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New Journal of Chemistry

Volumn 33, Issue 1, 2009, Pages 148-156

Probing multivalency for the inhibition of an enzyme: Glycogen phosphorylase as a case study

(6) Cecioni, Samy a Argintaru, Oana Andreea a Docsa, Tibor b Gergely, Pál b Praly, Jean Pierre a Vidal, Sébastien a

a UNIVERSITÉ LYON 1 (France)

b UNIVERSITY OF DEBRECEN (Hungary)

Author keywords

[No Author keywords available]

Indexed keywords

1,3,5 TRIS 4' 2'' [3''' C (BNETA DEXTRO GLUCOPYROSYL) 1 ''',2''',4''' OXADIAZOL 5''' YL]ETHYL 1',2',3' TRIAZOL 1' YLMETHYLBENZENE; 1,3,5 TRIS[3' C (BETA DEXTRO GLUCOPYRANOSYL) 1',2',4' OXADIAZOL 5' YL] BENZENE; 3 C (BETA DEXTRO GLUCOPYRANOSYL) 5 (BUT 1'' YN 4'' YL) 1,2,4 OXADIAZOLE; 5 [2 (1''' BENZYL 1''',2''',3''' TRIAZOL 4''' YL)ETHYL] 3 C (BETA DEXTRO GLUCOPYRANOSYL) 1,2,4 OXADIAZOLE; ENZYME INHIBITOR; GLYCOGEN PHOSPHORYLASE; ION; UNCLASSIFIED DRUG;

ARTICLE; DRUG PROTEIN BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME BINDING; ENZYME INHIBITION; PHARMACOPHORE; PRIORITY JOURNAL;

EID: 58149144765 PISSN: 11440546 EISSN: 13699261 Source Type: Journal
DOI: 10.1039/b812540f Document Type: Article

Times cited : (30)

References (58)

1
- 2342466734
- S. Wild G. Roglic A. Green R. Sicree H. King Diabetes Care 2004 27 1047
- (2004) Diabetes Care , vol.27 , pp. 1047
- Wild, S.¹ Roglic, G.² Green, A.³ Sicree, R.⁴ King, H.⁵

2
- 0035856920
- P. Zimmet K. G. M. M. Alberti J. Shaw Nature 2001 414 782
- (2001) Nature , vol.414 , pp. 782
- Zimmet, P.¹ Alberti, K.G.M.M.² Shaw, J.³

3
- 0035857020
- D. E. Moller Nature 2001 414 821
- (2001) Nature , vol.414 , pp. 821
- Moller, D.E.¹

4
- 0038408484
- N. Morral Trends Endocrinol. Metab. 2003 14 169
- (2003) Trends Endocrinol. Metab. , vol.14 , pp. 169
- Morral, N.¹

5
- 36549069114
- L. Agius Best Pract. Res. Clin. Metab. 2007 21 587
- (2007) Best Pract. Res. Clin. Metab. , vol.21 , pp. 587
- Agius, L.¹

6
- 3843079807
- B. R. Henke J. Med. Chem. 2004 47 4118
- (2004) J. Med. Chem. , vol.47 , pp. 4118
- Henke, B.R.¹

7
- 33750511973
- C. Fievet J.-C. Fruchart B. Staels Curr. Opin. Pharmacol. 2006 6 606
- (2006) Curr. Opin. Pharmacol. , vol.6 , pp. 606
- Fievet, C.¹ Fruchart, J.-C.² Staels, B.³

8
- 3843121153
- L. B. Knudsen J. Med. Chem. 2004 47 4128
- (2004) J. Med. Chem. , vol.47 , pp. 4128
- Knudsen, L.B.¹

9
- 15044362439
- M. A. Nauck J. J. Meier Regul. Pept. 2005 128 135
- (2005) Regul. Pept. , vol.128 , pp. 135
- Nauck, M.A.¹ Meier, J.J.²

10
- 3843072211
- A. E. Weber J. Med. Chem. 2004 47 4135
- (2004) J. Med. Chem. , vol.47 , pp. 4135
- Weber, A.E.¹

11
- 33749834648
- A. Barnett Int. J. Clin. Pract. 2006 60 1454
- (2006) Int. J. Clin. Pract. , vol.60 , pp. 1454
- Barnett, A.¹

