SCOPUS 정보 검색 플랫폼

Volumn 62, Issue , 2013, Pages 556-563

Synthesis of tacrine-lophine hybrids via one-pot four component reaction and biological evaluation as acetyl- and butyrylcholinesterase inhibitors

(10) Da Costa, Jessé Sobieski a Lopes, João Paulo Bizarro a Russowsky, Dennis a Petzhold, Cesar Liberato a Borges, Antonio César De Amorim a Ceschi, Marco Antonio a Konrath, Eduardo a Batassini, Cristiane a Lunardi, Paula Santana a Gonçalves, Carlos Alberto Saraiva a

a FEDERAL UNIVERSITY OF RIO GRANDE DO SUL (Brazil)

Author keywords

AChE inhibitory activity; Four component reaction; Indium trichloride; Lophine; Tacrine

Indexed keywords

9 AMINOALKYLAMINO 1,2,3,4TETRAHYDROACRIDINE; ACETYLCHOLINESTERASE; ALDEHYDE; CHOLINESTERASE INHIBITOR; IMIDAZOLE DERIVATIVE; TACRINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CATALYST; DRUG SYNTHESIS; HUMAN; HYBRID; IC 50; NONHUMAN; POLYMERIZATION;

ACETYLCHOLINESTERASE; ANIMALS; BUTYRYLCHOLINESTERASE; CHOLINESTERASE INHIBITORS; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; IMIDAZOLES; MALE; MOLECULAR STRUCTURE; RATS; RATS, WISTAR; STRUCTURE-ACTIVITY RELATIONSHIP; TACRINE;

EID: 84873735631 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2013.01.029 Document Type: Article

Times cited : (52)

References (35)

1
- 33750705653
- M. Goedert, and M.G. Spillantini Science 314 2006 777 781
- (2006) Science , vol.314 , pp. 777-781
- Goedert, M.¹ Spillantini, M.G.²

2
- 0042433479
- A.V. Terry Jr., and J.J. Buccafusco J. Pharmacol. Exp. Ther. 306 2003 821 827
- (2003) J. Pharmacol. Exp. Ther. , vol.306 , pp. 821-827
- Terry, Jr.A.V.¹ Buccafusco, J.J.²

3
- 0034125843
- R.T. Bartus Exp. Neurol. 163 2000 495 529
- (2000) Exp. Neurol. , vol.163 , pp. 495-529
- Bartus, R.T.¹

4
- 80052939127
- S. Rizzo, A. Bisi, M. Bartolini, F. Mancini, F. Belluti, S. Gobbi, V. Andrisano, and A. Rampa Eur. J. Med. Chem. 46 2011 4336 4343
- (2011) Eur. J. Med. Chem. , vol.46 , pp. 4336-4343
- Rizzo, S.¹ Bisi, A.² Bartolini, M.³ Mancini, F.⁴ Belluti, F.⁵ Gobbi, S.⁶ Andrisano, V.⁷ Rampa, A.⁸

5
- 79952140384
- M. Kozurkova, S. Hamulakova, Z. Gazova, H. Paulikova, and P. Kristian Pharmaceuticals 4 2011 382 418
- (2011) Pharmaceuticals , vol.4 , pp. 382-418
- Kozurkova, M.¹ Hamulakova, S.² Gazova, Z.³ Paulikova, H.⁴ Kristian, P.⁵

6
- 79959538767
- J.J. Bornstein, T.J. Eckroat, J.L. Houghton, C.K. Jones, K.D. Green, and S. Garneau-Tsodikova Med. Chem. Commun. 2 2011 406 412
- (2011) Med. Chem. Commun. , vol.2 , pp. 406-412
- Bornstein, J.J.¹ Eckroat, T.J.² Houghton, J.L.³ Jones, C.K.⁴ Green, K.D.⁵ Garneau-Tsodikova, S.⁶

7
- 78650901081
- C. Ronco, L. Jean, H. Outaabout, and P.Y. Renard Eur. J. Org. Chem. 2011 302 310
- (2011) Eur. J. Org. Chem. , pp. 302-310
- Ronco, C.¹ Jean, L.² Outaabout, H.³ Renard, P.Y.⁴

8
- 68949197617
- R.T. Delfino, T.S. Ribeiro, and J.D. Figueroa-Villar J. Braz. Chem. Soc. 20 2009 407 428
- (2009) J. Braz. Chem. Soc. , vol.20 , pp. 407-428
- Delfino, R.T.¹ Ribeiro, T.S.² Figueroa-Villar, J.D.³

