-
1
-
-
0003702649
-
-
ACS, Washinton, DC
-
(a) Kingston, H.M.; Haswell, S.J. Microwave Enhance Chemistry, ACS, Washinton, DC, 1997;
-
(1997)
Microwave Enhance Chemistry
-
-
Kingston, H.M.1
Haswell, S.J.2
-
9
-
-
0032330265
-
-
(d) Gabriel, C.; Gabriel, S.; Grant, E.H.; Halstead, B.S.J.; Mingos, D.M.P. Chem. Soc. Rev., 1998, 27, 213;
-
(1998)
Chem. Soc. Rev
, vol.27
, pp. 213
-
-
Gabriel, C.1
Gabriel, S.2
Grant, E.H.3
Halstead, B.S.J.4
Mingos, D.M.P.5
-
10
-
-
0345963038
-
-
(e) Elander, N.; Jones, J.R.; Lu, S.-Y.; Stone-Elander, S. Chem. Soc. Rev., 2000, 29, 239;
-
(2000)
Chem. Soc. Rev
, vol.29
, pp. 239
-
-
Elander, N.1
Jones, J.R.2
Lu, S.-Y.3
Stone-Elander, S.4
-
11
-
-
12344252096
-
-
(f) Lidström, P.; Tieney, J.; Wathey, B.; Westmann, J. Tetrahedron, 2001, 57, 735.
-
(2001)
Tetrahedron
, vol.57
, pp. 735
-
-
Lidström, P.1
Tieney, J.2
Wathey, B.3
Westmann, J.4
-
13
-
-
0141988603
-
-
(h) Swamy, M.K.; Yeh, W.B.; Lin, M.J.; Sun, C.M. Curr. Med. Chem., 2003, 10, 2403.
-
(2003)
Curr. Med. Chem
, vol.10
, pp. 2403
-
-
Swamy, M.K.1
Yeh, W.B.2
Lin, M.J.3
Sun, C.M.4
-
16
-
-
0030477258
-
-
(b) Balkenhohl, F.; von dem Bussche-Huennefeld, C; Lansky, A.; Zechel, C. Angew. Chem. Int. Ed. Engl., 1996, 35, 2288.
-
(1996)
Angew. Chem. Int. Ed. Engl
, vol.35
, pp. 2288
-
-
Balkenhohl, F.1
von dem2
Bussche-Huennefeld, C.3
Lansky, A.4
Zechel, C.5
-
19
-
-
0041461964
-
-
(c) Lew, A.; Krutzik, P.O.; Hart, M.E.; Chamberlain, A.R. J. Comb. Chem., 2002, 4, 95.
-
(2002)
J. Comb. Chem
, vol.4
, pp. 95
-
-
Lew, A.1
Krutzik, P.O.2
Hart, M.E.3
Chamberlain, A.R.4
-
20
-
-
0038066071
-
-
(d) Lidstrom, P.; Westman, J.; Lewis, A. Comb. Chem. High Throughput Screen., 2002, 5, 441.
-
(2002)
Comb. Chem. High Throughput Screen
, vol.5
, pp. 441
-
-
Lidstrom, P.1
Westman, J.2
Lewis, A.3
-
22
-
-
0141988603
-
-
(f) Swamy, M.K.; Yeh, W.B.; Lin, M.J.; Sun, C.M. Curr. Med. Chem., 2003, 10, 2403.
-
(2003)
Curr. Med. Chem
, vol.10
, pp. 2403
-
-
Swamy, M.K.1
Yeh, W.B.2
Lin, M.J.3
Sun, C.M.4
-
25
-
-
34047205297
-
-
(c) Kremsner, J.M.; Stadler, A.; Kappe, C.O. J. Comb. Chem., 2007, 9, 285.
-
(2007)
J. Comb. Chem
, vol.9
, pp. 285
-
-
Kremsner, J.M.1
Stadler, A.2
Kappe, C.O.3
-
27
-
-
0036294671
-
-
(b) Santagada, V.; Perissutti, E.; Caliendo, G. Curr. Med. Chem., 2002, 9, 1251.
-
(2002)
Curr. Med. Chem
, vol.9
, pp. 1251
-
-
Santagada, V.1
Perissutti, E.2
Caliendo, G.3
-
28
-
-
0037085575
-
-
(c) Wathey, B.; Tierney, J.; Lidström, P.; Westman, J.; Drug. Discov. Today, 2002, 7, 373.