12
- 34249902025
- D. J. Drucker Diabetes Care 2007 30 1335
- (2007) Diabetes Care , vol.30 , pp. 1335
- Drucker, D.J.¹

13
- 85047684646
- B. J. Goldstein J. Clin. Endocrinol. Metab. 2002 87 2474
- (2002) J. Clin. Endocrinol. Metab. , vol.87 , pp. 2474
- Goldstein, B.J.¹

14
- 3843121119
- R. Hooft van Huijsduijnen W. H. B. Sauer A. Bombrun D. Swinnen J. Med. Chem. 2004 47 4142
- (2004) J. Med. Chem. , vol.47 , pp. 4142
- Hooft Van Huijsduijnen, R.¹ Sauer, W.H.B.² Bombrun, A.³ Swinnen, D.⁴

15
- 21244444303
- L. Bialy H. Waldmann Angew. Chem., Int. Ed. 2005 44 3814
- (2005) Angew. Chem., Int. Ed. , vol.44 , pp. 3814
- Bialy, L.¹ Waldmann, H.²

16
- 0035110957
- J. L. Treadway P. Mendys D. J. Hoover Exp. Opin. Invest. Drugs 2001 10 439
- (2001) Exp. Opin. Invest. Drugs , vol.10 , pp. 439
- Treadway, J.L.¹ Mendys, P.² Hoover, D.J.³

17
- 0036889606
- N. G. Oikonomakos Curr. Protein Pept. Sci. 2002 3 561
- (2002) Curr. Protein Pept. Sci. , vol.3 , pp. 561
- Oikonomakos, N.G.¹

18
- 0037648878
- L. Somsak V. Nagy Z. Hadady T. Docsa P. Gergely Curr. Pharm. Des. 2003 9 1177
- (2003) Curr. Pharm. Des. , vol.9 , pp. 1177
- Somsak, L.¹ Nagy, V.² Hadady, Z.³ Docsa, T.⁴ Gergely, P.⁵

19
- 23644444478
- D. J. Baker J. A. Timmons P. L. Greenhaff Diabetes 2005 54 2453
- (2005) Diabetes , vol.54 , pp. 2453
- Baker, D.J.¹ Timmons, J.A.² Greenhaff, P.L.³

20
- 24644517553
- L. Somsák V. Nagy Z. Hadady N. Felfoldi T. Docsa P. Gergely Front. Med. Chem. 2005 2 253
- (2005) Front. Med. Chem. , vol.2 , pp. 253
- Somsák, L.¹ Nagy, V.² Hadady, Z.³ Felfoldi, N.⁴ Docsa, T.⁵ Gergely, P.⁶

21
- 41949086319
- N. G. Oikonomakos L. Somsák Curr. Opin. Invest. Drugs 2008 9 379
- (2008) Curr. Opin. Invest. Drugs , vol.9 , pp. 379
- Oikonomakos, N.G.¹ Somsák, L.²

22
- 9544234747
- R. J. Fletterick S. R. Sprang Acc. Chem. Res. 1982 15 361
- (1982) Acc. Chem. Res. , vol.15 , pp. 361
- Fletterick, R.J.¹ Sprang, S.R.²

23
- 0024290703
- S. R. Sprang K. R. Acharya E. J. Goldsmith D. I. Stuart K. Varvill R. J. Fletterick N. B. Madsen L. N. Johnson Nature 1988 336 215
- (1988) Nature , vol.336 , pp. 215
- Sprang, S.R.¹ Acharya, K.R.² Goldsmith, E.J.³ Stuart, D.I.⁴ Varvill, K.⁵ Fletterick, R.J.⁶ Madsen, N.B.⁷ Johnson, L.N.⁸

24
- 0024322304
- D. Barford L. N. Johnson Nature 1989 340 609
- (1989) Nature , vol.340 , pp. 609
- Barford, D.¹ Johnson, L.N.²

25
- 0034660681
- N. G. Oikonomakos V. T. Skamnaki K. E. Tsitsanou N. G Gavalas L. N. Johnson Structure 2000 8 575
- (2000) Structure , vol.8 , pp. 575
- Oikonomakos, N.G.¹ Skamnaki, V.T.² Tsitsanou, K.E.³ Gavalas, N.G.⁴ Johnson, L.N.⁵

