SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry

Volumn 18, Issue 21, 2010, Pages 7331-7337

3-O-Arylmethylgalangin, a novel isostere for anti-HCV 1,3-diketoacids (DKAs)

(5) Lee, Hyo Seon a Park, Kwang Su a Lee, Bokhui a Kim, Dong Eun a Chong, Youhoon a

a Konkuk University (South Korea)

Author keywords

1,3 Diketoacid; 3 O Arylmethylgalangin; Hepatitis C Virus (HCV); Isostere

Indexed keywords

GALANGIN; GALANGIN DERIVATIVE; INTEGRASE; NONSTRUCTURAL PROTEIN 5B; UNCLASSIFIED DRUG;

ANTIVIRAL ACTIVITY; ARTICLE; CHELATION; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; HEPATITIS C VIRUS; NONHUMAN; STRUCTURE ACTIVITY RELATION;

ANTIVIRAL AGENTS; CELL LINE, TUMOR; FLAVONOIDS; HEPACIVIRUS; HUMANS; KETO ACIDS; PROTEASE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP; VIRAL NONSTRUCTURAL PROTEINS;

HEPATITIS C VIRUS;

EID: 77958018258 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2010.09.021 Document Type: Article

Times cited : (8)

References (25)

1
- 0034723439
- D.J. Hazuda, P. Felock, M. Witmer, A. Wolfe, KI. Stillmock, J.A. Grobler, A. Espeseth, L. Gabryelski, W. Schleif, C. Blau, and M.D. Miller Science 287 2000 646
- (2000) Science , vol.287 , pp. 646
- Hazuda, D.J.¹ Felock, P.² Witmer, M.³ Wolfe, A.⁴ Stillmock, K.I.⁵ Grobler, J.A.⁶ Espeseth, A.⁷ Gabryelski, L.⁸ Schleif, W.⁹ Blau, C.¹⁰ Miller, M.D.¹¹

2
- 0037076324
- J.A. Grobler, K. Stillmock, B. Hu, M. Witmer, P. Felock, A.S. Espeseth, A. Wolfe, M. Egbertson, M. Bourgeois, J. Melamed, J.S. Wai, S. Young, J. Vacca, and D.J. Hazuda Proc. Natl. Acad. Sci. U.S.A. 99 2002 6661
- (2002) Proc. Natl. Acad. Sci. U.S.A. , vol.99 , pp. 6661
- Grobler, J.A.¹ Stillmock, K.² Hu, B.³ Witmer, M.⁴ Felock, P.⁵ Espeseth, A.S.⁶ Wolfe, A.⁷ Egbertson, M.⁸ Bourgeois, M.⁹ Melamed, J.¹⁰ Wai, J.S.¹¹ Young, S.¹² Vacca, J.¹³ Hazuda, D.J.¹⁴

3
- 33751014050
- V. Summa, A. Petrocchi, V.G. Matassa, C. Gardelli, E. Muraglia, M. Rowley, O.G. Paz, R. Laufer, E. Monteagudo, and P. Pace J. Med. Chem. 49 2006 6646
- (2006) J. Med. Chem. , vol.49 , pp. 6646
- Summa, V.¹ Petrocchi, A.² Matassa, V.G.³ Gardelli, C.⁴ Muraglia, E.⁵ Rowley, M.⁶ Paz, O.G.⁷ Laufer, R.⁸ Monteagudo, E.⁹ Pace, P.¹⁰

4
- 27444447888
- M.L. Barreca, S. Ferro, A. Rao, L.D. Luca, M. Zappala, A.M. Monforte, Z. Debyser, M. Witvrouw, and A. Chimirri J. Med. Chem. 48 2005 7084
- (2005) J. Med. Chem. , vol.48 , pp. 7084
- Barreca, M.L.¹ Ferro, S.² Rao, A.³ Luca, L.D.⁴ Zappala, M.⁵ Monforte, A.M.⁶ Debyser, Z.⁷ Witvrouw, M.⁸ Chimirri, A.⁹

