Ivermectin antagonizes ethanol inhibition in purinergic P2X4 receptors

Journal of Pharmacology and Experimental Therapeutics

Volumn 334, Issue 3, 2010, Pages 720-728

  Asatryan, Liana ^a   Popova, Maya ^a   Perkins, Daya ^a   Trudell, James R ^b   Alkana, Ronald L ^a   Davies, Daryl L ^a  

^a UNIVERSITY OF SOUTHERN CALIFORNIA   (United States)

^b STANFORD UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINE TRIPHOSPHATE; ALCOHOL; IVERMECTIN; PURINERGIC P2X4 RECEPTOR; ANTHELMINTIC AGENT; CENTRAL DEPRESSANT AGENT; COMPLEMENTARY RNA; METHIONINE; P2RX4 PROTEIN, RAT; PURINERGIC P2 RECEPTOR; PURINERGIC P2 RECEPTOR ANTAGONIST;

ANIMAL CELL; ARTICLE; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; CRYSTAL STRUCTURE; NONHUMAN; NUCLEOTIDE SEQUENCE; OOCYTE; PRIORITY JOURNAL; PROTEIN EXPRESSION; SENSITIVITY ANALYSIS; SUBSTITUTION REACTION; VOLTAGE CLAMP; X RAY ANALYSIS; XENOPUS; ZEBRA FISH; ANIMAL; ANTAGONISTS AND INHIBITORS; BIOTINYLATION; CHEMICAL STRUCTURE; CHEMISTRY; DRUG EFFECTS; METABOLISM; PATCH CLAMP TECHNIQUE; RAT; SITE DIRECTED MUTAGENESIS; WESTERN BLOTTING; X RAY CRYSTALLOGRAPHY;

ADENOSINE TRIPHOSPHATE; ANIMALS; ANTHELMINTICS; BIOTINYLATION; BLOTTING, WESTERN; CENTRAL NERVOUS SYSTEM DEPRESSANTS; CRYSTALLOGRAPHY, X-RAY; ETHANOL; IVERMECTIN; METHIONINE; MODELS, MOLECULAR; MUTAGENESIS, SITE-DIRECTED; OOCYTES; PATCH-CLAMP TECHNIQUES; PURINERGIC P2 RECEPTOR ANTAGONISTS; RATS; RECEPTORS, PURINERGIC P2; RECEPTORS, PURINERGIC P2X4; RNA, COMPLEMENTARY; XENOPUS; ZEBRAFISH;

EID: 77956257859     PISSN: 00223565     EISSN: 15210103     Source Type: Journal    
DOI: 10.1124/jpet.110.167908     Document Type: Article

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