SCOPUS 정보 검색 플랫폼

Volumn 4, Issue 1, 2013, Pages 140-144

The design and synthesis of 5- and 6-isoxazolylbenzimidazoles as selective inhibitors of the BET bromodomains

(12) Hay, Duncan a Fedorov, Oleg a Filippakopoulos, Panagis a Martin, Sarah a Philpott, Martin a Picaud, Sarah a Hewings, David S b Uttakar, Sagar a Heightman, Tom D a Conway, Stuart J b Knapp, Stefan a Brennan, Paul E a

a UNIVERSITY OF OXFORD (United Kingdom)

b UNIVERSITY OF OXFORD (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

5 ISOXAZOLYLBENZIMIDAZOLE DERIVATIVE; 6 ISOXAZOLYLBENZIMIDAZOLE DERIVATIVE; BENZIMIDAZOLE DERIVATIVE; BROMODOMAIN CONTAINING PROTEIN; IBET 762; JQ 1; PROTEIN DERIVATIVE; PROTEIN INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG DESIGN; DRUG POTENCY; DRUG SELECTIVITY; DRUG SYNTHESIS; PRIORITY JOURNAL; PROTEIN DOMAIN;

EID: 84871738620 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c2md20189e Document Type: Article

Times cited : (63)

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