5
- 13044295993
- Y. Goldgur, R. Craigie, G.H. Cohen, T. Fujiwara, T. Yoshinage, T. Fujishita, H. Sugimoto, T. Endo, H. Murai, and D.R. Davies Proc. Natl. Acad. Sci. U.S.A. 96 1999 13040
- (1999) Proc. Natl. Acad. Sci. U.S.A. , vol.96 , pp. 13040
- Goldgur, Y.¹ Craigie, R.² Cohen, G.H.³ Fujiwara, T.⁴ Yoshinage, T.⁵ Fujishita, T.⁶ Sugimoto, H.⁷ Endo, T.⁸ Murai, H.⁹ Davies, D.R.¹⁰

6
- 0037434509
- L. Zhuang, J.S. Wai, M.W. Embrey, T.E. Fisher, M.S. Egbertson, L.S. Payne, J.P. Guare Jr., J.P. Vacca, D.J. Hazuda, P.J. Felock, A.L. Wolfe, K.A. Stillmock, M.V. Witmer, G. Moyer, W.A. Schleif, L.J. Gabryelski, Y.M. Leonard, J.J. Lynch Jr., S.R. Michelson, and S.D. Young J. Med. Chem. 46 2003 453
- (2003) J. Med. Chem. , vol.46 , pp. 453
- Zhuang, L.¹ Wai, J.S.² Embrey, M.W.³ Fisher, T.E.⁴ Egbertson, M.S.⁵ Payne, L.S.⁶ Guare Jr., J.P.⁷ Vacca, J.P.⁸ Hazuda, D.J.⁹ Felock, P.J.¹⁰ Wolfe, A.L.¹¹ Stillmock, K.A.¹² Witmer, M.V.¹³ Moyer, G.¹⁴ Schleif, W.A.¹⁵ Gabryelski, L.J.¹⁶ Leonard, Y.M.¹⁷ Lynch Jr., J.J.¹⁸ Michelson, S.R.¹⁹ Young, S.D.²⁰ more..

7
- 3843108916
- D.J. Hazuda, N.J. Anthony, R.P. Gomez, S.M. Jolly, J.S. Wai, L. Zhuang, T.E. Fisher, M. Embrey, J.P. Guare Jr., M.S. Egbertson, J.P. Vacca, J.R. Huff, P.J. Felock, M.V. Witmer, K.A. Stillmock, R. Danovich, J. Grobler, M.D. Miller, A.S. Espeseth, L. Jin, I.-W. Chen, J.H. Lin, K. Kassahun, J.D. Ellis, B.K. Wong, W. Xu, P.G. Pearson, W.A. Schleif, R. Cortese, E. Emini, V. Summa, M.K. Holloway, and S.D. Young Proc. Natl. Acad. Sci. U.S.A. 101 2004 11233
- (2004) Proc. Natl. Acad. Sci. U.S.A. , vol.101 , pp. 11233
- Hazuda, D.J.¹ Anthony, N.J.² Gomez, R.P.³ Jolly, S.M.⁴ Wai, J.S.⁵ Zhuang, L.⁶ Fisher, T.E.⁷ Embrey, M.⁸ Guare Jr., J.P.⁹ Egbertson, M.S.¹⁰ Vacca, J.P.¹¹ Huff, J.R.¹² Felock, P.J.¹³ Witmer, M.V.¹⁴ Stillmock, K.A.¹⁵ Danovich, R.¹⁶ Grobler, J.¹⁷ Miller, M.D.¹⁸ Espeseth, A.S.¹⁹ Jin, L.²⁰ more..

8
- 3242769788
- D.J. Hazuda, S.D. Young, J.P. Guare, N.J. Anthony, R.P. Gomez, J.S. Wai, J.P. Vacca, L. Handt, S.L. Motzel, H.J. Klein, G. Dornadula, R.M. Danovich, M.V. Witmer, K.A.A. Wilson, L. Tussey, W.A. Schleif, L.S. Gabryelski, L. Jin, M.D. Miller, D.R. CAsimiro, E.A. Emini, and J.W. Shiver Science 305 2004 528
- (2004) Science , vol.305 , pp. 528
- Hazuda, D.J.¹ Young, S.D.² Guare, J.P.³ Anthony, N.J.⁴ Gomez, R.P.⁵ Wai, J.S.⁶ Vacca, J.P.⁷ Handt, L.⁸ Motzel, S.L.⁹ Klein, H.J.¹⁰ Dornadula, G.¹¹ Danovich, R.M.¹² Witmer, M.V.¹³ Wilson, K.A.A.¹⁴ Tussey, L.¹⁵ Schleif, W.A.¹⁶ Gabryelski, L.S.¹⁷ Jin, L.¹⁸ Miller, M.D.¹⁹ Casimiro, D.R.²⁰ Emini, E.A.²¹ Shiver, J.W.²² more..