9
- 65649137775
- D.A. Smith Am. J. Health-syst. Pharm. 66 2009 899 907
- (2009) Am. J. Health-syst. Pharm. , vol.66 , pp. 899-907
- Smith, D.A.¹

10
- 84856914519
- M.I. Fernández-Bachiller, C. Pérez, L. Monjas, J. Rademann, and M.I. Rodríguez-Franco J. Med. Chem. 55 2012 1303 1317
- (2012) J. Med. Chem. , vol.55 , pp. 1303-1317
- Fernández-Bachiller, M.I.¹ Pérez, C.² Monjas, L.³ Rademann, J.⁴ Rodríguez-Franco, M.I.⁵

11
- 59249084336
- G.T. Grossberg, V. Pejovic, M.L. Miller, and S.M. Graham Dement. Geriatr. Cogn. Disord. 27 2009 164 172
- (2009) Dement. Geriatr. Cogn. Disord. , vol.27 , pp. 164-172
- Grossberg, G.T.¹ Pejovic, V.² Miller, M.L.³ Graham, S.M.⁴

12
- 0018129338
- E.K. Perry, R.H. Perry, G. Blessed, and B.E. Tomlinson Neuropathol. Appl. Neurobiol. 4 1978 273 277
- (1978) Neuropathol. Appl. Neurobiol. , vol.4 , pp. 273-277
- Perry, E.K.¹ Perry, R.H.² Blessed, G.³ Tomlinson, B.E.⁴

13
- 0025778840
- J.L. Sussman, M. Harel, F. Frolow, C. Oefner, A. Goldman, L. Toker, and I. Silman Science 253 1991 872 879
- (1991) Science , vol.253 , pp. 872-879
- Sussman, J.L.¹ Harel, M.² Frolow, F.³ Oefner, C.⁴ Goldman, A.⁵ Toker, L.⁶ Silman, I.⁷

14
- 0142039868
- Y. Nicolet, O. Lockridge, P. Masson, J.C. Fontecilla-Camps, and F. Nachon J. Biol. Chem. 278 2003 41141 41147
- (2003) J. Biol. Chem. , vol.278 , pp. 41141-41147
- Nicolet, Y.¹ Lockridge, O.² Masson, P.³ Fontecilla-Camps, J.C.⁴ Nachon, F.⁵

15
- 0029817834
- Y.P. Pang, P. Quiram, T. Jelacic, F. Hong, and S. Brimijoin J. Biol. Chem. 271 1996 23646 23649
- (1996) J. Biol. Chem. , vol.271 , pp. 23646-23649
- Pang, Y.P.¹ Quiram, P.² Jelacic, T.³ Hong, F.⁴ Brimijoin, S.⁵

16
- 45749135895
- P. Camps, X. Formosa, C. Galdeano, T. Gómez, D. Muñoz-Torrero, M. Scarpellini, E. Viayna, A. Badia, M.V. Clos, A. Camins, M. Pallàs, M. Bartolini, F. Mancini, V. Andrisano, J. Estelrich, M. Lizondo, A. Bidon-Chanal, and F.J. Luque J. Med. Chem. 51 2008 3588 3598
- (2008) J. Med. Chem. , vol.51 , pp. 3588-3598
- Camps, P.¹ Formosa, X.² Galdeano, C.³ Gómez, T.⁴ Muñoz-Torrero, D.⁵ Scarpellini, M.⁶ Viayna, E.⁷ Badia, A.⁸ Clos, M.V.⁹ Camins, A.¹⁰ Pallàs, M.¹¹ Bartolini, M.¹² Mancini, F.¹³ Andrisano, V.¹⁴ Estelrich, J.¹⁵ Lizondo, M.¹⁶ Bidon-Chanal, A.¹⁷ Luque, F.J.¹⁸

17
- 0032054003
- A. Badia, J.E. Baños, P. Camps, J. Contreras, D.M. Görbig, D. Muñoz-Torrero, M. Simón, and N.M. Vivas Bioorg. Med. Chem. 6 1998 427 440
- (1998) Bioorg. Med. Chem. , vol.6 , pp. 427-440
- Badia, A.¹ Baños, J.E.² Camps, P.³ Contreras, J.⁴ Görbig, D.M.⁵ Muñoz-Torrero, D.⁶ Simón, M.⁷ Vivas, N.M.⁸

