Hits, leads and drugs against malaria through diversity-oriented synthesis

Future Medicinal Chemistry

Volumn 4, Issue 18, 2012, Pages 2279-2294

  Dandapani, Sivaraman ^a   Comer, Eamon ^a   Duvall, Jeremy R ^a   Munoz, Benito ^a  

^a BROAD INSTITUTE OF MIT AND HARVARD   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINO 3,5 DIMETHYLISOXAZOYL UREA DERIVATIVE; AMINE; ANILINE; ANTIMALARIAL AGENT; ARTEMISININ DERIVATIVE; INDOLE DERIVATIVE; NITD 609; SPIROAZEPINEINDOLE; UNCLASSIFIED DRUG; UREA DERIVATIVE;

AQUEOUS SOLUTION; CHEMICAL STRUCTURE; CHEMOTHERAPY; DIVERSITY ORIENTED SYNTHESIS; DRUG HALF LIFE; DRUG SYNTHESIS; ENZYME METABOLISM; GROWTH INHIBITION; HIGH THROUGHPUT SCREENING; MALARIA; NONHUMAN; PHARMACOPHORE; PHENOTYPE; PLASMODIUM BERGHEI; PLASMODIUM FALCIPARUM; PLASMODIUM MALARIAE INFECTION; PRIORITY JOURNAL; REVIEW; RING CLOSING METATHESIS; STEREOCHEMISTRY; STEREOISOMERISM; STRUCTURE ACTIVITY RELATION;

ANIMALS; ANTIMALARIALS; DRUG DISCOVERY; HUMANS; MALARIA; PLASMODIUM; PLASMODIUM FALCIPARUM;

EID: 84871080255     PISSN: 17568919     EISSN: 17568927     Source Type: Journal    
DOI: 10.4155/fmc.12.178     Document Type: Review

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