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Volumn 3, Issue 3, 2008, Pages 473-477

Carbonic anhydrase inhibitors: Binding of indanesulfonamides to the human isoform II

(6) D'Ambrosio, Katia a Masereel, Bernard b Thiry, Anne b Scozzafava, Andrea c Supuran, Claudiu T c De Simone, Giuseppina a

a CNR (Italy)

b UNIVERSITY OF NAMUR (Belgium)

c UNIVERSITY OF FLORENCE (Italy)

Author keywords

Carbonic anhydrase II; Enzyme inhibitor complexes; Medicinal chemistry; Sulfonamide design; X ray structure

Indexed keywords

CARBONATE DEHYDRATASE II; CARBONATE DEHYDRATASE INHIBITOR; INDAN DERIVATIVE; ISOPROTEIN; SULFONAMIDE;

ARTICLE; BINDING SITE; CHEMISTRY; CONFORMATION; DRUG ANTAGONISM; HUMAN; METABOLISM; STRUCTURE ACTIVITY RELATION; X RAY CRYSTALLOGRAPHY;

BINDING SITES; CARBONIC ANHYDRASE II; CARBONIC ANHYDRASE INHIBITORS; CRYSTALLOGRAPHY, X-RAY; HUMANS; INDANS; MOLECULAR CONFORMATION; PROTEIN ISOFORMS; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES;

EID: 48049109465 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200700274 Document Type: Article

Times cited : (10)

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