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Volumn 7, Issue 6, 2011, Pages 704-710

Synthesis and in vitro leishmanicidal activity of disulfide derivatives

Author keywords

Disulfides; Leishmanicidal activity; Synthesis

Indexed keywords

ANTILEISHMANIAL AGENT; BIS(2 BENZIMIDAZOLE)DISULFIDE; BIS(2 PYRIDYL)DISULFIDE; BIS(4 HYDROXYPHENYL)DISULFIDE; BIS(4 METHYLPHENYL)DISULFIDE; DISULFIDE; N [2 [[2 (ACETYLAMINO)PHENYL]DISULFANYL]PHENYL]ACETAMIDE; PENTAMIDINE; UNCLASSIFIED DRUG;

EID: 80755176746     PISSN: 15734064     EISSN: 18756638     Source Type: Journal    
DOI: 10.2174/157340611797928460     Document Type: Article
Times cited : (25)

References (45)
  • 1
    • 80755160559 scopus 로고
    • In: Kiple KF editor. The Cambridge history of human disease. Cambridge: Cambridge University Press
    • Allison, M.J. Leishmaniasis. In: Kiple KF, editor. The Cambridge history of human disease. Cambridge: Cambridge University Press, 1993.
    • (1993) Leishmaniasis
    • Allison, M.J.1
  • 2
    • 84970795837 scopus 로고
    • On the possibility of the occurrence of trypanosomiasis in India
    • Leishaman, W.B. On the possibility of the occurrence of trypanosomiasis in India. Brit. Med. J., 1903, 1, 1252-1254.
    • (1903) Brit. Med. J. , vol.1 , pp. 1252-1254
    • Leishaman, W.B.1
  • 3
    • 0000269479 scopus 로고
    • On the possibility of the occurrence of trypanosomiasis in India
    • Donovan, C. On the possibility of the occurrence of trypanosomiasis in India. Brit. Med. J., 1903, 2, 79-82.
    • (1903) Brit. Med. J. , vol.2 , pp. 79-82
    • Donovan, C.1
  • 6
    • 0030883946 scopus 로고    scopus 로고
    • The current status of antiparasite chemotherapy
    • Croft, S.L. The current status of antiparasite chemotherapy. Parasitology, 1997, 114, S3-S15.
    • (1997) Parasitology , vol.114
    • Croft, S.L.1
  • 8
    • 0023734112 scopus 로고
    • Recent developments in the chemotherapy of leishmaniasis
    • Croft, S.L. Recent developments in the chemotherapy of leishmaniasis. Trends Pharmacol. Sci., 1988, 9, 376-381.
    • (1988) Trends Pharmacol. Sci. , vol.9 , pp. 376-381
    • Croft, S.L.1
  • 9
    • 0024004690 scopus 로고
    • Chemotherapy of leishmaniasis: Biochemical mechanisms, clinical efficacy, and future strategies
    • Berman, J.D. Chemotherapy of leishmaniasis: Biochemical mechanisms, clinical efficacy, and future strategies. Rev. Infect. Dis., 1988, 10, 560-586.
    • (1988) Rev. Infect. Dis. , vol.10 , pp. 560-586
    • Berman, J.D.1
  • 12
    • 77950860253 scopus 로고    scopus 로고
    • Synthesis and biological evaluation of new [1,2,4]triazino[5,6-b]indol-3- ylthio-1,3,5-triazines and [1,2,4]triazino[5,6-b]indol-3-ylthio-pyrimidines against Leishmania donovani
    • Leena, G.; Naresh, S.; Aditya, V.; Saumya, S.; Suman, G.; Neena, G.; Prem, M.S. C. Synthesis and biological evaluation of new [1,2,4]triazino[5,6-b] indol-3-ylthio-1,3,5-triazines and [1,2,4]triazino[5,6-b]indol-3-ylthio- pyrimidines against Leishmania donovani. Eur. J. Med. Chem., 2010, 45, 2359-2365;
    • (2010) Eur. J. Med. Chem. , vol.45 , pp. 2359-2365
    • Leena, G.1    Naresh, S.2    Aditya, V.3    Saumya, S.4    Suman, G.5    Neena, G.6    Prem, M.S.C.7
  • 14
    • 70349643110 scopus 로고    scopus 로고
