Functional properties of internalization-deficient P2X4 receptors reveal a novel mechanism of ligand-gated channel facilitation by ivermectin

Molecular Pharmacology

Volumn 69, Issue 2, 2006, Pages 576-587

  Toulmé, Estelle ^a   Soto, Florentina ^b,c   Garret, Maurice ^a   Boué Grabot, Eric ^a  

^a CNRS   (France)

^b MAX PLANCK INSTITUTE OF EXPERIMENTAL MEDICINE   (Germany)

^c SAINT LOUIS UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ACETYLCHOLINE; ACETYLCHOLINE DERIVATIVE; ADENOSINE TRIPHOSPHATE; CELL SURFACE RECEPTOR; CLATHRIN; EPIDERMAL GROWTH FACTOR RECEPTOR PATHWAY SUBSTRATE 15; IVERMECTIN; NICOTINIC ALPHA7 ACETYLCHOLINE; PURINE P2X4 RECEPTOR; TRANSCRIPTION FACTOR AP 2; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CELL MEMBRANE; CONTROLLED STUDY; ENDOCYTOSIS; FEMALE; ION PERMEABILITY; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN TRANSPORT; RAT; SIGNAL TRANSDUCTION;

ADENOSINE TRIPHOSPHATE; AMINO ACID MOTIFS; ANIMALS; ANTIPARASITIC AGENTS; CELL MEMBRANE; ENDOCYTOSIS; HUMANS; ION CHANNEL GATING; ION CHANNELS; IVERMECTIN; LIGANDS; MUTATION; OOCYTES; PERMEABILITY; RATS; RECEPTORS, NICOTINIC; RECEPTORS, PURINERGIC P2;

EID: 31044446583     PISSN: 0026895X     EISSN: 15210111     Source Type: Journal    
DOI: 10.1124/mol.105.018812     Document Type: Article

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