26
- 0034602424
- N. G. Oikonomakos J. B. Schnier S. E. Zographos V. T. Skamnaki K. E. Tsitsanou L. N. Johnson J. Biol. Chem. 2000 275 34566
- (2000) J. Biol. Chem. , vol.275 , pp. 34566
- Oikonomakos, N.G.¹ Schnier, J.B.² Zographos, S.E.³ Skamnaki, V.T.⁴ Tsitsanou, K.E.⁵ Johnson, L.N.⁶

27
- 2942544255
- M. N. Kosmopoulou D. D. Leonidas E. D. Chrysina N. Bischler G. Eisenbrand C. E. Sakarellos R. Pauptit N. G. Oikonomakos Eur. J. Biochem. 2004 271 2280
- (2004) Eur. J. Biochem. , vol.271 , pp. 2280
- Kosmopoulou, M.N.¹ Leonidas, D.D.² Chrysina, E.D.³ Bischler, N.⁴ Eisenbrand, G.⁵ Sakarellos, C.E.⁶ Pauptit, R.⁷ Oikonomakos, N.G.⁸

28
- 26444555541
- T. Klabunde K. U. Wendt D. Kadereit V. Brachvogel H. J. Burger A. W. Herling N. G. Oikonomakos M. N. Kosmopoulou D. Schmoll E. Sarubbi E. von Roedern K. Schonafinger E. Defossa J. Med. Chem. 2005 48 6178
- (2005) J. Med. Chem. , vol.48 , pp. 6178
- Klabunde, T.¹ Wendt, K.U.² Kadereit, D.³ Brachvogel, V.⁴ Burger, H.J.⁵ Herling, A.W.⁶ Oikonomakos, N.G.⁷ Kosmopoulou, M.N.⁸ Schmoll, D.⁹ Sarubbi, E.¹⁰ Von Roedern, E.¹¹ Schonafinger, K.¹² Defossa, E.¹³

29
- 33746906704
- B. R. Henke S. M. Sparks Mini-Rev. Med. Chem. 2006 6 845
- (2006) Mini-Rev. Med. Chem. , vol.6 , pp. 845
- Henke, B.R.¹ Sparks, S.M.²

30
- 33645794959
- D. J. Baker P. L. Greenhaff J. A. Timmons Exp. Opin. Ther. Pat. 2006 16 459
- (2006) Exp. Opin. Ther. Pat. , vol.16 , pp. 459
- Baker, D.J.¹ Greenhaff, P.L.² Timmons, J.A.³

31
- 33846236476
- A. M. Birch P. W. Kenny N. G. Oikonomakos L. Otterbein P. Schofield P. R. O. Whittamore D. P. Whalley Bioorg. Med. Chem. Lett. 2007 17 394
- (2007) Bioorg. Med. Chem. Lett. , vol.17 , pp. 394
- Birch, A.M.¹ Kenny, P.W.² Oikonomakos, N.G.³ Otterbein, L.⁴ Schofield, P.⁵ Whittamore, P.R.O.⁶ Whalley, D.P.⁷

32
- 18344387526
- N. G. Oikonomakos M. N. Kosmopoulou S. E. Zographos D. D. Leonidas E. D. Chrysina L. Somsak V. Nagy J.-P. Praly T. Docsa B. Toth P. Gergely Eur. J. Biochem. 2002 269 1684
- (2002) Eur. J. Biochem. , vol.269 , pp. 1684
- Oikonomakos, N.G.¹ Kosmopoulou, M.N.² Zographos, S.E.³ Leonidas, D.D.⁴ Chrysina, E.D.⁵ Somsak, L.⁶ Nagy, V.⁷ Praly, J.-P.⁸ Docsa, T.⁹ Toth, B.¹⁰ Gergely, P.¹¹

33
- 33748803362
- M. Benltifa S. Vidal B. Fenet M. Msaddek P. G. Goekjian J.-P. Praly A. Brunyánszki T. Docsa P. Gergely Eur. J. Org. Chem. 2006 4242
- (2006) Eur. J. Org. Chem. , pp. 4242
- Benltifa, M.¹ Vidal, S.² Fenet, B.³ Msaddek, M.⁴ Goekjian, P.G.⁵ Praly, J.-P.⁶ Brunyánszki, A.⁷ Docsa, T.⁸ Gergely, P.⁹

