SCOPUS 정보 검색 플랫폼

Volumn 4, Issue 2, 2013, Pages 432-442

The advantage of biosensor analysis over enzyme inhibition studies for slow dissociating inhibitors-characterization of hydroxamate-based matrix metalloproteinase-12 inhibitors

(7) Gossas, Thomas a Nordström, Helena a Xu, Ming Hua b Sun, Zhi Hua c Lin, Guo Qiang c Wallberg, Hans d Danielson, U Helena a

a UPPSALA UNIVERSITY (Sweden)

b SHANGHAI INSTITUTE OF MATERIA MEDICA (China)

c SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY (China)

d MEDIVIR AB (Sweden)

Author keywords

[No Author keywords available]

Indexed keywords

2 (4 BROMOPHENETHYL) 4 TERT BUTOXY 4 OXOBUTANOIC ACID; 3 [1 (METHYLAMINO) 1 OXO 3 PHENYLPROPAN 2 YLCARBAMOYL] 5 [4 (PYRIDIN 3 YL)PHENYL]PENTANOIC ACID; 4 BENZYL 3 [4 (4 BROMOPHENYL)BUTANOYL]OXAZOLIDIN 2 ONE; CARBOXYLIC ACID DERIVATIVE; HYDROXAMIC ACID DERIVATIVE; ILOMASTAT; MACROPHAGE ELASTASE; MATRIX METALLOPROTEINASE 12 INHIBITOR; MATRIX METALLOPROTEINASE INHIBITOR; N4 HYDROXY N1 [1 (METHYLAMINO) 1 OXO 3 PHENYLPROPAN 2 YL] 2 [4 (PYRIDIN 3 YL)PHENETHYL]SUCCINAMIDE; TERT BUTYL 3 (4 BENZYL 2 OXOOXAZOLIDINE 3 CARBONYL) 5 (4 BROMOPHENYL)PENTANOATE; TERT BUTYL 3 [1 (METHYLAMINO) 1 OXO 3 PHENYLPROPAN 2 YLCARBAMOYL] 5 [4 (PYRIDIN 3 YL)PHENYL]PENTANOATE; TERT BUTYL 5 (4 BROMOPHENYL) 3 [1 (METHYLAMINO) 1 OXO 3 PHENYLPROPAN 2 YLCARBAMOYL]PENTANOATE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; BIOSENSOR; CONTROLLED STUDY; DISSOCIATION; DRUG POTENCY; DRUG SYNTHESIS; ENZYME INHIBITION; ENZYME KINETICS; HUMAN; IC 50; INTERMETHOD COMPARISON; PRIORITY JOURNAL; STEADY STATE;

EID: 84876724694 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c2md20268a Document Type: Article

Times cited : (8)

References (35)

1
- 0345864015
- N. D. Rawlings D. P. Tolle A. J. Barrett Nucleic Acids Res. 2004 32 D160 D164
- (2004) Nucleic Acids Res. , vol.32
- Rawlings, N.D.¹ Tolle, D.P.² Barrett, A.J.³

2
- 0037447192
- G. L. Snider Am. J. Respir. Crit. Care Med. 2003 167 1045 1046
- (2003) Am. J. Respir. Crit. Care Med. , vol.167 , pp. 1045-1046
- Snider, G.L.¹

3
- 5644277560
- M. Liu H. Sun X. Wang T. Koike H. Mishima K. Ikeda T. Watanabe N. Ochiai J. Fan Arthritis Rheum. 2004 50 3112 3117
- (2004) Arthritis Rheum. , vol.50 , pp. 3112-3117
- Liu, M.¹ Sun, H.² Wang, X.³ Koike, T.⁴ Mishima, H.⁵ Ikeda, K.⁶ Watanabe, T.⁷ Ochiai, N.⁸ Fan, J.⁹

4
- 33748308883
- B. Turk Nat. Rev. Drug Discovery 2006 5 785 799
- (2006) Nat. Rev. Drug Discovery , vol.5 , pp. 785-799
- Turk, B.¹

5
- 0037192458
- L. M. Coussens B. Fingleton L. M. Matrisian Science 2002 295 2387 2392
- (2002) Science , vol.295 , pp. 2387-2392
- Coussens, L.M.¹ Fingleton, B.² Matrisian, L.M.³

6
- 33645738383
- C. M. Overall O. Kleifeld Br. J. Cancer 2006 94 941 946
- (2006) Br. J. Cancer , vol.94 , pp. 941-946
- Overall, C.M.¹ Kleifeld, O.²

