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Angewandte Chemie - International Edition

Volumn 47, Issue 23, 2008, Pages 4331-4334

Azadipeptide nitriles: Highly potent and proteolytically stable inhibitors of papain-like cysteine proteases

(4) Löser, Reik a,c Frizler, Maxim a Schilling, Klaus b Gütschow, Michael a

a UNIVERSITY OF BONN (Germany)

b FRIEDRICH SCHILLER UNIVERSITY JENA (Germany)

c UNIVERSITY OF QUEENSLAND (Australia)

Author keywords

Azapeptides; Enzyme inhibitors; Hydrazides; Nitriles

Indexed keywords

AZAPEPTIDES; ENZYME INHIBITORS; HYDRAZIDES; NITRILES;

CYANIDES;

CYSTEINE PROTEINASE INHIBITOR; DIPEPTIDE; HETEROCYCLIC COMPOUND; NITRILE; PAPAIN;

ARTICLE; CHEMISTRY; DRUG ANTAGONISM; HUMAN; SYNTHESIS;

AZA COMPOUNDS; CYSTEINE PROTEINASE INHIBITORS; DIPEPTIDES; HUMANS; NITRILES; PAPAIN;

EID: 46749119861 PISSN: 14337851 EISSN: None Source Type: Journal
DOI: 10.1002/anie.200705858 Document Type: Article

Times cited : (74)

References (30)

1
- 0036882393
- Review
- Review: F. Lecaille, J. Kaleta, D. Brömme, Chem. Rev. 2002, 102, 4459-4488.
- (2002) Chem. Rev , vol.102 , pp. 4459-4488
- Lecaille, F.¹ Kaleta, J.² Brömme, D.³

2
- 10844291804
- a) K. Ravanko, K. Järvinen, J. Helin, N. Kalkkinen, E. Hölttä, Cancer Res. 2004, 64, 8831-8838;
- (2004) Cancer Res , vol.64 , pp. 8831-8838
- Ravanko, K.¹ Järvinen, K.² Helin, J.³ Kalkkinen, N.⁴ Hölttä, E.⁵

3
- 0036329099
- b) K. Saegusa, N. Ishimura, K. Yanagi, R. Arakaki, K. Ogawa, I. Saito, N. Katunuma, Y. Hayashi, J. Clin. Invest. 2002, 110, 361-369;
- (2002) J. Clin. Invest , vol.110 , pp. 361-369
- Saegusa, K.¹ Ishimura, N.² Yanagi, K.³ Arakaki, R.⁴ Ogawa, K.⁵ Saito, I.⁶ Katunuma, N.⁷ Hayashi, Y.⁸

4
- 0030026637
- c) D. Brömme, K. Okamoto, B. B. Wang, S. Biroc, J. Biol. Chem. 1996, 271, 2126-2132.
- (1996) J. Biol. Chem , vol.271 , pp. 2126-2132
- Brömme, D.¹ Okamoto, K.² Wang, B.B.³ Biroc, S.⁴

5
- 33845339435
- Reviews: a
- Reviews: a) G. Abbenante, D. P. Fairlie, Med. Chem. 2005, 1, 71-104;
- (2005) Med. Chem , vol.1 , pp. 71-104
- Abbenante, G.¹ Fairlie, D.P.²

6
- 33646188959
- b) R. Vicik, M. Busemann, K. Baumann, T. Schirmeister, Curr. Top. Med. Chem. 2006, 6, 331-353;
- (2006) Curr. Top. Med. Chem , vol.6 , pp. 331-353
- Vicik, R.¹ Busemann, M.² Baumann, K.³ Schirmeister, T.⁴

7
- 33947604810
- c) O. Vasiljeva, T. Reinheckel, C. Peters, D. Turk, V. Turk, B. Turk, Curr. Pharm. Des. 2007, 13, 387-403.
- (2007) Curr. Pharm. Des , vol.13 , pp. 387-403
- Vasiljeva, O.¹ Reinheckel, T.² Peters, C.³ Turk, D.⁴ Turk, V.⁵ Turk, B.⁶

