-
6
-
-
0032732615
-
-
77er(1999) 291:1204-1209.
-
Kim RB, Leake B, Cvetkovic M, Roden MM, Nadeau J, Walubo A, Wilkinson GR: Modulation by drugs of human hepatic sodium-dependent bile acid transporter (sodium taurocholate cotransporting polypeptlde) activity. J PharmacolExp 77)er(1999) 291:1204-1209.
-
Leake B, Cvetkovic M, Roden MM, Nadeau J, Walubo A, Wilkinson GR: Modulation by Drugs of Human Hepatic Sodium-dependent Bile Acid Transporter (Sodium Taurocholate Cotransporting Polypeptlde) Activity. J PharmacolExp
-
-
Kim, R.B.1
-
11
-
-
0029876335
-
-
(1996) 270:F326-F331.
-
Kanai N, Lu R, Bao Y, Wolkoff AW, Vore M, Schuster VL: Estradiol 17-D-glucuronide is a high-affinity substrate for oatp organic anion transporter. Am J Physiol (1996) 270:F326-F331.
-
Lu R, Bao Y, Wolkoff AW, Vore M, Schuster VL: Estradiol 17-D-glucuronide Is A High-affinity Substrate for Oatp Organic Anion Transporter. Am J Physiol
-
-
Kanai, N.1
-
14
-
-
15844387507
-
-
(1996) 24:380-384.
-
Eckhardt U, Horz JA, Petzinger E, Stüber W, Reers M, Dickneite G, Daniel H, Wagener M, Hagenbuch B, Stieger B, Meier PJ: The peptide-based thrombin inhibitor CRC 220 is a new substrate of the basolateral rat liver organic aniontransporting polypeptide. Hepatology (1996) 24:380-384.
-
Horz JA, Petzinger E, Stüber W, Reers M, Dickneite G, Daniel H, Wagener M, Hagenbuch B, Stieger B, Meier PJ: the Peptide-based Thrombin Inhibitor CRC 220 Is A New Substrate of the Basolateral Rat Liver Organic Aniontransporting Polypeptide. Hepatology
-
-
Eckhardt, U.1
-
19
-
-
15444342300
-
-
(1998) 273:22395-22401.
-
Abe T, Kakyo M, Sakagami H, Tokui T, Nishio T, Tanemoto M, Nomura H, Hebert SC, Matsuno S, Kondo H, Yawo H: Molecular characterization and tissue distribution of a new organic anion transporter subtype (Oatp3) that transports thyroid hormones and taurocholate and comparison with Oatp2. J Biol Chem (1998) 273:22395-22401.
-
Kakyo M, Sakagami H, Tokui T, Nishio T, Tanemoto M, Nomura H, Hebert SC, Matsuno S, Kondo H, Yawo H: Molecular Characterization and Tissue Distribution of A New Organic Anion Transporter Subtype (Oatp3) That Transports Thyroid Hormones and Taurocholate and Comparison with Oatp2. J Biol Chem
-
-
Abe, T.1
-
20
-
-
0040368659
-
-
Chem (1999)274:17159-17163.
-
Abe T, Kakyo M, Tokui T, Nakagomi R, Nishio T, Nakai D, Nomura H, Unno M, Suzuki M, Naitoh T, Matsuno S, Yawo H: Identification of a novel gene family encoding human liverspecific organic anion transporter LST-1. J Biol Chem (1999)274:17159-17163.
-
Kakyo M, Tokui T, Nakagomi R, Nishio T, Nakai D, Nomura H, Unno M, Suzuki M, Naitoh T, Matsuno S, Yawo H: Identification of A Novel Gene Family Encoding Human Liverspecific Organic Anion Transporter LST-1. J Biol
-
-
Abe, T.1
-
21
-
-
85119810909
-
-
(1999) 117:770-775.
-
Kakyo M, Unno M, Tokui T, Nakagomi R, Nishio T, Iwasashi H, Nakai D, Seki M, Suzuki M, Naitoh T, Matsuno S, Yawo H, Abe T: Molecular characterization and functional regulation of a novel rat liver-specific organic anion transporter rlst-1. Gastroenterology (1999) 117:770-775.
-
Unno M, Tokui T, Nakagomi R, Nishio T, Iwasashi H, Nakai D, Seki M, Suzuki M, Naitoh T, Matsuno S, Yawo H, Abe T: Molecular Characterization and Functional Regulation of A Novel Rat Liver-specific Organic Anion Transporter Rlst-1. Gastroenterology
-
-
Kakyo, M.1
-
23
-
-
0029078231
-
-
Sc/ence(1995) 268:866-869.
