SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 24, 2012, Pages 7715-7718

Fluorescent nitrile-based inhibitors of cysteine cathepsins

(3) Frizler, Maxim a Mertens, Matthias D a Gütschow, Michael a

a UNIVERSITY OF BONN (Germany)

Author keywords

Azadipeptide nitriles; Coumarins; Cysteine cathepsins; Dipeptide nitriles; Fluorescent probes

Indexed keywords

AZADIPEPTIDE NITRILE DERIVATIVE; CYSTEINE PROTEINASE INHIBITOR; DIPEPTIDE NITRILE DERIVATIVE; NITRILE; UNCLASSIFIED DRUG;

ARTICLE; BIOLOGICAL ACTIVITY; DRUG DESIGN; DRUG STRUCTURE; DRUG SYNTHESIS; SPECTROSCOPY;

CATHEPSINS; CYSTEINE PROTEINASE INHIBITORS; DIPEPTIDES; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DESIGN; FLUORESCENCE; MOLECULAR STRUCTURE; NITRILES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84870244736 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.09.086 Document Type: Article

Times cited : (15)

References (33)

1
- 0036882393
- F. Lecaille, J. Kaleta, and D. Brömme Chem. Rev. 102 2002 4459
- (2002) Chem. Rev. , vol.102 , pp. 4459
- Lecaille, F.¹ Kaleta, J.² Brömme, D.³

2
- 77949483288
- M. Frizler, M. Stirnberg, M.T. Sisay, and M. Gütschow Curr. Top. Med. Chem. 10 2010 294
- (2010) Curr. Top. Med. Chem. , vol.10 , pp. 294
- Frizler, M.¹ Stirnberg, M.² Sisay, M.T.³ Gütschow, M.⁴

3
- 77952502923
- W.C. Black Curr. Top. Med. Chem. 10 2010 745
- (2010) Curr. Top. Med. Chem. , vol.10 , pp. 745
- Black, W.C.¹

4
- 46749119861
- R. Löser, M. Frizler, K. Schilling, and M. Gütschow Angew. Chem. Int. Ed. 47 2008 4331
- (2008) Angew. Chem. Int. Ed. , vol.47 , pp. 4331
- Löser, R.¹ Frizler, M.² Schilling, K.³ Gütschow, M.⁴

5
- 72049088495
- R. Löser, J. Gut, P.J. Rosenthal, M. Frizler, M. Gütschow, and K.T. Andrews Bioorg. Med. Chem. Lett. 20 2010 252
- (2010) Bioorg. Med. Chem. Lett. , vol.20 , pp. 252
- Löser, R.¹ Gut, J.² Rosenthal, P.J.³ Frizler, M.⁴ Gütschow, M.⁵ Andrews, K.T.⁶

6
- 78651072739
- M. Frizler, F. Lohr, N. Furtmann, J. Kläs, and M. Gütschow J. Med. Chem. 54 2011 396
- (2011) J. Med. Chem. , vol.54 , pp. 396
- Frizler, M.¹ Lohr, F.² Furtmann, N.³ Kläs, J.⁴ Gütschow, M.⁵

7
- 80053188665
- M. Frizler, F. Lohr, M. Lülsdorff, and M. Gütschow Chem. Eur. J. 17 2011 11419
- (2011) Chem. Eur. J. , vol.17 , pp. 11419
- Frizler, M.¹ Lohr, F.² Lülsdorff, M.³ Gütschow, M.⁴

8
- 78049405461
- Y. Loh, H. Shi, M. Hu, and S.Q. Yao Chem. Commun. 46 2010 8407
- (2010) Chem. Commun. , vol.46 , pp. 8407
- Loh, Y.¹ Shi, H.² Hu, M.³ Yao, S.Q.⁴

9
- 32644474873
- M. Skoumal, G. Haberhauer, G. Kolarz, G. Hawa, W. Woloszczuk, and A. Klingler Arthritis Res. Ther. 7 2005 R65
- (2005) Arthritis Res. Ther. , vol.7 , pp. 65
- Skoumal, M.¹ Haberhauer, G.² Kolarz, G.³ Hawa, G.⁴ Woloszczuk, W.⁵ Klingler, A.⁶

