-
1
-
-
84937424396
-
Über die Bildung von Isochinolin-derivaten durch Einwirkung von Methylal auf Phenyl-thylamin, Phenyl-alanin und Tyrosin
-
Pictet, A.; Spengler, T.T. Über die Bildung von Isochinolin-derivaten durch Einwirkung von Methylal auf Phenyl-thylamin, Phenyl-alanin und Tyrosin. Ber. Dtsch. Chem. Ges., 1911, 44, 2030-2036.
-
(1911)
Ber. Dtsch. Chem. Ges.
, vol.44
, pp. 2030-2036
-
-
Pictet, A.1
Spengler, T.T.2
-
2
-
-
0347089132
-
The Pictet-Spengler reaction in solid-phase combinatorial chemistry
-
Nielsen, T.E.; Diness, F.; Meldal, M. The Pictet-Spengler reaction in solid-phase combinatorial chemistry. Curr. Opin. Drug. Discov. Devel., 2003, 6, 801-814.
-
(2003)
Curr. Opin. Drug. Discov. Devel.
, vol.6
, pp. 801-814
-
-
Nielsen, T.E.1
Diness, F.2
Meldal, M.3
-
3
-
-
2942574530
-
Chiral heterocycles by iminium ion cyclization
-
Royer, J.; Bonin, M.; Micouin, L. Chiral heterocycles by iminium ion cyclization. Chem. Rev., 2004, 104, 2311-2352.
-
(2004)
Chem. Rev.
, vol.104
, pp. 2311-2352
-
-
Royer, J.1
Bonin, M.2
Micouin, L.3
-
4
-
-
33845476736
-
The Pictet-Spengler reaction: Efficient carboncarbon bond forming reaction in heterocyclic synthesis
-
Youn, S.W. The Pictet-Spengler reaction: efficient carboncarbon bond forming reaction in heterocyclic synthesis. Org. Prep. Proced. Int., 2006, 38, 505-591.
-
(2006)
Org. Prep. Proced. Int.
, vol.38
, pp. 505-591
-
-
Youn, S.W.1
-
5
-
-
0030575349
-
Solid phase synthesis of tetrahydroisoquinolines & tetrahydroimidazopyridines
-
Hutchins, S.M.; Chapman, K.T. Solid phase synthesis of tetrahydroisoquinolines & tetrahydroimidazopyridines. Tetrahedron Lett., 1996, 37, 4865-4868.
-
(1996)
Tetrahedron Lett.
, vol.37
, pp. 4865-4868
-
-
Hutchins, S.M.1
Chapman, K.T.2
-
6
-
-
0037127752
-
Synthesis of protoberberines using a silyl-directed Pictet-Spengler cyclization
-
Cutter, P.S.; Miller, R.B.; Schore, N.E. Synthesis of protoberberines using a silyl-directed Pictet-Spengler cyclization. Tetrahedron, 2002, 58, 1471-1478.
-
(2002)
Tetrahedron
, vol.58
, pp. 1471-1478
-
-
Cutter, P.S.1
Miller, R.B.2
Schore, N.E.3
-
7
-
-
0037010827
-
Synthesis of optically pure pyrroloquinolones via Pictet-Spengler and Winterfeldt reactions
-
Jiang, W.; Sui, Z.; Chen, X. Synthesis of optically pure pyrroloquinolones via Pictet-Spengler and Winterfeldt reactions. Tetrahedron Lett., 2002, 43, 8941-8945.
-
(2002)
Tetrahedron Lett.
, vol.43
, pp. 8941-8945
-
-
Jiang, W.1
Sui, Z.2
Chen, X.3
-
8
-
-
0034725771
-
Biomimetic Total Synthesis of (β)-Spirotryprostatin B and related studies
-
Wang, H.; Ganesan, A.A. Biomimetic Total Synthesis of (β)-Spirotryprostatin B and related studies. J. Org. Chem., 2000, 65, 4685-4693.
-
(2000)
J. Org. Chem.
, vol.65
, pp. 4685-4693
-
-
Wang, H.1
Ganesan, A.A.2
-
9
-
-
0028145369
-
Asymmetric steering of the Pictet-Spengler reaction by means of amino acid esters as chiral auxiliary groups
-
Waldmann, H.; Schmidt, G.; Jansen, M.; Geb, J. Asymmetric steering of the Pictet-Spengler reaction by means of amino acid esters as chiral auxiliary groups. Tetrahedron, 1994, 50, 11865-11884.
-
(1994)
Tetrahedron
, vol.50
, pp. 11865-11884
-
-
Waldmann, H.1
Schmidt, G.2
Jansen, M.3
Geb, J.4
-
10
-
-
0032418941
-
First Synthesis of 5,6-Dihydro-4H-furo[3,2-f]pyrrolo[1,2-a][1,4]diazepines
-
Feng, X.; Lancelot, J.C.; Gillard, A.C.; Landelle, H.; Rault, S. First Synthesis of 5,6-Dihydro-4H-furo[3,2-f]pyrrolo[1,2-a][1,4]diazepines. J. Heterocycl. Chem., 1998, 35, 1313-1316.
-
(1998)
J. Heterocycl. Chem.
, vol.35
, pp. 1313-1316
-
-
Feng, X.1
Lancelot, J.C.2
Gillard, A.C.3
Landelle, H.4
Rault, S.5
-
11
-
-
0034714249
-
Pictet-Spengler/palladium catalyzed allenylation and carbonylation processes
-
Grigg, R.; MacLachlan, W.S.; MacPherson, D.T.; Sridharan, V.; Suganthan, S.; Pett, M.T.; Zhang, J. Pictet-Spengler/palladium catalyzed allenylation and carbonylation processes. Tetrahedron, 2000, 56, 6585-6594.
-
(2000)
Tetrahedron
, vol.56
, pp. 6585-6594
-
-
Grigg, R.1
McLachlan, W.S.2
McPherson, D.T.3
Sridharan, V.4
Suganthan, S.5
Pett, M.T.6
Zhang, J.7
-
12
-
-
0034697136
-
Synthesis of tetrahydro-γ-carbolines and STUDIES of the Pictet-Spengler reaction
-
Ducrot, P.; Rabhi, C.; Thal, C. Synthesis of tetrahydro-γ-carbolines and STUDIES of the Pictet-Spengler reaction. Tetrahedron, 2000, 56, 2683-2692.
-
(2000)
Tetrahedron
, vol.56
, pp. 2683-2692
-
-
Ducrot, P.1
Rabhi, C.2
Thal, C.3
-
13
-
-
0036109208
-
Investigation of PictetβSpengler type reactions of Secologanin with histamine and its benzyl derivative
-
Beke, G.; Szabo, L.F.; Podanyi, B. Investigation of PictetβSpengler type reactions of Secologanin with histamine and its benzyl derivative. J. Nat. Prod., 2002, 65, 649-655.
-
(2002)
J. Nat. Prod.
, vol.65
, pp. 649-655
-
-
Beke, G.1
Szabo, L.F.2
Podanyi, B.3
-
14
-
-
0031013399
-
Enantiospecific formation of trans 1,3-Disubstituted Tetrahydro-γ-carbolines by the PictetβSpengler reaction and Conversion of Cis Diastereomers into their trans counterparts by Scission of the C-1/N-2 Bond
-
Cox, E.D.; Hamaker, L.K.; Yu, P.; Czerwinski, K.M.; Deng, L.; Bennett, D.W.; Cook, J.M. Enantiospecific formation of trans 1,3-Disubstituted Tetrahydro-γ-carbolines by the PictetβSpengler reaction and Conversion of Cis Diastereomers into their trans counterparts by Scission of the C-1/N-2 Bond. J. Org. Chem., 1997, 62, 44-61.
-
(1997)
J. Org. Chem.
, vol.62
, pp. 44-61
-
-
Cox, E.D.1
Hamaker, L.K.2
Yu, P.3
Czerwinski, K.M.4
Deng, L.5
Bennett, D.W.6
Cook, J.M.7
-
15
-
-
0000489863
-
Chiral lewis acid-mediated enantioselective PictetβSpengler REACTION of Nb-Hydroxytryptamine with Aldehydes
-
Yamada, H.; Kawate, T.; Matsumizu, M.; Nishida, A.; Yamaguchi, K.; Nakgawa, M. chiral lewis acid-mediated enantioselective PictetβSpengler REACTION of Nb-Hydroxytryptamine with Aldehydes. J. Org. Chem., 1998, 63, 6348-6354.
-
(1998)
J. Org. Chem.
, vol.63
, pp. 6348-6354
-
-
Yamada, H.1
Kawate, T.2
Matsumizu, M.3
Nishida, A.4
Yamaguchi, K.5
Nakgawa, M.6
-
16
-
-
0035840111
-
Modified Pictet-Spengler reaction A highly diastereoselective approach to 1,2,3-trisubstituted-1,2,3,4-tetrahydro-γ-carbolines using perhydro-1,3-heterocycles
-
Singh, K.; Deb, P.K.; Venugopalan, P. Modified Pictet-Spengler reaction. A highly diastereoselective approach to 1,2,3-trisubstituted-1,2,3,4-tetrahydro-γ-carbolines using perhydro-1,3-heterocycles. Tetrahedron, 2001, 57, 7939-7949.
-
(2001)
Tetrahedron
, vol.57
, pp. 7939-7949
-
-
Singh, K.1
Deb, P.K.2
Venugopalan, P.3
-
17
-
-
0023022922
-
Enantioselective synthesis of isoquinoline alkaloids
-
Czarnocki, Z.; MacLean, D.B.; Szarek, W.A. Enantioselective synthesis of isoquinoline alkaloids. Can. J. Chem., 1986, 64, 2205-2210.
