-
1
-
-
0032576426
-
-
Mocroft, A.; Vella, S.; Benfield, T. L.; Chiesi, A.; Miller, V.; Gargalianos, P.; d'Arminio Monforte, A.; Yust, I.; Bruun, J. N.; Phillips, A. N.; Lundgren, J. D. Lancet 1998, 352, 1725-1730.
-
(1998)
Lancet
, vol.352
, pp. 1725-1730
-
-
Mocroft, A.1
Vella, S.2
Benfield, T.L.3
Chiesi, A.4
Miller, V.5
Gargalianos, P.6
D'Arminio Monforte, A.7
Yust, I.8
Bruun, J.N.9
Phillips, A.N.10
Lundgren, J.D.11
-
2
-
-
2642709177
-
-
Palella, F. J., Jr.; Delaney, K. M.; Moorman, A. C.; Loveless, M. O.; Fuhrer, J.; Satten, G. A.; Aschman, D. J.; Holmberg, S. D. N. Engl. J. Med. 1998, 338, 853-860.
-
(1998)
N. Engl. J. Med.
, vol.338
, pp. 853-860
-
-
Palella Jr., F.J.1
Delaney, K.M.2
Moorman, A.C.3
Loveless, M.O.4
Fuhrer, J.5
Satten, G.A.6
Aschman, D.J.7
Holmberg, S.D.8
-
4
-
-
0035922595
-
-
Fellay, J.; Boubaker, K.; Ledergerber, B.; Bernasconi, E.; Furrer, H.; Battegay, M.; Hirschel, B.; Vernazza, P.; Francioli, P.; Greub, G.; Flepp, M.; Telenti, A. Lancet 2001, 358, 1322-1327.
-
(2001)
Lancet
, vol.358
, pp. 1322-1327
-
-
Fellay, J.1
Boubaker, K.2
Ledergerber, B.3
Bernasconi, E.4
Furrer, H.5
Battegay, M.6
Hirschel, B.7
Vernazza, P.8
Francioli, P.9
Greub, G.10
Flepp, M.11
Telenti, A.12
-
5
-
-
4744361049
-
-
UNAIDS, Geneva
-
Joint United Nations Programme on HIV/AIDS (UNAIDS). 2004 Report on the Global AIDS Epidemic. http://www.unaids.org (UNAIDS, Geneva, 2004).
-
(2004)
2004 Report on the Global AIDS Epidemic
-
-
-
6
-
-
14444280615
-
-
Alterman, M.; Björsne, M.; Mühlman, A.; Classon, B.; Kvarnström, I.; Danielson, H.; Markgren, P. O.; Nillroth, U.; Unge, T.; Hallberg, A.; Samuelsson, B. J. Med. Chem. 1998, 41, 3782-3792.
-
(1998)
J. Med. Chem.
, vol.41
, pp. 3782-3792
-
-
Alterman, M.1
Björsne, M.2
Mühlman, A.3
Classon, B.4
Kvarnström, I.5
Danielson, H.6
Markgren, P.O.7
Nillroth, U.8
Unge, T.9
Hallberg, A.10
Samuelsson, B.11
-
7
-
-
0033598384
-
-
Alterman, M.; Andersson, H. O.; Garg, N.; Ahlsen, G.; Lövgren, S.; Classon, B.; Danielson, U. H.; Kvarnström, I.; Vrang, L.; Unge, T.; Samuelsson, B.; Hallberg, A. J. Med. Chem. 1999, 42, 3835-3844.
-
(1999)
J. Med. Chem.
, vol.42
, pp. 3835-3844
-
-
Alterman, M.1
Andersson, H.O.2
Garg, N.3
Ahlsen, G.4
Lövgren, S.5
Classon, B.6
Danielson, U.H.7
Kvarnström, I.8
Vrang, L.9
Unge, T.10
Samuelsson, B.11
Hallberg, A.12
-
8
-
-
8444233969
-
-
Morimoto, T.; Kakiuchi, K. Angew. Chem., Int. Ed. 2004, 43, 5580-5588.
-
(2004)
Angew. Chem., Int. Ed.
, vol.43
, pp. 5580-5588
-
-
Morimoto, T.1
Kakiuchi, K.2
-
9
-
-
0036514950
-
-
Kaiser, N.-F. K.; Hallberg, A.; Larhed, M. J. Comb. Chem. 2002, 4, 109-111.
-
(2002)
J. Comb. Chem.
, vol.4
, pp. 109-111
-
-
Kaiser, N.-F.K.1
Hallberg, A.2
Larhed, M.3
-
12
-
-
0036738330
-
-
Larhed, M.; Moberg, C.; Hallberg, A. Acc. Chem. Res. 2002, 35, 717-727.
-
(2002)
Acc. Chem. Res.
, vol.35
, pp. 717-727
-
-
Larhed, M.1
Moberg, C.2
Hallberg, A.3
-
13
-
-
4644273521
-
-
Ersmark, K.; Larhed, M.; Wannberg, J. Curr. Opin. Drug Discovery Devel. 2004, 7, 417-427.
-
(2004)
Curr. Opin. Drug Discovery Devel.
, vol.7
, pp. 417-427
-
-
Ersmark, K.1
Larhed, M.2
Wannberg, J.3
-
14
-
-
22844452022
-
-
In press
-
Wannberg, J.; Dallinger, D.; Kappe, C. O.; Larhed, M. J. Comb. Chem. 2005, 7, In press.
-
(2005)
J. Comb. Chem.
, pp. 7
-
-
Wannberg, J.1
Dallinger, D.2
Kappe, C.O.3
Larhed, M.4
-
16
-
-
33750236967
-
-
Herrmann, W. A.; Brossmer, C.; Öfele, K.; Reisinger, C. P.; Priermeier, T.; Beller, M.; Fischer, H. Angew. Chem., Int. Ed. 1995, 34, 1844-1848.
-
(1995)
Angew. Chem., Int. Ed.
, vol.34
, pp. 1844-1848
-
-
Herrmann, W.A.1
Brossmer, C.2
Öfele, K.3
Reisinger, C.P.4
Priermeier, T.5
Beller, M.6
Fischer, H.7
-
18
-
-
22844451537
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-
note
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Employing the o-iodo starting material 4, competing mono dehalogenation resulted in small amounts (<10%) of non-symmetric monoamidation products.
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19
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22844448144
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note
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Full conversion of 10 was not achieved with 3-chloroaniline as the nucleophile, which explains the relatively low isolated yield of 61 (24%).
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20
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22844448612
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note
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No traces of inhibitor 4 or the corresponding dehalogenated arene was detected by LC/MS or NMR of the purified compounds.
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-
-
-
21
-
-
0031944861
-
-
Danielson, H.; Lindgren, M. T.; Markgren, P. O.; Nillroth, U. Adv. Exp. Med. Biol. 1998, 436, 99-103.
-
(1998)
Adv. Exp. Med. Biol.
, vol.436
, pp. 99-103
-
-
Danielson, H.1
Lindgren, M.T.2
Markgren, P.O.3
Nillroth, U.4
-
22
-
-
0030664454
-
-
Nillroth, U.; Vrang, L.; Markgren, P. O.; Hulten, J.; Hallberg, A.; Danielson, U. H. Antimicrob. Agents Chemother. 1997, 41, 2383-2388.
-
(1997)
Antimicrob. Agents Chemother.
, vol.41
, pp. 2383-2388
-
-
Nillroth, U.1
Vrang, L.2
Markgren, P.O.3
Hulten, J.4
Hallberg, A.5
Danielson, U.H.6
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