10
- 41849102403
- M. Skoumal, G. Haberhauer, G. Kolarz, G. Hawa, W. Woloszczuk, A. Klingler, F. Varga, and K. Klaushofer Rheumatol. Int. 28 2008 637
- (2008) Rheumatol. Int. , vol.28 , pp. 637
- Skoumal, M.¹ Haberhauer, G.² Kolarz, G.³ Hawa, G.⁴ Woloszczuk, W.⁵ Klingler, A.⁶ Varga, F.⁷ Klaushofer, K.⁸

11
- 59049103199
- Y. Liu, X. Li, D. Peng, Z. Tan, H. Liu, Y. Qing, Y. Xue, and G.P. Shi Am. J. Cardiol. 103 2009 476
- (2009) Am. J. Cardiol. , vol.103 , pp. 476
- Liu, Y.¹ Li, X.² Peng, D.³ Tan, Z.⁴ Liu, H.⁵ Qing, Y.⁶ Xue, Y.⁷ Shi, G.P.⁸

12
- 80755146088
- J.A. Gormley, S.M. Hegarty, A. O'Grady, M.R. Stevenson, R.E. Burden, H.L. Barrett, C.J. Scott, J.A. Johnston, R.H. Wilson, E.W. Kay, P.G. Johnston, and S.A. Olwill Br. J. Cancer. 105 2011 1487
- (2011) Br. J. Cancer. , vol.105 , pp. 1487
- Gormley, J.A.¹ Hegarty, S.M.² O'Grady, A.³ Stevenson, M.R.⁴ Burden, R.E.⁵ Barrett, H.L.⁶ Scott, C.J.⁷ Johnston, J.A.⁸ Wilson, R.H.⁹ Kay, E.W.¹⁰ Johnston, P.G.¹¹ Olwill, S.A.¹²

13
- 80052773481
- E. Jobs, E. Ingelsson, U. Risérus, E. Nerpin, M. Jobs, J. Sundström, S. Basu, A. Larsson, L. Lind, and J. Ärnlöv JAMA 306 2011 1113
- (2011) JAMA , vol.306 , pp. 1113
- Jobs, E.¹ Ingelsson, E.² Risérus, U.³ Nerpin, E.⁴ Jobs, M.⁵ Sundström, J.⁶ Basu, S.⁷ Larsson, A.⁸ Lind, L.⁹ Ärnlöv, J.¹⁰

14
- 78650727555
- M.A. Nouh, M.M. Mohamed, M. El-Shinawi, M.A. Shaalan, D. Cavallo-Medved, H.M. Khaled, and B.F. Sloane J. Transl. Med. 9 2011 1
- (2011) J. Transl. Med. , vol.9 , pp. 1
- Nouh, M.A.¹ Mohamed, M.M.² El-Shinawi, M.³ Shaalan, M.A.⁴ Cavallo-Medved, D.⁵ Khaled, H.M.⁶ Sloane, B.F.⁷

15
- 38049057786
- A. Watzke, G. Kosec, M. Kindermann, V. Jeske, H.P. Nestler, V. Turk, B. Turk, and K.U. Wendt Angew. Chem. Int. Ed. 47 2008 406
- (2008) Angew. Chem. Int. Ed. , vol.47 , pp. 406
- Watzke, A.¹ Kosec, G.² Kindermann, M.³ Jeske, V.⁴ Nestler, H.P.⁵ Turk, V.⁶ Turk, B.⁷ Wendt, K.U.⁸

16
- 79551503110
- D. Caglič, A. Globisch, M. Kindermann, N.H. Lim, V. Jeske, H.P. Juretschke, E. Bartnik, K.U. Weithmann, H. Nagase, B. Turk, and K.U. Wendt Bioorg. Med. Chem. 19 2011 1055
- (2011) Bioorg. Med. Chem. , vol.19 , pp. 1055
- Caglič, D.¹ Globisch, A.² Kindermann, M.³ Lim, N.H.⁴ Jeske, V.⁵ Juretschke, H.P.⁶ Bartnik, E.⁷ Weithmann, K.U.⁸ Nagase, H.⁹ Turk, B.¹⁰ Wendt, K.U.¹¹

