Improving the apo-state detergent stability of NTS1 with CHESS for pharmacological and structural studies

Biochimica et Biophysica Acta - Biomembranes

Volumn 1838, Issue 11, 2014, Pages 2817-2824

  Scott, Daniel J ^a,b   Kummer, Lutz ^a   Egloff, Pascal ^a   Bathgate, Ross A D ^b   Plückthun, Andreas ^a  

^a UNIVERSITY OF ZURICH   (Switzerland)

^b UNIVERSITY OF MELBOURNE   (Australia)

Author keywords

Detergent; Directed evolution; Encapsulation; G protein coupled receptor; Stabilization; Thermostability

Indexed keywords

DETERGENT; G PROTEIN COUPLED RECEPTOR; NEUROTENSIN RECEPTOR; NEUROTENSIN RECEPTOR 1; UNCLASSIFIED DRUG;

ARTICLE; CELL ENCAPSULATION; CELLULAR HIGH THROUGHPUT ENCAPSULATION SOLUBILIZATION AND SCREENING; CONTROLLED STUDY; CRYSTAL STRUCTURE; DRUG DEVELOPMENT; FEASIBILITY STUDY; HIGH THROUGHPUT SCREENING; HUMAN; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING ASSAY; SOLUBILIZATION; THERMOSTABILITY;

EID: 84905615352     PISSN: 00052736     EISSN: 18792642     Source Type: Journal    
DOI: 10.1016/j.bbamem.2014.07.015     Document Type: Article

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