    • Discovery of novel antileishmanial agents in an attempt to synthesize pentamidine-aplysinopsin hybrid molecule
    • Sharad, P.; Chauhan, S.C.; Chauhan, P.M.S.; Shakya, N.; Verma, A.; Gupta, S. Discovery of novel antileishmanial agents in an attempt to synthesize pentamidine-aplysinopsin hybrid molecule. J. Med. Chem., 2009, 52, 5793-5802.
    • (2009) J. Med. Chem. , vol.52 , pp. 5793-5802
    • Sharad, P.1    Chauhan, S.C.2    Chauhan, P.M.S.3    Shakya, N.4    Verma, A.5    Gupta, S.6
  • 16
    • 6044272951 scopus 로고    scopus 로고
    • Antileishmanial pyrazolopyridine derivatives: Synthesis and structure-activity relationship analysis
    • DOI 10.1021/jm0401006
    • de Mello, H.; Echevarria, A.; Bernardino, A. M.; Canto-Cavalheiro, M.; Leon, L.L. Antileishmanial pyrazolopyridine derivatives: Synthesis and structure-activity relationship analysis. J. Med. Chem., 2004, 47, 5427-5432. (Pubitemid 39382792)
    • (2004) Journal of Medicinal Chemistry , vol.47 , Issue.22 , pp. 5427-5432
    • De Mello, H.1    Echevarria, A.2    Bernardino, A.M.3    Canto-Cavalheiro, M.4    Leon, L.L.5
  • 18
    • 0036946453 scopus 로고    scopus 로고
    • Synthesis, and biological evaluation of new 1,3,4-thiadiazolium-2- phenylamine derivatives against Leishmania amazonensis promastigotes and amastigotes
    • DOI 10.1016/S0223-5234(02)01401-0, PII S0223523402014010
    • da Silva, E.F.; Canto-Cavalheiro, M.M.; Braz, V.R.; Cysne-Finkelstein, L.; Leon, L. L.; Echevarria, A. Synthesis, and biological evaluation of new 1,3,4-thiazolium-2-phenylamine derivatives against Leishmania amazonensis promastigotes. Eur. J. Med. Chem., 2002, 37, 979-984. (Pubitemid 36355835)
    • (2002) European Journal of Medicinal Chemistry , vol.37 , Issue.12 , pp. 979-984
    • Da Silva, E.F.1    Canto-Cavalheiro, M.M.2    Braz, V.R.3    Cysne-Finkelstein, L.4    Leon, L.L.5    Echevarria, A.6
  • 20
    • 79751488230 scopus 로고    scopus 로고
    • Synthesis, leishmanicidal and enzyme inhibitory activities of quinoline-4-carboxylic acid
    • Khan, K.M.; Saied, S.; Mughal, U.R.; Munawar, M.; Samreen, Khan, A.; Perveen, S. Synthesis, leishmanicidal and enzyme inhibitory activities of quinoline-4-carboxylic acid. J. Chem. Soc. Pak., 2009, 31, 809-818.
    • (2009) J. Chem. Soc. Pak. , vol.31 , pp. 809-818
    • Khan, K.M.1    Saied, S.2    Mughal, U.R.3    Munawar, M.4    Samreen Khan, A.5    Perveen, S.6
  • 21
    • 68049108342 scopus 로고    scopus 로고
    • Vitro antileishmanial activities of germatarnyl and silicon incorporated diorganotin derivatives: Synthesis and spectroscopic properties
    • Salma, U.; Mazhar, M.; Imtiaz-ud-Din; Ali, S.; Khan K.M. In vitro antileishmanial activities of germatarnyl and silicon incorporated diorganotin derivatives: Synthesis and spectroscopic properties. J. Enzyme Inhib. Med. Chem., 2009, 24, 413-419.
    • (2009) J. Enzyme Inhib. Med. Chem. , vol.24 , pp. 413-419
    • Salma, U.1    Mazhar, M.2    Imtiaz-Ud-Din Ali, S.3    Khan, K.M.4
  • 22
    • 66149137584 scopus 로고    scopus 로고
    • Leishmanicidal potential of Nsubstituted morpholine derivatives: Synthesis and structure-activity relationships