-
(2002)
Drug. Discov. Today
, vol.7
, pp. 373
-
-
Wathey, B.1
Tierney, J.2
Lidström, P.3
Westman, J.4
-
29
-
-
1542752259
-
-
(d) Al-Obeidi, F.; Austin, R.E. Okonya, J.F.; Bond, D.R.S. Mini-Rev. Med. Chem., 2003, 3, 449
-
(2003)
Mini-Rev. Med. Chem
, vol.3
, pp. 449
-
-
Al-Obeidi, F.1
Austin, R.E.2
Okonya, J.F.3
Bond, D.R.S.4
-
31
-
-
34247641289
-
-
(f) Alcázar, J.; Diels, G; Schoentjes, B. Mini-Rev. Med. Chem., 2007, 7, 345.
-
(2007)
Mini-Rev. Med. Chem
, vol.7
, pp. 345
-
-
Alcázar, J.1
Diels, G.2
Schoentjes, B.3
-
32
-
-
0034345903
-
-
(a) Cléophax, J.; Liagre, M.; Loupy, A,; Petit, A. Org. Process Res. Develop., 2000, 4, 498.
-
(2000)
Org. Process Res. Develop
, vol.4
, pp. 498
-
-
Cléophax, J.1
Liagre, M.2
Loupy, A.3
Petit, A.4
-
33
-
-
0141922655
-
-
(b) Stadler, A.; Yousefi, B.H.; Dallinger, D.; Walla, P.; Van der Eycken, E.; Kaval, N.; Kappe, C.O. Org. Process Res. Develop., 2003, 7, 707.
-
(2003)
Org. Process Res. Develop
, vol.7
, pp. 707
-
-
Stadler, A.1
Yousefi, B.H.2
Dallinger, D.3
Walla, P.4
Van der Eycken, E.5
Kaval, N.6
Kappe, C.O.7
-
35
-
-
25144446828
-
-
(d) Loones, K.T.J.; Maes, B. U.W.; Rombouts, G.; Hostyna, S.; Diels, G. Tetrahedron, 2005, 61, 10338.
-
(2005)
Tetrahedron
, vol.61
, pp. 10338
-
-
Loones, K.T.J.1
Maes, B.U.W.2
Rombouts, G.3
Hostyna, S.4
Diels, G.5
-
36
-
-
33947208419
-
-
(e) Díaz-Ortiz, A.; de la Hoz, A.; Alcázar, J.; Carrillo, J.R.; Herrero, M.A.; Fontana, A.; Muñoz, J.M. Comb. Chem. High Throughput Screen., 2007, 10, 163.
-
(2007)
Comb. Chem. High Throughput Screen
, vol.10
, pp. 163
-
-
Díaz-Ortiz, A.1
de la Hoz, A.2
Alcázar, J.3
Carrillo, J.R.4
Herrero, M.A.5
Fontana, A.6
Muñoz, J.M.7
-
37
-
-
0035674634
-
-
(a) Caliendo, G.; Fiorino, F.; Perissutti, E.; Severino, B.; Gessi, S.; Cattabriga, E.; Borea, P.A.; Santagada, V. Eur. J. Med. Chem., 2001, 36, 873.
-
(2001)
Eur. J. Med. Chem
, vol.36
, pp. 873
-
-
Caliendo, G.1
Fiorino, F.2
Perissutti, E.3
Severino, B.4
Gessi, S.5
Cattabriga, E.6
Borea, P.A.7
Santagada, V.8
-
38
-
-
0036020059
-
-
(b) Caliendo, G.; Fiorino, F.; Perissutti, E.; Severino, B.; Scolaro, D.; Gessi, S.; Cattabriga, E.; Borea, P.A.; Santagada, V. Eur. J. Pharm. Sci., 2002, 16, 15.
-
(2002)
Eur. J. Pharm. Sci
, vol.16
, pp. 15
-
-
Caliendo, G.1
Fiorino, F.2
Perissutti, E.3
Severino, B.4
Scolaro, D.5
Gessi, S.6
Cattabriga, E.7
Borea, P.A.8
Santagada, V.9
-
39
-
-
5144228817
-
-
Cotas, S.J.; Schulz, M.J.; Carson, J.R.; Codd, E.E.; Hlasta, D.J.; Pitis, P.M.; Stone, D.J.; Zhang, S.P.; Colburn, R.W.; Dax, S.L. Biorg. Med. Chem. Lett., 2004, 14, 5493.