7
- 33644545381
- C. M. Overall O. Kleifeld Nat. Rev. Cancer 2006 6 227 239
- (2006) Nat. Rev. Cancer , vol.6 , pp. 227-239
- Overall, C.M.¹ Kleifeld, O.²

8
- 45749114201
- H. Nordström T. Gossas M. Hämäläinen P. Källblad S. Nyström H. Wallberg U. H. Danielson J. Med. Chem. 2008 51 3449 3459
- (2008) J. Med. Chem. , vol.51 , pp. 3449-3459
- Nordström, H.¹ Gossas, T.² Hämäläinen, M.³ Källblad, P.⁴ Nyström, S.⁵ Wallberg, H.⁶ Danielson, U.H.⁷

9
- 17944369447
- J. I. Levin J. Chen M. Du M. Hogan S. Kincaid F. C. Nelson A. M. Venkatesan T. Wehr A. Zask J. DiJoseph L. M. Killar S. Skala A. Sung M. Sharr C. Roth G. Jin R. Cowling K. M. Mohler R. A. Black C. J. March J. S. Skotnicki Bioorg. Med. Chem. Lett. 2001 11 2189 2192
- (2001) Bioorg. Med. Chem. Lett. , vol.11 , pp. 2189-2192
- Levin, J.I.¹ Chen, J.² Du, M.³ Hogan, M.⁴ Kincaid, S.⁵ Nelson, F.C.⁶ Venkatesan, A.M.⁷ Wehr, T.⁸ Zask, A.⁹ Dijoseph, J.¹⁰ Killar, L.M.¹¹ Skala, S.¹² Sung, A.¹³ Sharr, M.¹⁴ Roth, C.¹⁵ Jin, G.¹⁶ Cowling, R.¹⁷ Mohler, K.M.¹⁸ Black, R.A.¹⁹ March, C.J.²⁰ Skotnicki, J.S.²¹ more..

10
- 0032505173
- S. Pikul K. L. McDow Dunham N. G. Almstead B. De M. G. Natchus M. V. Anastasio S. J. McPhail C. E. Snider Y. O. Taiwo T. Rydel C. M. Dunaway F. Gu G. E. Mieling J. Med. Chem. 1998 41 3568 3571
- (1998) J. Med. Chem. , vol.41 , pp. 3568-3571
- Pikul, S.¹ McDow Dunham, K.L.² Almstead, N.G.³ De, B.⁴ Natchus, M.G.⁵ Anastasio, M.V.⁶ McPhail, S.J.⁷ Snider, C.E.⁸ Taiwo, Y.O.⁹ Rydel, T.¹⁰ Dunaway, C.M.¹¹ Gu, F.¹² Mieling, G.E.¹³

11
- 0032499266
- M. Yamamoto H. Tsujishita N. Hori Y. Ohishi S. Inoue S. Ikeda Y. Okada J. Med. Chem. 1998 41 1209 1217
- (1998) J. Med. Chem. , vol.41 , pp. 1209-1217
- Yamamoto, M.¹ Tsujishita, H.² Hori, N.³ Ohishi, Y.⁴ Inoue, S.⁵ Ikeda, S.⁶ Okada, Y.⁷

12
- 15444343493
- D. E. Levy F. Lapierre W. Liang W. Ye C. W. Lange X. Li D. Grobelny M. Casabonne D. Tyrrell K. Holme A. Nadzan R. E. Galardy J. Med. Chem. 1998 41 199 223
- (1998) J. Med. Chem. , vol.41 , pp. 199-223
- Levy, D.E.¹ Lapierre, F.² Liang, W.³ Ye, W.⁴ Lange, C.W.⁵ Li, X.⁶ Grobelny, D.⁷ Casabonne, M.⁸ Tyrrell, D.⁹ Holme, K.¹⁰ Nadzan, A.¹¹ Galardy, R.E.¹²

13
- 0343484958
- P. O. Markgren M. Hamalainen U. H. Danielson Anal. Biochem. 2000 279 71 78
- (2000) Anal. Biochem. , vol.279 , pp. 71-78
- Markgren, P.O.¹ Hamalainen, M.² Danielson, U.H.³

14
- 31144460354
- R. Karlsson P. S. Katsamba H. Nordin E. Pol D. G. Myszka Anal. Biochem. 2006 349 136 147
- (2006) Anal. Biochem. , vol.349 , pp. 136-147
- Karlsson, R.¹ Katsamba, P.S.² Nordin, H.³ Pol, E.⁴ Myszka, D.G.⁵

