300
, pp. 13-21
-
-
Ramos, R.1
Gaisford, S.2
Buckton, G.3
-
138
-
-
0032703825
-
The detection of amorphous material in a nominally crystalline drug using modulated temperature DSC - a case study
-
Saklatvala, R., Royall, P.G. and Craig, D.Q.M. (1999) The detection of amorphous material in a nominally crystalline drug using modulated temperature DSC - a case study. Int. J. Pharm., 192, 55-62.
-
(1999)
Int. J. Pharm
, vol.192
, pp. 55-62
-
-
Saklatvala, R.1
Royall, P.G.2
Craig, D.Q.M.3
-
139
-
-
1842557588
-
The potential of high speed DSC (hyper-DSC) for the detection and quantification of small amounts of amorphous content in predominantly crystalline samples
-
Saunders, M., Podluii, K., Shergill, S. et al. (2004) The potential of high speed DSC (hyper-DSC) for the detection and quantification of small amounts of amorphous content in predominantly crystalline samples. Int. J. Pharm., 274, 35-40.
-
(2004)
Int. J. Pharm
, vol.274
, pp. 35-40
-
-
Saunders, M.1
Podluii, K.2
Shergill, S.3
-
140
-
-
77954312924
-
Determination of low levels of amorphous content in inhalation grade lactose by moisture sorption isotherms
-
Vollenbroek, J., Hebbink, G.A., Ziffels, S. and Steckel, H. (2010) Determination of low levels of amorphous content in inhalation grade lactose by moisture sorption isotherms. Int. J. Pharm., 395, 62-70.
-
(2010)
Int. J. Pharm
, vol.395
, pp. 62-70
-
-
Vollenbroek, J.1
Hebbink, G.A.2
Ziffels, S.3
Steckel, H.4
-
141
-
-
0014699523
-
Non-symmetrical dielectric relaxation behaviour arising from a simple empirical decay function
-
Williams, G. and Watts, D.C. (1970) Non-symmetrical dielectric relaxation behaviour arising from a simple empirical decay function. Trans. Fara. Soc., 66, 80-85.
-
(1970)
Trans. Fara. Soc
, vol.66
, pp. 80-85
-
-
Williams, G.1
Watts, D.C.2
-
142
-
-
0003689329
-
-
2nd edn, John Wiley & Sons, Ltd
-
Connors, K.A., Amidon, G.L. and Stella, V.J. (1986) Chemical Stability of Pharmaceuticals, 2nd edn, John Wiley & Sons, Ltd. ISBN 0-4718-8795-X.
-
(1986)
Chemical Stability of Pharmaceuticals
-
-
Connors, K.A.1
Amidon, G.L.2
Stella, V.J.3
-
143
-
-
37049148254
-
Mechanism and kinetics of carboxylic ester hydrolysis and carboxyl esterification
-
Day, J.N.E. and Ingold, C.K. (1941) Mechanism and kinetics of carboxylic ester hydrolysis and carboxyl esterification. Trans. Faraday Soc., 37, 686-705.
-
(1941)
Trans. Faraday Soc
, vol.37
, pp. 686-705
-
-
Day, J.N.E.1
Ingold, C.K.2
-
144
-
-
50249162817
-
Autoxidation of etheric oils used in pharmacy
-
Fryklöf, L.-E. (1954) Autoxidation of etheric oils used in pharmacy. Farm. Rev., 53, 317-335.
-
(1954)
Farm. Rev
, vol.53
, pp. 317-335
-
-
Fryklöf, L.-E.1
-
145
-
-
0017437920
-
Humidity fixed of binary saturated aqueous solutions
-
Greenspan, L. (1977) Humidity fixed of binary saturated aqueous solutions. J. Res. Natl Bur. Stand., 81A (1977) 89-96.
-
(1977)
J. Res. Natl Bur. Stand
, vol.81 A
, Issue.1977
, pp. 89-96
-
-
Greenspan, L.1
-
146
-
-
0344014812
-
Storage conditions for stability testing (Part 2)
-
Grimm, W. (1986) Storage conditions for stability testing (Part 2). Drugs Made in Germany, 29, 39-47.
-
(1986)
Drugs Made in Germany
, vol.29
, pp. 39-47
-
-
Grimm, W.1
-
147
-
-
0031954253
-
Extension of the International Conference on Harmonisation Tripartite Guidelines for stability testing of new drug substances and products to countries of Climatic Zones III and IV
-
Grimm, W. (1998) Extension of the International Conference on Harmonisation Tripartite Guidelines for stability testing of new drug substances and products to countries of Climatic Zones III and IV. Drug Dev. Ind. Pharm., 24, 313-325.
-
(1998)
Drug Dev. Ind. Pharm
, vol.24
, pp. 313-325
-
-
Grimm, W.1
-
151
-
-
84949755804
-
-
Processed photographic colour films and paper prints -methods for measuring image stability
-
ISO 10977 (1993) Photography. Processed photographic colour films and paper prints -methods for measuring image stability.