-
(1986)
Can. J. Chem.
, vol.64
, pp. 2205-2210
-
-
Czarnocki, Z.1
McLean, D.B.2
Szarek, W.A.3
-
18
-
-
0343986494
-
Pictet-Spengler reaction of Biogenic amines with (2R)-N-Glyoxyloylbornane-10,2-sultam. enantioselective Synthesis of (S)-(+)-N-Methylcalycotomine and (R)-(+)-Xylopinine
-
Czarnocki, Z.; Arazzńy, Z. Pictet-Spengler reaction of Biogenic amines with (2R)-N-Glyoxyloylbornane-10,2-sultam. enantioselective Synthesis of (S)-(+)-N-Methylcalycotomine and (R)-(+)-Xylopinine. Heterocycles, 1999, 51, 2871-2879.
-
(1999)
Heterocycles
, vol.51
, pp. 2871-2879
-
-
Czarnocki, Z.1
Arazzńy, Z.2
-
19
-
-
0001251131
-
Recent Progress in the Enatioselective Synthesis of Isoquinoline Alkaloids
-
Rozwadowska, M.D. Recent Progress in the Enatioselective Synthesis of Isoquinoline Alkaloids. Heterocycles, 1994, 39, 903-931.
-
(1994)
Heterocycles
, vol.39
, pp. 903-931
-
-
Rozwadowska, M.D.1
-
20
-
-
0029617352
-
Pictet-Spengler reaction of biogenic amines with (2R)-N-Glyoxyloylbornane-10,2-sultam. Enantioselective of synthesis of (S)-(+)-N-methylcalycotomine
-
Czarnocki, Z.; Mieckzkowsi, J.B.; Kiegiel, J.; Arazńy, Z. Pictet-Spengler reaction of biogenic amines with (2R)-N-Glyoxyloylbornane-10,2-sultam. Enantioselective of synthesis of (S)-(+)-N-methylcalycotomine. Tetrahyedron Asymmetry, 1995, 6, 2899-2902.
-
(1995)
Tetrahyedron Asymmetry
, vol.6
, pp. 2899-2902
-
-
Czarnocki, Z.1
Mieckzkowsi, J.B.2
Kiegiel, J.3
Arazńy, Z.4
-
21
-
-
0013592304
-
Enantioselective synthesis of 1-substituted tetrahydroisoquinoline-1-carboxylic acids
-
Czarnocki, Z.; Suh, D.; MacLean, D.B.; Hultin, P.G.; Szarek, W.A. Enantioselective synthesis of 1-substituted tetrahydroisoquinoline-1-carboxylic acids. Can. J. Chem., 1992, 70, 1555-1561.
-
(1992)
Can. J. Chem.
, vol.70
, pp. 1555-1561
-
-
Czarnocki, Z.1
Suh, D.2
McLean, D.B.3
Hultin, P.G.4
Szarek, W.A.5
-
22
-
-
0346365498
-
Studies on the intramolecular oxa-Pictet-Spengler rearrangement of 5-aryl-1,3-dioxolanes to 4-hydroxyisochromans
-
Bianchi, D.A.; Rua, F.; Kaufman, T.S. Studies on the intramolecular oxa-Pictet-Spengler rearrangement of 5-aryl-1,3-dioxolanes to 4-hydroxyisochromans. Tetrahedron Lett., 2004, 45, 411-415.
-
(2004)
Tetrahedron Lett.
, vol.45
, pp. 411-415
-
-
Bianchi, D.A.1
Rua, F.2
Kaufman, T.S.3
-
23
-
-
4744372596
-
Synthesis of tetrahydro-γ-carbolinediketopiperazines in [bdmim][PF6] ionic liquid accelerated by controlled microwave heating
-
Yen, Y.H.; Chu, Y.H. Synthesis of tetrahydro-γ-carbolinediketopiperazines in [bdmim][PF6] ionic liquid accelerated by controlled microwave heating. Tetrahedron Lett., 2004, 45, 8137-8140.
-
(2004)
Tetrahedron Lett.
, vol.45
, pp. 8137-8140
-
-
Yen, Y.H.1
Chu, Y.H.2
-
24
-
-
3242791871
-
Pictet Spengler-type reactions in 3-arylmethylpiperazine-2,5-diones Synthesis of pyrazinotetrahydroisoquinolines
-
Gonzalez, J.F.; Cuesta, E.; Avendano, C. Pictet Spengler-type reactions in 3-arylmethylpiperazine-2,5-diones. Synthesis of pyrazinotetrahydroisoquinolines. Tetrahedron, 2004, 60, 6319-6326.
-
(2004)
Tetrahedron
, vol.60
, pp. 6319-6326
-
-
Gonzalez, J.F.1
Cuesta, E.2
Avendano, C.3
-
25
-
-
5644266177
-
One-step preparation of 1-substituted tetrahydroisoquinolines via the Pictet-Spengler reaction using zeolite catalysts
-
Hegedus, A.; Hell, Z. One-step preparation of 1-substituted tetrahydroisoquinolines via the Pictet-Spengler reaction using zeolite catalysts. Tetrahedron Lett., 2004, 45, 8553-8555.
-
(2004)
Tetrahedron Lett.
, vol.45
, pp. 8553-8555
-
-
Hegedus, A.1
Hell, Z.2
-
26
-
-
4143121319
-
Solid-Phase synthesis of 1,2,3,4-tetrahydroisoquinoline derivatives employing support-bound tyrosine esters in the pictetβspengler reaction
-
Kane, T.R.; Ly, C.Q.; Kelly, D.E.; Dener, J.M. Solid-Phase synthesis of 1,2,3,4-tetrahydroisoquinoline derivatives employing support-bound tyrosine esters in the pictetβspengler reaction. J. Comb. Chem., 2004, 6, 564-572.
-
(2004)
J. Comb. Chem.
, vol.6
, pp. 564-572
-
-
Kane, T.R.1
Ly, C.Q.2
Kelly, D.E.3
Dener, J.M.4
-
27
-
-
0842306887
-
Regiospecific, enantiospecific total synthesis of the 12-Alkoxysubstituted indole alkaloids, (+)-12-Methoxy-Na-methylvellosimine, (+)-12-Methoxyaffinisine, and (β)-Fuchsiaefoline
-
Zhou, H.; Liao, X.; Cook, J.M. Regiospecific, enantiospecific total synthesis of the 12-Alkoxysubstituted indole alkaloids, (+)-12-Methoxy-Na-methylvellosimine, (+)-12-Methoxyaffinisine, and (β)-Fuchsiaefoline. Org. Lett., 2004, 6, 249-252.
-
(2004)
Org. Lett.
, vol.6
, pp. 249-252
-
-
Zhou, H.1
Liao, X.2
Cook, J.M.3
-
28
-
-
22844431920
-
Solid-Phase synthesis of pyrroloisoquinolines via the intramolecular N-Acyliminium PictetβSpengler reaction
-
Nielsen, T.E.; Meldal, M. Solid-Phase synthesis of pyrroloisoquinolines via the intramolecular N-Acyliminium PictetβSpengler reaction. J. Comb. Chem., 2005, 7, 599-610.
-
(2005)
J. Comb. Chem.
, vol.7
, pp. 599-610
-
-
Nielsen, T.E.1
Meldal, M.2
-
29
-
-
0028834658
-
Solid phase synthesis of 1,2,3,4-tetrahydro-γ-carbolines; implications for combinatorial chemistry
-
Kaljuste, K.; Unden, A. Solid phase synthesis of 1,2,3,4-tetrahydro-γ-carbolines; implications for combinatorial chemistry. Tetrahedron Lett., 1995, 36, 9211-9214.
-
(1995)
Tetrahedron Lett.
, vol.36
, pp. 9211-9214
-
-
Kaljuste, K.1
Unden, A.2
-
30
-
-
0037048495
-
Pictet-Spengler synthesis of tetrahydro-γ-carbolines using vinylsulfonylmethyl resin
-
Connors, R.V.; Zhang, A.J.; Shuttleworth, S.J. Pictet-Spengler synthesis of tetrahydro-γ-carbolines using vinylsulfonylmethyl resin. Tetrahedron Lett., 2002, 43, 6661-6663.
-
(2002)
Tetrahedron Lett.
, vol.43
, pp. 6661-6663
-
-
Connors, R.V.1
Zhang, A.J.2
Shuttleworth, S.J.3
-
31
-
-
0034606938
-
Solid phase sequential 1,3-dipolar cycloaddition-Pictet-Spengler reactions
-
Dondas, H.A.; Grigg, R.; MacLachlan, W.S.; MacPherson, D.T.; Markandu, J.; Sridharan, V.; Suganthan, S. Solid phase sequential 1,3-dipolar cycloaddition-Pictet-Spengler reactions. Tetrahedron Lett., 2000, 41, 967-970.
-
(2000)
Tetrahedron Lett.
, vol.41
, pp. 967-970
-
-
Dondas, H.A.1
Grigg, R.2
McLachlan, W.S.3
McPherson, D.T.4
Markandu, J.5
Sridharan, V.6
Suganthan, S.7
-
32
-
-
0036831374
-
Solid-Phase synthesis of tetrahydro-γ-carbolinehydantoins via the N-Acyliminium pictetβspengler reaction and cyclative cleavage
-
Bonnet, D.; Ganesan, A. Solid-Phase synthesis of tetrahydro-γ-carbolinehydantoins via the N-Acyliminium pictetβspengler reaction and cyclative cleavage. J. Comb. Chem., 2002, 4, 546-548.