8
- 0035924180
- a) P. D. Greenspan, K. L. Clark, R. A. Tommasi, S. D. Cowen, L. W. McQuire, D. L. Farley, J. H. van Duzer, R. L. Goldberg, H. Zhou, Z. Du, J. J. Fitt, D. E. Coppa, Z. Fang, W. Macchia, L. Zhu, M. P. Capparelli, R. Goldstein, A. M. Wigg, J. R. Doughty, R. S. Bohacek, A. K. Knap, J. Med. Chem. 2001, 44, 4524-4534;
- (2001) J. Med. Chem , vol.44 , pp. 4524-4534
- Greenspan, P.D.¹ Clark, K.L.² Tommasi, R.A.³ Cowen, S.D.⁴ McQuire, L.W.⁵ Farley, D.L.⁶ van Duzer, J.H.⁷ Goldberg, R.L.⁸ Zhou, H.⁹ Du, Z.¹⁰ Fitt, J.J.¹¹ Coppa, D.E.¹² Fang, Z.¹³ Macchia, W.¹⁴ Zhu, L.¹⁵ Capparelli, M.P.¹⁶ Goldstein, R.¹⁷ Wigg, A.M.¹⁸ Doughty, J.R.¹⁹ Bohacek, R.S.²⁰ Knap, A.K.²¹ more..

9
- 33646829091
- b) J. Bondebjerg, H. Fuglsang, K. Rosendal Valeur, J. Pedersen, L. Naerum, Bioorg. Med. Chem. Lett. 2006, 16, 3614-3617;
- (2006) Bioorg. Med. Chem. Lett , vol.16 , pp. 3614-3617
- Bondebjerg, J.¹ Fuglsang, H.² Rosendal Valeur, K.³ Pedersen, J.⁴ Naerum, L.⁵

10
- 33750125526
- c) A. W. Patterson, W. J. L. Wood, M. Hornsby, S. Lesley, G. Spraggon, J. A. Ellman, J. Med. Chem. 2006, 49, 6298-6307.
- (2006) J. Med. Chem , vol.49 , pp. 6298-6307
- Patterson, A.W.¹ Wood, W.J.L.² Hornsby, M.³ Lesley, S.⁴ Spraggon, G.⁵ Ellman, J.A.⁶

11
- 0001146727
- J. B. Moon, R. S. Coleman, R.-P. Hanzlik, J. Am. Chem. Soc. 1986, 108, 1350-1351.
- (1986) J. Am. Chem. Soc , vol.108 , pp. 1350-1351
- Moon, J.B.¹ Coleman, R.S.² Hanzlik, R.-P.³

12
- 14744297865
- Review
- Review: A. Zega, Curr. Med. Chem. 2005, 12, 589-597.
- (2005) Curr. Med. Chem , vol.12 , pp. 589-597
- Zega, A.¹

13
- 0001215147
- Review
- a) Review: J. Gante, Angew. Chem. 1994, 106, 1780-1802;
- (1994) Angew. Chem , vol.106 , pp. 1780-1802
- Gante, J.¹

14
- 0028038601
- Angew. Chem. Int. Ed. Engl. 1994, 33, 1699-1720;
- (1994) Angew. Chem. Int. Ed. Engl , vol.33 , pp. 1699-1720

15
- 0037068629
- b) E. Wieczerzak, P. Drabik, L. Lankiewicz, S. Oldziej, Z. Grzonka, M. Abrahamson, A. Grubb, D. Brömme, J. Med. Chem. 2002, 45, 4202-4211;
- (2002) J. Med. Chem , vol.45 , pp. 4202-4211
- Wieczerzak, E.¹ Drabik, P.² Lankiewicz, L.³ Oldziej, S.⁴ Grzonka, Z.⁵ Abrahamson, M.⁶ Grubb, A.⁷ Brömme, D.⁸

16
- 33745314454
- c) S. H. L. Verhelst, M. D. Witte, S. Arastu-Kapur, M. Fonovic, M. Bogyo, ChemBioChem 2006, 7, 943-950.
- (2006) ChemBioChem , vol.7 , pp. 943-950
- Verhelst, S.H.L.¹ Witte, M.D.² Arastu-Kapur, S.³ Fonovic, M.⁴ Bogyo, M.⁵

17
- 0035804301
- J.-P. Falgueyret, R. M. Oballa, O. Okamoto, G. Wesolowski, Y. Aubin, R. M. Rydzewski, P. Prasit, D. Riendeau, S: B. Rodan, M. D. Percival, J. Med. Chem. 2001, 44, 94-104;
- a) J.-P. Falgueyret, R. M. Oballa, O. Okamoto, G. Wesolowski, Y. Aubin, R. M. Rydzewski, P. Prasit, D. Riendeau, S: B. Rodan, M. D. Percival, J. Med. Chem. 2001, 44, 94-104;

