-
1
-
-
0036908594
-
Estrogen receptor dimerization: Ligand binding regulates dimer affinity and dimer dissociation rate
-
Tamrazi, A., Carlson, K. E., Daniels, J. R., Hurth, K. M., and Katzenellenbogen, J. A. (2002) Estrogen receptor dimerization: ligand binding regulates dimer affinity and dimer dissociation rate Mol. Endocrinol. 16, 2706-2719
-
(2002)
Mol. Endocrinol.
, vol.16
, pp. 2706-2719
-
-
Tamrazi, A.1
Carlson, K.E.2
Daniels, J.R.3
Hurth, K.M.4
Katzenellenbogen, J.A.5
-
2
-
-
0033305430
-
Coactivator peptides have a differential stabilizing effect on the binding of estrogens and antiestrogens with the estrogen receptor
-
Gee, A. C., Carlson, K. E., Martini, P. G., Katzenellenbogen, B. S., and Katzenellenbogen, J. A. (1999) Coactivator peptides have a differential stabilizing effect on the binding of estrogens and antiestrogens with the estrogen receptor Mol. Endocrinol. 13, 1912-23
-
(1999)
Mol. Endocrinol.
, vol.13
, pp. 1912-1923
-
-
Gee, A.C.1
Carlson, K.E.2
Martini, P.G.3
Katzenellenbogen, B.S.4
Katzenellenbogen, J.A.5
-
3
-
-
72449169864
-
Inhibitors of Nuclear Hormone Receptor/Coactivator Interactions
-
Moore, T. W. and Katzenellenbogen, J. A. (2009) Inhibitors of Nuclear Hormone Receptor/Coactivator Interactions Annu. Rep. Med. Chem. 44, 443-457
-
(2009)
Annu. Rep. Med. Chem.
, vol.44
, pp. 443-457
-
-
Moore, T.W.1
Katzenellenbogen, J.A.2
-
4
-
-
84908243878
-
Targeting the nuclear receptor-cofactor interaction, in
-
(, Eds.) Wiley-VCH, Weinheim, Germany.
-
Vaz, B., Mocklinghoff, S., and Brunsveld, L. (2008) Targeting the nuclear receptor-cofactor interaction, in Nuclear Receptors as Drug Targets (Ottow, F. and Weinmann, H., Eds.) pp 25 - 45, Wiley-VCH, Weinheim, Germany.
-
(2008)
Nuclear Receptors As Drug Targets
, pp. 25-45
-
-
Vaz, B.1
Mocklinghoff, S.2
Brunsveld, L.3
Ottow, F.4
Weinmann, H.5
-
5
-
-
0035400820
-
Preventing estrogen receptor action with dimer-interface peptides
-
Yudt, M. R. and Koide, S. (2001) Preventing estrogen receptor action with dimer-interface peptides Steroids 66, 549-58
-
(2001)
Steroids
, vol.66
, pp. 549-558
-
-
Yudt, M.R.1
Koide, S.2
-
6
-
-
77950442251
-
Minireview: Not picking pockets: Nuclear receptor alternate-site modulators (NRAMs)
-
Moore, T. W., Mayne, C. G., and Katzenellenbogen, J. A. (2010) Minireview: not picking pockets: nuclear receptor alternate-site modulators (NRAMs) Mol. Endocrinol. 24, 683-695
-
(2010)
Mol. Endocrinol.
, vol.24
, pp. 683-695
-
-
Moore, T.W.1
Mayne, C.G.2
Katzenellenbogen, J.A.3
-
7
-
-
0032446607
-
The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen
-
Shiau, A. K., Barstad, D., Loria, P. M., Cheng, L., Kushner, P. J., Agard, D. A., and Greene, G. L. (1998) The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen Cell 95, 927-37
-
(1998)
Cell
, vol.95
, pp. 927-937
-
-
Shiau, A.K.1
Barstad, D.2
Loria, P.M.3
Cheng, L.4
Kushner, P.J.5
Agard, D.A.6
Greene, G.L.7
-
8
-
-
54549083372
-
Blocking estrogen signaling after the hormone: Pyrimidine-core inhibitors of estrogen receptor-coactivator binding
-
Parent, A. A., Gunther, J. R., and Katzenellenbogen, J. A. (2008) Blocking estrogen signaling after the hormone: pyrimidine-core inhibitors of estrogen receptor-coactivator binding J. Med. Chem. 51, 6512-6530
-
(2008)