-
Kanai N, Lu R, Satriano JA, Bao Y, Wolkoff AW, Schuster VL: Identification and characterization of a prostaglandin transporter. Sc/ence(1995) 268:866-869.
-
Lu R, Satriano JA, Bao Y, Wolkoff AW, Schuster VL: Identification and Characterization of A Prostaglandin Transporter.
-
-
Kanai, N.1
-
24
-
-
0029739973
-
-
(1996) 98:1142-1149.
-
Lu R, Kanai N, Bao Y, Schuster VL: Cloning, in vitro expression, and tissue distribution of a human prostaglandin transporter cDNA (hPGT). J Clin Invest (1996) 98:1142-1149.
-
Kanai N, Bao Y, Schuster VL: Cloning, in Vitro Expression, and Tissue Distribution of A Human Prostaglandin Transporter CDNA (HPGT). J Clin Invest
-
-
Lu, R.1
-
26
-
-
0028333611
-
-
/Vafure(1994) 368:563-566.
-
Fei Y-J, Kanai Y, Nussberger S, Ganapathy V, Leibach FH, Romero MF, Singh SK, Boron WF, Hediger MA: Expression cloning of a mammalian proton-coupled oligopeptide transporter. /Vafure(1994) 368:563-566.
-
Kanai Y, Nussberger S, Ganapathy V, Leibach FH, Romero MF, Singh SK, Boron WF, Hediger MA: Expression Cloning of A Mammalian Proton-coupled Oligopeptide Transporter.
-
-
Fei, Y.-J.1
-
27
-
-
0028920129
-
-
Chem (1995)270:6456-6463.
-
Liang R, Fei Y-J, Prasad PD, Ramamoorthy S, Han H, YangFeng TL, Hediger MA, Ganapathy V, Leibach FH: Human intestinal H'/peptide cotransporter. Cloning, functional expression, and chromosomal localization. J Biol Chem (1995)270:6456-6463.
-
Fei Y-J, Prasad PD, Ramamoorthy S, Han H, YangFeng TL, Hediger MA, Ganapathy V, Leibach FH: Human Intestinal H'/peptide Cotransporter. Cloning, Functional Expression, and Chromosomal Localization. J Biol
-
-
Liang, R.1
-
30
-
-
0027363563
-
-
(1993) 75:451-462.
-
Smit JJ, Schinkel AH, Oude Elferink RP, Groen AK, Wagenaar E, van Deemter L, Mol CA, Ottenhoff R, van der Lugt NM, van Roon MA, van der Valk MA, Offerhaus GJA, Berns AJ, Borst P: Homozygous disruption of the murine mdr2 P-glycoprotein gene leads to a complete absence of phospholipid from bile and to liver disease. Cell (1993) 75:451-462.
-
Schinkel AH, Oude Elferink RP, Groen AK, Wagenaar E, Van Deemter L, Mol CA, Ottenhoff R, Van der Lugt NM, Van Roon MA, Van der Valk MA, Offerhaus GJA, Berns AJ, Borst P: Homozygous Disruption of the Murine Mdr2 P-glycoprotein Gene Leads to A Complete Absence of Phospholipid from Bile and to Liver Disease. Cell
-
-
Smit, J.J.1
-
31
-
-
0000712439
-
-
(1989) 86:695-698.
-
Cordon-Cardo C, O'Brien JP, Casals D, Rittman-Grauer L, Biedier JL, Melarned MR, Bertino JR: Multidrug-resistance gene (Pglycoprotein) is expressed by endothelial cells at blood-brain barrier sites. Proc Nail Acad Sci USA (1989) 86:695-698.
-
O'Brien JP, Casals D, Rittman-Grauer L, Biedier JL, Melarned MR, Bertino JR: Multidrug-resistance Gene (Pglycoprotein) Is Expressed by Endothelial Cells at Blood-brain Barrier Sites. Proc Nail Acad Sci USA
-
-
Cordon-Cardo, C.1
-
33
-
-
0032907322
-
-
(1999) 16:408-414.
-
Kim RB, Wandel C, Leake B, Cvetkovic M, Fromm MF, Dempsey PJ, Roden MM, Belas F, Chaudhary AK, Roden DM, Wood AJ, Wilkinson GR: Interrelationship between substrates and inhibitors of human CYP3A and Pglycoprotein. Pharm Res (1999) 16:408-414.
