Erratum: Corrigendum to "development of methyl isoxazoleazepines as inhibitors of BET" [Bioorganic and Medicinal Chemistry Letters (2015) 25 9 (1842-1848) 10.1016/j.bmcl.2015.03.045];Development of methyl isoxazoleazepines as inhibitors of BET

Bioorganic and Medicinal Chemistry Letters

Volumn 25, Issue 9, 2015, Pages 1842-1848

  Hewitt, Michael C ^a   Leblanc, Yves ^a   Gehling, Victor S ^a   Vaswani, Rishi G ^a   Côté, Alexandre ^a   Nasveschuk, Christopher G ^a   Taylor, Alexander M ^a   Harmange, Jean Christophe ^a   Audia, James E ^a   Pardo, Eneida ^a   Cummings, Rich ^a   Joshi, Shivangi ^a   Sandy, Peter ^a   Mertz, Jennifer A ^a   Sims, Robert J ^a   Bergeron, Louise ^a   Bryant, Barbara M ^a   Bellon, Steve ^a   Poy, Florence ^a   Jayaran, Hariharan ^a   Tang, Yong ^a   Albrecht, Brian K ^a   more..

^a Department of Structural Biology   (United States)

Author keywords

BET inhibitors; Bromodomains; Isoxazoles; MYC; Unbound clearance

Indexed keywords

AZEPINE DERIVATIVE; BRD2 PROTEIN, HUMAN; BRD3 PROTEIN, HUMAN; BRD4 PROTEIN, HUMAN; BRDT PROTEIN, HUMAN; METHYL ISOXAZOLEAZEPINE; NUCLEAR PROTEIN; OXAZOLE DERIVATIVE; PROTEIN SERINE THREONINE KINASE; RNA BINDING PROTEIN; TRANSCRIPTION FACTOR;

ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; CHEMISTRY; DOSE RESPONSE; DRUG DESIGN; HUMAN; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

AZEPINES; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DESIGN; HUMANS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; NUCLEAR PROTEINS; OXAZOLES; PROTEIN-SERINE-THREONINE KINASES; RNA-BINDING PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP; TRANSCRIPTION FACTORS;

EID: 84937762548     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2015.06.064     Document Type: Erratum

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