9
- 52449097240
- V. Summa, A. Petrocchi, F. Bonelli, B. Crescenzi, M. Donghi, M. Ferrara, F. Fiore, C. Gardelli, O.G. Paz, D.J. Hazuda, P. Jones, O. Kinzel, R. Laufer, E. Monteagudo, E. Muraglia, E. Nizi, F. Orvieto, P. Pace, G. Pescatore, R. Scarpelli, K. Stillmock, M.V. Witmer, and M. Rowley J. Med. Chem. 51 2008 5843
- (2008) J. Med. Chem. , vol.51 , pp. 5843
- Summa, V.¹ Petrocchi, A.² Bonelli, F.³ Crescenzi, B.⁴ Donghi, M.⁵ Ferrara, M.⁶ Fiore, F.⁷ Gardelli, C.⁸ Paz, O.G.⁹ Hazuda, D.J.¹⁰ Jones, P.¹¹ Kinzel, O.¹² Laufer, R.¹³ Monteagudo, E.¹⁴ Muraglia, E.¹⁵ Nizi, E.¹⁶ Orvieto, F.¹⁷ Pace, P.¹⁸ Pescatore, G.¹⁹ Scarpelli, R.²⁰ more..

10
- 68549115378
- M. Sato, H. Kawakami, T. Motomura, H. Aramaki, T. Matsuda, M. Yamashita, Y. Ito, Y. Matsuzaki, K. Yamataka, S. Ikeda, and H. Shinkai J. Med. Chem. 52 2009 4869
- (2009) J. Med. Chem. , vol.52 , pp. 4869
- Sato, M.¹ Kawakami, H.² Motomura, T.³ Aramaki, H.⁴ Matsuda, T.⁵ Yamashita, M.⁶ Ito, Y.⁷ Matsuzaki, Y.⁸ Yamataka, K.⁹ Ikeda, S.¹⁰ Shinkai, H.¹¹

11
- 0347361643
- V. Summa, A. Petrocchi, P. Pace, V.G. Matassa, R. De Francesco, S. Altamura, L. Tomei, U. Koch, and P. Neuner J. Med. Chem. 47 2004 14
- (2004) J. Med. Chem. , vol.47 , pp. 14
- Summa, V.¹ Petrocchi, A.² Pace, P.³ Matassa, V.G.⁴ De Francesco, R.⁵ Altamura, S.⁶ Tomei, L.⁷ Koch, U.⁸ Neuner, P.⁹

12
- 33751357565
- J. Kim, J.H. Han, and Y. Chong Bull. Korean Chem. Soc. 27 2006 1919
- (2006) Bull. Korean Chem. Soc. , vol.27 , pp. 1919
- Kim, J.¹ Han, J.H.² Chong, Y.³

13
- 34548454840
- J. Kim, and Y. Chong Mol. Simul. 32 2006 1131
- (2006) Mol. Simul. , vol.32 , pp. 1131
- Kim, J.¹ Chong, Y.²

14
- 48649084902
- J. Kim, K.-S. Kim, H.S. Lee, K.-S. Park, S.Y. Park, S.-Y. Kang, S.J. Lee, H.S. Park, D.-E. Kim, and Y. Chong Bioorg. Med. Chem. Lett. 18 2008 4661
- (2008) Bioorg. Med. Chem. Lett. , vol.18 , pp. 4661
- Kim, J.¹ Kim, K.-S.² Lee, H.S.³ Park, K.-S.⁴ Park, S.Y.⁵ Kang, S.-Y.⁶ Lee, S.J.⁷ Park, H.S.⁸ Kim, D.-E.⁹ Chong, Y.¹⁰

15
- 0024364268
- I.B. Afanas'ev, A.I. Dorozhko, A.V. Brodskii, V.A. Kostyuk, and A.I. Potapovitch Biochem. Pharmacol. 38 1989 1763
- (1989) Biochem. Pharmacol. , vol.38 , pp. 1763
- Afanas'Ev, I.B.¹ Dorozhko, A.I.² Brodskii, A.V.³ Kostyuk, V.A.⁴ Potapovitch, A.I.⁵

