Structural mechanism of ligand activation in human GABA B receptor

Nature

Volumn 504, Issue 7479, 2013, Pages 254-259

  Geng, Yong ^a   Bush, Martin ^a   Mosyak, Lidia ^a   Wang, Feng ^a   Fan, Qing R ^a,b  

^a Och Spine at New York Presbyterian Hospitals   (United States)

^b NewYork Presbyterian Hospital   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOBUTYRIC ACID B RECEPTOR; 4 AMINOBUTYRIC ACID B RECEPTOR 1; 4 AMINOBUTYRIC ACID B RECEPTOR 2; UNCLASSIFIED DRUG;

BIOCHEMISTRY; BRAIN; CRYSTAL STRUCTURE; HOMINID; INHIBITOR; LIGAND; NEUROLOGY; PHYSIOLOGY; PROTEIN;

ARTICLE; CONFORMATIONAL TRANSITION; CRYSTAL STRUCTURE; HUMAN; HUMAN CELL; PRIORITY JOURNAL;

APOPROTEINS; BINDING SITES; CRYSTALLOGRAPHY, X-RAY; DISULFIDES; GABA-B RECEPTOR AGONISTS; GABA-B RECEPTOR ANTAGONISTS; HUMANS; LIGANDS; MODELS, MOLECULAR; PROTEIN MULTIMERIZATION; PROTEIN STRUCTURE, TERTIARY; PROTEIN SUBUNITS; RECEPTORS, GABA-B; SUBSTRATE SPECIFICITY;

EID: 84890434896     PISSN: 00280836     EISSN: 14764687     Source Type: Journal    
DOI: 10.1038/nature12725     Document Type: Article

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