A structural insight into the reorientation of transmembrane domains 3 and 5 during family A G protein-coupled receptor activation

Molecular Pharmacology

Volumn 79, Issue 2, 2011, Pages 262-269

  Sansuk, Kamonchanok ^a   Deupi, Xavier ^b,c   Torrecillas, Ivan R ^b   Jongejan, Aldo ^a   Nijmeijer, Saskia ^a   Bakker, Remko A ^a,d   Pardo, Leonardo ^b   Leurs, Rob ^a  

^a VU UNIVERSITY AMSTERDAM   (Netherlands)

^b UNIVERSITAT AUTÒNOMA DE BARCELONA   (Spain)

^c PAUL SCHERRER INSTITUTE   (Switzerland)

^d BOEHRINGER INGELHEIM PHARMA GMBH AND CO KG   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

G PROTEIN COUPLED RECEPTOR; HISTAMINE H1 RECEPTOR; ISOLEUCINE; PROLINE; THREONINE;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; HYDROPHOBICITY; MATHEMATICAL MODEL; MOLECULAR STABILITY; NONHUMAN; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN FAMILY; PROTEIN MOTIF; RECEPTOR UPREGULATION; SITE DIRECTED MUTAGENESIS; X RAY CRYSTALLOGRAPHY;

ANIMALS; CERCOPITHECUS AETHIOPS; COS CELLS; HUMANS; MEMBRANE PROTEINS; MODELS, MOLECULAR; MUTAGENESIS, SITE-DIRECTED; PROTEIN BINDING; RECEPTORS, G-PROTEIN-COUPLED;

EID: 78751487961     PISSN: 0026895X     EISSN: 15210111     Source Type: Journal    
DOI: 10.1124/mol.110.066068     Document Type: Article

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