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Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 8, 2014, Pages 1941-1943

Arylamino bisphosphonates: Potent and selective inhibitors of the tumor-associated carbonic anhydrase XII

(5) Tauro, Marilena a Loiodice, Fulvio a Ceruso, Mariangela b Supuran, Claudiu T b Tortorella, Paolo a

a UNIVERSITY OF BARI (Italy)

b UNIVERSITY OF FLORENCE (Italy)

Author keywords

Antitumor agent; Bisphosphonate; Carbonic anhydrase; Isoform selective inhibitor; Matrix metalloproteinase inhibitor

Indexed keywords

ACETAZOLAMIDE; ANTINEOPLASTIC AGENT; BISPHOSPHONIC ACID DERIVATIVE; CARBONATE DEHYDRATASE I; CARBONATE DEHYDRATASE II; CARBONATE DEHYDRATASE INHIBITOR; CARBONATE DEHYDRATASE IX; CARBONATE DEHYDRATASE XII; CARBONATE DEHYDRATASE XII INHIBITOR; CARBONATE DEHYDRATASE XIV; UNCLASSIFIED DRUG; ZOLEDRONIC ACID;

ARTICLE; DRUG SELECTIVITY; DRUG STRUCTURE; ENZYME ACTIVITY; ENZYME INHIBITION; HUMAN;

ANTITUMOR AGENT; BISPHOSPHONATE; CARBONIC ANHYDRASE; ISOFORM-SELECTIVE INHIBITOR; MATRIX METALLOPROTEINASE INHIBITOR;

ACETAZOLAMIDE; ANTINEOPLASTIC AGENTS; CARBONIC ANHYDRASE INHIBITORS; CARBONIC ANHYDRASES; DIPHOSPHONATES; DRUG DELIVERY SYSTEMS; ENZYME ACTIVATION; HUMANS; IMIDAZOLES; INHIBITORY CONCENTRATION 50; MOLECULAR STRUCTURE; PROTEIN ISOFORMS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84897487395 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2014.03.001 Document Type: Article

Times cited : (13)

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