15
- 33644796110
- R. A. Copeland Methods Biochem. Anal. 2005 46 1 265
- (2005) Methods Biochem. Anal. , vol.46 , pp. 1-265
- Copeland, R.A.¹

16
- 33748749807
- T. Gossas U. H. Danielson Biochem. J. 2006 398 393 398
- (2006) Biochem. J. , vol.398 , pp. 393-398
- Gossas, T.¹ Danielson, U.H.²

17
- 0038038524
- G. Rosenblum S. O. Meroueh O. Kleifeld S. Brown S. P. Singson R. Fridman S. Mobashery I. Sagi J. Biol. Chem. 2003 278 27009 27015
- (2003) J. Biol. Chem. , vol.278 , pp. 27009-27015
- Rosenblum, G.¹ Meroueh, S.O.² Kleifeld, O.³ Brown, S.⁴ Singson, S.P.⁵ Fridman, R.⁶ Mobashery, S.⁷ Sagi, I.⁸

18
- 0037202174
- F. J. Moy P. K. Chanda J. Chen S. Cosmi W. Edris J. I. Levin T. S. Rush J. Wilhelm R. Powers J. Am. Chem. Soc. 2002 124 12658 12659
- (2002) J. Am. Chem. Soc. , vol.124 , pp. 12658-12659
- Moy, F.J.¹ Chanda, P.K.² Chen, J.³ Cosmi, S.⁴ Edris, W.⁵ Levin, J.I.⁶ Rush, T.S.⁷ Wilhelm, J.⁸ Powers, R.⁹

19
- 0023728105
- J. F. Morrison C. T. Walsh Adv. Enzymol. Relat. Areas Mol. Biol. 1988 61 201 301
- (1988) Adv. Enzymol. Relat. Areas Mol. Biol. , vol.61 , pp. 201-301
- Morrison, J.F.¹ Walsh, C.T.²

20
- 0014454095
- J. F. Morrison Biochim. Biophys. Acta 1969 185 269 286
- (1969) Biochim. Biophys. Acta , vol.185 , pp. 269-286
- Morrison, J.F.¹

21
- 77956225829
- M. Elinder P. Selhorst G. Vanham B. Öberg L. Vrang U. H. Danielson Biochem. Pharmacol. 2010 80 1133 1140
- (2010) Biochem. Pharmacol. , vol.80 , pp. 1133-1140
- Elinder, M.¹ Selhorst, P.² Vanham, G.³ Öberg, B.⁴ Vrang, L.⁵ Danielson, U.H.⁶

22
- 15244345731
- C. Lombard J. Saulnier J. Wallach Biochimie 2005 87 265 272
- (2005) Biochimie , vol.87 , pp. 265-272
- Lombard, C.¹ Saulnier, J.² Wallach, J.³

23
- 34948864524
- R. Johnson A. G. Pavlovsky D. F. Ortwine F. Prior C. F. Man D. A. Bornemeier C. A. Banotai W. T. Mueller P. McConnell C. Yan V. Baragi C. Lesch W. H. Roark M. Wilson K. Datta R. Guzman H. K. Dyer J. Biol. Chem. 2007 282 27781 27791
- (2007) J. Biol. Chem. , vol.282 , pp. 27781-27791
- Johnson, R.¹ Pavlovsky, A.G.² Ortwine, D.F.³ Prior, F.⁴ Man, C.F.⁵ Bornemeier, D.A.⁶ Banotai, C.A.⁷ Mueller, W.T.⁸ McConnell, P.⁹ Yan, C.¹⁰ Baragi, V.¹¹ Lesch, C.¹² Roark, W.H.¹³ Wilson, M.¹⁴ Datta, K.¹⁵ Guzman, R.¹⁶ Dyer, H.K.¹⁷

24
- 0346639256
- M. Tegoni F. Dallavalle M. Amelia Santos J. Inorg. Biochem. 2004 98 209 218
- (2004) J. Inorg. Biochem. , vol.98 , pp. 209-218
- Tegoni, M.¹ Dallavalle, F.² Amelia Santos, M.³

25
- 0037192860
- M. M. Bernardo S. Brown Z. H. Li R. Fridman S. Mobashery J. Biol. Chem. 2002 277 11201 11207
- (2002) J. Biol. Chem. , vol.277 , pp. 11201-11207
- Bernardo, M.M.¹ Brown, S.² Li, Z.H.³ Fridman, R.⁴ Mobashery, S.⁵