16
- 0028117768
- I. Morel, G. Lescoat, P. Cillard, and J. Cillard Methods Enzymol. 234 1994 437
- (1994) Methods Enzymol. , vol.234 , pp. 437
- Morel, I.¹ Lescoat, G.² Cillard, P.³ Cillard, J.⁴

17
- 0030593711
- N.J. Miller, C. Castellucio, L. Tijburg, and C. Rice-Evans FEBS Lett. 392 1996 40
- (1996) FEBS Lett. , vol.392 , pp. 40
- Miller, N.J.¹ Castellucio, C.² Tijburg, L.³ Rice-Evans, C.⁴

18
- 52749096335
- J. Kim, H.S. Lee, K.-S. Park, and Y. Chong Bull. Korean Chem. Soc. 29 2008 1667
- (2008) Bull. Korean Chem. Soc. , vol.29 , pp. 1667
- Kim, J.¹ Lee, H.S.² Park, K.-S.³ Chong, Y.⁴

19
- 7044253372
- T.T. Dao, S.B. Kim, K.-S. Sin, S. Kim, H.P. Kim, and H. Park Arch. Pharm. Res. 27 2004 278
- (2004) Arch. Pharm. Res. , vol.27 , pp. 278
- Dao, T.T.¹ Kim, S.B.² Sin, K.-S.³ Kim, S.⁴ Kim, H.P.⁵ Park, H.⁶

20
- 0000778391
- L.W. McGarry, and M.R. Detty J. Org. Chem. 55 1990 4349
- (1990) J. Org. Chem. , vol.55 , pp. 4349
- McGarry, L.W.¹ Detty, M.R.²

21
- 0038467627
- R.A. Love, H.E. Parge, X. Yu, M.J. Hickey, W. Diehl, J. Gao, H. Wriggers, A. Ekker, L. Wang, J.A. Thomson, P.S. Dragovich, and S.A. Fuhrman J. Virol. 77 2003 7575
- (2003) J. Virol. , vol.77 , pp. 7575
- Love, R.A.¹ Parge, H.E.² Yu, X.³ Hickey, M.J.⁴ Diehl, W.⁵ Gao, J.⁶ Wriggers, H.⁷ Ekker, A.⁸ Wang, L.⁹ Thomson, J.A.¹⁰ Dragovich, P.S.¹¹ Fuhrman, S.A.¹²

22
- 0345188811
- V. Lohmann, F. Korner, J. Koch, U. Herian, L. Theilmann, and R. Bartenschlager Science 285 1999 110
- (1999) Science , vol.285 , pp. 110
- Lohmann, V.¹ Korner, F.² Koch, J.³ Herian, U.⁴ Theilmann, L.⁵ Bartenschlager, R.⁶

23
- 0037716580
- J.M. Vroljk, A. Kaul, B.E. Hansen, V. Lohmann, B.L. Haagmans, S.W. Schalm, and R. Bartenschlager J. Virol. Methods 110 2003 201
- (2003) J. Virol. Methods , vol.110 , pp. 201
- Vroljk, J.M.¹ Kaul, A.² Hansen, B.E.³ Lohmann, V.⁴ Haagmans, B.L.⁵ Schalm, S.W.⁶ Bartenschlager, R.⁷

24
- 38649113265
- A. Gozdek, I. Zhukov, A. Polkowska, J. Poznanski, A. Stankiewicz-Drogon, J.M. Pawlowicz, W. Zagorski-Ostoja, P. Borowski, and A. Boguszewska-Chachulska Antimicrob. Agents Chemother. 52 2008 393
- (2008) Antimicrob. Agents Chemother. , vol.52 , pp. 393
- Gozdek, A.¹ Zhukov, I.² Polkowska, A.³ Poznanski, J.⁴ Stankiewicz-Drogon, A.⁵ Pawlowicz, J.M.⁶ Zagorski-Ostoja, W.⁷ Borowski, P.⁸ Boguszewska-Chachulska, A.⁹

25
- 34447631178
- T. Kirschberg, and J. Parrish Curr. Opin. Drug Discov. Dev. 10 2007 460
- (2007) Curr. Opin. Drug Discov. Dev. , vol.10 , pp. 460
- Kirschberg, T.¹ Parrish, J.²

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.