Affinity selection-mass spectrometry and its emerging application to the high throughput screening of G protein-coupled receptors

Combinatorial Chemistry and High Throughput Screening

Volumn 11, Issue 6, 2008, Pages 427-438

  Whitehurst, Charles E ^a   Annis, D Allen ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ATROPINE; G PROTEIN COUPLED RECEPTOR; N [2 [2 (DIPROPYLAMINOMETHYL) 1 PIPERIDYL]ETHYL] 5,11 DIHYDRO 6 OXO 6H PYRIDO[2,3 B][1,4]BENZODIAZEPINE 11 CARBOXAMIDE; NGD 3346; NGD 3348; NGD 3350; OTENZEPAD;

AFFINITY SELECTION MASS SPECTROMETRY; ALLOSTERISM; COMPLEX FORMATION; CONTROLLED STUDY; DRUG EFFICACY; DRUG TARGETING; FLUORESCENCE; HIGH THROUGHPUT SCREENING; HUMAN; INTERMETHOD COMPARISON; LIGAND BINDING; MASS SPECTROMETRY; PRIORITY JOURNAL; PROTEIN PURIFICATION; PROTEIN TARGETING; REVIEW;

BINDING, COMPETITIVE; COMBINATORIAL CHEMISTRY TECHNIQUES; DRUG EVALUATION, PRECLINICAL; HUMANS; MASS SPECTROMETRY; RECEPTORS, G-PROTEIN-COUPLED;

EID: 47049102615     PISSN: 13862073     EISSN: None     Source Type: Journal    
DOI: 10.2174/138620708784911447     Document Type: Review

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