J. Med. Chem.
, vol.51
, pp. 6512-6530
-
-
Parent, A.A.1
Gunther, J.R.2
Katzenellenbogen, J.A.3
-
9
-
-
1642581072
-
Design, synthesis, and in vitro biological evaluation of small molecule inhibitors of estrogen receptor α coactivator binding
-
Rodriguez, A. L., Tamrazi, A., Collins, M. L., and Katzenellenbogen, J. A. (2004) Design, synthesis, and in vitro biological evaluation of small molecule inhibitors of estrogen receptor α coactivator binding J. Med. Chem. 47, 600-611
-
(2004)
J. Med. Chem.
, vol.47
, pp. 600-611
-
-
Rodriguez, A.L.1
Tamrazi, A.2
Collins, M.L.3
Katzenellenbogen, J.A.4
-
10
-
-
3142781225
-
Small-molecule inhibitors of protein-protein interactions: Progressing towards the dream
-
Arkin, M. R. and Wells, J. A. (2004) Small-molecule inhibitors of protein-protein interactions: progressing towards the dream Nat. Rev. Drug Discovery 3, 301-17
-
(2004)
Nat. Rev. Drug Discovery
, vol.3
, pp. 301-317
-
-
Arkin, M.R.1
Wells, J.A.2
-
11
-
-
37249004920
-
Reaching for high-hanging fruit in drug discovery at protein-protein interfaces
-
Wells, J. A. and McClendon, C. L. (2007) Reaching for high-hanging fruit in drug discovery at protein-protein interfaces Nature 450, 1001-9
-
(2007)
Nature
, vol.450
, pp. 1001-1009
-
-
Wells, J.A.1
McClendon, C.L.2
-
12
-
-
7444221875
-
Harnessing chaperones to generate small-molecule inhibitors of amyloid beta aggregation
-
Gestwicki, J. E., Crabtree, G. R., and Graef, I. A. (2004) Harnessing chaperones to generate small-molecule inhibitors of amyloid beta aggregation Science 306, 865-869
-
(2004)
Science
, vol.306
, pp. 865-869
-
-
Gestwicki, J.E.1
Crabtree, G.R.2
Graef, I.A.3
-
13
-
-
36048962201
-
Chemical control over protein-protein interactions: Beyond inhibitors
-
Gestwicki, J. E. and Marinec, P. S. (2007) Chemical control over protein-protein interactions: beyond inhibitors Comb. Chem. High Throughput Screen. 10, 667-75
-
(2007)
Comb. Chem. High Throughput Screen.
, vol.10
, pp. 667-675
-
-
Gestwicki, J.E.1
Marinec, P.S.2
-
14
-
-
42049121934
-
Crosstalk between the estrogen receptor and the HER tyrosine kinase receptor family: Molecular mechanism and clinical implications for endocrine therapy resistance
-
Arpino, G., Wiechmann, L., Osborne, C. K., and Schiff, R. (2008) Crosstalk between the estrogen receptor and the HER tyrosine kinase receptor family: molecular mechanism and clinical implications for endocrine therapy resistance Endocr. Rev. 29, 217-33
-
(2008)
Endocr. Rev.
, vol.29
, pp. 217-233
-
-
Arpino, G.1
Wiechmann, L.2
Osborne, C.K.3
Schiff, R.4
-
15
-
-
0031059270
-
The estradiol pharmacophore: Ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding site
-
Anstead, G. M., Carlson, K. E., and Katzenellenbogen, J. A. (1997) The estradiol pharmacophore: Ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding site Steroids 62, 268-303
-
(1997)
Steroids
, vol.62
, pp. 268-303
-
-
Anstead, G.M.1
Carlson, K.E.2
Katzenellenbogen, J.A.3
-
16
-
-
0033096995
-
Comparative QSAR analysis of estrogen receptor ligands
-
Gao, H., Katzenellenbogen, J. A., Garg, R., and Hansch, C. (1999) Comparative QSAR analysis of estrogen receptor ligands Chem. Rev. 99, 723-744
-
(1999)
Chem. Rev.