-
(2002)
J. Comb. Chem.
, vol.4
, pp. 546-548
-
-
Bonnet, D.1
Ganesan, A.2
-
33
-
-
85031233356
-
HR22C16: A potent small-molecule probe for the dynamics of cell division
-
Klein, C.; Ostrech, J.M.; Nefzi, A. HR22C16: A potent small-molecule probe for the dynamics of cell division. Tetrahedron Lett., 2003, 44, 2211-2215.
-
(2003)
Tetrahedron Lett.
, vol.44
, pp. 2211-2215
-
-
Klein, C.1
Ostrech, J.M.2
Nefzi, A.3
-
34
-
-
0038343601
-
Solid phase synthesis of tetrahydroisoquinolines & tetrahydroimidazopyridines
-
Hotha, S.; Yarrow, J.C.; Yang, J.G.; Garret, S.; Renduchintala, K.V.; Mayer, T.U.; Kapoor, T.M. Solid phase synthesis of tetrahydroisoquinolines & tetrahydroimidazopyridines. Angew Chem. Int. Ed., 2003, 42, 2379-2382.
-
(2003)
Angew Chem. Int. Ed.
, vol.42
, pp. 2379-2382
-
-
Hotha, S.1
Yarrow, J.C.2
Yang, J.G.3
Garret, S.4
Renduchintala, K.V.5
Mayer, T.U.6
Kapoor, T.M.7
-
35
-
-
0000802968
-
Study of the Pictet-Spengler reaction in aprotic media: Synthesis of the. beta.-galactosidase inhibitor, pyridindolol
-
Soerens, D.; Sandrin, J.; Ungemach, F.; Mokry, P.; Nu, G.S.; Yamanaka, E.; Hutchkins, L.; DiPierro, M.; Cook, J. M. Study of the Pictet-Spengler reaction in aprotic media: synthesis of the. beta.-galactosidase inhibitor, pyridindolol. J. Org. Chem., 1979, 44, 535-545.
-
(1979)
J. Org. Chem.
, vol.44
, pp. 535-545
-
-
Soerens, D.1
Sandrin, J.2
Ungemach, F.3
Mokry, P.4
Nu, G.S.5
Yamanaka, E.6
Hutchkins, L.7
DiPierro, M.8
Cook, J.M.9
-
36
-
-
0001476198
-
Synthesis of 1,2,3,4-Tetrahydro-γ-carbolines
-
Sandrin, J.; Soerens, D.; Mokry, P.; Cook, J.M. Synthesis of 1,2,3,4-Tetrahydro-γ-carbolines. Heterocycles, 1977, 6, 1133-1139.
-
(1977)
Heterocycles
, vol.6
, pp. 1133-1139
-
-
Sandrin, J.1
Soerens, D.2
Mokry, P.3
Cook, J.M.4
-
37
-
-
0030581372
-
Chiral ligands derived from Abrine. 3. Asymmetric Pictet-Spengler reaction of Abrine methyl ester and synthesis of chiral 1,2,3,4-tetrahydro-β-carbolines as promoters in addition of diethylzinc toward aromatic aldehydes
-
Dai, W.M.; Zhu, H.J.; Hao, X.J. Chiral ligands derived from Abrine. 3. Asymmetric Pictet-Spengler reaction of Abrine methyl ester and synthesis of chiral 1,2,3,4-tetrahydro-β-carbolines as promoters in addition of diethylzinc toward aromatic aldehydes. Tetrahedron Lett, 1996, 37, 5971-5974.
-
(1996)
Tetrahedron Lett
, vol.37
, pp. 5971-5974
-
-
Dai, W.M.1
Zhu, H.J.2
Hao, X.J.3
-
38
-
-
0026670664
-
Mechanism driven trans stereospecificity in the Pictet-Spengler reaction Stereospecific formation of trans-1,2,3-trisubstituted-tetrahydro β-carbolines by condensation of Nb-diphenylmethyl tryptophan isopropyl esters wtm aldehydes
-
Czerwinski, K.M.; Deng, L.; Cook, J.M. Mechanism driven trans stereospecificity in the Pictet-Spengler reaction. Stereospecific formation of trans-1,2,3-trisubstituted-tetrahydro β-carbolines by condensation of Nb-diphenylmethyl tryptophan isopropyl esters wtm aldehydes. Tetrahedron Lett., 1994, 33, 4721-4724.
-
(1994)
Tetrahedron Lett.
, vol.33
, pp. 4721-4724
-
-
Czerwinski, K.M.1
Deng, L.2
Cook, J.M.3
-
39
-
-
0003351386
-
Stereospecificity in the pictetspengler reaction Enantiospecific synthesis of (6S,10S)-(-)-5-Methyl-9-oxo-12-benzyl-6,7,8,9,10,11-hexahydro-6,10-imino -5H-cyclooct[b]indole, a template for preparation of macroline/sarpagine alkaloids
-
Zhang, L.H.; Bi, Y.Z.; Yu, F.X.; Menzia, G.; Cook, J.M. Stereospecificity in the pictetspengler reaction. Enantiospecific synthesis of (6S,10S)-(-)-5-Methyl-9-oxo-12-benzyl-6,7,8,9,10,11-hexahydro-6,10-imino -5H-cyclooct[b]indole, a template for preparation of macroline/sarpagine alkaloids. Heterocycles, 1992, 34, 517-547.
-
(1992)
Heterocycles
, vol.34
, pp. 517-547
-
-
Zhang, L.H.1
Bi, Y.Z.2
Yu, F.X.3
Menzia, G.4
Cook, J.M.5
-
40
-
-
0000801022
-
Stereospecific synthesis of trans-1,3-disubstituted-1,2,3,4-tetrahydro-. beta.-carbolines
-
Ungemach, F.; DiPierro, M.; Weber, R.; Cook, J.M. Stereospecific synthesis of trans-1,3-disubstituted-1,2,3,4-tetrahydro-. beta.-carbolines. J. Org. Chem., 1981, 46, 164-168.
-
(1981)
J. Org. Chem.
, vol.46
, pp. 164-168
-
-
Ungemach, F.1
DiPierro, M.2
Weber, R.3
Cook, J.M.4
-
41
-
-
33845471906
-
Pictet-Spengler reactions in aprotic media
-
Jawdosiuk, M.; Cook, J.M. Pictet-Spengler reactions in aprotic media. J. Org. Chem., 1984, 49, 2699-2701.
-
(1984)
J. Org. Chem.
, vol.49
, pp. 2699-2701
-
-
Jawdosiuk, M.1
Cook, J.M.2
-
42
-
-
0011551580
-
The N-Acyliminium PictetβSpengler condensation as a multicomponent combinatorial reaction on solid phase and its application to the synthesis of demethoxyfumitremorgin C analogues
-
Wang, H.; Ganesan, A. The N-Acyliminium PictetβSpengler condensation as a multicomponent combinatorial reaction on solid phase and its application to the synthesis of demethoxyfumitremorgin C analogues. Org Lett., 1999, 1, 1647-1649.
-
(1999)
Org Lett.
, vol.1
, pp. 1647-1649
-
-
Wang, H.1
Ganesan, A.2
-
43
-
-
0035810396
-
Diastereoselective synthesis of 1-benzyltetrahydroisoquinoline derivatives from amino acids via 1,4 chirality transfer. Part 1
-
Zawadzka, A.; Leniewski, A.; Maurin, J.K.; Wojtasiewicz, K.; Czarnocki, Z. Diastereoselective synthesis of 1-benzyltetrahydroisoquinoline derivatives from amino acids via 1,4 chirality transfer. Part 1. Org. Lett., 2001, 3, 997-999.
-
(2001)
Org. Lett.
, vol.3
, pp. 997-999
-
-
Zawadzka, A.1
Leniewski, A.2
Maurin, J.K.3
Wojtasiewicz, K.4
Czarnocki, Z.5
-
44
-
-
0035842128
-
Enantiopure tetrahydroisoquinolines via N-sulfinyl Pictet-Spengler reactions
-
Gremmen, C.; Wanner, M.J.; Koommen, G.J. Enantiopure tetrahydroisoquinolines via N-sulfinyl Pictet-Spengler reactions. Tetrahedron Lett., 2001, 42, 8885-8888.
-
(2001)
Tetrahedron Lett.
, vol.42
, pp. 8885-8888
-
-
Gremmen, C.1
Wanner, M.J.2
Koommen, G.J.3
-
45
-
-
0000219741
-
Enantiopure tetrahydro-γ-carbolines via pictetβspengler reactions with N-Sulfinyl tryptamines
-
Gremmen, C.; Willemse, B.; Wanner, M.J.; Koomen G.J. Enantiopure tetrahydro-γ-carbolines via pictetβspengler reactions with N-Sulfinyl tryptamines. Org. Lett., 2000, 2, 1955-1958.
-
(2000)
Org. Lett.
, vol.2
, pp. 1955-1958
-
-
Gremmen, C.1
Willemse, B.2
Wanner, M.J.3
Koomen, G.J.4
-
46
-
-
37049130362
-
Further cyclisation reactions of 1-arylpyrroles
-
Cheeseman, G.W.H.; Rafiq, M. Further cyclisation reactions of 1-arylpyrroles. J. Chem. Soc., 1971, 2732-2734.