-
Wandel C, Leake B, Cvetkovic M, Fromm MF, Dempsey PJ, Roden MM, Belas F, Chaudhary AK, Roden DM, Wood AJ, Wilkinson GR: Interrelationship between Substrates and Inhibitors of Human CYP3A and Pglycoprotein. Pharm Res
-
-
Kim, R.B.1
-
36
-
-
0032518290
-
-
(1998) 101:289-294.
-
Kim RB, Fromm MF, Wandel C, Leake B, Wood AJ, Roden DM, Wilkinson GR: The drug transporter P-glycoprotein limits oral absorption and brain entry of HIV-1 protease Inhibitors. J Clin Invest (1998) 101:289-294.
-
Fromm MF, Wandel C, Leake B, Wood AJ, Roden DM, Wilkinson GR: the Drug Transporter P-glycoprotein Limits Oral Absorption and Brain Entry of HIV-1 Protease Inhibitors. J Clin Invest
-
-
Kim, R.B.1
-
38
-
-
0028229150
-
-
77:491 -502.
-
Schinkel AH, Smit JJ, van Tellingen O, Beijnen JH, Wagenaar E, van Deemter L, Mol ÇA, van der Valk MA, RobanusMaandag EC, Riele HPJ, Berns AJ, Borst P: Disruption of the mouse mdrla P-glycoprotein gene leads to a deficiency in the blood-brain barrier and to increased sensitivity to drugs. Cell (1994) 77:491 -502.
-
Smit JJ, Van Tellingen O, Beijnen JH, Wagenaar E, Van Deemter L, Mol ÇA, Van der Valk MA, RobanusMaandag EC, Riele HPJ, Berns AJ, Borst P: Disruption of the Mouse Mdrla P-glycoprotein Gene Leads to A Deficiency in the Blood-brain Barrier and to Increased Sensitivity to Drugs. Cell (1994)
-
-
Schinkel, A.H.1
-
40
-
-
0028825399
-
-
(1995) 96:1698-1705.
-
Schinkel AH, Wagenaar E, van Deemter L, Mol CA, Borst P: Absence of the mdrla P-glycoprotein in mice affects tissue distribution and pharmacokinetics of dexamethasone, digoxin, and cyclosporin A. J Clin /nvesf (1995) 96:1698-1705.
-
Wagenaar E, Van Deemter L, Mol CA, Borst P: Absence of the Mdrla P-glycoprotein in Mice Affects Tissue Distribution and Pharmacokinetics of Dexamethasone, Digoxin, and Cyclosporin A. J Clin /Nvesf
-
-
Schinkel, A.H.1
-
46
-
-
0345411341
-
-
(1999) 59:3944-3948.
-
Wandel C, Kim RB, Kajiji S, Guengerich P, Guengerich FP, Wilkinson GR, Wood AJ: P-glycoprotein and cytochrome P450 3A inhibition: Dissociation of inhibitory potencies. Cancer Res (1999) 59:3944-3948.
-
Kim RB, Kajiji S, Guengerich P, Guengerich FP, Wilkinson GR, Wood AJ: P-glycoprotein and Cytochrome P450 3A Inhibition: Dissociation of Inhibitory Potencies. Cancer Res
-
-
Wandel, C.1
-
47
-
-
0029981430
-
-
(1996) 271:1126-1128.
-
Paulusma CC, Bosma PJ, Zaman GJ, Bakker CT, Otter M, Scheffer GL, Scheper RJ, Borst P, Oude Elferink RP: Congenital jaundice in rats with a mutation in a multidrug resistance-associated protein gene. Science (1996) 271:1126-1128.
-
Bosma PJ, Zaman GJ, Bakker CT, Otter M, Scheffer GL, Scheper RJ, Borst P, Oude Elferink RP: Congenital Jaundice in Rats with A Mutation in A Multidrug Resistance-associated Protein Gene. Science
-
-
Paulusma, C.C.1
-
48
-
-
0030994468
-
-
(1997) 25:1539-1542.
-
Paulusma CG, Kool M, Bosma PJ, Scheffer GL, ter Borg F, Scheper RJ, Tytgat GN, Borst P, Baas F, Oude Elferink RP: A mutation in the human canalicular multispecific organic anion transporter gène causes thé Dubin-Jonnson syndrome. Hepatology (1997) 25:1539-1542.