18
- 19944407105
- b) D. G. Barrett, D. N. Deaton, A. M. Hassell, R. B. McFayden, A. B. Miller, L. R. Miller, J. A. Payne, L. M. Shewchuk, D. H. Willard Jr. , L. L. Wright, Bioorg. Med. Chem. Lett. 2005, 15, 3039-3043.
- (2005) Bioorg. Med. Chem. Lett , vol.15 , pp. 3039-3043
- Barrett, D.G.¹ Deaton, D.N.² Hassell, A.M.³ McFayden, R.B.⁴ Miller, A.B.⁵ Miller, L.R.⁶ Payne, J.A.⁷ Shewchuk, L.M.⁸ Willard Jr., D.H.⁹ Wright, L.L.¹⁰

19
- 28144443719
- R. Löser, K. Schilling, E. Dimmig, M. Gütschow, J. Med. Chem. 2005, 48, 7688-7707.
- (2005) J. Med. Chem , vol.48 , pp. 7688-7707
- Löser, R.¹ Schilling, K.² Dimmig, E.³ Gütschow, M.⁴

20
- 0023728105
- J. F. Morrison, C. T. Walsh, Adv. Enzymol. Relat. Areas Mol. Biol. 1988, 61, 201-301.
- (1988) Adv. Enzymol. Relat. Areas Mol. Biol , vol.61 , pp. 201-301
- Morrison, J.F.¹ Walsh, C.T.²

21
- 0033226493
- J. D. A. Tyndall, D. P. Fairlie, J. Mol. Recognit. 1999, 12, 363-370.
- (1999) J. Mol. Recognit , vol.12 , pp. 363-370
- Tyndall, J.D.A.¹ Fairlie, D.P.²

22
- 85069795554
- G. A. Olah, S. C. Narang, A. P. Fung, B. G. B. Gupta, Synthesis 1980, 657-658.
- (1980) Synthesis , pp. 657-658
- Olah, G.A.¹ Narang, S.C.² Fung, A.P.³ Gupta, B.G.B.⁴

23
- 33750116951
- Review
- Review: A. F. Abdel-Magid, S. J. Mehrman, Org. Process Res. Dev. 2006, 10, 971-1031.
- (2006) Org. Process Res. Dev , vol.10 , pp. 971-1031
- Abdel-Magid, A.F.¹ Mehrman, S.J.²

24
- 0025803608
- R. Calabretta, C. Gallina, C. Giordano, Synthesis 1991, 536-539.
- (1991) Synthesis , pp. 536-539
- Calabretta, R.¹ Gallina, C.² Giordano, C.³

25
- 0038721888
- S. Caddick, D. B. Judd, A. K. de Lewis, M. T. Reich, M. R. V. Williams, Tetrahedron 2003, 59, 5417-5423.
- (2003) Tetrahedron , vol.59 , pp. 5417-5423
- Caddick, S.¹ Judd, D.B.² de Lewis, A.K.³ Reich, M.T.⁴ Williams, M.R.V.⁵

26
- 0037163336
- M. E. Casarini, F. Ghelfi, E. Libertini, U. M. Pagnoni, A. F. Parsons, Tetrahedron 2002, 58, 7925-7932.
- (2002) Tetrahedron , vol.58 , pp. 7925-7932
- Casarini, M.E.¹ Ghelfi, F.² Libertini, E.³ Pagnoni, U.M.⁴ Parsons, A.F.⁵

27
- 5744232410
- Review
- a) Review: S. Sagan, P. Karoyan, O. Lequin, G. Chassaing, S. Lavielle, Curr. Med. Chem. 2004, 11, 2799-2822;
- (2004) Curr. Med. Chem , vol.11 , pp. 2799-2822
- Sagan, S.¹ Karoyan, P.² Lequin, O.³ Chassaing, G.⁴ Lavielle, S.⁵

28
- 0016753995
- b) S. A. Bizzozero, B. O. Zweifel, FEBS Lett. 1975, 59, 105-108;
- (1975) FEBS Lett , vol.59 , pp. 105-108
- Bizzozero, S.A.¹ Zweifel, B.O.²

29
- 0032738396
- c) A. Bianco, D. Kaiser, G. Jung, J. Pept. Res. 1999, 54, 544-548.
- (1999) J. Pept. Res , vol.54 , pp. 544-548
- Bianco, A.¹ Kaiser, D.² Jung, G.³

30
- 70449169903
- B. Borgström, A. Dahlqvist, G. Lundh, J. Sjövall, J. Clin. Invest. 1957, 36, 1521-1536.
- (1957) J. Clin. Invest , vol.36 , pp. 1521-1536
- Borgström, B.¹ Dahlqvist, A.² Lundh, G.³ Sjövall, J.⁴

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