-
(1971)
J. Chem. Soc.
, pp. 2732-2734
-
-
Cheeseman, G.W.H.1
Rafiq, M.2
-
47
-
-
84980231074
-
Mannich Reactions Synthesis of 4,5-Dihydropyrrolo[1,2-a]quinoxalines, 2,3,4,5-Tetrahydro-1H-pyrrolo[1,2-a][1,4]diazepines and 5,6-Dihydro-4H-pyrrolo[1,2-a][1,4]benzodiazepines
-
Raines, S.; Chai, S.Y.; Palopoli, F.P. Mannich Reactions. Synthesis of 4,5-Dihydropyrrolo[1,2-a]quinoxalines, 2,3,4,5-Tetrahydro-1H-pyrrolo[1,2-a][1,4]diazepines and 5,6-Dihydro-4H-pyrrolo[1,2-a][1,4]benzodiazepines. J. Heterocyclic Chem., 1976, 13, 711-716.
-
(1976)
J. Heterocyclic Chem.
, vol.13
, pp. 711-716
-
-
Raines, S.1
Chai, S.Y.2
Palopoli, F.P.3
-
48
-
-
0028886751
-
Pictet-Spengler reaction in trifluoroacetic acid Large scale synthesis of pyridoindolobenzodiazepine as an atypical antipsychotic agent
-
Zhang, L.H.; Meier, W.; Wats, E.; Costell, T.D.; Ma, P.; Ensinger, C.L.; Rodgers, J.M.; Jacobson, I. C.; Rajagopalan, P. Pictet-Spengler reaction in trifluoroacetic acid. Large scale synthesis of pyridoindolobenzodiazepine as an atypical antipsychotic agent. Tetrahedron Lett., 1995, 36, 8387-8391.
-
(1995)
Tetrahedron Lett.
, vol.36
, pp. 8387-8391
-
-
Zhang, L.H.1
Meier, W.2
Wats, E.3
Costell, T.D.4
Ma, P.5
Ensinger, C.L.6
Rodgers, J.M.7
Jacobson, I.C.8
Rajagopalan, P.9
-
49
-
-
0036889626
-
2-(Dimethylaminomethyl)-tetrahydroisoxazolopyridobenzazepine derivatives. Synthesis of a new 5-HT2C antagonist with potential anxiolytic properties
-
Andres, J.I.; Alonso, J.M.; Fernandez, J.; Iturrino, L.; Martinez, P.; Meert, T.F.; Sipido, V.K. 2-(Dimethylaminomethyl)-tetrahydroisoxazolopyridobenzazepine derivatives. Synthesis of a new 5-HT2C antagonist with potential anxiolytic properties. Bioorg. Med. Chem. Lett. 2002, 12, 3573-3577.
-
(2002)
Bioorg. Med. Chem. Lett.
, vol.12
, pp. 3573-3577
-
-
Andres, J.I.1
Alonso, J.M.2
Fernandez, J.3
Iturrino, L.4
Martinez, P.5
Meert, T.F.6
Sipido, V.K.7
-
50
-
-
17144384747
-
A Modified strategy for pictetβspengler reaction leading to the synthesis of imidazoquinoxalines on solid phase
-
Kundu, B.; Sawant, D.; Chhabra, R. A Modified strategy for pictetβspengler reaction leading to the synthesis of imidazoquinoxalines on solid phase. J. Comb. Chem., 2005, 7, 317-321.
-
(2005)
J. Comb. Chem.
, vol.7
, pp. 317-321
-
-
Kundu, B.1
Sawant, D.2
Chhabra, R.3
-
51
-
-
20344383734
-
New application of pictetβspengler reaction leading to the synthesis of an unusual seven-membered heterocyclic ring system
-
Kundu, B.; Sawant, D.; Partani, P.; Kesarwani, A.P. New application of pictetβspengler reaction leading to the synthesis of an unusual seven-membered heterocyclic ring system. J. Org. Chem., 2005, 70, 4889-4892.
-
(2005)
J. Org. Chem.
, vol.70
, pp. 4889-4892
-
-
Kundu, B.1
Sawant, D.2
Partani, P.3
Kesarwani, A.P.4
-
52
-
-
33644914455
-
Application of modified Pictet-Spengler reaction for the synthesis of thiazolo-and pyrazolo-quinolines
-
Duggineni, S.; Sawant, D.; Kundu, B. Application of modified Pictet-Spengler reaction for the synthesis of thiazolo-and pyrazolo-quinolines. Tetrahedron, 2006, 62, 3228-3241.
-
(2006)
Tetrahedron
, vol.62
, pp. 3228-3241
-
-
Duggineni, S.1
Sawant, D.2
Kundu, B.3
-
53
-
-
34948840010
-
Synthesis of Novel N-Rich Polycyclic Skeletons Based on Azoles and Pyridines
-
Sharma, S.; Saha, B.; Sawant, D.; Kundu, B. Synthesis of Novel N-Rich Polycyclic Skeletons Based on Azoles and Pyridines. J. Comb. Chem., 2007, 9, 783-792.
-
(2007)
J. Comb. Chem.
, vol.9
, pp. 783-792
-
-
Sharma, S.1
Saha, B.2
Sawant, D.3
Kundu, B.4
-
54
-
-
48049111168
-
Application of the Pictet-Spengler reaction to aryl amine substrates linked to deactivated aromatic heterosystems
-
Saha, B.; Sharma, S.; Sawant, D.; Kundu, B. Application of the Pictet-Spengler reaction to aryl amine substrates linked to deactivated aromatic heterosystems. Tetrahedron, 2008, 64, 8676-8684.
-
(2008)
Tetrahedron
, vol.64
, pp. 8676-8684
-
-
Saha, B.1
Sharma, S.2
Sawant, D.3
Kundu, B.4
-
55
-
-
58649119073
-
New route to the synthesis of the isocryptolepine alkaloid and its related skeletons using a modified pictetspengler reaction
-
Agarwal, P.K.; Sawant, D.; Sharma, S.; Kundu, B. New route to the synthesis of the isocryptolepine alkaloid and its related skeletons using a modified pictetspengler reaction. Eur. J. Org. Chem., 2009, 2, 292-303.
-
(2009)
Eur. J. Org. Chem.
, vol.2
, pp. 292-303
-
-
Agarwal, P.K.1
Sawant, D.2
Sharma, S.3
Kundu, B.4
-
56
-
-
58149170443
-
Application of the Pictet-Spengler reaction to aryl amine-based substrates having pyrimidine as a α-nucleophile: Synthesis of pyrimidoquinolines with structural analogy to benzonaphthyridines present in alkaloids
-
Agarwal, P.K.; Sharma, S.K.; Sawant, D.; Kundu, B. Application of the Pictet-Spengler reaction to aryl amine-based substrates having pyrimidine as a α-nucleophile: synthesis of pyrimidoquinolines with structural analogy to benzonaphthyridines present in alkaloids. Tetrahedron, 2009, 65, 1153-1161.
-
(2009)
Tetrahedron
, vol.65
, pp. 1153-1161
-
-
Agarwal, P.K.1
Sharma, S.K.2
Sawant, D.3
Kundu, B.4
-
57
-
-
63449115780
-
Application of 7-endo-trig Pictet-Spengler cyclization to the formation of the benzazepine Ring: Synthesis of benzazepinoindoles
-
Sharma, S.K.; Sharma, S.; Agarwal, P.K.; Kundu, B. Application of 7-endo-trig Pictet-Spengler cyclization to the formation of the benzazepine Ring: synthesis of benzazepinoindoles. Eur. J. Org. Chem., 2009, 9, 1309-1312.
-
(2009)
Eur. J. Org. Chem.
, vol.9
, pp. 1309-1312
-
-
Sharma, S.K.1
Sharma, S.2
Agarwal, P.K.3
Kundu, B.4
-
58
-
-
72149120610
-
Regioselective intramolecular electrophilic substitution reactions involving α-deficient pyridine substrates: A new entry to pyridoquinazolines and benzo[h][1,6]naphthyridines
-
Agarwal, P.K.; Saifuddin, M.; Kundu, B. Regioselective intramolecular electrophilic substitution reactions involving α-deficient pyridine substrates: a new entry to pyridoquinazolines and benzo[h][1,6]naphthyridines. Tetrahedron, 2010, 66, 862-870.
-
(2010)
Tetrahedron
, vol.66
, pp. 862-870
-
-
Agarwal, P.K.1
Saifuddin, M.2
Kundu, B.3
-
59
-
-
67549112170
-
A new entry to phenanthridine ring systems via sequential application of Suzuki and the modified Pictet-Spengler reactions
-
Mandadapu, K.A.; Saifuddin, M.; Agarwal, P.K. A new entry to phenanthridine ring systems via sequential application of Suzuki and the modified Pictet-Spengler reactions. Org. Biomol. Chem., 2009, 7, 2796-2803.
-
(2009)
Org. Biomol. Chem.
, vol.7
, pp. 2796-2803
-
-
Mandadapu, K.A.1
Saifuddin, M.2
Agarwal, P.K.3
-
60
-
-
28244479033
-
Solid-Phase synthesis of 2-Aminoquinazolinone derivatives with Two-and Three-Point diversity
-
Kundu, B.; Partani, P.; Duggineni, S.; Sawant, D. Solid-Phase synthesis of 2-Aminoquinazolinone derivatives with Two-and Three-Point diversity. J. Comb. Chem., 2005, 7, 909-915.
-
(2005)
J. Comb. Chem.
, vol.7
, pp. 909-915
-
-
Kundu, B.1
Partani, P.2
Duggineni, S.3
Sawant, D.4
-
61
-
-
67650692766
-
Application of the modified pictetβspengler cyclization reaction for the preparation of an imidazopyrazine ring: Synthesis of new Pyrido-and Pyrimidoimidazopyrazines
-
Sharma, S.; Kundu, B. Application of the modified pictetβspengler cyclization reaction for the preparation of an imidazopyrazine ring: Synthesis of new Pyrido-and Pyrimidoimidazopyrazines. J. Comb. Chem., 2009, 11, 720-731.