18
- 77955510495
- P. Camps, X. Formosa, C. Galdeano, T. Gómez, D. Muñoz-Torrero, L. Ramírez, E. Viayna, E. Gómez, N. Isambert, R. Lavilla, A. Badia, M.V. Clos, M. Bartolini, F. Mancini, V. Andrisano, A. Bidon-Chanal, O. Huertas, T. Dafni, and F.J. Luque Chem. Biol. Interact. 187 2010 411 415
- (2010) Chem. Biol. Interact. , vol.187 , pp. 411-415
- Camps, P.¹ Formosa, X.² Galdeano, C.³ Gómez, T.⁴ Muñoz-Torrero, D.⁵ Ramírez, L.⁶ Viayna, E.⁷ Gómez, E.⁸ Isambert, N.⁹ Lavilla, R.¹⁰ Badia, A.¹¹ Clos, M.V.¹² Bartolini, M.¹³ Mancini, F.¹⁴ Andrisano, V.¹⁵ Bidon-Chanal, A.¹⁶ Huertas, O.¹⁷ Dafni, T.¹⁸ Luque, F.J.¹⁹

19
- 69949089936
- P. Camps, X. Formosa, C. Galdeano, D. Muñoz-Torrero, L. Ramírez, E. Gómez, N. Isambert, R. Lavilla, A. Badia, M.V. Clos, M. Bartolini, F. Mancini, V. Andrisano, M.P. Arce, M.I. Rodríguez-Franco, O. Huertas, T. Dafni, and F.J. Luque J. Med. Chem. 52 2009 5365 5379
- (2009) J. Med. Chem. , vol.52 , pp. 5365-5379
- Camps, P.¹ Formosa, X.² Galdeano, C.³ Muñoz-Torrero, D.⁴ Ramírez, L.⁵ Gómez, E.⁶ Isambert, N.⁷ Lavilla, R.⁸ Badia, A.⁹ Clos, M.V.¹⁰ Bartolini, M.¹¹ Mancini, F.¹² Andrisano, V.¹³ Arce, M.P.¹⁴ Rodríguez-Franco, M.I.¹⁵ Huertas, O.¹⁶ Dafni, T.¹⁷ Luque, F.J.¹⁸

20
- 8544243477
- D. Shao, C. Zou, C. Luo, X. Tang, and Y. Li Bioorg. Med. Chem. Lett. 14 2004 4639 4642
- (2004) Bioorg. Med. Chem. Lett. , vol.14 , pp. 4639-4642
- Shao, D.¹ Zou, C.² Luo, C.³ Tang, X.⁴ Li, Y.⁵

21
- 27644561204
- D. Alonso, I. Dorronsoro, L. Rubio, P. Muñoz, E. García-Palomero, M. Del Monte, A. Bidon-Chanal, M. Orozco, F.J. Luque, A. Castro, M. Medina, and A. Martínez Bioorg. Med. Chem. 13 2005 6588 6597
- (2005) Bioorg. Med. Chem. , vol.13 , pp. 6588-6597
- Alonso, D.¹ Dorronsoro, I.² Rubio, L.³ Muñoz, P.⁴ García-Palomero, E.⁵ Del Monte, M.⁶ Bidon-Chanal, A.⁷ Orozco, M.⁸ Luque, F.J.⁹ Castro, A.¹⁰ Medina, M.¹¹ Martínez, A.¹²

22
- 28544451677
- P. Muñoz-Ruiz, L. Rubio, E. García-Palomero, I. Dorronsoro, M. del Monte-Millán, R. Valenzuela, P. Usán, C. de Austria, M. Bartolini, V. Andrisano, A. Bidon-Chanal, M. Orozco, F.J. Luque, M. Medina, and A. Martínez J. Med. Chem. 48 2005 7223 7233
- (2005) J. Med. Chem. , vol.48 , pp. 7223-7233
- Muñoz-Ruiz, P.¹ Rubio, L.² García-Palomero, E.³ Dorronsoro, I.⁴ Del Monte-Millán, M.⁵ Valenzuela, R.⁶ Usán, P.⁷ De Austria, C.⁸ Bartolini, M.⁹ Andrisano, V.¹⁰ Bidon-Chanal, A.¹¹ Orozco, M.¹² Luque, F.J.¹³ Medina, M.¹⁴ Martínez, A.¹⁵

23
- 84860838525
- D. Antequera, M. Bolos, C. Spuch, C. Pascual, I. Ferrer, M.I. Fernandez-Bachiller, M.I. Rodríguez-Franco, and E. Carro Neurobiol. Dis. 46 2012 682 691
- (2012) Neurobiol. Dis. , vol.46 , pp. 682-691
- Antequera, D.¹ Bolos, M.² Spuch, C.³ Pascual, C.⁴ Ferrer, I.⁵ Fernandez-Bachiller, M.I.⁶ Rodríguez-Franco, M.I.⁷ Carro, E.⁸