, vol.99
, pp. 723-744
-
-
Gao, H.1
Katzenellenbogen, J.A.2
Garg, R.3
Hansch, C.4
-
17
-
-
5244370033
-
Safe and convenient procedure for solvent purification
-
Pangborn, A. B., Giardello, M. A., Grubbs, R. H., Rosen, R. K., and Timmers, F. J. (1996) Safe and convenient procedure for solvent purification Organometallics 15, 1518-1520
-
(1996)
Organometallics
, vol.15
, pp. 1518-1520
-
-
Pangborn, A.B.1
Giardello, M.A.2
Grubbs, R.H.3
Rosen, R.K.4
Timmers, F.J.5
-
18
-
-
0002714675
-
Rapid chromatographic technique for preparative separations with moderate resolution
-
Still, W. C., Kahn, M., and Mitra, A. (1978) Rapid chromatographic technique for preparative separations with moderate resolution J. Org. Chem. 43, 2923-25
-
(1978)
J. Org. Chem.
, vol.43
, pp. 2923-2925
-
-
Still, W.C.1
Kahn, M.2
Mitra, A.3
-
19
-
-
0001019593
-
Design, synthesis, and kinetic evaluation of high-affinity FKBP Ligands and the X-ray crystal-structures of their complexes with FKBP12
-
Holt, D. A., Luengo, J. I., Yamashita, D. S., Oh, H. J., Konialian, A. L., Yen, H. K., Rozamus, L. W., Brandt, M., Bossard, M. J., Levy, M. A., Eggleston, D. S., Liang, J., Schultz, L. W., Stout, T. J., and Clardy, J. (1993) Design, synthesis, and kinetic evaluation of high-affinity FKBP Ligands and the X-ray crystal-structures of their complexes with FKBP12 J. Am. Chem. Soc. 115, 9925-9938
-
(1993)
J. Am. Chem. Soc.
, vol.115
, pp. 9925-9938
-
-
Holt, D.A.1
Luengo, J.I.2
Yamashita, D.S.3
Oh, H.J.4
Konialian, A.L.5
Yen, H.K.6
Rozamus, L.W.7
Brandt, M.8
Bossard, M.J.9
Levy, M.A.10
Eggleston, D.S.11
Liang, J.12
Schultz, L.W.13
Stout, T.J.14
Clardy, J.15
-
20
-
-
0031683101
-
Synthesis and activity of bivalent FKBP12 ligands for the regulated dimerization of proteins
-
Keenan, T., Yaeger, D. R., Courage, N. L., Rollins, C. T., Pavone, M. E., Rivera, V. M., Yang, W., Guo, T., Amara, J. F., Clackson, T., Gilman, M., and Holt, D. A. (1998) Synthesis and activity of bivalent FKBP12 ligands for the regulated dimerization of proteins Bioorg. Med. Chem. 6, 1309-35
-
(1998)
Bioorg. Med. Chem.
, vol.6
, pp. 1309-1335
-
-
Keenan, T.1
Yaeger, D.R.2
Courage, N.L.3
Rollins, C.T.4
Pavone, M.E.5
Rivera, V.M.6
Yang, W.7
Guo, T.8
Amara, J.F.9
Clackson, T.10
Gilman, M.11
Holt, D.A.12
-
21
-
-
0030734795
-
Altered ligand binding properties and enhanced stability of a constitutively active estrogen receptor: Evidence that an open pocket conformation is required for ligand interaction
-
Carlson, K. E., Choi, I., Gee, A., Katzenellenbogen, B. S., and Katzenellenbogen, J. A. (1997) Altered ligand binding properties and enhanced stability of a constitutively active estrogen receptor: Evidence that an open pocket conformation is required for ligand interaction Biochemistry 36, 14897-14905
-
(1997)
Biochemistry
, vol.36
, pp. 14897-14905
-
-
Carlson, K.E.1
Choi, I.2
Gee, A.3
Katzenellenbogen, B.S.4
Katzenellenbogen, J.A.5
-
22
-
-
0033548071
-
The FKBP12-rapamycin-binding domain is required for FKBP12-rapamycin- associated protein kinase activity and G(1) progression
-
Vilella-Bach, M., Nuzzi, P., Fang, Y. M., and Chen, J. (1999) The FKBP12-rapamycin-binding domain is required for FKBP12-rapamycin-associated protein kinase activity and G(1) progression J. Biol. Chem. 274, 4266-4272
-
(1999)
J. Biol. Chem.
, vol.274
, pp. 4266-4272
-
-
Vilella-Bach, M.1
Nuzzi, P.2
Fang, Y.M.3
Chen, J.4
-
23
-
-
61849123737
-
A set of time-resolved fluorescence resonance energy transfer assays for the discovery of inhibitors of estrogen receptor-coactivator binding
-
Gunther, J. R., Du, Y., Rhoden, E., Lewis, I., Revennaugh, B., Moore, T. W., Kim, S. H., Dingledine, R., Fu, H., and Katzenellenbogen, J. A. (2009) A set of time-resolved fluorescence resonance energy transfer assays for the discovery of inhibitors of estrogen receptor-coactivator binding J. Biomol. Screen. 14, 181-193
-
(2009)