34
- 33746316409
- M. Benltifa S. Vidal D. Gueyrard P. G. Goekjian M. Msaddek J.-P. Praly Tetrahedron Lett. 2006 47 6143
- (2006) Tetrahedron Lett. , vol.47 , pp. 6143
- Benltifa, M.¹ Vidal, S.² Gueyrard, D.³ Goekjian, P.G.⁴ Msaddek, M.⁵ Praly, J.-P.⁶

35
- 33846564497
- L. He Y. Z. Zhang M. Tanoh G.-R. Chen J.-P. Praly E. D. Chrysina C. Tiraidis M. Kosmopoulou D. D. Leonidas N. G. Oikonomakos Eur. J. Org. Chem. 2007 596
- (2007) Eur. J. Org. Chem. , pp. 596
- He, L.¹ Zhang, Y.Z.² Tanoh, M.³ Chen, G.-R.⁴ Praly, J.-P.⁵ Chrysina, E.D.⁶ Tiraidis, C.⁷ Kosmopoulou, M.⁸ Leonidas, D.D.⁹ Oikonomakos, N.G.¹⁰

36
- 11144317860
- H. L. Handl J. Vagner H. Han E. Mash V. J. Hruby R. J. Gillies Exp. Opin. Ther. Targets 2004 8 565 586
- (2004) Exp. Opin. Ther. Targets , vol.8 , pp. 565-586
- Handl, H.L.¹ Vagner, J.² Han, H.³ Mash, E.⁴ Hruby, V.J.⁵ Gillies, R.J.⁶

37
- 9644275467
- S. J. F. Macdonald K. G. Watson R. Cameron D. K. Chalmers D. A. Demaine R. J. Fenton D. Gower J. N. Hamblin S. Hamilton G. J. Hart G. G. A. Inglis B. Jin H. T. Jones D. B. McConnell A. M. Mason V. Nguyen I. J. Owens N. Parry P. A. Reece S. E. Shanahan D. Smith W.-Y. Wu S. P. Tucker Antimicrob. Agents Chemother. 2004 48 4542
- (2004) Antimicrob. Agents Chemother. , vol.48 , pp. 4542
- MacDonald, S.J.F.¹ Watson, K.G.² Cameron, R.³ Chalmers, D.K.⁴ Demaine, D.A.⁵ Fenton, R.J.⁶ Gower, D.⁷ Hamblin, J.N.⁸ Hamilton, S.⁹ Hart, G.J.¹⁰ Inglis, G.G.A.¹¹ Jin, B.¹² Jones, H.T.¹³ McConnell, D.B.¹⁴ Mason, A.M.¹⁵ Nguyen, V.¹⁶ Owens, I.J.¹⁷ Parry, N.¹⁸ Reece, P.A.¹⁹ Shanahan, S.E.²⁰ more..

38
- 58149155969
- S. J. F. MacDonald R. Cameron D. A. Demaine R. J. Fenton G. Foster D. Gower J. N. Hamblin S. Hamilton G. J. Hart A. P. Hill G. G. A. Inglis B. Jin H. T. Jones D. McConnell J. McKimm-Breschkin G. Mills V. Nguyen I. J. Owens N. Parry S. E. Shanahan D. Smith K. G. Watson W.-Y. Wu S. P. Tucker J. Med. Chem. 2005 48 2694
- (2005) J. Med. Chem. , vol.48 , pp. 2694
- MacDonald, S.J.F.¹ Cameron, R.² Demaine, D.A.³ Fenton, R.J.⁴ Foster, G.⁵ Gower, D.⁶ Hamblin, J.N.⁷ Hamilton, S.⁸ Hart, G.J.⁹ Hill, A.P.¹⁰ Inglis, G.G.A.¹¹ Jin, B.¹² Jones, H.T.¹³ McConnell, D.¹⁴ McKimm-Breschkin, J.¹⁵ Mills, G.¹⁶ Nguyen, V.¹⁷ Owens, I.J.¹⁸ Parry, N.¹⁹ Shanahan, S.E.²⁰ more..