-
(2004)
Biorg. Med. Chem. Lett
, vol.14
, pp. 5493
-
-
Cotas, S.J.1
Schulz, M.J.2
Carson, J.R.3
Codd, E.E.4
Hlasta, D.J.5
Pitis, P.M.6
Stone, D.J.7
Zhang, S.P.8
Colburn, R.W.9
Dax, S.L.10
-
40
-
-
4644248658
-
-
Caliendo, G.; Perissutti, E.; Santagada, V.; Fiorino, F.; Severino, B.; Cirillo, D.; d'Emmanuele de Villa Bianca, R.; Loppolis, L.; Pinto, A.; Sorrentino, R. Eur. J. Med. Chem., 2004, 39, 815.
-
(2004)
Eur. J. Med. Chem
, vol.39
, pp. 815
-
-
Caliendo, G.1
Perissutti, E.2
Santagada, V.3
Fiorino, F.4
Severino, B.5
Cirillo, D.6
d'Emmanuele de Villa Bianca, R.7
Loppolis, L.8
Pinto, A.9
Sorrentino, R.10
-
41
-
-
0033598384
-
-
(a) Alterman, M.; Andersson, H.O.; Garg, N.; Ahlsen, G.; Loevgren, S.; Classon, B.; Danielson, U.H.; Kvarnstroem, I.; Vrang, L.; Unge, T.; Samuelsson, B.; Hallberg, A. J. Med. Chem., 1999, 42, 3835;
-
(1999)
J. Med. Chem
, vol.42
, pp. 3835
-
-
Alterman, M.1
Andersson, H.O.2
Garg, N.3
Ahlsen, G.4
Loevgren, S.5
Classon, B.6
Danielson, U.H.7
Kvarnstroem, I.8
Vrang, L.9
Unge, T.10
Samuelsson, B.11
Hallberg, A.12
-
42
-
-
22844442612
-
-
(b) Wannberg, J.; Kaiser, N.F.K.; Vrang, L.; Samuelsson, B.; Larhed, M.; Hallberg, A. J. Comb. Chem., 2005, 7, 611;
-
(2005)
J. Comb. Chem
, vol.7
, pp. 611
-
-
Wannberg, J.1
Kaiser, N.F.K.2
Vrang, L.3
Samuelsson, B.4
Larhed, M.5
Hallberg, A.6
-
43
-
-
33745179573
-
-
(c) Wannberg, J.; Sabnis, Y.A.; Vrang, L.; Samuelsson, B.; Karlén, A.; Hallberg, A.; Larhed, M. Biorg. Med. Chem., 2006, 14, 5303.
-
(2006)
Biorg. Med. Chem
, vol.14
, pp. 5303
-
-
Wannberg, J.1
Sabnis, Y.A.2
Vrang, L.3
Samuelsson, B.4
Karlén, A.5
Hallberg, A.6
Larhed, M.7
-
45
-
-
29144440875
-
-
Manetti, F.; Este, J.A.; Clotet-Codina, I.; Armand-Ugon, M.; Maga, G.; Crespan, E.; Cancio, R.; Mugnaini, C.; Bernardini, C.; Togninelli, A.; Carmi, C.; Alongi, M.; Petricci, E.; Massa, S.; Corelli, F.; Botta, M. J. Med. Chem., 2005, 48, 8000.
-
(2005)
J. Med. Chem
, vol.48
, pp. 8000
-
-
Manetti, F.1
Este, J.A.2
Clotet-Codina, I.3
Armand-Ugon, M.4
Maga, G.5
Crespan, E.6
Cancio, R.7
Mugnaini, C.8
Bernardini, C.9
Togninelli, A.10
Carmi, C.11
Alongi, M.12
Petricci, E.13
Massa, S.14
Corelli, F.15
Botta, M.16
-
46
-
-
9144243695
-
-
Ersmark, K.; Feierberg, I.; Bjelic, S.; Hamelink, E.; Hackett, F.; Blackman, M.J.; Hulten, J.; Samuelsson, B.; Qvist, J.; Hallberg, A. J. Med. Chem., 2004, 47, 110.
