64Cu-AMD3100-A novel imaging agent for targeting chemokine receptor CXCR4

Bioorganic and Medicinal Chemistry

Volumn 17, Issue 4, 2009, Pages 1486-1493

  Jacobson, Orit ^a   Weiss, Ido D ^b   Szajek, Lawrence ^c   Farber, Joshua M ^b   Kiesewetter, Dale O ^a  

^a NATIONAL INSTITUTE OF BIOMEDICAL IMAGING AND BIOENGINEERING   (United States)

^b NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES   (United States)

^c NATIONAL INSTITUTES OF HEALTH   (United States)

Author keywords

AMD3100; Copper 64; CXCR4; PET

Indexed keywords

CHEMOKINE RECEPTOR CXCR4; CONTRAST MEDIUM; COPPER 64; PLERIXAFOR; COPPER; DIAGNOSTIC AGENT; HETEROCYCLIC COMPOUND; RADIOPHARMACEUTICAL AGENT;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; BINDING AFFINITY; CELL MIGRATION; CONTROLLED STUDY; DRUG ACCUMULATION; DRUG CLEARANCE; DRUG DISTRIBUTION; DRUG RECEPTOR BINDING; KIDNEY CLEARANCE; MOUSE; NONHUMAN; TUMOR DIAGNOSIS; ANIMAL; C57BL MOUSE; CALCIUM SIGNALING; CHEMISTRY; DIAGNOSTIC IMAGING; DRUG ANTAGONISM; DRUG EFFECT; HUMAN; ISOTOPE LABELING; LEUKEMIA CELL LINE; METABOLISM; METHODOLOGY; POSITRON EMISSION TOMOGRAPHY; PROTEIN BINDING; SIGNAL TRANSDUCTION; SYNTHESIS; TUMOR CELL LINE;

ANIMALS; CALCIUM SIGNALING; CELL LINE, TUMOR; COPPER RADIOISOTOPES; DIAGNOSTIC IMAGING; HETEROCYCLIC COMPOUNDS; HUMANS; ISOTOPE LABELING; JURKAT CELLS; MICE; MICE, INBRED C57BL; POSITRON-EMISSION TOMOGRAPHY; PROTEIN BINDING; RADIOPHARMACEUTICALS; RECEPTORS, CXCR4; SIGNAL TRANSDUCTION;

EID: 60049083843     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2009.01.014     Document Type: Article

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