    • Khan, K.M.; Khan, M.Z.; Taha, M.; Maharvi, G.M.; Saify, Z.S.; Perveen, S.; Choudhary, M.I. Leishmanicidal potential of Nsubstituted morpholine derivatives: Synthesis and structure-activity relationships. Nat. Prod. Res., 2009, 23, 479-484.
    • (2009) Nat. Prod. Res. , vol.23 , pp. 479-484
    • Khan, K.M.1    Khan, M.Z.2    Taha, M.3    Maharvi, G.M.4    Saify, Z.S.5    Perveen, S.6    Choudhary, M.I.7
  • 24
    • 0001379039 scopus 로고
    • Boron trifluoride catalyzed addition of disulfides to alkenes
    • Caserio, M.C.; Fisher, C.L.; Kim, J.K. Boron trifluoride catalyzed addition of disulfides to alkenes. J. Org. Chem., 1985, 50, 4390-4393.
    • (1985) J. Org. Chem. , vol.50 , pp. 4390-4393
    • Caserio, M.C.1    Fisher, C.L.2    Kim, J.K.3
  • 25
    • 37049074738 scopus 로고
    • 1,2-Disulphenylation of alkenes induced by a hypervalent iodine (III) reagent [PhIOTfOH]
    • Kitamura, T.; Matsuyuki, J.-I.; Taniguchi, H. 1,2-Disulphenylation of alkenes induced by a hypervalent iodine (III) reagent [PhIOTfOH]. J. Chem. Soc. Perkin Trans., 1991, 1, 1607-1608.
    • (1991) J. Chem. Soc. Perkin Trans. , vol.1 , pp. 1607-1608
    • Kitamura, T.1    Matsuyuki, J.-I.2    Taniguchi, H.3
  • 27
    • 0017615827 scopus 로고
    • Artificial hybrid protein containing a toxic protein fragment and a cell membrane receptor binding moiety in a disulfide conjugate. I. Synthesis of diphtheria toxin fragment A-S-S human placental lactogen with methyl 5 bromovalerimidate
    • Chang, T.-M.; Dazord, A.; Neville Jr, D.M. Artificial hybrid protein containing a toxic protein fragment and a cell membrane receptor-binding moiety in a disulfide conjugate I Synthesis of diphtheria toxin fragment A-S-S-human placental lactogen with methyl-5-bromovalerimidate. J. Biol. Chem., 1977, 252, 1505-1514. (Pubitemid 8047761)
    • (1977) Journal of Biological Chemistry , vol.252 , Issue.4 , pp. 1505-1514
    • Chang, T.M.1    Neville Jr., D.M.2
  • 28
    • 0034524904 scopus 로고    scopus 로고
    • Disulfide bond mutations in follicle-stimulating hormone result in uncoupling of biological activity from intracellular behavior
    • DOI 10.1210/en.141.12.4751
    • Hiróoka, T.; Maassen, D.; Berger, P.; Boime, I. Disulfide bond mutations in follicle-stimulating hormone result in uncoupling of biological activity from intracellular behaviour. Endocrinology, 2000, 141, 4751-4756. (Pubitemid 32055155)
    • (2000) Endocrinology , vol.141 , Issue.12 , pp. 4751-4756
    • Hiro'oka, T.1    Maassen, D.2    Berger, P.3    Boime, I.4
  • 31
    • 0023130309 scopus 로고
    • Antifungal activity of ajoene derived from garlic
    • Yoshida, S., Kasuga, S.; Hayashi, N.; Ushiroguchi, T.; Matsuura, H.; Nakagawa, S. Antifungal activity of ajoene derived from garlic. Appl. Environ. Microbiol., 1987, 53, 615-617. (Pubitemid 17017558)
    • (1987) Applied and Environmental Microbiology , vol.53 , Issue.3 , pp. 615-617
    • Yoshida, S.1    Kasuga, S.2    Hayashi, N.3
  • 33
    • 0029660277 scopus 로고    scopus 로고
    • Inhibation of microbial growth by ajoene , A sulfurcontaining compound derived from garlic
    • Naganawa, R.; Iwata, N.; Ishikawa, K.; Fukuda, H.; Fujino, T.; Suzuki, A. Inhibation of microbial growth by ajoene , A sulfurcontaining compound derived from garlic. Appl. Environ. Microbiol., 1996, 63, 4238-4242.
    • (1996) Appl. Environ. Microbiol. , vol.63 , pp. 4238-4242