J. Biomol. Screen.
, vol.14
, pp. 181-193
-
-
Gunther, J.R.1
Du, Y.2
Rhoden, E.3
Lewis, I.4
Revennaugh, B.5
Moore, T.W.6
Kim, S.H.7
Dingledine, R.8
Fu, H.9
Katzenellenbogen, J.A.10
-
24
-
-
0004752110
-
Novel ligands that function as selective estrogens or antiestrogens for estrogen receptor-alpha or estrogen receptor-beta
-
Sun, J., Meyers, M. J., Fink, B. E., Rajendran, R., Katzenellenbogen, J. A., and Katzenellenbogen, B. S. (1999) Novel ligands that function as selective estrogens or antiestrogens for estrogen receptor-alpha or estrogen receptor-beta Endocrinology 140, 800-804
-
(1999)
Endocrinology
, vol.140
, pp. 800-804
-
-
Sun, J.1
Meyers, M.J.2
Fink, B.E.3
Rajendran, R.4
Katzenellenbogen, J.A.5
Katzenellenbogen, B.S.6
-
25
-
-
0033490140
-
Expression of the estrogen receptor-associated immunophilins, cyclophilin 40 and FKBP52, in breast cancer
-
Ward, B. K., Mark, P. J., Ingram, D. M., Minchin, R. F., and Ratajczak, T. (1999) Expression of the estrogen receptor-associated immunophilins, cyclophilin 40 and FKBP52, in breast cancer Breast Cancer Res. Treat. 58, 267-80
-
(1999)
Breast Cancer Res. Treat.
, vol.58
, pp. 267-280
-
-
Ward, B.K.1
Mark, P.J.2
Ingram, D.M.3
Minchin, R.F.4
Ratajczak, T.5
-
26
-
-
13144276290
-
Redesigning an FKBP-ligand interface to generate chemical dimerizers with novel specificity
-
Clackson, T., Yang, W., Rozamus, L. W., Hatada, M., Amara, J. F., Rollins, C. T., Stevenson, L. F., Magari, S. R., Wood, S. A., Courage, N. L., Lu, X., Cerasoli, F., Jr., Gilman, M., and Holt, D. A. (1998) Redesigning an FKBP-ligand interface to generate chemical dimerizers with novel specificity Proc. Natl. Acad. Sci. U.S.A. 95, 10437-42
-
(1998)
Proc. Natl. Acad. Sci. U.S.A.
, vol.95
, pp. 10437-10442
-
-
Clackson, T.1
Yang, W.2
Rozamus, L.W.3
Hatada, M.4
Amara, J.F.5
Rollins, C.T.6
Stevenson, L.F.7
Magari, S.R.8
Wood, S.A.9
Courage, N.L.10
Lu, X.11
Cerasoli, Jr.F.12
Gilman, M.13
Holt, D.A.14
-
27
-
-
0015867364
-
Studies on uterine, cytoplasmic estrogen binding protein - Thermal-stability and ligand dissociation rate - Assay of empty and filled sites by exchange
-
Katzenellenbogen, J. A., Johnson, H. J., and Carlson, K. E. (1973) Studies on uterine, cytoplasmic estrogen binding protein-thermal-stability and ligand dissociation rate-assay of empty and filled sites by exchange Biochemistry 12, 4092-4099
-
(1973)
Biochemistry
, vol.12
, pp. 4092-4099
-
-
Katzenellenbogen, J.A.1
Johnson, H.J.2
Carlson, K.E.3
-
28
-
-
34547653666
-
Structural plasticity in the oestrogen receptor ligand-binding domain
-
Nettles, K. W., Bruning, J. B., Gil, G., O'Neill, E. E., Nowak, J., Guo, Y., Kim, Y., DeSombre, E. R., Dilis, R., Hanson, R. N., Joachimiak, A., and Greene, G. L. (2007) Structural plasticity in the oestrogen receptor ligand-binding domain EMBO Rep. 8, 563-8
-
(2007)
EMBO Rep.
