SCOPUS 정보 검색 플랫폼

Volumn 46, Issue 11, 2011, Pages 5598-5608

A class of novel N-(1-methyl-β-carboline-3-carbonyl)-N′- (aminoacid-acyl)-hydrazines: Aromatization leaded design, synthesis, in vitro anti-platelet aggregation/in vivo anti-thrombotic evaluation and 3D QSAR analysis

(8) Li, Chunyu a Zhang, Xiaoyi a Zhao, Ming a Wang, Yuji a Wu, Jianhui a Liu, Jiawang a Zheng, Meiqing a Peng, Shiqi a

a CAPITAL MEDICAL UNIVERSITY (China)

Author keywords

Carboline; 3D QSAR; Anti platelet aggregation; Anti thrombotic activity; Aromatization

Indexed keywords

1 METHYL 1,2,3,4 TETRAHYDRO BETA CARBOLINE 3 CARBOXYLIC ACID METHYL ESTER; 1 METHYL BETA CARBOLINE 3 CARBONYLHYDRAZINE; 1 METHYL BETA CARBOLINE 3 CARBOXYLIC ACID METHYL ESTER; 1,2,3,4 TETRAHYDRO 1 METHYL BETA CARBOLINE 3 CARBOXYLIC ACID; ANTITHROMBOCYTIC AGENT; N (1 METHYL BETA CARBOLINE 3 CARBONYL) N' (AMINOACID ACYL)HYDRAZINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; AROMATIZATION; ARTICLE; CONTROLLED STUDY; DRUG DESIGN; DRUG SCREENING; DRUG SYNTHESIS; IN VITRO STUDY; IN VIVO STUDY; NONHUMAN; QUANTITATIVE STRUCTURE ACTIVITY RELATION; RAT; THROMBOCYTE AGGREGATION INHIBITION;

ANIMALS; CHEMISTRY TECHNIQUES, SYNTHETIC; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DESIGN; FIBRINOLYTIC AGENTS; HYDRAZINES; MALE; MODELS, MOLECULAR; MOLECULAR CONFORMATION; PLATELET AGGREGATION; PLATELET AGGREGATION INHIBITORS; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; RATS; SWINE; THROMBOSIS;

EID: 80054923928 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2011.09.027 Document Type: Article

Times cited : (23)

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