-
(1993)
Photography
-
-
-
152
-
-
0033051354
-
Trends in stability testing, with emphasis on stability during distribution and storage
-
Kommanaboyina, B. and Rhodes, C.T. (1999) Trends in stability testing, with emphasis on stability during distribution and storage. Drug. Dev. Ind. Pharm., 25, 857-868.
-
(1999)
Drug. Dev. Ind. Pharm
, vol.25
, pp. 857-868
-
-
Kommanaboyina, B.1
Rhodes, C.T.2
-
153
-
-
34250459937
-
Stability of d-cycloserine in aqueous solutions at high concentrations
-
Kondrat'eva, A.P., Bruns, B.P. and Libinson, G.S. (1971) Stability of d-cycloserine in aqueous solutions at high concentrations. Pharm. Chem. J., 5, 356-360.
-
(1971)
Pharm. Chem. J
, vol.5
, pp. 356-360
-
-
Kondrat'eva, A.P.1
Bruns, B.P.2
Libinson, G.S.3
-
154
-
-
0019850513
-
Stability of procaine hydrochloride in a buffered cardioplegia formulation
-
Loucas, S.P., Mehl, B., Litwak, R.S. and Jurado, R.A. (1981) Stability of procaine hydrochloride in a buffered cardioplegia formulation. Am. J. Hosp. Pharm., 38, 1924-1928.
-
(1981)
Am. J. Hosp. Pharm
, vol.38
, pp. 1924-1928
-
-
Loucas, S.P.1
Mehl, B.2
Litwak, R.S.3
Jurado, R.A.4
-
156
-
-
33846385383
-
Modification of the crystal habit of celecoxib for improved processability
-
Banga, S., Chawla, G., Varandani, D. and Mehta, B.R. (2007) Modification of the crystal habit of celecoxib for improved processability. J. Pharm. Pharmacol., 59, 29-39.
-
(2007)
J. Pharm. Pharmacol
, vol.59
, pp. 29-39
-
-
Banga, S.1
Chawla, G.2
Varandani, D.3
Mehta, B.R.4
-
157
-
-
0035206815
-
Particle size distribution, Part 1, representations of particle shape, size and distribution
-
Brittain, H.G. (2001) Particle size distribution, Part 1, representations of particle shape, size and distribution. Pharm. Technol., 25, 38-45.
-
(2001)
Pharm. Technol
, vol.25
, pp. 38-45
-
-
Brittain, H.G.1
-
158
-
-
0026749510
-
Crystal habit modifications and altered tableting characteristics
-
Kaul, D., Nguyen, N.T. and Venkataram, S. (1992) Crystal habit modifications and altered tableting characteristics. Int. J. Pharm., 88, 345-350.
-
(1992)
Int. J. Pharm
, vol.88
, pp. 345-350
-
-
Kaul, D.1
Nguyen, N.T.2
Venkataram, S.3
-
159
-
-
0037026268
-
Crystal habit and tableting behavior
-
Rasenack, N. andMüller, B.W. (2002) Crystal habit and tableting behavior. Int. J. Pharm., 244, 45-57.
-
(2002)
Int. J. Pharm
, vol.244
, pp. 45-57
-
-
Rasenack, N.1
Müller, B.W.2
-
160
-
-
0000496231
-
Evaluating flow properties of solids
-
Carr, R.L. (1965) Evaluating flow properties of solids. Chem. Engng, 72, 163-167.
-
(1965)
Chem. Engng
, vol.72
, pp. 163-167
-
-
Carr, R.L.1
-
161
-
-
0002737830
-
Friction conditions in a mass of metal powder
-
Hausner, H.H. (1967) Friction conditions in a mass of metal powder. Int. J. Powder Metall., 3, 7-13.
-
(1967)
Int. J. Powder Metall
, vol.3
, pp. 7-13
-
-
Hausner, H.H.1
-
162
-
-
84984087501
-
Some angular properties of magnesia and their relevance to material handling
-
Jones, T.M. and Pilpel, N. (1966) Some angular properties of magnesia and their relevance to material handling. J. Pharm. Pharmacol., 18, 182T.
-
(1966)
J. Pharm. Pharmacol
, vol.18
, pp. 182T
-
-
Jones, T.M.1
Pilpel, N.2
-
164
-
-
0028025198
-
Effect of moisture sorption on tableting characteristics of spray dried (15% amorphous) lactose
-
Sebhatu, T., Elamin, A.A. and Ahlneck, C. (1994) Effect of moisture sorption on tableting characteristics of spray dried (15% amorphous) lactose. Pharm. Res., 11, 1233-1238.
-
(1994)
Pharm. Res
, vol.11
, pp. 1233-1238
-
-
Sebhatu, T.1
Elamin, A.A.2
Ahlneck, C.3
|