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Journal of Biological Chemistry

Volumn 277, Issue 13, 2002, Pages 11201-11207

Design, synthesis, and characterization of potent, slow-binding inhibitors that are selective for gelatinases

(5) Margarida Bernardo, M a Brown, Stephen a Li, Zhi Hong b Fridman, Rafael c Mobashery, Shahriar a,c

a Department of Pathology ^* (United States)

b Department of Departments of Chemistry Pharmacology and Biochemistry and Molecular Biology (United States)

c WAYNE STATE UNIVERSITY (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ENZYME INHIBITION; ENZYMES; MOLECULAR WEIGHT; TUMORS;

ANGIOGENESIS;

BIOCHEMISTRY;

4 (4 PHENOXYPHENYLSULFONYL)BUTANE 1,2 DITHIOL; 5 (4 PHENOXYPHENYLSULFONYL)PENTANE 1,2 DITHIOL; GELATINASE A; GELATINASE INHIBITOR; MARIMASTAT; MATRIX METALLOPROTEINASE INHIBITOR; METALLOPROTEINASE; STROMELYSIN; TISSUE INHIBITOR OF METALLOPROTEINASE 2; UNCLASSIFIED DRUG;

ARTICLE; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG BINDING; DRUG DESIGN; DRUG INHIBITION; DRUG POTENCY; DRUG SELECTIVITY; DRUG SYNTHESIS; ENZYME ACTIVATION; HUMAN; HUMAN CELL; PRIORITY JOURNAL;

CATALYTIC DOMAIN; ENZYME INHIBITORS; GELATINASES; HELA CELLS; HUMANS; RECOMBINANT PROTEINS; SPECTROMETRY, FLUORESCENCE;

FELIS CATUS;

EID: 0037192860 PISSN: 00219258 EISSN: None Source Type: Journal
DOI: 10.1074/jbc.M111021200 Document Type: Article

Times cited : (75)

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