-
(2009)
J. Comb. Chem.
, vol.11
, pp. 720-731
-
-
Sharma, S.1
Kundu, B.2
-
62
-
-
33846382303
-
Water as an efficient medium for the synthesis of tetrahydro-β-carbolines via Pictet-Spengler reactions
-
Saha, B.; Sharma, S.; Sawant, D.; Kundu, B. Water as an efficient medium for the synthesis of tetrahydro-β-carbolines via Pictet-Spengler reactions. Tetrahedron Lett., 2007, 48, 1379-1383.
-
(2007)
Tetrahedron Lett.
, vol.48
, pp. 1379-1383
-
-
Saha, B.1
Sharma, S.2
Sawant, D.3
Kundu, B.4
-
63
-
-
77956387439
-
Water-Accelerated cationic α-(7-endo) cyclisation: Application to indole-based peri-annulated polyheterocycles
-
Saifuddin, M.; Agarwal, P.K.; Sharma, S.; Mandadapu, K.A.; Gupta, S.; Harit, V.K. Water-Accelerated cationic α-(7-endo) cyclisation: Application to indole-based peri-annulated polyheterocycles. Eur. J. Org. Chem., 2010, 26, 5108-5117.
-
(2010)
Eur. J. Org. Chem.
, vol.26
, pp. 5108-5117
-
-
Saifuddin, M.1
Agarwal, P.K.2
Sharma, S.3
Mandadapu, K.A.4
Gupta, S.5
Harit, V.K.6
-
64
-
-
33947153856
-
Synthesis of novel substituted naphthoquino[b]-benzo[e][1,4]diazepines via Pictet-Spengler cyclisation
-
Wang, X.L.; Zheng, X.F.; Liu, R.H.; Reiner, J.; Chang, J.B. Synthesis of novel substituted naphthoquino[b]-benzo[e][1,4]diazepines via Pictet-Spengler cyclisation. Tetrahedron, 2007, 63, 3389-3394.
-
(2007)
Tetrahedron
, vol.63
, pp. 3389-3394
-
-
Wang, X.L.1
Zheng, X.F.2
Liu, R.H.3
Reiner, J.4
Chang, J.B.5
-
65
-
-
11144324252
-
-
Katritzky, A.R., Rees, C, W., Eds.; Pergamon Press Ltd.: London
-
Katritzky, A.R. In Comprehensive Heterocyclic Chemistry; Katritzky, A.R., Rees, C. W., Eds.; Pergamon Press Ltd.: London, 1984, 41-110.
-
(1984)
In Comprehensive Heterocyclic Chemistry
, pp. 41-110
-
-
Katritzky, A.R.1
-
66
-
-
53849135238
-
New strategies for the synthesis of pyrimidine derivatives
-
For a recent review see
-
For a recent review see: Hill M.D.; Movassaghi, M. New strategies for the synthesis of pyrimidine derivatives. Chem. Eur. J., 2008, 14, 6836-6844.
-
(2008)
Chem. Eur. J.
, vol.14
, pp. 6836-6844
-
-
Hill, M.D.1
Movassaghi, M.2
-
67
-
-
84943378078
-
-
Katritzky, A.R., Rees, C.W., Eds.; Pergamon Press Ltd.: London
-
Metzger, J.V. In Comprehensive Heterocyclic Chemistry; Katritzky, A.R., Rees, C.W., Eds.; Pergamon Press Ltd.: London, 1984, 235-330.
-
(1984)
In Comprehensive Heterocyclic Chemistry
, pp. 235-330
-
-
Metzger, J.V.1
-
68
-
-
4243241249
-
The Pictet-Spengler condensation: A new direction for an old reaction
-
Cox, E.D.; Cook, J. The Pictet-Spengler condensation: a new direction for an old reaction. Chem. Rev., 1995, 95, 1797-1842.
-
(1995)
Chem. Rev.
, vol.95
, pp. 1797-1842
-
-
Cox, E.D.1
Cook, J.2
-
69
-
-
0037366605
-
The combinatorial synthesis of bicyclic privileged structures or privileged substructures
-
For a review on privileged structures as starting point for library synthesis, see
-
For a review on privileged structures as starting point for library synthesis, see: Horton, D.A.; Bourne, G.T.; Smythe, M.L. The combinatorial synthesis of bicyclic privileged structures or privileged substructures. Chem. Rev., 2003, 103, 893-930.
-
(2003)
Chem. Rev.
, vol.103
, pp. 893-930
-
-
Horton, D.A.1
Bourne, G.T.2
Smythe, M.L.3
-
70
-
-
4644316145
-
Effects of new ubiquinone-imidazo[2,1-b]thiazoles on mitochondrial complex I (NADHubiquinone reductase) and on mitochondrial permeability transition pore
-
Andreani, A.; Granaiola, M.; Leoni, A.; Locatelli, A.; Morigi, R.; Rambaldi, M.; Recanatini, M.; Lenaz, G.; Fato, R.; Bergamini, C. Effects of new ubiquinone-imidazo[2,1-b]thiazoles on mitochondrial complex I (NADHubiquinone reductase) and on mitochondrial permeability transition pore. Bioorg. Med. Chem., 2004, 12, 5525-5532.
-
(2004)
Bioorg. Med. Chem.
, vol.12
, pp. 5525-5532
-
-
Andreani, A.1
Granaiola, M.2
Leoni, A.3
Locatelli, A.4
Morigi, R.5
Rambaldi, M.6
Recanatini, M.7
Lenaz, G.8
Fato, R.9
Bergamini, C.10
-
71
-
-
33645893175
-
Optimization of 2-aminothiazole derivatives as CCR4 antagonists
-
Wang, X.; Xu, F.; Xu, Q.; Mahmud, H.; Houze, J.; Zhu, L.; Akerman, M.; Tonn, G.; Tang, l.; McMaster, B.E.; Dairaghi, d.J.; Schall, T.J.; Collins, T.L.; Medina, J.C. Optimization of 2-aminothiazole derivatives as CCR4 antagonists. Bioorg. Med. Chem. Lett., 2006, 16, 2800-2803.
-
(2006)
Bioorg. Med. Chem. Lett.
, vol.16
, pp. 2800-2803
-
-
Wang, X.1
Xu, F.2
Xu, Q.3
Mahmud, H.4
Houze, J.5
Zhu, L.6
Akerman, M.7
Tonn, G.8
Tang, L.9
McMaster, B.E.10
Dairaghi, D.J.11
Schall, T.J.12
Collins, T.L.13
Medina, J.C.14
-
72
-
-
0032693483
-
6-Thienyl and 6-phenylimidazo[2,1-b]thiazoles as inhibitors of mitochondrial NADH dehydrogenase
-
Andreani, A.; Rambaldi, M.; Leoni, A.; Morigi, R.; Locatelli, A.; Ghelli, A.; Esposti, M.D.; Ratta, M.; Benelli, B.; Degli Espoti, M. 6-Thienyl and 6-phenylimidazo[2,1-b]thiazoles as inhibitors of mitochondrial NADH dehydrogenase. Eur. J. Med. Chem., 1999, 34, 883-889.
-
(1999)
Eur. J. Med. Chem.
, vol.34
, pp. 883-889
-
-
Andreani, A.1
Rambaldi, M.2
Leoni, A.3
Morigi, R.4
Locatelli, A.5
Ghelli, A.6
Esposti, M.D.7
Ratta, M.8
Benelli, B.9
Degli Espoti, M.10
-
73
-
-
38349075672
-
Use of the Pictet-Spengler reaction for the synthesis of 1,4-disubstituted-1,2,3,4-tetrahydro-α-carbolines and 1,4-disubstituted-α-carbolines: Formation of α-carbolines
-
Kusurkar, R.S.; Alkobati, N.A.H.; Gokule, A.S.; Puranik, V.G. Use of the Pictet-Spengler reaction for the synthesis of 1,4-disubstituted-1,2,3,4-tetrahydro-α-carbolines and 1,4-disubstituted-α-carbolines: formation of α-carbolines. Tetrahedron, 2008, 64, 1654-1662
-
(2008)
Tetrahedron
, vol.64
, pp. 1654-1662
-
-
Kusurkar, R.S.1
Alkobati, N.A.H.2
Gokule, A.S.3
Puranik, V.G.4
-
74
-
-
0000223992
-
-
(Katritzky, A.R., Rees, C.W., Eds.), Pergamon Press, London
-
Jones, R.A. In Comprehensive Heterocyclic Chemistry (Katritzky, A.R., Rees, C.W., Eds.), Pergamon Press, London, 1984, vol. 4, pp. 205-206.
-
(1984)
In Comprehensive Heterocyclic Chemistry
, vol.4
, pp. 205-206
-
-
Jones, R.A.1
-
75
-
-
26444617730
-
-
(Brossi, A., Ed.), Academic Press, San Diego, chapter 7
-
Gribble, G.W. The Alkaloids (Brossi, A., Ed.), Academic Press, San Diego, 1990, vol. 39, chapter 7
-
(1990)
The Alkaloids
, vol.39
-
-
Gribble, G.W.1
-
76
-
-
85038478846
-
-
(Blum M.S. Ed.), Alaken, Ft. Collins (Colorado, USA)
-
Pezzuto, J.M. Chemistry and Toxicology of Diverse Classes of Alkaloids (Blum M.S. Ed.), Alaken, Ft. Collins (Colorado, USA), 1996, pp. 1-119.