24
- 73849108496
- D.S. Pisoni, J.S. da Costa, D. Gamba, C.L. Petzhold, A.C.A. Borges, M.A. Ceschi, P. Lunardi, and C.A.S. Gonçalves Eur. J. Med. Chem. 45 2010 526 535
- (2010) Eur. J. Med. Chem. , vol.45 , pp. 526-535
- Pisoni, D.S.¹ Da Costa, J.S.² Gamba, D.³ Petzhold, C.L.⁴ Borges, A.C.A.⁵ Ceschi, M.A.⁶ Lunardi, P.⁷ Gonçalves, C.A.S.⁸

25
- 76249124586
- J.S. da Costa, D.S. Pisoni, C.B. da Silva, C.L. Petzhold, D. Russowsky, and M.A. Ceschi J. Braz. Chem. Soc. 20 2009 1448 1454
- (2009) J. Braz. Chem. Soc. , vol.20 , pp. 1448-1454
- Da Costa, J.S.¹ Pisoni, D.S.² Da Silva, C.B.³ Petzhold, C.L.⁴ Russowsky, D.⁵ Ceschi, M.A.⁶

26
- 84856143985
- M.V. Marques, M.M. Ruthner, L.A.M. Fontoura, and D. Russowsky J. Braz. Chem. Soc. 23 2012 171 179
- (2012) J. Braz. Chem. Soc. , vol.23 , pp. 171-179
- Marques, M.V.¹ Ruthner, M.M.² Fontoura, L.A.M.³ Russowsky, D.⁴

27
- 79953328346
- C.S. Schwalm, M.A. Ceschi, and D. Russowsky J. Braz. Chem. Soc. 22 2011 623 636
- (2011) J. Braz. Chem. Soc. , vol.22 , pp. 623-636
- Schwalm, C.S.¹ Ceschi, M.A.² Russowsky, D.³

28
- 70350516103
- S. Samai, G.C. Nandi, P. Singh, and M.S. Singh Tetrahedron 65 2009 10155 10161
- (2009) Tetrahedron , vol.65 , pp. 10155-10161
- Samai, S.¹ Nandi, G.C.² Singh, P.³ Singh, M.S.⁴

29
- 40049097415
- S. Das Sharma, P. Hazarika, and D. Konwar Tetrahedron Lett. 49 2008 2216 2220
- (2008) Tetrahedron Lett. , vol.49 , pp. 2216-2220
- Das Sharma, S.¹ Hazarika, P.² Konwar, D.³

30
- 0034635805
- M.K. Hu, and C.F. Lu Tetrahedron Lett. 41 2000 1815 1818
- (2000) Tetrahedron Lett. , vol.41 , pp. 1815-1818
- Hu, M.K.¹ Lu, C.F.²

31
- 0035128448
- M.K. Hu J. Pharm. Pharmacol. 53 2001 83 88
- (2001) J. Pharm. Pharmacol. , vol.53 , pp. 83-88
- Hu, M.K.¹

32
- 78651472058
- W. Luo, Y.P. Li, Y. He, S.L. Huang, J.H. Tan, T.M. Ou, D. Li, L.Q. Gu, and Z.S. Huang Bioorg. Med. Chem. 19 2011 763 770
- (2011) Bioorg. Med. Chem. , vol.19 , pp. 763-770
- Luo, W.¹ Li, Y.P.² He, Y.³ Huang, S.L.⁴ Tan, J.H.⁵ Ou, T.M.⁶ Li, D.⁷ Gu, L.Q.⁸ Huang, Z.S.⁹

33
- 64149111560
- D. Yanover, and M. Kaftory Acta Cryst. E65 2009 o711
- (2009) Acta Cryst. , vol.E65 , pp. 711
- Yanover, D.¹ Kaftory, M.²

34
- 33644811612
- G.L. Ellman, K.D. Courtney, V. Andres, and R.M. Featherstone Biochem. Pharmacol. 7 1961 88 95
- (1961) Biochem. Pharmacol. , vol.7 , pp. 88-95
- Ellman, G.L.¹ Courtney, K.D.² Andres, V.³ Featherstone, R.M.⁴

35
- 0017613512
- A simplification of the protein assay method of Lowry et al. which is more generally applicable
- G.L. Peterson A simplification of the protein assay method of Lowry et al. which is more generally applicable Anal. Biochem. 83 1977 346 356
- (1977) Anal. Biochem. , vol.83 , pp. 346-356
- Peterson, G.L.¹

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.