Solid–phase synthesis and bioevaluation of Lupeol–based libraries as antimalarial agents

Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 20, 2002, Pages 2803-2806

  Srinivasan, T ^a   Srivastava, G K ^a   Pathak, A ^a   Batra, S ^a   Raj, K ^a   Singh, Kshipra ^a   Puri, S K ^a   Kundu, B ^a  

^a CENTRAL DRUG RESEARCH INSTITUTE   (India)

Author keywords

[No Author keywords available]

Indexed keywords

ALIPHATIC DICARBOXYLIC ACID; ALKENE DERIVATIVE; AMIDE; ANTIMALARIAL AGENT; CHLOROQUINE; LUPEOL; POLYMER;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIMALARIAL ACTIVITY; ARTICLE; COMBINATORIAL LIBRARY; CONTROLLED STUDY; DRUG EFFECT; DRUG EFFICACY; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; FEMALE; MALE; MINIMUM INHIBITORY CONCENTRATION; MOUSE; NONHUMAN; PARASITEMIA; PLASMODIUM FALCIPARUM; SURVIVAL TIME; TREATMENT OUTCOME;

ANIMALS; ANTIMALARIALS; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; COMBINATORIAL CHEMISTRY TECHNIQUES; INDICATORS AND REAGENTS; MAGNETIC RESONANCE SPECTROSCOPY; MALARIA; MICE; PLASMODIUM BERGHEI; PLASMODIUM FALCIPARUM; SPECTROMETRY, MASS, FAST ATOM BOMBARDMENT; TRITERPENES;

PLASMODIUM FALCIPARUM;

EID: 0037152474     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)00623-6     Document Type: Article

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