-
(1996)
Chemistry and Toxicology of Diverse Classes of Alkaloids
, pp. 1-119
-
-
Pezzuto, J.M.1
-
77
-
-
0242528072
-
The action of acyl cyanides on 2-and 1: 2-substituted indoles. Part II. Derivatives of 2-oaminophenylindole
-
Kiang, A.K.; Mann, A.F.; Prior, A.F.; Topham, A. The action of acyl cyanides on 2-and 1: 2-substituted indoles. Part II. Derivatives of 2-oaminophenylindole. J. Chem. Soc., 1956, 1319-1331.
-
(1956)
J. Chem. Soc.
, pp. 1319-1331
-
-
Kiang, A.K.1
Mann, A.F.2
Prior, A.F.3
Topham, A.4
-
78
-
-
2742543376
-
-
Duncan, R. L.; Helsey, G. C.; Boswell, R. F. J. Heterocycl. Chem., 1973, 10, 65-70.
-
(1973)
J. Heterocycl. Chem.
, vol.10
, pp. 65-70
-
-
Duncan, R.L.1
Helsey, G.C.2
Boswell, R.F.3
-
79
-
-
0037368393
-
Design of antineoplastic agents based on the '2-phenylnaphthalene-type' structural pattern-synthesis and biological activity studies of 11H-indolo[3.2-c]quinoline derivatives
-
He, L.; Chang, H.X.; Chou, T.C.; Savaraj, N.; Cheng, C.C. Design of antineoplastic agents based on the '2-phenylnaphthalene-type' structural pattern-synthesis and biological activity studies of 11H-indolo[3.2-c]quinoline derivatives. Eur. J. Med. Chem., 2003, 38, 101-107.
-
(2003)
Eur. J. Med. Chem.
, vol.38
, pp. 101-107
-
-
He, L.1
Chang, H.X.2
Chou, T.C.3
Savaraj, N.4
Cheng, C.C.5
-
80
-
-
53849100355
-
Auto-Tandem catalysis: Synthesis of substituted 11H-Indolo [3,2-c]quinolines via palladium-catalyzed intermolecular C_N and intramolecular C_C bond formation
-
Meyers, C.; Rombouts, G.; Loones, K.T.J.; Coelho, A.; Maes, B.U.W. Auto-Tandem catalysis: synthesis of substituted 11H-Indolo [3,2-c]quinolines via palladium-catalyzed intermolecular C_N and intramolecular C_C bond formation. Adv. Synth. Catal., 2008, 350, 465-470.
-
(2008)
Adv. Synth. Catal.
, vol.350
, pp. 465-470
-
-
Meyers, C.1
Rombouts, G.2
Loones, K.T.J.3
Coelho, A.4
Maes, B.U.W.5
-
81
-
-
38849090728
-
Synthesis of novel pyrimidine fused 8-Membered heterocycles via iminium ion cyclization reactions
-
Che, X.; Zheng, L.; Dang, Q.; Bai, X. Synthesis of novel pyrimidine fused 8-Membered heterocycles via iminium ion cyclization reactions. J. Org. Chem., 2008, 73, 1147-1149.
-
(2008)
J. Org. Chem.
, vol.73
, pp. 1147-1149
-
-
Che, X.1
Zheng, L.2
Dang, Q.3
Bai, X.4
-
82
-
-
28244493092
-
Novel heterocyclic scaffold consisting of indole-fused pteridines
-
Zheng, L.; Xiang, J.; Daang, Q.D.; Bai, X. Novel heterocyclic scaffold consisting of indole-fused pteridines. J. Comb. Chem., 2005, 7, 813-815.
-
(2005)
J. Comb. Chem.
, vol.7
, pp. 813-815
-
-
Zheng, L.1
Xiang, J.2
Daang, Q.D.3
Bai, X.4
-
83
-
-
34447621974
-
Heck-like coupling and Pictet-Spengler reaction for the synthesis of benzothieno[3,2-c]quinolines
-
David, E.; Pellet-Rostaing, S.; Lemaire, M. Heck-like coupling and Pictet-Spengler reaction for the synthesis of benzothieno[3,2-c]quinolines. Tetrahedron, 2007, 63, 8999-9006.
-
(2007)
Tetrahedron
, vol.63
, pp. 8999-9006
-
-
David, E.1
Pellet-Rostaing, S.2
Lemaire, M.3
-
84
-
-
2942708002
-
A new entry to the substituted pyrrolo[3,2-c]quinoline derivatives of biological interest by intramolecular heteroannulation of internal imines
-
Testa, M.L.; Lamartina, L.; Mingoia, F. A new entry to the substituted pyrrolo[3,2-c]quinoline derivatives of biological interest by intramolecular heteroannulation of internal imines. Tetrahedron, 2004, 60, 5873-5880.
-
(2004)
Tetrahedron
, vol.60
, pp. 5873-5880
-
-
Testa, M.L.1
Lamartina, L.2
Mingoia, F.3
-
85
-
-
84990131664
-
-
Katritzky, A.R., Ed.; Pergamon Press, London
-
Katritzky, A.R. In Comprehensive Heterocyclic Chemistry; Katritzky, A.R., Ed.; Pergamon Press, London, 1984; Vol. 3, pp. 68-71.
-
(1984)
In Comprehensive Heterocyclic Chemistry
, vol.3
, pp. 68-71
-
-
Katritzky, A.R.1
-
86
-
-
4344713238
-
Highly enantioselective catalytic acylpictet βspengler reactions
-
Taylor, M.S.; Jacobsen, E.N. highly enantioselective catalytic acylpictet βspengler reactions. J. Am. Chem. Soc., 2004, 126, 10558-10559.
-
(2004)
J. Am. Chem. Soc.
, vol.126
, pp. 10558-10559
-
-
Taylor, M.S.1
Jacobsen, E.N.2
-
87
-
-
0037425327
-
Highly efficient Lewis acid-catalysed Pictet-Spengler reactions discovered by parallel screening
-
Srinivasan, N.; Ganesan, A. Highly efficient Lewis acid-catalysed Pictet-Spengler reactions discovered by parallel screening. Chem. Commun., 2003, 916-917.
-
(2003)
Chem. Commun.
, pp. 916-917
-
-
Srinivasan, N.1
Ganesan, A.2
-
88
-
-
0037433930
-
General approach for the total synthesis of the sarpagine related indole alkaloids (+)-Na-methyl-16-epipericyclivine, (β)-alkaloid Q3 and (β)-panarine via the asymmetric Pictet-Spengler reaction
-
Yu, J.; Wearing, X.Z.; Cook, J. M. General approach for the total synthesis of the sarpagine related indole alkaloids (+)-Na-methyl-16-epipericyclivine, (β)-alkaloid Q3 and (β)-panarine via the asymmetric Pictet-Spengler reaction. Tetrahedron Lett., 2003, 44, 543-547.
-
(2003)
Tetrahedron Lett.
, vol.44
, pp. 543-547
-
-
Yu, J.1
Wearing, X.Z.2
Cook, J.M.3
-
89
-
-
19544381560
-
Silicon-Directed oxa-PictetβSpengler cyclization and an unusual dimerization of 2-Trimethylsilanyl tryptophols
-
Zhang, X.; Li, X.; Lanter, J. C.; Sui, Z. Silicon-Directed oxa-PictetβSpengler cyclization and an unusual dimerization of 2-Trimethylsilanyl tryptophols. Org. Lett., 2005, 7, 2043-2046.
-
(2005)
Org. Lett.
, vol.7
, pp. 2043-2046
-
-
Zhang, X.1
Li, X.2
Lanter, J.C.3
Sui, Z.4
-
90
-
-
0024239320
-
Methods for drug discovery: Development of potent, selective, orally effective cholecystokinin antagonists
-
Evans, B.E.; Rittle, K.E.; Bock, M.G.; DiPardo, R.M.; Freidinger, R.M.; Whitter, W.L.; Lundell, G.F.; Veber, D.F.; Anderson, P.S. Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonists. J. Med. Chem., 1988, 31, 2235-2246.
-
(1988)
J. Med. Chem.
, vol.31
, pp. 2235-2246
-
-
Evans, B.E.1
Rittle, K.E.2
Bock, M.G.3
DiPardo, R.M.4
Freidinger, R.M.5
Whitter, W.L.6
Lundell, G.F.7
Veber, D.F.8
Anderson, P.S.9
-
91
-
-
0033606988
-
New 4-Point pharmacophore method for molecular similarity and diversity applications: Overview of the method and applications, including a novel approach to the design of combinatorial libraries containing privileged substructures
-
Mason, J.S.; Morize, I.; Menard, P.R.; Cheney, D.L.; Hulme, C.; Labaudiniere, R.F. New 4-Point pharmacophore method for molecular similarity and diversity applications: overview of the method and applications, including a novel approach to the design of combinatorial libraries containing privileged substructures. J. Med. Chem., 1999, 42, 3251-3264.
-
(1999)
J. Med. Chem.
, vol.42
, pp. 3251-3264
-
-
Mason, J.S.1
Morize, I.2
Menard, P.R.3
Cheney, D.L.4
Hulme, C.5
Labaudiniere, R.F.6
-
92
-
-
0034684250
-
Natural product-like combinatorial libraries based on privileged structures. 1. General Principles and Solid-Phase Synthesis of Benzopyrans
-
Nicolaou, K.C.; Pfefferkorn, J. A.; Roecker, A.J.; Cao, G.-Q.; Barluenga, S.; Mitchell, H. J. Natural product-like combinatorial libraries based on privileged structures. 1. General Principles and Solid-Phase Synthesis of Benzopyrans. J. Am. Chem. Soc., 2000, 122, 9939-9953.