-
Kool M, Bosma PJ, Scheffer GL, ter Borg F, Scheper RJ, Tytgat GN, Borst P, Baas F, Oude Elferink RP: A Mutation in the Human Canalicular Multispecific Organic Anion Transporter Gène Causes thé Dubin-Jonnson Syndrome. Hepatology
-
-
Paulusma, C.G.1
-
50
-
-
0031866357
-
-
(1998) 53:1068-1075.
-
Hirohashi T, Suzuki H, Ito K, Ogawa K, Kume K, Shimizu T, Sugiyama Y: Hepatic expression of multidrug resistanceassociated protein-like proteins maintained in Eisal hyperbilirubinemic rats. Mol Pharmacol (1998) 53:1068-1075.
-
Suzuki H, Ito K, Ogawa K, Kume K, Shimizu T, Sugiyama Y: Hepatic Expression of Multidrug Resistanceassociated Protein-like Proteins Maintained in Eisal Hyperbilirubinemic Rats. Mol Pharmacol
-
-
Hirohashi, T.1
-
51
-
-
0032922395
-
-
(1999) 1415:369-374.
-
Fromm MF, Leake B, Roden DM, Wilkinson GR, Kim RB: Human MRP3 transporter: Identification of the S'-flanking region, genomic organization and alternative splice variants. Biochim Biophys Acta (1999) 1415:369-374.
-
Leake B, Roden DM, Wilkinson GR, Kim RB: Human MRP3 Transporter: Identification of the S'-flanking Region, Genomic Organization and Alternative Splice Variants. Biochim Biophys Acta
-
-
Fromm, M.F.1
-
53
-
-
0032540277
-
-
(1998) 273:1004610050.
-
Gerloff T, Stieger B, Hagenbuch B, Madon J, Landmann L, Roth J, Hofmann AF, Meier PJ: The sister of Pglycoprotein represents the canalicular bile salt export pump of mammalian liver. J Biol Chem (1998) 273:1004610050.
-
Stieger B, Hagenbuch B, Madon J, Landmann L, Roth J, Hofmann AF, Meier PJ: the Sister of Pglycoprotein Represents the Canalicular Bile Salt Export Pump of Mammalian Liver. J Biol Chem
-
-
Gerloff, T.1
-
54
-
-
17344366172
-
-
Genet (1998)20:233-238.
-
Strautnieks SS, Bull LN, Knisely AS, Kocoshis SA, Dahl N, Amell H, Sokal E, Dahan K, Childs S, Ling V, Tanner MS, Kagalwalla AF, Nemeth A, Pawlowska J, Baker A, MieliVergani G, Freimer NB, Gardiner RM, Thompson RJ: A gene encoding a liver-specific ABC transporter Is mutated in progressive familial intrahepatic cholestasis. Nature Genet (1998)20:233-238.
-
Bull LN, Knisely AS, Kocoshis SA, Dahl N, Amell H, Sokal E, Dahan K, Childs S, Ling V, Tanner MS, Kagalwalla AF, Nemeth A, Pawlowska J, Baker A, MieliVergani G, Freimer NB, Gardiner RM, Thompson RJ: A Gene Encoding A Liver-specific ABC Transporter Is Mutated in Progressive Familial Intrahepatic Cholestasis. Nature
-
-
Strautnieks, S.S.1
-
55
-
-
85119790707
-
-
(1999) 117:688-695.
-
Reichel C, Gao B, Van Montfoort J, Cattori V, Rahner C, Hagenbuch B, Stieger B, Kamisako T, Meier PJ: Localization and function of the organic aniontransporting polypeptide Oatp2 in rat liver. Gastroenterology (1999) 117:688-695.
-
Gao B, Van Montfoort J, Cattori V, Rahner C, Hagenbuch B, Stieger B, Kamisako T, Meier PJ: Localization and Function of the Organic Aniontransporting Polypeptide Oatp2 in Rat Liver. Gastroenterology
-
-
Reichel, C.1
-
56
-
-
0032813028
-
-
T/7er(1999) 290:1107-1115.
-
Akhteruzzaman S, Kato Y, Kouzuki H, Suzuki H, Hisaka A, Stieger B, Meier PJ, Sugiyama Y: Carrier-mediated hepatic uptake of peptidic endothelin antagonists in rats. J PharmacolExp T/7er(1999) 290:1107-1115.
-
Kato Y, Kouzuki H, Suzuki H, Hisaka A, Stieger B, Meier PJ, Sugiyama Y: Carrier-mediated Hepatic Uptake of Peptidic Endothelin Antagonists in Rats. J PharmacolExp
-
-
Akhteruzzaman, S.1
|