Synthesis by microwave irradiation of a substituted benzoxazine parallel library with preferential relaxant activity for guinea pig trachealis

European Journal of Medicinal Chemistry

Volumn 39, Issue 10, 2004, Pages 815-826

  Caliendo, Giuseppe ^a   Perissutti, Elisa ^a   Santagada, Vincenzo ^a   Fiorino, Ferdinando ^a   Severino, Beatrice ^a   Cirillo, Donatella ^a   D'Emmanuele Di Villa Bianca, Roberta ^a   Lippolis, Laura ^b   Pinto, Aldo ^b   Sorrentino, Raffaella ^a  

^a UNIVERSITY OF NAPLES FEDERICO II   (Italy)

^b UNIVERSITY OF SALERNO   (Italy)

Author keywords

ATP sensitive potassium channels; Benzoxazine; Microwave; Parallel synthesis; Relaxant activity

Indexed keywords

BENZOXAZINE DERIVATIVE; CARBACHOL; CROMAKALIM; PHENYLEPHRINE; POTASSIUM CHANNEL STIMULATING AGENT;

ANIMAL TISSUE; AORTA; ARTICLE; CHEMICAL REACTION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG EFFECT; DRUG SYNTHESIS; GUINEA PIG; MICROWAVE IRRADIATION; NONHUMAN; REACTION ANALYSIS; SMOOTH MUSCLE RELAXATION; TRACHEA; VASODILATATION;

ANIMALS; AORTA; BENZOXAZINES; GUINEA PIGS; MALE; MICROWAVES; MUSCLE RELAXATION; RATS; RATS, WISTAR; TRACHEA; VASODILATION;

EID: 4644248658     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejmech.2004.05.003     Document Type: Article

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