-
(2000)
J. Am. Chem. Soc.
, vol.122
, pp. 9939-9953
-
-
Nicolaou, K.C.1
Pfefferkorn, J.A.2
Roecker, A.J.3
Cao, G.-Q.4
Barluenga, S.5
Mitchell, H.J.6
-
93
-
-
0042121318
-
Medicinal chemistry of target family-directed masterkeys
-
Muller, G. Medicinal chemistry of target family-directed masterkeys. Drug Discov. Today, 2003, 8, 681-691.
-
(2003)
Drug Discov. Today
, vol.8
, pp. 681-691
-
-
Muller, G.1
-
94
-
-
33644876210
-
DrugBank: A comprehensive resource for in silico drug discovery and exploration
-
Wishart, D.S.; Knox, C.; Guo, A.C.; Shrivastava, S.; Hassanali, M.; Stothard, P.; Chang, Z.; Woolsey, J. DrugBank: a comprehensive resource for in silico drug discovery and exploration. Nucleic Acids Res., 2006, D668-D672.
-
(2006)
Nucleic Acids Res.
-
-
Wishart, D.S.1
Knox, C.2
Guo, A.C.3
Shrivastava, S.4
Hassanali, M.5
Stothard, P.6
Chang, Z.7
Woolsey, J.8
-
95
-
-
4444269491
-
Voriconazole: Therapeutic review of a new azole antifungal
-
Herbrecht, R. Voriconazole: therapeutic review of a new azole antifungal. Expert Rev. Anti Infect. Ther., 2004, 485-497.
-
(2004)
Expert Rev. Anti Infect. Ther.
, pp. 485-497
-
-
Herbrecht, R.1
-
96
-
-
34548488008
-
Pyrimidine as antiinflammatory agent: A review
-
Amir, M.; Javed, S.A.; Kumar, H. Pyrimidine as antiinflammatory agent: A review. Indian J. Pharm. Sci., 2007, 69, 337-343.
-
(2007)
Indian J. Pharm. Sci.
, vol.69
, pp. 337-343
-
-
Amir, M.1
Javed, S.A.2
Kumar, H.3
-
97
-
-
0002014103
-
-
Katritzky, A. R., Rees, C, W., Eds.; Pergamon: Oxford, New York, NY
-
Katritzky, A.R. In Comprehensive Heterocyclic Chemistry; Katritzky, A. R., Rees, C. W., Eds.; Pergamon: Oxford, New York, NY, 1984; Vol. 2, pp. 29-31.
-
(1984)
In Comprehensive Heterocyclic Chemistry
, vol.2
, pp. 29-31
-
-
Katritzky, A.R.1
-
98
-
-
0038729563
-
Microwave enhanced formation of electron rich arylboronates
-
Appukkuttan, P.; Van der Eycken, E.; Dehaen, W. Microwave enhanced formation of electron rich arylboronates. Synlett, 2003, 8, 1204-1206.
-
(2003)
Synlett
, vol.8
, pp. 1204-1206
-
-
Appukkuttan, P.1
van der Eycken, E.2
Dehaen, W.3
-
99
-
-
0001899311
-
Lithiation of methoxypyridines directed by. alpha.-amino alkoxides
-
Comins, D.L.; Killpack, M.O. Lithiation of methoxypyridines directed by. alpha.-amino alkoxides. J. Org. Chem., 1990, 55, 69-73.
-
(1990)
J. Org. Chem.
, vol.55
, pp. 69-73
-
-
Comins, D.L.1
Killpack, M.O.2
-
100
-
-
0030743362
-
Electrophilic aromatic substitution on pyridine rings Intramolecular cyclization using N-Acyliminium ions
-
Brodney, M.A.; Padwa, A. Electrophilic aromatic substitution on pyridine rings. Intramolecular cyclization using N-Acyliminium ions. Tetrahedron Lett., 1997, 38, 6153-6156.
-
(1997)
Tetrahedron Lett.
, vol.38
, pp. 6153-6156
-
-
Brodney, M.A.1
Padwa, A.2
-
101
-
-
0020406552
-
Isolation and structure of aaptamine a novel heteroaromatic substance possessing γ-blocking activity from the sea sponge
-
Nakamura, H.; Kobayashi, J.; Ohizumi, Y. Isolation and structure of aaptamine a novel heteroaromatic substance possessing γ-blocking activity from the sea sponge. Tetrahedron Lett., 1982, 23, 5555-5558.
-
(1982)
Tetrahedron Lett.
, vol.23
, pp. 5555-5558
-
-
Nakamura, H.1
Kobayashi, J.2
Ohizumi, Y.3
-
102
-
-
33750308939
-
Electrophilic allylations and benzylations of indoles in neutral aqueous or alcoholic solutions
-
Westermaier, M.; Mayr, H. Electrophilic allylations and benzylations of indoles in neutral aqueous or alcoholic solutions. Org. Lett., 2006, 8, 4791-4794.
-
(2006)
Org. Lett.
, vol.8
, pp. 4791-4794
-
-
Westermaier, M.1
Mayr, H.2
-
103
-
-
0036944830
-
Synthesis of Cryptolepine and Cryptotackieine from a Common Intermediate
-
Ho, T.L.; Jou, D. G. Synthesis of Cryptolepine and Cryptotackieine from a Common Intermediate. Helv. Chim. Acta, 2002, 85, 3823-3827.
-
(2002)
Helv. Chim. Acta
, vol.85
, pp. 3823-3827
-
-
Ho, T.L.1
Jou, D.G.2
-
104
-
-
48349088650
-
Synthesis of new pyrrolobenzazepines via pictet-spengler cyclization
-
Gracia, S.; Schulz, J.; Pellet-Rostaing, S. Synthesis of new pyrrolobenzazepines via pictet-spengler cyclization. Synlett, 2008, 1852-1856.
-
(2008)
Synlett
, pp. 1852-1856
-
-
Gracia, S.1
Schulz, J.2
Pellet-Rostaing, S.3
-
105
-
-
34347394771
-
Cu-FeCl3 one pot multicomponent reaction leading to the synthesis of N-aryl/alkyl triazoles in water
-
Saha, B.; Sharma, S.; Sawant, D.; Kundu, B. Cu-FeCl3 one pot multicomponent reaction leading to the synthesis of N-aryl/alkyl triazoles in water. Synlett, 2007, 1591-94.
-
(2007)
Synlett
, pp. 1591-1594
-
-
Saha, B.1
Sharma, S.2
Sawant, D.3
Kundu, B.4
-
106
-
-
33846382303
-
Water as an efficient medium for the synthesis of tetrahydro-aa-carbolines via Pictet-Spengler reactions
-
Saha, B.; Sharma, S.; Sawant, D.; Kundu, B. Water as an efficient medium for the synthesis of tetrahydro-aa-carbolines via Pictet-Spengler reactions. Tetrahedron Lett., 2007, 48, 1379-1382.
-
(2007)
Tetrahedron Lett.
, vol.48
, pp. 1379-1382
-
-
Saha, B.1
Sharma, S.2
Sawant, D.3
Kundu, B.4
-
107
-
-
27744581943
-
Preparation of substituted Pyrimido[4,5-b]-1,4-benzoxazepines, thiazepines, and diazepines via a pictetβspengler cyclization
-
Duncton, M.A.J.; Smith II, L.M.; Burdzovic-Wizeman, S.; Burns, A.; Liu, H.; Mao, Y.; Wong, W.C.; Kiselyov, A.S. Preparation of substituted Pyrimido[4,5-b]-1,4-benzoxazepines, thiazepines, and diazepines via a pictetβspengler cyclization. J. Org. Chem., 2005, 70, 9629-9631.
-
(2005)
J. Org. Chem.
, vol.70
, pp. 9629-9631
-
-
Duncton, M.A.J.1
Smith II, L.M.2
Burdzovic-Wizeman, S.3
Burns, A.4
Liu, H.5
Mao, Y.6
Wong, W.C.7
Kiselyov, A.S.8
-
108
-
-
33744455765
-
Design and synthesis of a tetracyclic pyrimidine-fused benzodiazepine library
-
Zheng, L.; Xiang, J.; Dang, Q.; Guo, S.; Bai, X. Design and synthesis of a tetracyclic pyrimidine-fused benzodiazepine library. J. Comb. Chem., 2006, 8, 381-387.
-
(2006)
J. Comb. Chem.
, vol.8
, pp. 381-387
-
-
Zheng, L.1
Xiang, J.2
Dang, Q.3
Guo, S.4
Bai, X.5
-
109
-
-
33750495371
-
Modification at the C9 position of the marine natural product isoaaptamine and the impact on HIV-1, mycobacterial, and tumor cell activity
-
Gul, W.; Hammond, N. L.; Yousaf, M.; Bowling, J. J.; Schinazi, R. F.; Wirtz, S. S.; Andrews, G. A.; Cuevas, C.; Hamann, M. T. Modification at the C9 position of the marine natural product isoaaptamine and the impact on HIV-1, mycobacterial, and tumor cell activity. Bioorg. Med. Chem. 2006, 14, 8495-8505.
-
(2006)
Bioorg. Med. Chem.