17
- 79951577371
- A. Veilleux, W.C. Black, J.Y. Gauthier, C. Mellon, M.D. Percival, P. Tawa, and J.P. Falgueyret Anal. Biochem. 411 2011 43
- (2011) Anal. Biochem. , vol.411 , pp. 43
- Veilleux, A.¹ Black, W.C.² Gauthier, J.Y.³ Mellon, C.⁴ Percival, M.D.⁵ Tawa, P.⁶ Falgueyret, J.P.⁷

18
- 79961083293
- M.G. Paulick, and M. Bogyo ACS Chem. Biol. 6 2011 563
- (2011) ACS Chem. Biol. , vol.6 , pp. 563
- Paulick, M.G.¹ Bogyo, M.²

19
- 84861610305
- M. Verdoes, L.E. Edgington, F.A. Scheeren, M. Leyva, G. Blum, K. Weiskopf, M.H. Bachmann, J.A. Ellman, and M. Bogyo Chem. Biol. 19 2012 619
- (2012) Chem. Biol. , vol.19 , pp. 619
- Verdoes, M.¹ Edgington, L.E.² Scheeren, F.A.³ Leyva, M.⁴ Blum, G.⁵ Weiskopf, K.⁶ Bachmann, M.H.⁷ Ellman, J.A.⁸ Bogyo, M.⁹

20
- 84862650253
- F. Fan, S. Nie, D. Yang, M. Luo, H. Shi, and Y.H. Zhang Bioconjug. Chem. 23 2012 1309
- (2012) Bioconjug. Chem. , vol.23 , pp. 1309
- Fan, F.¹ Nie, S.² Yang, D.³ Luo, M.⁴ Shi, H.⁵ Zhang, Y.H.⁶

21
- 84861153498
- P.Y. Yang, M. Wang, L. Li, H. Wu, C.Y. He, and S.Q. Yao Chem. Eur. J. 18 2012 6528
- (2012) Chem. Eur. J. , vol.18 , pp. 6528
- Yang, P.Y.¹ Wang, M.² Li, L.³ Wu, H.⁴ He, C.Y.⁵ Yao, S.Q.⁶

22
- 0037463416
- A. Song, X. Wang, and K.S. Lam Tetrahedron Lett. 44 2003 1755
- (2003) Tetrahedron Lett. , vol.44 , pp. 1755
- Song, A.¹ Wang, X.² Lam, K.S.³

23
- 20044390256
- M.E. Jung, and G. Piizzi Chem. Rev. 105 2005 1735
- (2005) Chem. Rev. , vol.105 , pp. 1735
- Jung, M.E.¹ Piizzi, G.²

24
- 79955005064
- S. Fustero, V. Rodrigo, M. Sánchez-Roselló, C. del Pozo, J. Timoneda, M. Frizler, M.T. Sisay, J. Bajorath, L.P. Calle, F.J. Cañada, J. Jiménez-Barbero, and M. Gütschow Chem. Eur. J. 17 2011 5256
- (2011) Chem. Eur. J. , vol.17 , pp. 5256
- Fustero, S.¹ Rodrigo, V.² Sánchez-Roselló, M.³ Del Pozo, C.⁴ Timoneda, J.⁵ Frizler, M.⁶ Sisay, M.T.⁷ Bajorath, J.⁸ Calle, L.P.⁹ Cañada, F.J.¹⁰ Jiménez-Barbero, J.¹¹ Gütschow, M.¹²

25
- 40849096399
- G. Wells, M. Suggitt, M. Coffils, M.A. Baig, P.W. Howard, P.M. Loadman, J.A. Hartley, T.C. Jenkins, and D.E. Thurston Bioorg. Med. Chem. Lett. 18 2008 2147
- (2008) Bioorg. Med. Chem. Lett. , vol.18 , pp. 2147
- Wells, G.¹ Suggitt, M.² Coffils, M.³ Baig, M.A.⁴ Howard, P.W.⁵ Loadman, P.M.⁶ Hartley, J.A.⁷ Jenkins, T.C.⁸ Thurston, D.E.⁹

