Roles of ectodomain and transmembrane regions in ethanol and agonist action in purinergic P2X2 and P2X3 receptors

Neuropharmacology

Volumn 55, Issue 5, 2008, Pages 835-843

  Asatryan, Liana ^a   Popova, Maya ^a   Woodward, John J ^b   King, Brian F ^c   Alkana, Ronald L ^a   Davies, Daryl L ^a  

^a UNIVERSITY OF SOUTHERN CALIFORNIA   (United States)

^b MEDICAL UNIVERSITY OF SOUTH CAROLINA   (United States)

^c UNIVERSITY COLLEGE LONDON   (United Kingdom)

Author keywords

Alcohol; Chimeric receptors; Electrophysiology; Purinergic P2X receptors; Sites of ethanol action; Xenopus oocytes

Indexed keywords

ADENOSINE TRIPHOSPHATE; ALCOHOL; ALPHA,BETA METHYLENEADENOSINE TRIPHOSPHATE; COMPLEMENTARY RNA; ION CHANNEL; PURINERGIC P2X2 RECEPTOR; PURINERGIC P2X3 RECEPTOR;

AGONIST; ANIMAL CELL; ARTICLE; BINDING SITE; CHANNEL GATING; CHIMERA; CONCENTRATION RESPONSE; CONTROLLED STUDY; ELECTROPHYSIOLOGY; LONG TERM POTENTIATION; NEUROTRANSMITTER RELEASE; NOCICEPTION; NONHUMAN; NUCLEOTIDE SEQUENCE; OOCYTE; POINT MUTATION; PRIORITY JOURNAL; RECEPTOR DOWN REGULATION; RECEPTOR UPREGULATION; RNA SYNTHESIS; SYNAPTIC TRANSMISSION; VOLTAGE CLAMP; WILD TYPE; XENOPUS LAEVIS;

ADENOSINE TRIPHOSPHATE; ANIMALS; CENTRAL NERVOUS SYSTEM DEPRESSANTS; DOSE-RESPONSE RELATIONSHIP, DRUG; ETHANOL; MEMBRANE POTENTIALS; MUTATION; OOCYTES; PATCH-CLAMP TECHNIQUES; PROTEIN STRUCTURE, TERTIARY; RECEPTORS, PURINERGIC P2; XENOPUS LAEVIS;

EID: 50849130216     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.neuropharm.2008.06.044     Document Type: Article

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