Carrier-mediated hepatic uptake of peptidic endothelin antagonists in rats

Journal of Pharmacology and Experimental Therapeutics

Volumn 290, Issue 3, 1999, Pages 1107-1115

  Akhteruzzaman, Sharif ^a   Kato, Yukio ^a   Kouzuki, Hirokazu ^a   Suzuki, Hiroshi ^a   Hisaka, Akihiro ^b   Stieger, Bruno ^c   Meier, Peter J ^c   Sugiyama, Yuichi ^a  

^a UNIVERSITY OF TOKYO   (Japan)

^b BANYU PHARMACEUTICAL CO LTD   (Japan)

^c UNIVERSITY HOSPITAL ZURICH   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

BQ 518; BQ 587; CYCLO(DEXTRO TRYPTOPHYL DEXTRO ASPARTYL HYDROXYPROLYL (N(ALPHA),N(EPSILON) DIMETHYL LYSINE) DEXTRO VALYLLEUCYL); CYCLO(DEXTRO TRYPTOPHYL DEXTRO ASPARTYLPROLYL DEXTRO 2 (2 THIENYL)GLYCINE; CYCLO(DEXTRO TRYPTOPHYL DEXTRO ASPARTYLPROLYL DEXTRO VALYLLEUCYL); ENDOTHELIN RECEPTOR ANTAGONIST; PERHYDRO 1 AZEPINYLCARBONYLLEUCYL DEXTRO TRYPTOPHYL DEXTRO TRYPTOPHAN; UNCLASSIFIED DRUG;

ACTIVE TRANSPORT; ANIMAL CELL; ARTICLE; COMPETITIVE INHIBITION; DRUG UPTAKE; ISOTOPE LABELING; LIVER CELL; MALE; NONHUMAN; PEPTIDE ANALYSIS; PRIORITY JOURNAL; RAT; RECEPTOR BLOCKING; VASCULAR ENDOTHELIUM;

ANESTHETICS, INHALATION; ANIMALS; ANTIHYPERTENSIVE AGENTS; AZEPINES; BINDING, COMPETITIVE; BIOLOGICAL TRANSPORT, ACTIVE; CARRIER PROTEINS; CELLS, CULTURED; COS CELLS; ETHERS; HYDROCARBONS, FLUORINATED; KINETICS; LIVER; MALE; OLIGOPEPTIDES; PEPTIDES; PEPTIDES, CYCLIC; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, ENDOTHELIN; TRANSFECTION;

EID: 0032813028     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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