, vol.8
, pp. 563-568
-
-
Nettles, K.W.1
Bruning, J.B.2
Gil, G.3
O'Neill, E.E.4
Nowak, J.5
Guo, Y.6
Kim, Y.7
Desombre, E.R.8
Dilis, R.9
Hanson, R.N.10
Joachimiak, A.11
Greene, G.L.12
-
29
-
-
55749112475
-
Synthesis and biological evaluation of guanylhydrazone coactivator binding inhibitors for the estrogen receptor
-
LaFrate, A. L., Gunther, J. R., Carlson, K. E., and Katzenellenbogen, J. A. (2008) Synthesis and biological evaluation of guanylhydrazone coactivator binding inhibitors for the estrogen receptor Bioorg. Med. Chem. 16, 10075-10084
-
(2008)
Bioorg. Med. Chem.
, vol.16
, pp. 10075-10084
-
-
Lafrate, A.L.1
Gunther, J.R.2
Carlson, K.E.3
Katzenellenbogen, J.A.4
-
30
-
-
2442502910
-
Identification of novel estrogen receptor α antagonists
-
Shao, D., Berrodin, T. J., Manas, E., Hauze, D., Powers, R., Bapat, A., Gonder, D., Winneker, R. C., and Frail, D. E. (2004) Identification of novel estrogen receptor α antagonists J. Steroid Biochem. Mol. Biol. 88, 351-360
-
(2004)
J. Steroid Biochem. Mol. Biol.
, vol.88
, pp. 351-360
-
-
Shao, D.1
Berrodin, T.J.2
Manas, E.3
Hauze, D.4
Powers, R.5
Bapat, A.6
Gonder, D.7
Winneker, R.C.8
Frail, D.E.9
-
31
-
-
57349133187
-
Simulating oligomerization at experimental concentrations and long timescales: A Markov state model approach
-
Kelley, N. W., Vishal, V., Krafft, G. A., and Pande, V. S. (2008) Simulating oligomerization at experimental concentrations and long timescales: A Markov state model approach J. Chem. Phys. 129, 214707
-
(2008)
J. Chem. Phys.
, vol.129
, pp. 214707
-
-
Kelley, N.W.1
Vishal, V.2
Krafft, G.A.3
Pande, V.S.4
-
32
-
-
0030611858
-
Soluble amyloid Abeta-(1-40) exists as a stable dimer at low concentrations
-
Garzon-Rodriguez, W., Sepulveda-Becerra, M., Milton, S., and Glabe, C. G. (1997) Soluble amyloid Abeta-(1-40) exists as a stable dimer at low concentrations J. Biol. Chem. 272, 21037-44
-
(1997)
J. Biol. Chem.
, vol.272
, pp. 21037-21044
-
-
Garzon-Rodriguez, W.1
Sepulveda-Becerra, M.2
Milton, S.3
Glabe, C.G.4
-
33
-
-
77949905345
-
Fibrillar oligomers nucleate the oligomerization of monomeric amyloid beta but do not seed fibril formation
-
Wu, J. W., Breydo, L., Isas, J. M., Lee, J., Kuznetsov, Y. G., Langen, R., and Glabe, C. Fibrillar oligomers nucleate the oligomerization of monomeric amyloid beta but do not seed fibril formation J. Biol. Chem. 285, 6071-9
-
J. Biol. Chem.
, vol.285
, pp. 6071-6079
-
-
Wu, J.W.1
Breydo, L.2
Isas, J.M.3
Lee, J.4
Kuznetsov, Y.G.5
Langen, R.6
Glabe, C.7
-
34
-
-
51649107127
-
Rational design of novel antiandrogens for neutralizing androgen receptor function in hormone refractory prostate cancer
-
Singh, P., Hallur, G., Anchoori, R. K., Bakare, O., Kageyama, Y., Khan, S. R., and Isaacs, J. T. (2008) Rational design of novel antiandrogens for neutralizing androgen receptor function in hormone refractory prostate cancer Prostate 68, 1570-81
-
(2008)
Prostate
, vol.68
, pp. 1570-1581
-
-
Singh, P.1
Hallur, G.2
Anchoori, R.K.3
Bakare, O.4
Kageyama, Y.5
Khan, S.R.6
Isaacs, J.T.7
-
35
-
-
43949096905
-
Bifunctional molecules evade cytochrome P(450) metabolism by forming protective complexes with FK506-binding protein
-
Marinec, P. S., Lancia, J. K., and Gestwicki, J. E. (2008) Bifunctional molecules evade cytochrome P(450) metabolism by forming protective complexes with FK506-binding protein Mol. Biosyst. 4, 571-8
-
(2008)
Mol. Biosyst.