26
- 22844434878
- A. C. Dublanchet P. Ducrot C. Andrianjara M. O'Gara R. Morales D. Compere A. Denis S. Blais P. Cluzeau K. Courte J. Hamon F. Moreau M. L. Prunet A. Tertre Bioorg. Med. Chem. Lett. 2005 15 3787 3790
- (2005) Bioorg. Med. Chem. Lett. , vol.15 , pp. 3787-3790
- Dublanchet, A.C.¹ Ducrot, P.² Andrianjara, C.³ O'Gara, M.⁴ Morales, R.⁵ Compere, D.⁶ Denis, A.⁷ Blais, S.⁸ Cluzeau, P.⁹ Courte, K.¹⁰ Hamon, J.¹¹ Moreau, F.¹² Prunet, M.L.¹³ Tertre, A.¹⁴

27
- 15244350894
- P. Cuniasse L. Devel A. Makaritis F. Beau D. Georgiadis M. Matziari A. Yiotakis V. Dive Biochimie 2005 87 393 402
- (2005) Biochimie , vol.87 , pp. 393-402
- Cuniasse, P.¹ Devel, L.² Makaritis, A.³ Beau, F.⁴ Georgiadis, D.⁵ Matziari, M.⁶ Yiotakis, A.⁷ Dive, V.⁸

28
- 0035965125
- R. Lang A. Kocourek M. Braun H. Tschesche R. Huber W. Bode K. Maskos J. Mol. Biol. 2001 312 731 742
- (2001) J. Mol. Biol. , vol.312 , pp. 731-742
- Lang, R.¹ Kocourek, A.² Braun, M.³ Tschesche, H.⁴ Huber, R.⁵ Bode, W.⁶ Maskos, K.⁷

29
- 0035965133
- H. Nar K. Werle M. M. Bauer H. Dollinger B. Jung J. Mol. Biol. 2001 312 743 751
- (2001) J. Mol. Biol. , vol.312 , pp. 743-751
- Nar, H.¹ Werle, K.² Bauer, M.M.³ Dollinger, H.⁴ Jung, B.⁵

30
- 33748325882
- R. A. Copeland D. L. Pompliano T. D. Meek Nat. Rev. Drug Discovery 2006 5 730 739
- (2006) Nat. Rev. Drug Discovery , vol.5 , pp. 730-739
- Copeland, R.A.¹ Pompliano, D.L.² Meek, T.D.³

31
- 3843152629
- R. Morales S. Perrier J. M. Florent J. Beltra S. Dufour I. De Mendez P. Manceau A. Tertre F. Moreau D. Compere A. C. Dublanchet M. O'Gara J. Mol. Biol. 2004 341 1063 1076
- (2004) J. Mol. Biol. , vol.341 , pp. 1063-1076
- Morales, R.¹ Perrier, S.² Florent, J.M.³ Beltra, J.⁴ Dufour, S.⁵ De Mendez, I.⁶ Manceau, P.⁷ Tertre, A.⁸ Moreau, F.⁹ Compere, D.¹⁰ Dublanchet, A.C.¹¹ O'Gara, M.¹²

32
- 0035871240
- P. O. Markgren M. T. Lindgren K. Gertow R. Karlsson M. Hämäläinen U. H. Danielson Anal. Biochem. 2001 291 207 218
- (2001) Anal. Biochem. , vol.291 , pp. 207-218
- Markgren, P.O.¹ Lindgren, M.T.² Gertow, K.³ Karlsson, R.⁴ Hämälä inen, M.⁵ Danielson, U.H.⁶

33
- 0026153423
- E. Stenberg B. Persson H. Roos C. Urbaniczky J. Colloid Interface Sci. 1991 143 513 526
- (1991) J. Colloid Interface Sci. , vol.143 , pp. 513-526
- Stenberg, E.¹ Persson, B.² Roos, H.³ Urbaniczky, C.⁴

34
- 0032899689
- C. T. Goudar J. R. Sonnad R. G. Duggleby Biochim. Biophys. Acta 1999 1429 377 383
- (1999) Biochim. Biophys. Acta , vol.1429 , pp. 377-383
- Goudar, C.T.¹ Sonnad, J.R.² Duggleby, R.G.³

35
- 21444436092
- R. M. Corless G. H. Gonnett D. E. G. Hare D. J. Jeffrey D. E. Knuth Adv. Comput. Math. 1996 5 329 359
- (1996) Adv. Comput. Math. , vol.5 , pp. 329-359
- Corless, R.M.¹ Gonnett, G.H.² Hare, D.E.G.³ Jeffrey, D.J.⁴ Knuth, D.E.⁵

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