26
- 43049105748
- K. Kuromochi, S. Yukizawa, S. Ikeda, T. Sunoki, S. Arai, R. Matsui, A. Morita, Y. Mizushina, K. Sakaguchi, F. Sugawara, M. Ikekita, and S. Kobayashi Bioorg. Med. Chem. 16 2008 5039
- (2008) Bioorg. Med. Chem. , vol.16 , pp. 5039
- Kuromochi, K.¹ Yukizawa, S.² Ikeda, S.³ Sunoki, T.⁴ Arai, S.⁵ Matsui, R.⁶ Morita, A.⁷ Mizushina, Y.⁸ Sakaguchi, K.⁹ Sugawara, F.¹⁰ Ikekita, M.¹¹ Kobayashi, S.¹²

27
- 33947588806
- D. Schweitzer, J. Zhu, G. Jarori, J. Tanaka, T. Higa, V.J. Davisson, and P. Helquist Bioorg. Med. Chem. 15 2007 3208
- (2007) Bioorg. Med. Chem. , vol.15 , pp. 3208
- Schweitzer, D.¹ Zhu, J.² Jarori, G.³ Tanaka, J.⁴ Higa, T.⁵ Davisson, V.J.⁶ Helquist, P.⁷

28
- 34548502668
- A.G. Shilabin, N. Kasanah, D.E. Wedge, and M.T. Hamann J. Med. Chem. 50 2007 4340
- (2007) J. Med. Chem. , vol.50 , pp. 4340
- Shilabin, A.G.¹ Kasanah, N.² Wedge, D.E.³ Hamann, M.T.⁴

29
- 83755171532
- H.J. Cho, H.Y. Gee, K.H. Baek, S.K. Ko, J.M. Park, H. Lee, N.D. Kim, M.G. Lee, and I. Shin J. Am. Chem. Soc. 21 2011 20267
- (2011) J. Am. Chem. Soc. , vol.21 , pp. 20267
- Cho, H.J.¹ Gee, H.Y.² Baek, K.H.³ Ko, S.K.⁴ Park, J.M.⁵ Lee, H.⁶ Kim, N.D.⁷ Lee, M.G.⁸ Shin, I.⁹

30
- 84857745980
- G. Leriche, G. Budin, Z. Darwich, D. Weltin, Y. Mély, A.S. Klymchenko, and A. Wagner Chem. Commun. 48 2012 3224
- (2012) Chem. Commun. , vol.48 , pp. 3224
- Leriche, G.¹ Budin, G.² Darwich, Z.³ Weltin, D.⁴ Mély, Y.⁵ Klymchenko, A.S.⁶ Wagner, A.⁷

31
- 77951682590
- R.S. Agnes, F. Jernigan, J.R. Shell, V. Sharma, and D.S. Lawrence J. Am. Soc. Chem. 132 2010 6075
- (2010) J. Am. Soc. Chem. , vol.132 , pp. 6075
- Agnes, R.S.¹ Jernigan, F.² Shell, J.R.³ Sharma, V.⁴ Lawrence, D.S.⁵

32
- 83355160776
- C.L. Ho, S.L. Koh, M.L. Chuah, Z. Luo, W.J. Tan, D.K. Low, and Z.X. Liang ChemBioChem 12 2011 2753
- (2011) ChemBioChem , vol.12 , pp. 2753
- Ho, C.L.¹ Koh, S.L.² Chuah, M.L.³ Luo, Z.⁴ Tan, W.J.⁵ Low, D.K.⁶ Liang, Z.X.⁷

33
- 79751523412
- J.W. Hanes, D. Chatterjee, E.V. Soriano, S.E. Ealick, and T.P. Begley Chem. Commun. 47 2011 2273
- (2011) Chem. Commun. , vol.47 , pp. 2273
- Hanes, J.W.¹ Chatterjee, D.² Soriano, E.V.³ Ealick, S.E.⁴ Begley, T.P.⁵

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.