, vol.4
, pp. 571-578
-
-
Marinec, P.S.1
Lancia, J.K.2
Gestwicki, J.E.3
-
36
-
-
0342460407
-
Cytotoxic Oestrogens and Antioestrogens: Concepts, Progress and Evaluation, in
-
(, Eds.) Bailliere Tindall, London.
-
Katzenellenbogen, J. A. and Zablocki, J. A. (1987) Cytotoxic Oestrogens and Antioestrogens: Concepts, Progress and Evaluation, in Pharmacology and clinical uses of inhibitors of hormone secretion and action (Furr, B. J. A. and Wakeling, A. E., Eds.) pp 41 - 59, Bailliere Tindall, London.
-
(1987)
Pharmacology and Clinical Uses of Inhibitors of Hormone Secretion and Action
, pp. 41-59
-
-
Katzenellenbogen, J.A.1
Zablocki, J.A.2
Furr, B.J.A.3
Wakeling, A.E.4
-
37
-
-
58149528026
-
A bifunctional platinum(II) antitumor agent that forms DNA adducts with affinity for the estrogen receptor
-
Kim, E., Rye, P. T., Essigmann, J. M., and Croy, R. G. (2009) A bifunctional platinum(II) antitumor agent that forms DNA adducts with affinity for the estrogen receptor J. Inorg. Biochem. 103, 256-261
-
(2009)
J. Inorg. Biochem.
, vol.103
, pp. 256-261
-
-
Kim, E.1
Rye, P.T.2
Essigmann, J.M.3
Croy, R.G.4
-
38
-
-
0037028969
-
A rationally designed genotoxin that selectively destroys estrogen receptor-positive breast cancer cells
-
Mitra, K., Marquis, J. C., Hillier, S. M., Rye, P. T., Zayas, B., Lee, A. S., Essigmann, J. M., and Croy, R. G. (2002) A rationally designed genotoxin that selectively destroys estrogen receptor-positive breast cancer cells J. Am. Chem. Soc. 124, 1862-1863
-
(2002)
J. Am. Chem. Soc.
, vol.124
, pp. 1862-1863
-
-
Mitra, K.1
Marquis, J.C.2
Hillier, S.M.3
Rye, P.T.4
Zayas, B.5
Lee, A.S.6
Essigmann, J.M.7
Croy, R.G.8
-
39
-
-
0030466324
-
Synthesis and biological activity of DNA damaging agents that form decoy binding sites for the estrogen receptor
-
Rink, S. M., Yarema, K. J., Solomon, M. S., Paige, L. A., Tadayoni-Rebek, B. M., Essigmann, J. M., and Croy, R. G. (1996) Synthesis and biological activity of DNA damaging agents that form decoy binding sites for the estrogen receptor Proc. Natl. Acad. Sci. U.S.A. 93, 15063-15068
-
(1996)
Proc. Natl. Acad. Sci. U.S.A.
, vol.93
, pp. 15063-15068
-
-
Rink, S.M.1
Yarema, K.J.2
Solomon, M.S.3
Paige, L.A.4
Tadayoni-Rebek, B.M.5
Essigmann, J.M.6
Croy, R.G.7
-
40
-
-
0003008238
-
Synthesis and evaluation of geldanamycin-estradiol hybrids
-
Kuduk, S. D., Zheng, F. F., Sepp-Lorenzino, L., Rosen, N., and Danishefsky, S. J. (1999) Synthesis and evaluation of geldanamycin-estradiol hybrids Bioorg. Med. Chem. Lett. 9, 1233-8
-
(1999)
Bioorg. Med. Chem. Lett.
, vol.9
, pp. 1233-1238
-
-
Kuduk, S.D.1
Zheng, F.F.2
Sepp-Lorenzino, L.3
Rosen, N.4
Danishefsky, S.J.5
-
41
-
-
0037414262
-
Synthesis of a β-estradiol-biotin chimera that potently heterodimerizes estrogen receptor and streptavidin proteins in a yeast three-hybrid system
-
Hussey, S. L., Muddana, S. S., and Peterson, B. R. (2003) Synthesis of a β-estradiol-biotin chimera that potently heterodimerizes estrogen receptor and streptavidin proteins in a yeast three-hybrid system J. Am. Chem. Soc. 125, 3692-3693
-
(2003)
J. Am. Chem. Soc.
, vol.125
, pp. 3692-3693
-
-
Hussey, S.L.1
Muddana, S.S.2
Peterson, B.R.3
|