-
(2004)
J. Med. Chem
, vol.47
, pp. 110
-
-
Ersmark, K.1
Feierberg, I.2
Bjelic, S.3
Hamelink, E.4
Hackett, F.5
Blackman, M.J.6
Hulten, J.7
Samuelsson, B.8
Qvist, J.9
Hallberg, A.10
-
47
-
-
21144448631
-
-
Souers, A.J.; Gao, J.; Wodka, D.; Judd, A.S.; Mulhern, M.M.; Napier, J.J.; Brune, M.E.; Bush, E.N.; Brodjian, S.J.; Dayton, B.D.; Shapiro, R.; Hernandez, L.E.; Marsh, K.C.; Sham, H.L.; Collins, C.A.; Kym, P.R. Bioorg. Med. Chem. Lett., 2005, 15, 2752.
-
(2005)
Bioorg. Med. Chem. Lett
, vol.15
, pp. 2752
-
-
Souers, A.J.1
Gao, J.2
Wodka, D.3
Judd, A.S.4
Mulhern, M.M.5
Napier, J.J.6
Brune, M.E.7
Bush, E.N.8
Brodjian, S.J.9
Dayton, B.D.10
Shapiro, R.11
Hernandez, L.E.12
Marsh, K.C.13
Sham, H.L.14
Collins, C.A.15
Kym, P.R.16
-
48
-
-
33749005650
-
-
Manetti, F.; Magnani, M.; Castagnolo, D.; Passalacqua, L.; Botta, M.; Corelli, F.; Saddi, M.; Deidda, D.; and De Logu, A.: ChemMedChem, 2006, 1, 973
-
(2006)
ChemMedChem
, vol.1
, pp. 973
-
-
Manetti, F.1
Magnani, M.2
Castagnolo, D.3
Passalacqua, L.4
Botta, M.5
Corelli, F.6
Saddi, M.7
Deidda, D.8
De Logu, A.9
-
49
-
-
20944432485
-
-
Kutterer, K.M.; K., Davis, J.M.; Singh, G.; Yang, Y.; Hu, W.; Severin, A.; Rasmussen, B.A.; Krishnamurthy, G.; Failli, A.; Katz, A.H. Bioorg. Med. Chem. Lett., 2005, 15, 2527.
-
Kutterer, K.M.; K., Davis, J.M.; Singh, G.; Yang, Y.; Hu, W.; Severin, A.; Rasmussen, B.A.; Krishnamurthy, G.; Failli, A.; Katz, A.H. Bioorg. Med. Chem. Lett., 2005, 15, 2527.
-
-
-
-
50
-
-
31544457663
-
-
Liu, J.-F.; Kaselj, M.; Isome, Y.; Ye, P.; Sargent, K.; Sprague, K.; Cherrak, D.; Wilson, C. J.; Si, Y.; Yohannes, D.; Ng, S.-C. J. Comb. Chem., 2006, 8, 7.
-
(2006)
J. Comb. Chem
, vol.8
, pp. 7
-
-
Liu, J.-F.1
Kaselj, M.2
Isome, Y.3
Ye, P.4
Sargent, K.5
Sprague, K.6
Cherrak, D.7
Wilson, C.J.8
Si, Y.9
Yohannes, D.10
Ng, S.-C.11
-
51
-
-
33744798761
-
-
Gong, Y.; Barbay, J.K.; Dyatkin, A.B.; Miskowski, T.A.; Kimball, E.S.; Prouty, S.M.; Fisher, M.C.; Santulli, R.J.; Scheneider, C.R.; Wallace, N.H.; Ballentine, S.A.; Hageman, W.E.; Masucci, J.A.; Maryanoff, B.E.; Damiano, B.P.; Andrade-Gordon, P.; Hlasta, D.J.; Hornby, P.J.; He, W. J. Med. Chem., 2006, 49, 3402.
-
(2006)
J. Med. Chem
, vol.49
, pp. 3402
-
-
Gong, Y.1
Barbay, J.K.2
Dyatkin, A.B.3
Miskowski, T.A.4
Kimball, E.S.5
Prouty, S.M.6
Fisher, M.C.7
Santulli, R.J.8
Scheneider, C.R.9
Wallace, N.H.10
Ballentine, S.A.11
Hageman, W.E.12
Masucci, J.A.13
Maryanoff, B.E.14
Damiano, B.P.15
Andrade-Gordon, P.16
Hlasta, D.J.17
Hornby, P.J.18
He, W.19
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