Carbonic anhydrase activators: Activation of the β-carbonic anhydrase from the pathogenic yeast Candida glabrata with amines and amino acids

Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 5, 2010, Pages 1701-1704

  Innocenti, Alessio ^a   Leewattanapasuk, Worraanong ^b   Manole, Gheorghe ^c   Scozzafava, Andrea ^a   Mühlschlegel, Fritz A ^b   Supuran, Claudiu T ^a  

^a UNIVERSITY OF FLORENCE   (Italy)

^b UNIVERSITY OF KENT   (United Kingdom)

^c V Babes National Institute of Pathology   (Romania)

Author keywords

Activator; Amine; Amino acid; Candida glabrata; Carbonic anhydrase

Indexed keywords

1 (2 AMINOETHYL) PIPERAZINE; 2 (2 PYRIDYL)ETHYLAMINE; 2 PYRIDYL METHYLAMINE; 4 (2 AMINOETHYL) MORPHOLINE; ADRENALIN; AMINE; AMINO ACID; AMINOETHYL PIPERAZINE; BETA CARBONIC ANHYDRASE; CARBONATE DEHYDRATASE; DOPA; DOPAMINE; HISTAMINE; HISTIDINE; LEVODOPA; MORPHOLINE; PHENYLALANINE; PYRIDYL ALKYL AMINE; SEROTONIN; TRYPTOPHAN; UNCLASSIFIED DRUG;

ARTICLE; CANDIDA GLABRATA; CATALYSIS; ENZYME ACTIVATION; ENZYME MECHANISM; GENETIC CODE; NONHUMAN; PATHOGENESIS;

AMINES; AMINO ACIDS; CANDIDA GLABRATA; CARBONIC ANHYDRASES; CATALYTIC DOMAIN; ENZYME ACTIVATION; HUMANS; KINETICS; MODELS, MOLECULAR; RECOMBINANT PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP;

CANDIDA GLABRATA; FUNGI;

EID: 76649128714     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.01.054     Document Type: Article

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