SCOPUS 정보 검색 플랫폼

Volumn 12, Issue 20, 2014, Pages 3288-3302

Synthesis and biological evaluation of dual action cyclo-RGD/SMAC mimetic conjugates targeting αvβ3/α vβ5 integrins and IAP proteins

(11) Mingozzi, M a Manzoni, L b Arosio, D b Dal Corso, A a Manzotti, M a Innamorati, F a Pignataro, L a Lecis, D c Delia, D c Seneci, P a Gennari, C a

a UNIVERSITY OF MILAN (Italy)

b CNR (Italy)

c NATIONAL CANCER INSTITUTE (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

BINDING ENERGY; GLYCOPROTEINS; PROTEINS;

ANCHOR POINT; BINDING AFFINITIES; BINDING STRENGTH; BIOLOGICAL EVALUATION; DUAL ACTION; MOLECULAR TARGETS; RATIONAL DESIGN; SEPARATE UNIT;

CHELATION;

ALPHAVBETA5 INTEGRIN; ANTINEOPLASTIC AGENT; CYCLIC ARGININE-GLYCINE-ASPARTIC ACID PEPTIDE; CYCLOPEPTIDE; DOXORUBICIN; INHIBITOR OF APOPTOSIS PROTEIN; LIGAND; MITOCHONDRIAL PROTEIN; PROTEIN BINDING; VITRONECTIN; VITRONECTIN RECEPTOR;

ANIMAL; BIOTINYLATION; BOVINE; CELL FREE SYSTEM; CHEMISTRY; DIMERIZATION; DRUG EFFECTS; HUMAN; IC50; METABOLISM; SYNTHESIS; TUMOR CELL LINE;

ANIMALS; ANTINEOPLASTIC AGENTS; BIOTINYLATION; CATTLE; CELL LINE, TUMOR; CELL-FREE SYSTEM; DIMERIZATION; DOXORUBICIN; HUMANS; INHIBITOR OF APOPTOSIS PROTEINS; INHIBITORY CONCENTRATION 50; INTEGRIN ALPHAVBETA3; LIGANDS; MITOCHONDRIAL PROTEINS; PEPTIDES, CYCLIC; PROTEIN BINDING; RECEPTORS, VITRONECTIN; VITRONECTIN;

EID: 84899090315 PISSN: 14770520 EISSN: None Source Type: Journal
DOI: 10.1039/c4ob00207e Document Type: Article

Times cited : (24)

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