, vol.14
, pp. 8495-8505
-
-
Gul, W.1
Hammond, N.L.2
Yousaf, M.3
Bowling, J.J.4
Schinazi, R.F.5
Wirtz, S.S.6
Andrews, G.A.7
Cuevas, C.8
Hamann, M.T.9
-
110
-
-
12144287559
-
Isolation and X-ray crystal structure determination of isoaaptamine from the republic of singapore Hymeniacidon sp. and conversion to the phosphate prodrug hystatin 1
-
Antineoplastic Agents. 380
-
Pettit, G. R.; Hoffmann, H.; McNulty, J.; Higgs, K. C.; Murphy, A.; Molloy, D. J.; Herald, D. L.; Williams, M. D.; Pettit, R. K.; Doubek, D. L.; Hooper, J. N. A.; Albright, L.; Schmidt, J. M.; Chapuis, J.-C.; Tackett, L. P. Antineoplastic Agents. 380. Isolation and X-ray crystal structure determination of isoaaptamine from the republic of singapore Hymeniacidon sp. and conversion to the phosphate prodrug hystatin 1. J. Nat. Prod. 2004, 67, 506-509.
-
(2004)
J. Nat. Prod.
, vol.67
, pp. 506-509
-
-
Pettit, G.R.1
Hoffmann, H.2
McNulty, J.3
Higgs, K.C.4
Murphy, A.5
Molloy, D.J.6
Herald, D.L.7
Williams, M.D.8
Pettit, R.K.9
Doubek, D.L.10
Hooper, J.N.A.11
Albright, L.12
Schmidt, J.M.13
Chapuis, J.-C.14
Tackett, L.P.15
-
111
-
-
0037451847
-
Discovery and SAR of novel [and]Naphthyridines as potent inhibitors of spleen tyrosine kinase (SYK)
-
Cywin, C. L.; Zhao, B.-P.; McNeil, D. W.; Hrapchak, M.; Prokopowicz, A. S., III; Goldberg, D. R.; Morwick, T. M.; Gao, A.; Jakes, S.; Kashem, M.; Magolda, R. L.; Soll, R. M.; Player, M. R.; Bobko, M. A.; Rinker, J.; DesJarlais, R. L.; Winters, M. P. Discovery and SAR of novel [and]Naphthyridines as potent inhibitors of spleen tyrosine kinase (SYK). Bioorg. Med. Chem. Lett. 2003, 13, 1415-1418.
-
(2003)
Bioorg. Med. Chem. Lett.
, vol.13
, pp. 1415-1418
-
-
Cywin, C.L.1
Zhao, B.-P.2
McNeil, D.W.3
Hrapchak, M.4
Prokopowicz III, A.S.5
Goldberg, D.R.6
Morwick, T.M.7
Gao, A.8
Jakes, S.9
Kashem, M.10
Magolda, R.L.11
Soll, R.M.12
Player, M.R.13
Bobko, M.A.14
Rinker, J.15
DesJarlais, R.L.16
Winters, M.P.17
-
112
-
-
0035137292
-
Marine natural products
-
Faulkner, D. J. Marine natural products. Nat. Prod. Rep., 2001, 18, 1-49.
-
(2001)
Nat. Prod. Rep.
, vol.18
, pp. 1-49
-
-
Faulkner, D.J.1
-
113
-
-
18244400107
-
Synthesis and in vitro and in vivo antitumor activity of 2-Phenylpyrroloquinolin-4-ones
-
Ferlin, M. G.; Chiarelotto, G.; Gasparotto, V.; Via, L. D.; Pezzi, V.; Barzon, L.; Palù, G.; Castagliuolo, I. Synthesis and in vitro and in vivo antitumor activity of 2-Phenylpyrroloquinolin-4-ones. J. Med. Chem., 2005, 48, 3417-3427.
-
(2005)
J. Med. Chem.
, vol.48
, pp. 3417-3427
-
-
Ferlin, M.G.1
Chiarelotto, G.2
Gasparotto, V.3
Via, L.D.4
Pezzi, V.5
Barzon, L.6
Palù, G.7
Castagliuolo, I.8
-
114
-
-
33746864043
-
Practical methodologies for the synthesis of indoles
-
Humphrey, G. R.; Kuethe, J. T. Practical methodologies for the synthesis of indoles. Chem. Rev., 2006, 106, 2875-2911.
-
(2006)
Chem. Rev.
, vol.106
, pp. 2875-2911
-
-
Humphrey, G.R.1
Kuethe, J.T.2
-
115
-
-
2942598364
-
Synthesis of polyheterocyclic nitrogen-containing marine natural products
-
Fernández, D.; Ahaidar, A.; Danelón, G.; Cironi, P.; Marfil, M.; Pérez, O.; Cuevas, C.; Albericio, F.; Joule, J. A.; Álvarez, M. Synthesis of polyheterocyclic nitrogen-containing marine natural products. Monatsh. Chem. 2004, 135, 615-627.
-
(2004)
Monatsh. Chem.
, vol.135
, pp. 615-627
-
-
Fernández, D.1
Ahaidar, A.2
Danelón, G.3
Cironi, P.4
Marfil, M.5
Pérez, O.6
Cuevas, C.7
Albericio, F.8
Joule, J.A.9
Álvarez, M.10
-
116
-
-
0036286613
-
The recent impact of solid-phase synthesis on medicinally relevant benzoannelated nitrogen heterocycles
-
Bräse, S.; Gil, C.; Knepper, K. The recent impact of solid-phase synthesis on medicinally relevant benzoannelated nitrogen heterocycles. Bioorg. Med. Chem., 2002, 10, 2415-2434.
-
(2002)
Bioorg. Med. Chem.
, vol.10
, pp. 2415-2434
-
-
Bräse, S.1
Gil, C.2
Knepper, K.3
-
117
-
-
2942580883
-
Aromaticity as a cornerstone of heterocyclic chemistry
-
Balaban, A. T.; Oniciu, D. C.; Katritzky, A. R. Aromaticity as a cornerstone of heterocyclic chemistry. Chem. Rev., 2004, 104, 2777-2812.
-
(2004)
Chem. Rev.
, vol.104
, pp. 2777-2812
-
-
Balaban, A.T.1
Oniciu, D.C.2
Katritzky, A.R.3
-
118
-
-
29244491409
-
Simple indole alkaloids and those with a nonrearranged monoterpenoid unit
-
Kawasaki, T.; Higuchi, K. Simple indole alkaloids and those with a nonrearranged monoterpenoid unit. Nat. Prod. Rep., 2005, 22, 761-793.
-
(2005)
Nat. Prod. Rep.
, vol.22
, pp. 761-793
-
-
Kawasaki, T.1
Higuchi, K.2
-
119
-
-
0028845177
-
Regioselective metalation of 9-Methoxymethyl-β-carboline-3-carboxamides with amidomagnesium Chlorides
-
Schlecker, W.; Huth, A.; Ottow, E.; Mulzer, J. Regioselective metalation of 9-Methoxymethyl-β-carboline-3-carboxamides with amidomagnesium Chlorides. Synthesis 1995, 1225-1227.
-
(1995)
Synthesis
, pp. 1225-1227
-
-
Schlecker, W.1
Huth, A.2
Ottow, E.3
Mulzer, J.4
-
120
-
-
37049078455
-
Iminophosphorane-mediated annelation of a pyridine or pyrimidine ring into an indole ring: Synthesis of β-, γ-carbolines and pyrimido[4,5-b]indole derivatives
-
Molina, P.; Fresneda, P. M. Iminophosphorane-mediated annelation of a pyridine or pyrimidine ring into an indole ring: synthesis of β-, γ-carbolines and pyrimido[4,5-b]indole derivatives J. Chem. Soc., Perkin Trans. 1 1988, 1819-1822.
-
(1988)
J. Chem. Soc., Perkin Trans. 1
, pp. 1819-1822
-
-
Molina, P.1
Fresneda, P.M.2
-
121
-
-
0027996777
-
Iminophosphorane-mediated syntheses of the fascaplysin alkaloid of marine origin and nitramarine
-
Molina, P.; Fresneda, P. M.; Zafra, G. S.; Almendros, P. Iminophosphorane-mediated syntheses of the fascaplysin alkaloid of marine origin and nitramarine. Tetrahedron Lett., 1994, 35, 8851-8854.
-
(1994)
Tetrahedron Lett.
, vol.35
, pp. 8851-8854
-
-
Molina, P.1
Fresneda, P.M.2
Zafra, G.S.3
Almendros, P.4
-
122
-
-
0036093922
-
Synthesis of combinatorial libraries based on triterpenoid scaffolds
-
Pathak, A.; Singh, S. K.; Farooq Biabani, M.A.; Srivastava, S.; Kulshreshtha, D.K.; Puri, S. K.; Kundu, B. Synthesis of combinatorial libraries based on triterpenoid scaffolds. Comb. Chem. Highthroughput Screen., 2002, 5, 241-248.
-
(2002)
Comb. Chem. Highthroughput Screen.
, vol.5
, pp. 241-248
-
-
Pathak, A.1
Singh, S.K.2
Farooq Biabani, M.A.3
Srivastava, S.4
Kulshreshtha, D.K.5
Puri, S.K.6
Kundu, B.7
-
123
-
-
0037152474
-
Solid-phase synthesis and bioevaluation of Lupeolbased libraries as antimalarial agents
-
Srinivasan, T.; Srivastava, G. K.; Pathak, A.; S. Batra, Puri, S.K.; Raj K.; Kundu, B. Solid-phase synthesis and bioevaluation of Lupeolbased libraries as antimalarial agents. Bioorg. Med. Chem. Lett., 2002, 12, 2803-2806.
-
(2002)
Bioorg. Med. Chem. Lett.
, vol.12
, pp. 2803-2806
-
-
Srinivasan, T.1
Srivastava, G.K.2
Pathak, A.3
Batra, S.4
Puri, S.K.5
Raj, K.6
Kundu, B.7
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