39
- 10744221268
- K. G. Watson R. Cameron R. J. Fenton D. Gower S. Hamilton B. Jin G. Y. Krippner A. Luttick D. McConnell S. J. F. MacDonald A. M. Mason V. Nguyen S. P. Tucker W.-Y. Wu Bioorg. Med. Chem. Lett. 2004 14 1589 1592
- (2004) Bioorg. Med. Chem. Lett. , vol.14 , pp. 1589-1592
- Watson, K.G.¹ Cameron, R.² Fenton, R.J.³ Gower, D.⁴ Hamilton, S.⁵ Jin, B.⁶ Krippner, G.Y.⁷ Luttick, A.⁸ McConnell, D.⁹ MacDonald, S.J.F.¹⁰ Mason, A.M.¹¹ Nguyen, V.¹² Tucker, S.P.¹³ Wu, W.-Y.¹⁴

40
- 34447307403
- Y. Lu J. Gervay-Hague Carbohydr. Res. 2007 342 1636 1650
- (2007) Carbohydr. Res. , vol.342 , pp. 1636-1650
- Lu, Y.¹ Gervay-Hague, J.²

41
- 0001564454
- Y. F. Han C. P.-L. Li E. Chow H. Wang Y.-P. Pang P. R. Carlier Bioorg. Med. Chem. 1999 7 2569 2575
- (1999) Bioorg. Med. Chem. , vol.7 , pp. 2569-2575
- Han, Y.F.¹ Li, C.P.-L.² Chow, E.³ Wang, H.⁴ Pang, Y.-P.⁵ Carlier, P.R.⁶

42
- 0032546139
- B. A. Johns C. R. Johnson Tetrahedron Lett. 1998 39 749
- (1998) Tetrahedron Lett. , vol.39 , pp. 749
- Johns, B.A.¹ Johnson, C.R.²

43
- 0032835335
- A. Lohse K. B. Jensen K. Lundgren M. Bols Bioorg. Med. Chem. 1999 7 1965
- (1999) Bioorg. Med. Chem. , vol.7 , pp. 1965
- Lohse, A.¹ Jensen, K.B.² Lundgren, K.³ Bols, M.⁴

44
- 0035033274
- N. Schaschke G. Matschinerb F. Zettlb U. Marquardta A. Bergnera W. Bodea C. P. Sommerhoff L. Moroder Chem. Biol. 2001 8 313 327
- (2001) Chem. Biol. , vol.8 , pp. 313-327
- Schaschke, N.¹ Matschinerb, G.² Zettlb, F.³ Marquardta, U.⁴ Bergnera, A.⁵ Bodea, W.⁶ Sommerhoff, C.P.⁷ Moroder, L.⁸

45
- 0033827122
- V. L. Rath M. Ammirati D. E. Danley J. L. Ekstrom E. M. Gibbs T. R. Hynes A. M. Mathiowetz R. K. McPherson T. V. Olson J. L. Treadway D. J. Hoover Chem. Biol. 2000 7 677 682
- (2000) Chem. Biol. , vol.7 , pp. 677-682
- Rath, V.L.¹ Ammirati, M.² Danley, D.E.³ Ekstrom, J.L.⁴ Gibbs, E.M.⁵ Hynes, T.R.⁶ Mathiowetz, A.M.⁷ McPherson, R.K.⁸ Olson, T.V.⁹ Treadway, J.L.¹⁰ Hoover, D.J.¹¹

46
- 0034607764
- L. Somsak V. Nagy Tetrahedron: Asymmetry 2000 11 1719 1727
- (2000) Tetrahedron: Asymmetry , vol.11 , pp. 1719-1727
- Somsak, L.¹ Nagy, V.²

47
- 0035911020
- A. R. Gangloff J. Litvak E. J. Shelton D. Sperandio V. R. Wang K. D. Rice Tetrahedron Lett. 2001 42 1441 1443
- (2001) Tetrahedron Lett. , vol.42 , pp. 1441-1443
- Gangloff, A.R.¹ Litvak, J.² Shelton, E.J.³ Sperandio, D.⁴ Wang, V.R.⁵ Rice, K.D.⁶