    • Naganawa, R.1    Iwata, N.2    Ishikawa, K.3    Fukuda, H.4    Fujino, T.5    Suzuki, A.6
  • 34
    • 15044358936 scopus 로고    scopus 로고
    • Recent studies on bioactive natural products
    • Atta-Ur-Rahman, Choudhary, M.I. Recent studies on bioactive natural products. Pure Appl. Chem., 1999, 71, 1079-1081
    • (1999) Pure Appl. Chem. , vol.71 , pp. 1079-1081
    • Atta-Ur-Rahman1    Choudhary, M.I.2
  • 35
    • 0036020342 scopus 로고    scopus 로고
    • Antiproliferative and leishmanicidal effect of ajoene on various Leishmania species: Ultrastructural study
    • DOI 10.1007/s00436-002-0649-9
    • Ledezma E.; Jorquera, A.; Bendezú, H.; Vivas, J.; Péres, G. Antiproliferative and leishmanicidal effect of ajoene on various Leishmania species; Ultrastructural study. Parasitol Res., 2002, 88, 748-753 and references quoted therein. (Pubitemid 34762328)
    • (2002) Parasitology Research , vol.88 , Issue.8 , pp. 748-753
    • Ledezma, E.1    Jorquera, A.2    Bendezu, H.3    Vivas, J.4    Perez, G.5
  • 36
    • 57349102432 scopus 로고    scopus 로고
    • An expedient and selective approach towards disulfides using sodium bromate/sodium hydrogen sulfite reagent
    • Khan, K.M.; Ali, M.; Taha, M.; Perveen, S.; Choudhary, M.I.; Voelter. W. An expedient and selective approach towards disulfides using sodium bromate/sodium hydrogen sulfite reagent. Lett. Org. Chem., 2008, 5, 432-434.
    • (2008) Lett. Org. Chem. , vol.5 , pp. 432-434
    • Khan, K.M.1    Ali, M.2    Taha, M.3    Perveen, S.4    Choudhary, M.I.5    Voelter, W.6
  • 37
    • 69549097841 scopus 로고    scopus 로고
    • A mild and alternative approach towards symmetrical disulfides using H3IO5/NaHSO3 combination
    • Khan, K.M.; Taha, M.; Ali, M.; Perveen, S. A mild and alternative approach towards symmetrical disulfides using H3IO5/NaHSO3 combination. Lett. Org. Chem., 2009, 6, 319-320.
    • (2009) Lett. Org. Chem. , vol.6 , pp. 319-320
    • Khan, K.M.1    Taha, M.2    Ali, M.3    Perveen, S.4
  • 38
    • 77955936821 scopus 로고    scopus 로고
    • An improved method for the synthesis of disulfides by periodic acid and sodium hydrogen sulfite in water
    • Khan, K.M.; Taha, M.; Rahim, F.; Ali, M.; Jamil, W.; Perveen, S.; Choudhary, M.I. An improved method for the synthesis of disulfides by periodic acid and sodium hydrogen sulfite in water. Lett. Org. Chem., 2010, 7, 0000.
    • (2010) Lett. Org. Chem. , vol.7 , pp. 0000
    • Khan, K.M.1    Taha, M.2    Rahim, F.3    Ali, M.4    Jamil, W.5    Perveen, S.6    Choudhary, M.I.7
  • 41
    • 71749088187 scopus 로고    scopus 로고
    • 1,3,4-Oxadiazole-2(3H)-thione and its analogues: A new class of non-competitive nucleotide pyrophosphatases/phosphodiesterases 1 inhibitors
    • Khan, K.M.; Fatima, N.; Rasheed, M.; Jalil, S.; Ambreen, N.; Perveen, S.; Choudhary, M.I. 1,3,4-Oxadiazole-2(3H)-thione and its analogues: A new class of non-competitive nucleotide pyrophosphatases/phosphodiesterases 1 inhibitors. Bioorg. Med. Chem., 2009, 17, 7816-7822.
    • (2009) Bioorg. Med. Chem. , vol.17 , pp. 7816-7822
    • Khan, K.M.1    Fatima, N.2    Rasheed, M.3    Jalil, S.4    Ambreen, N.5    Perveen, S.6    Choudhary, M.I.7


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