48
- 15044363597
- Y. Wang R. L. Miller D. R. Sauer S. W. Djuric Org. Lett. 2005 7 925 928
- (2005) Org. Lett. , vol.7 , pp. 925-928
- Wang, Y.¹ Miller, R.L.² Sauer, D.R.³ Djuric, S.W.⁴

49
- 84945104463
- R. Huisgen R. Knorr L. Möbius G. Szeimies Chem. Ber. 1965 98 4014
- (1965) Chem. Ber. , vol.98 , pp. 4014
- Huisgen, R.¹ Knorr, R.² Möbius, L.³ Szeimies, G.⁴

50
- 84981452695
- R. Huisgen G. Szeimies L. Möbius Chem. Ber. 1967 100 2494
- (1967) Chem. Ber. , vol.100 , pp. 2494
- Huisgen, R.¹ Szeimies, G.² Möbius, L.³

51
- 0001716552
- R. Huisgen K. Fraunberg H. J. Sturm Tetrahedron Lett. 1969 10 2589
- (1969) Tetrahedron Lett. , vol.10 , pp. 2589
- Huisgen, R.¹ Fraunberg, K.² Sturm, H.J.³

52
- 0037099395
- V. V. Rostovtsev L. G. Green V. V. Fokin K. B. Sharpless Angew. Chem., Int. Ed. 2002 41 2596
- (2002) Angew. Chem., Int. Ed. , vol.41 , pp. 2596
- Rostovtsev, V.V.¹ Green, L.G.² Fokin, V.V.³ Sharpless, K.B.⁴

53
- 0037012920
- C. W. Tornoe C. Christensen M. Meldal J. Org. Chem. 2002 67 3057
- (2002) J. Org. Chem. , vol.67 , pp. 3057
- Tornoe, C.W.¹ Christensen, C.² Meldal, M.³

54
- 0001449887
- T. M. Garrett T. J. McMurry M. W. Hosseini Z. E. Reyes F. E. Hahn K. N. Raymond J. Am. Chem. Soc. 1991 113 2965 2977
- (1991) J. Am. Chem. Soc. , vol.113 , pp. 2965-2977
- Garrett, T.M.¹ McMurry, T.J.² Hosseini, M.W.³ Reyes, Z.E.⁴ Hahn, F.E.⁵ Raymond, K.N.⁶

55
- 77957003650
- E. H. Fischer E. G. Krebs Methods Enzymol. 1962 5 369
- (1962) Methods Enzymol. , vol.5 , pp. 369
- Fischer, E.H.¹ Krebs, E.G.²

56
- 0036132415
- N. G. Oikonomakos V. T. Skamnaki E. Osz L. Szilágyi L. Somsák T. Docsa B. Tóth P. Gergely Bioorg. Med. Chem. 2002 10 261
- (2002) Bioorg. Med. Chem. , vol.10 , pp. 261
- Oikonomakos, N.G.¹ Skamnaki, V.T.² Osz, E.³ Szilágyi, L.⁴ Somsák, L.⁵ Docsa, T.⁶ Tóth, B.⁷ Gergely, P.⁸

57
- 0033577776
- E. Osz L. Somsák L. Szilágyi L. Kovács T. Docsa B. Tóth P. Gergely Bioorg. Med. Chem. Lett. 1999 9 1385
- (1999) Bioorg. Med. Chem. Lett. , vol.9 , pp. 1385
- Osz, E.¹ Somsák, L.² Szilágyi, L.³ Kovács, L.⁴ Docsa, T.⁵ Tóth, B.⁶ Gergely, P.⁷

58
- 0035899177
- L. Somsák L. Kovács M. Tóth E. Osz L. Szilágyi Z. Györgydeák Z. Dinya T. Docsa B. Tóth P. Gergely J. Med. Chem. 2001 44 2843
- (2001) J. Med. Chem. , vol.44 , pp. 2843
- Somsák, L.¹ Kovács, L.² Tóth, M.³ Osz, E.⁴ Szilágyi, L.⁵ Györgydeák, Z.⁶ Dinya, Z.⁷ Docsa, T.⁸ Tóth, B.⁹ Gergely, P.¹⁰

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